NO20033883L - Heterosykliske derivater for behandling av kreft og andre proliferative sykdommer - Google Patents

Heterosykliske derivater for behandling av kreft og andre proliferative sykdommer

Info

Publication number
NO20033883L
NO20033883L NO20033883A NO20033883A NO20033883L NO 20033883 L NO20033883 L NO 20033883L NO 20033883 A NO20033883 A NO 20033883A NO 20033883 A NO20033883 A NO 20033883A NO 20033883 L NO20033883 L NO 20033883L
Authority
NO
Norway
Prior art keywords
cancer
treatment
proliferative diseases
heterocyclic derivatives
heterocyclic
Prior art date
Application number
NO20033883A
Other languages
English (en)
Norwegian (no)
Other versions
NO20033883D0 (no
Inventor
Magnus Pfahl
Hussein A Al-Shamma
Andrea Fanjul
David P M Pleynet
Lyle W Spruce
Torsten R Wiemann
Jason B Ibarra
Catherine Tachdjian
Original Assignee
Incyte San Diego Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Incyte San Diego Inc filed Critical Incyte San Diego Inc
Publication of NO20033883D0 publication Critical patent/NO20033883D0/no
Publication of NO20033883L publication Critical patent/NO20033883L/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D277/00Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/02Antineoplastic agents specific for leukemia
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D277/00Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/34Oxygen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/06Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/10Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing aromatic rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Hematology (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
NO20033883A 2001-03-07 2003-09-02 Heterosykliske derivater for behandling av kreft og andre proliferative sykdommer NO20033883L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US27475101P 2001-03-07 2001-03-07
PCT/US2002/007001 WO2002072009A2 (fr) 2001-03-07 2002-03-07 Derives heterocycliques pour le traitement du cancer et d'autres maladies proliferatives

Publications (2)

Publication Number Publication Date
NO20033883D0 NO20033883D0 (no) 2003-09-02
NO20033883L true NO20033883L (no) 2003-11-05

Family

ID=23049469

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20033883A NO20033883L (no) 2001-03-07 2003-09-02 Heterosykliske derivater for behandling av kreft og andre proliferative sykdommer

Country Status (12)

Country Link
US (1) US7153875B2 (fr)
EP (1) EP1385465A4 (fr)
JP (1) JP2005506290A (fr)
AU (1) AU2002252227A1 (fr)
BR (1) BR0207846A (fr)
CA (1) CA2440184A1 (fr)
EA (1) EA200300982A1 (fr)
IL (1) IL157740A0 (fr)
MX (1) MXPA03008117A (fr)
NO (1) NO20033883L (fr)
PL (1) PL373912A1 (fr)
WO (1) WO2002072009A2 (fr)

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WO2002072009A2 (fr) 2001-03-07 2002-09-19 Maxia Pharmaceuticals, Inc. Derives heterocycliques pour le traitement du cancer et d'autres maladies proliferatives
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EP1456187A4 (fr) * 2001-11-15 2005-02-09 Incyte San Diego Inc Heterocycles n-substitues pour le traitement de l'hypercholesterolemie, de la dyslipidemie et autres troubles du metabolisme, du cancer et de pathologies diverses
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US7196108B2 (en) * 2002-03-08 2007-03-27 Incyte San Diego Inc. Bicyclic heterocycles for the treatment of diabetes and other diseases
CA2520172C (fr) * 2003-03-27 2012-10-02 Lankenau Institute For Medical Research Nouvelles methodes pour le traitement du cancer avec un inhibiteur de l'indoleamine-2,3-dioxygenase
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AU2008326381B2 (en) * 2007-11-21 2014-10-23 Decode Genetics Ehf Biaryl PDE4 inhibitors for treating inflammation
CN102558088A (zh) * 2010-12-31 2012-07-11 中国科学院上海药物研究所 联苯亚甲基-2-硫代-4-噻唑酮类化合物及其制备方法和用途
KR102922092B1 (ko) * 2021-12-21 2026-02-03 주식회사 메디픽바이오 치환된 티아졸리딘디온 유도체 화합물 및 이를 포함하는 암의 예방 또는 치료용 약학적 조성물
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EP1456187A4 (fr) 2001-11-15 2005-02-09 Incyte San Diego Inc Heterocycles n-substitues pour le traitement de l'hypercholesterolemie, de la dyslipidemie et autres troubles du metabolisme, du cancer et de pathologies diverses
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Also Published As

Publication number Publication date
EP1385465A2 (fr) 2004-02-04
CA2440184A1 (fr) 2002-09-19
MXPA03008117A (es) 2004-11-12
EP1385465A4 (fr) 2005-09-07
PL373912A1 (en) 2005-09-19
BR0207846A (pt) 2005-09-13
WO2002072009A3 (fr) 2003-10-16
US7153875B2 (en) 2006-12-26
US20020143182A1 (en) 2002-10-03
JP2005506290A (ja) 2005-03-03
IL157740A0 (en) 2004-03-28
NO20033883D0 (no) 2003-09-02
AU2002252227A1 (en) 2002-09-24
EA200300982A1 (ru) 2004-12-30
WO2002072009A2 (fr) 2002-09-19

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