NO20032234L - Nye imidazolderivater, deres fremstilling og anvendelse - Google Patents

Nye imidazolderivater, deres fremstilling og anvendelse

Info

Publication number
NO20032234L
NO20032234L NO20032234A NO20032234A NO20032234L NO 20032234 L NO20032234 L NO 20032234L NO 20032234 A NO20032234 A NO 20032234A NO 20032234 A NO20032234 A NO 20032234A NO 20032234 L NO20032234 L NO 20032234L
Authority
NO
Norway
Prior art keywords
preparation
imidazole derivatives
novel imidazole
novel
derivatives
Prior art date
Application number
NO20032234A
Other languages
English (en)
Other versions
NO326366B1 (no
NO20032234D0 (no
Inventor
Akihiro Tasaka
Takenori Hitaka
Nobuyuki Matsunaga
Masami Kusaka
Mari Adachi
Isao Aoki
Akio Ojida
Original Assignee
Takeda Chemical Industries Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Takeda Chemical Industries Ltd filed Critical Takeda Chemical Industries Ltd
Publication of NO20032234D0 publication Critical patent/NO20032234D0/no
Publication of NO20032234L publication Critical patent/NO20032234L/no
Publication of NO326366B1 publication Critical patent/NO326366B1/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/64—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/08—Drugs for disorders of the urinary system of the prostate
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/28—Antiandrogens
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Endocrinology (AREA)
  • Diabetes (AREA)
  • Urology & Nephrology (AREA)
  • Reproductive Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Steroid Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Medicinal Preparation (AREA)
NO20032234A 2000-11-17 2003-05-16 Imidazolderivater, farmasoytiske preparater inneholdende slike samt deres fremstilling NO326366B1 (no)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
JP2000351780 2000-11-17
JP2001247618 2001-08-17
JP2001336880 2001-11-01
PCT/JP2001/010002 WO2002040484A2 (en) 2000-11-17 2001-11-16 Novel imidazole derivatives, production method thereof and use thereof

Publications (3)

Publication Number Publication Date
NO20032234D0 NO20032234D0 (no) 2003-05-16
NO20032234L true NO20032234L (no) 2003-07-16
NO326366B1 NO326366B1 (no) 2008-11-17

Family

ID=27345219

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20032234A NO326366B1 (no) 2000-11-17 2003-05-16 Imidazolderivater, farmasoytiske preparater inneholdende slike samt deres fremstilling

Country Status (26)

Country Link
US (1) US7141598B2 (no)
EP (2) EP1334106B1 (no)
JP (2) JP3753971B2 (no)
KR (3) KR20080002929A (no)
CN (3) CN100572363C (no)
AR (1) AR034854A1 (no)
AT (2) ATE327237T1 (no)
AU (3) AU2002214296C1 (no)
BR (1) BR0115306B1 (no)
CA (1) CA2429133C (no)
CY (1) CY1105423T1 (no)
DE (1) DE60119963T2 (no)
DK (1) DK1334106T3 (no)
ES (1) ES2260303T3 (no)
HU (1) HU229408B1 (no)
IL (2) IL155624A0 (no)
MX (1) MXPA03004347A (no)
MY (1) MY134929A (no)
NO (1) NO326366B1 (no)
NZ (1) NZ526387A (no)
PE (1) PE20020596A1 (no)
PL (1) PL204934B1 (no)
PT (1) PT1334106E (no)
SI (1) SI1334106T1 (no)
TW (1) TWI306099B (no)
WO (1) WO2002040484A2 (no)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN1639130B (zh) * 2002-01-10 2012-07-18 武田药品工业株式会社 制备稠合咪唑化合物的方法、稳定形式的里福马斯基试剂及其制备方法
WO2004075890A1 (ja) * 2003-02-26 2004-09-10 Takeda Pharmaceutical Company 安定化されたイミダゾール誘導体含有医薬組成物、イミダゾ－ル誘導体の安定化方法
JP4745616B2 (ja) * 2003-02-26 2011-08-10 武田薬品工業株式会社 安定化されたイミダゾール誘導体含有医薬組成物、イミダゾール誘導体の安定化方法
JP4837895B2 (ja) * 2003-03-17 2011-12-14 武田薬品工業株式会社 放出制御組成物
EP1607092A4 (en) * 2003-03-17 2010-12-15 Takeda Pharmaceutical COMPOSITIONS WITH CONTROLLED RELEASE
CN1980917B (zh) * 2004-05-03 2014-02-12 詹森药业有限公司 作为选择性雄激素受体调节剂（sarms）的新的吲哚衍生物
CA2568159A1 (en) * 2004-05-28 2005-12-15 Speedel Experimenta Ag Tetrahydro-imidazo [1,5-a] pyridin derivatives as aldosterone synthase inhibitors
WO2006093353A1 (ja) 2005-03-03 2006-09-08 Takeda Pharmaceutical Company Limited 放出制御組成物
GT200600381A (es) 2005-08-25 2007-03-28 Compuestos organicos
TW200804378A (en) * 2005-12-09 2008-01-16 Speedel Experimenta Ag Organic compounds
US7655683B2 (en) * 2006-02-10 2010-02-02 Janssen Pharmaceutica Nv Imidazolopyrazole derivatives useful as selective androgen receptor modulators
TW200804284A (en) * 2006-03-31 2008-01-16 Speedel Experimenta Ag Process for preparing 6,7-dihydro-5H-imidazo[1,5-a]pyridin-8-one
AR069079A1 (es) * 2007-10-29 2009-12-30 Takeda Pharmaceutical Farmaco para la prevencion o el tratamiento de cancer
CA3121743A1 (en) * 2009-01-15 2010-07-22 Incyte Holdings Corporation Processes for preparing jak inhibitors and related intermediate compounds
AR083916A1 (es) * 2010-11-18 2013-04-10 Takeda Pharmaceutical Metodo para tratar el cancer de mama y cancer de ovarios
CA2831548A1 (en) 2011-04-01 2012-10-04 Takeda Pharmaceutical Company Limited Solid preparation
SG195036A1 (en) * 2011-06-15 2013-12-30 Takeda Pharmaceutical Production method of imidazole derivatives

