NO20032956D0 - Tricykliske og heterocykliske derivatforbindelser og legemidler inneholdende disse forbindelsene som den aktive bestanddel - Google Patents

Tricykliske og heterocykliske derivatforbindelser og legemidler inneholdende disse forbindelsene som den aktive bestanddel

Info

Publication number: NO20032956D0
Authority: NO; Norway
Prior art keywords: compounds; active ingredient; ring; tricyclic; heterocyclic
Prior art date: 2000-12-28

Application number

NO20032956A

Other languages

English (en)

Other versions

NO326522B1 (no

NO20032956L (no

Inventor

Hisao Nakai

Yoshifumi Kagamiishi

Original Assignee

Ono Pharmaceutical Co

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-12-28

Filing date

2003-06-26

Publication date

2003-06-26

2003-06-26 Application filed by Ono Pharmaceutical Co filed Critical Ono Pharmaceutical Co

2003-06-26 Publication of NO20032956D0 publication Critical patent/NO20032956D0/no

2003-08-28 Publication of NO20032956L publication Critical patent/NO20032956L/no

2008-12-22 Publication of NO326522B1 publication Critical patent/NO326522B1/no

Links

125000000623 heterocyclic group Chemical group 0.000 title abstract 3
239000004480 active ingredient Substances 0.000 title abstract 2
150000001875 compounds Chemical class 0.000 title abstract 2
239000003814 drug Substances 0.000 title 1
229940079593 drug Drugs 0.000 title 1
IJGRMHOSHXDMSA-UHFFFAOYSA-N Atomic nitrogen Chemical compound N#N IJGRMHOSHXDMSA-UHFFFAOYSA-N 0.000 abstract 4
125000002837 carbocyclic group Chemical group 0.000 abstract 2
229910052757 nitrogen Inorganic materials 0.000 abstract 2
208000007848 Alcoholism Diseases 0.000 abstract 1
208000024827 Alzheimer disease Diseases 0.000 abstract 1
208000019901 Anxiety disease Diseases 0.000 abstract 1
108010056643 Corticotropin-Releasing Hormone Receptors Proteins 0.000 abstract 1
102100038018 Corticotropin-releasing factor receptor 1 Human genes 0.000 abstract 1
208000020401 Depressive disease Diseases 0.000 abstract 1
208000030814 Eating disease Diseases 0.000 abstract 1
208000019454 Feeding and Eating disease Diseases 0.000 abstract 1
208000008469 Peptic Ulcer Diseases 0.000 abstract 1
NINIDFKCEFEMDL-UHFFFAOYSA-N Sulfur Chemical compound [S] NINIDFKCEFEMDL-UHFFFAOYSA-N 0.000 abstract 1
125000003342 alkenyl group Chemical group 0.000 abstract 1
125000000217 alkyl group Chemical group 0.000 abstract 1
125000000304 alkynyl group Chemical group 0.000 abstract 1
230000003042 antagnostic effect Effects 0.000 abstract 1
230000036506 anxiety Effects 0.000 abstract 1
QVGXLLKOCUKJST-UHFFFAOYSA-N atomic oxygen Chemical compound [O] QVGXLLKOCUKJST-UHFFFAOYSA-N 0.000 abstract 1
235000014632 disordered eating Nutrition 0.000 abstract 1
206010013663 drug dependence Diseases 0.000 abstract 1
238000000034 method Methods 0.000 abstract 1
229910052760 oxygen Inorganic materials 0.000 abstract 1
239000001301 oxygen Substances 0.000 abstract 1
208000011906 peptic ulcer disease Diseases 0.000 abstract 1
208000028173 post-traumatic stress disease Diseases 0.000 abstract 1
230000002265 prevention Effects 0.000 abstract 1
150000003839 salts Chemical class 0.000 abstract 1
208000011117 substance-related disease Diseases 0.000 abstract 1
239000011593 sulfur Substances 0.000 abstract 1
229910052717 sulfur Inorganic materials 0.000 abstract 1
208000011580 syndromic disease Diseases 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
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- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
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- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/12—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains three hetero rings
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- C07D495/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
- C07D495/14—Ortho-condensed systems

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NO20032956A 2000-12-28 2003-06-26 Tricykliske og heterocykliske derivatforbindelser og farmasoytiske preparater inneholdende disse forbindelsene som den aktive bestanddel NO326522B1 (no)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
JP2000402517		2000-12-28
PCT/JP2001/011581 WO2002053565A1 (en)	2000-12-28	2001-12-27	Tricyclic and heterocyclic derivative compounds and drugs containing these compounds as the active ingredient

Publications (3)

Publication Number	Publication Date
NO20032956D0 true NO20032956D0 (no)	2003-06-26
NO20032956L NO20032956L (no)	2003-08-28
NO326522B1 NO326522B1 (no)	2008-12-22

Family

ID=18866787

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO20032956A NO326522B1 (no)	2000-12-28	2003-06-26	Tricykliske og heterocykliske derivatforbindelser og farmasoytiske preparater inneholdende disse forbindelsene som den aktive bestanddel

Country Status (24)

Country	Link
US (3)	US7034153B2 (no)
EP (2)	EP1832590B8 (no)
JP (2)	JP3528968B2 (no)
KR (1)	KR100843281B1 (no)
CN (2)	CN1274690C (no)
AT (2)	ATE375345T1 (no)
AU (1)	AU2002226674B2 (no)
BR (1)	BR0116609A (no)
CA (1)	CA2432148C (no)
CZ (1)	CZ20031777A3 (no)
DE (1)	DE60130924T2 (no)
DK (1)	DK1354884T3 (no)
ES (2)	ES2369837T3 (no)
HU (1)	HUP0303653A3 (no)
IL (2)	IL156609A0 (no)
MX (1)	MXPA03005913A (no)
NO (1)	NO326522B1 (no)
NZ (1)	NZ526712A (no)
PL (1)	PL363381A1 (no)
PT (1)	PT1354884E (no)
RU (1)	RU2291869C2 (no)
TW (1)	TWI293630B (no)
WO (1)	WO2002053565A1 (no)
ZA (1)	ZA200305003B (no)