Family Cites Families (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4728645A (en) * 1982-12-21 1988-03-01 Ciba-Geigy Corporation Substituted imidazo[1,5-A]pyridine derivatives and other substituted bicyclic derivatives, useful as aromatase inhibitors
NZ221729A (en) 1986-09-15 1989-07-27 Janssen Pharmaceutica Nv Imidazolyl methyl-substituted benzimidazole derivatives and pharmaceutical compositions
NZ224288A (en) 1987-04-22 1989-12-21 Merrell Dow Pharma 17b-(cyclopropylamino)androst-5-en-3b-ol and related compounds and methods using these for treatment of non-humans
US5057521A (en) * 1988-10-26 1991-10-15 Ciba-Geigy Corporation Use of bicyclic imidazole compounds for the treatment of hyperaldosteronism
US4966898A (en) 1989-08-15 1990-10-30 Merrell Dow Pharmaceuticals Inc. 4-substituted 17β-(cyclopropylamino)androst-5-en-3β-ol and related compounds useful as C17-20 lyase inhibitors
CA2104234A1 (en) 1991-03-01 1993-07-22 Denis R. Mckay Powder coating method for producing circuit board laminae and the like
CA2127689A1 (en) * 1992-01-27 1993-08-05 Marcel A. C. Janssen Pyrroloimidazolyl and imidazopyridinyl substituted 1h-benzimidazole derivatives as aromatase inhibitors
US5457102A (en) 1994-07-07 1995-10-10 Janssen Pharmaceutica, N.V. Pyrroloimidazolyl and imidazopyridinyl substituted 1H-benzimidazole derivatives
GB2265624B (en) 1992-03-31 1995-04-19 British Tech Group 17-substituted steroids useful in cancer treatment
GB9310635D0 (en) 1993-05-21 1993-07-07 Glaxo Group Ltd Chemical compounds
PL313769A1 (en) 1993-09-30 1996-07-22 Yamanouchi Pharma Co Ltd Azole derivative and pharmaceutical composition thereof
WO1996014090A1 (en) 1994-11-07 1996-05-17 Janssen Pharmaceutica N.V. Compositions comprising carbazoles and cyclodextrins
WO1997000257A1 (en) 1995-06-14 1997-01-03 Yamanouchi Pharmaceutical Co., Ltd. Fused imidazole derivatives and medicinal composition thereof
WO1998037070A1 (en) 1997-02-21 1998-08-27 Takeda Chemical Industries, Ltd. Fused ring compounds, process for producing the same and use thereof
IL133483A0 (en) 1997-10-02 2001-04-30 Yukijirushi Nyugyo Kabushiki K Novel dihydronaphthalene compounds and processes of producing the same
WO1999054309A1 (en) 1998-04-23 1999-10-28 Takeda Chemical Industries, Ltd. Naphthalene derivatives, their production and use
PE20010781A1 (es) * 1999-10-22 2001-08-08 Takeda Chemical Industries Ltd Compuestos 1-(1h-imidazol-4-il)-1-(naftil-2-sustituido)etanol, su produccion y utilizacion

Also Published As

Publication number Publication date
EP1681290B9 (en) 2013-06-19
IL155624A0 (en) 2003-11-23
BR0115306A (pt) 2004-02-10
US7141598B2 (en) 2006-11-28
EP1681290A3 (en) 2006-07-26
KR100725442B1 (ko) 2007-06-07
JP3753971B2 (ja) 2006-03-08
AU2002214296B2 (en) 2005-09-29
EP1681290B1 (en) 2011-11-16
AU2005225035A1 (en) 2005-11-10
CA2429133A1 (en) 2002-05-23
AU2005225035B2 (en) 2007-02-22
KR20080002929A (ko) 2008-01-04
DE60119963D1 (de) 2006-06-29
CN1474819A (zh) 2004-02-11
DE60119963T2 (de) 2006-10-05
PE20020596A1 (es) 2002-08-13
NO326366B1 (no) 2008-11-17
HU229408B1 (hu) 2013-12-30
AU1429602A (en) 2002-05-27
CA2429133C (en) 2009-08-18
NO20032234D0 (no) 2003-05-16
KR100809899B1 (ko) 2008-03-10
MY134929A (en) 2008-01-31
EP1334106B1 (en) 2006-05-24
US20040033935A1 (en) 2004-02-19
CN1680336A (zh) 2005-10-12
HUP0400549A2 (hu) 2004-06-28
CN1900079A (zh) 2007-01-24
KR20050105287A (ko) 2005-11-03
DK1334106T3 (da) 2006-09-18
IL155624A (en) 2006-12-31
NZ526387A (en) 2004-02-27
CN1329394C (zh) 2007-08-01
JP2006045239A (ja) 2006-02-16
JP2003201282A (ja) 2003-07-18
MXPA03004347A (es) 2004-05-04
JP4427496B2 (ja) 2010-03-10
CN100572363C (zh) 2009-12-23
TWI306099B (en) 2009-02-11
HUP0400549A3 (en) 2004-09-28
ES2260303T3 (es) 2006-11-01
PL362766A1 (en) 2004-11-02
EP1681290A2 (en) 2006-07-19
ATE533768T1 (de) 2011-12-15
BR0115306B1 (pt) 2013-12-24
KR20030048156A (ko) 2003-06-18
HK1056168A1 (en) 2004-02-06
WO2002040484A2 (en) 2002-05-23
SI1334106T1 (sl) 2006-10-31
PT1334106E (pt) 2006-08-31
AU2002214296C1 (en) 2006-04-13
AR034854A1 (es) 2004-03-24
ATE327237T1 (de) 2006-06-15
CY1105423T1 (el) 2010-04-28
WO2002040484A3 (en) 2002-09-26
EP1334106A2 (en) 2003-08-13
PL204934B1 (pl) 2010-02-26

Similar Documents

Publication Publication Date Title
NO20015113D0 (no) Nye forbindelser, deres fremstilling og anvendelse
NO20024742D0 (no) Heterocykliske forbindelser, deres fremstilling og anvendelse
NO20015362L (no) Heterocyklisk substituerte benzimidazoler, deres fremstilling og anvendelse derav
NO20021449L (no) Substituerte 2-tio-3,5-dicyano-4-aryl-6-aminopyridiner og deres anvendelse
NO20015156L (no) 5-pyridyl-1,3-azolforbindelser, deres fremstilling og anvendelse
NO20030596L (no) Benzimidazolderivater, deres fremstilling og terapeutiske anvendelse
NO20014603L (no) Tienopyrimidinforbindelser, deres fremstilling og anvendelse
DK1455785T3 (da) Substituerede 2-thio-3,5-dicyano-4-phenyl-6-aminopyridiner og deres anvendelse
NO20012567D0 (no) Azepinoindolderivater, fremstilling og anvendelse derav
NO20030302L (no) Nye heteroarylderivater og deres anvendelse som medikamenter
DK1419150T3 (da) 1-Phenylsulfonyl-1,3-dihydro-2H-indol-2-on-derivater, deres fremstilling og deres terapeutiske anvendelse
NO20031838D0 (no) Benzokazinonderivater, deres fremstilling og anvendelse
NO20025029L (no) Nye epotilonderivater, fremgangsmÕte for fremstilling derav og deres farmasöytiske anvendelse
DK1161434T3 (da) Pyridopyranoazepinderivater, deres fremstilling og terapeutiske anvendelse
NO20032234L (no) Nye imidazolderivater, deres fremstilling og anvendelse
NO20023146L (no) Substituerte fenyl-piperazinderivater, deres fremstilling og anvendelse
DK1043307T3 (da) 3-amino-3-arylpropan-1-ol-derivater, deres fremstilling og anvendelse
NO20052124D0 (no) Nye 1,4-diazabisykloalkanderivater, deres fremstilling og anvendelse
DK1525193T3 (da) Acylaminothiazolderivater, deres fremstilling og deres terapeutiske anvendelse
NO20024107L (no) Tienopyridin derivater, deres fremstilling og anvendelse
NO20025209L (no) Cyklipostiner, deres fremstilling og anvendelse
NO20023188D0 (no) Nye heteroarylderivater, deres fremstilling og anvendelse
NO20001782L (no) 3-amino-3-arylpropan-1-ol-derivater, deres fremstilling og anvendelse
NO20033965D0 (no) Caloporosidderivater, fremgangsmåte for deres fremstilling og deres anvendelse
DK1404663T3 (da) Eurotinoner og derivater deraf, fremgangsmåde til deres fremstilling og anvendelse heraf

Legal Events

Date Code Title Description
MM1K Lapsed by not paying the annual fees