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US6562965B1 (en) *	2000-07-06	2003-05-13	Bristol-Myers Squibb Pharma Company	Convergent synthesis of α-aryl-β-ketonitriles
ATE375345T1 (de) *	2000-12-28	2007-10-15	Ono Pharmaceutical Co	Cyclopenta(d)pyrazolo(1,5-a)pyrimidin-verbindun als crf-rezeptor antagonist
UA80295C2 (en) *	2002-09-06	2007-09-10	Biogen Inc	Pyrazolopyridines and using the same
US7129239B2 (en)	2002-10-28	2006-10-31	Pfizer Inc.	Purine compounds and uses thereof
US7247628B2 (en)	2002-12-12	2007-07-24	Pfizer, Inc.	Cannabinoid receptor ligands and uses thereof
US7329658B2 (en)	2003-02-06	2008-02-12	Pfizer Inc	Cannabinoid receptor ligands and uses thereof
US7176210B2 (en)	2003-02-10	2007-02-13	Pfizer Inc.	Cannabinoid receptor ligands and uses thereof
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Publication number	Publication date
EP1354884B1 (en)	2007-10-10
EP1832590A2 (en)	2007-09-12
KR20030070593A (ko)	2003-08-30
US20060122392A1 (en)	2006-06-08
CA2432148A1 (en)	2002-07-11
IL156609A (en)	2010-02-17
JP2004083597A (ja)	2004-03-18
KR100843281B1 (ko)	2008-07-09
TWI293630B (en)	2008-02-21
BR0116609A (pt)	2005-02-15
IL156609A0 (en)	2004-01-04
HUP0303653A2 (hu)	2004-03-01
EP1354884A4 (en)	2005-09-07
CZ20031777A3 (cs)	2003-10-15
CN1896076A (zh)	2007-01-17
RU2291869C2 (ru)	2007-01-20
US7034153B2 (en)	2006-04-25
JP4217968B2 (ja)	2009-02-04
US7459459B2 (en)	2008-12-02
ATE375345T1 (de)	2007-10-15
DE60130924T2 (de)	2008-07-17
PL363381A1 (en)	2004-11-15
WO2002053565A1 (en)	2002-07-11
HUP0303653A3 (en)	2006-05-29
ES2294047T3 (es)	2008-04-01
US20040072833A1 (en)	2004-04-15
NO326522B1 (no)	2008-12-22
CA2432148C (en)	2011-01-18
CN1274690C (zh)	2006-09-13
EP1832590A3 (en)	2007-11-14
EP1832590B8 (en)	2012-04-25
EP1832590B1 (en)	2011-09-28
ES2369837T3 (es)	2011-12-07
ZA200305003B (en)	2005-07-27
ATE526330T1 (de)	2011-10-15
US7807688B2 (en)	2010-10-05
EP1354884A1 (en)	2003-10-22
US20090137604A1 (en)	2009-05-28
PT1354884E (pt)	2007-12-24
JP3528968B2 (ja)	2004-05-24
DE60130924D1 (de)	2007-11-22
CN1491225A (zh)	2004-04-21
NZ526712A (en)	2005-03-24
NO20032956L (no)	2003-08-28
AU2002226674B2 (en)	2007-03-22
MXPA03005913A (es)	2005-04-19
JPWO2002053565A1 (ja)	2004-05-13
DK1354884T3 (da)	2008-03-03

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FI872864A0 (fi)	1987-06-29	Menetelmä farmaseuttisesti aktiivisten bentsimidatsolijohdannaisten valmistamiseksi
BG106095A (bg)	2002-06-28	Нови лекарствени състави на базата на антихолинергично активни съединения и бета-миметици
EP1595867A4 (en)	2008-05-21	PIPERIDINE DERIVATIVES AS AN ACTIVE ANTAGONIST AT THE RECIPE OF MELANIN CONCENTRATING HORMONE
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DK0842923T3 (da)	2006-06-19	Pyrrolderivater og lægemiddelpræparat
ATE78470T1 (de)	1992-08-15	Imidazolin-derivate und verfahren zu deren herstellung.
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NO941451D0 (no)	1994-04-21	Oksazolinderivat
EP1419771A4 (en)	2004-11-03	AGENTS FOR THE PREVENTION AND / OR TREATMENT OF DISEASES THAT ARE ATTRIBUTED TO ARTERIOSCLEROTIC EFFECT
EP1134216A4 (en)	2002-01-30	AGENTS AGAINST MEDICINE-RESISTANT BACTERIA AND ANTI-CHLAMYDIA AGENTS
DE60009517D1 (de)	2004-05-06	A-500359-derivate
ATE294780T1 (de)	2005-05-15	Arylpiperidin- und aryl-1,2,5,6- tetrahydropyridinamid-derivate mit 5ht1a rezeptor aktivität
UA81610C2 (ru)	2008-01-25	Изохинолиновые соединения, способ их получения и фармацевтическая композиция, которая их содержит
ATE319452T1 (de)	2006-03-15	Arzneimittel gegen essstörungen
DE69722630D1 (de)	2003-07-10	Therapeutisches mittel zur behandlung von nierenerkrankungen
SE8702697L (sv)	1988-01-02	Framstellning av lekemedel for behandling av ischemiska kerlsjukdomar
JPH0386823A (ja)	1991-04-11	抗うつ剤