NO20041008L - Karbazolderivater og anvendelse derav som NPY5 reseptor antagonister - Google Patents

Karbazolderivater og anvendelse derav som NPY5 reseptor antagonister

Info

Publication number
NO20041008L
NO20041008L NO20041008A NO20041008A NO20041008L NO 20041008 L NO20041008 L NO 20041008L NO 20041008 A NO20041008 A NO 20041008A NO 20041008 A NO20041008 A NO 20041008A NO 20041008 L NO20041008 L NO 20041008L
Authority
NO
Norway
Prior art keywords
receptor antagonists
carbazole derivatives
npy5 receptor
npy5
carbazole
Prior art date
Application number
NO20041008A
Other languages
English (en)
Inventor
Kevin Michael Foote
Michael Howard Block
Wayne Brailsford
Original Assignee
Astrazeneca Ab Global Ip
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab Global Ip filed Critical Astrazeneca Ab Global Ip
Publication of NO20041008L publication Critical patent/NO20041008L/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/06Antihyperlipidemics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Anesthesiology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
NO20041008A 2001-09-11 2004-03-10 Karbazolderivater og anvendelse derav som NPY5 reseptor antagonister NO20041008L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0121941.9A GB0121941D0 (en) 2001-09-11 2001-09-11 Chemical compounds
PCT/GB2002/004109 WO2003022849A1 (en) 2001-09-11 2002-09-09 Carbazole derivatives and their use as npy5 receptor antagonists

Publications (1)

Publication Number Publication Date
NO20041008L true NO20041008L (no) 2004-03-10

Family

ID=9921890

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20041008A NO20041008L (no) 2001-09-11 2004-03-10 Karbazolderivater og anvendelse derav som NPY5 reseptor antagonister

Country Status (14)

Country Link
US (1) US7408064B2 (no)
EP (1) EP1427729A1 (no)
JP (1) JP2005516892A (no)
KR (1) KR20040036939A (no)
CN (1) CN1653067A (no)
BR (1) BR0212484A (no)
CA (1) CA2459973A1 (no)
GB (1) GB0121941D0 (no)
IL (1) IL160771A0 (no)
MX (1) MXPA04002338A (no)
NO (1) NO20041008L (no)
NZ (1) NZ531678A (no)
WO (1) WO2003022849A1 (no)
ZA (1) ZA200401956B (no)

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EA201592263A1 (ru) 2013-06-05 2016-05-31 Синерджи Фармасьютикалз, Инк. Ультрачистые агонисты гуанилатциклазы c, способ их получения и использования
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Also Published As

Publication number Publication date
EP1427729A1 (en) 2004-06-16
ZA200401956B (en) 2005-04-15
MXPA04002338A (es) 2004-06-29
IL160771A0 (en) 2004-08-31
CA2459973A1 (en) 2003-03-20
JP2005516892A (ja) 2005-06-09
KR20040036939A (ko) 2004-05-03
BR0212484A (pt) 2004-08-24
WO2003022849A1 (en) 2003-03-20
CN1653067A (zh) 2005-08-10
GB0121941D0 (en) 2001-10-31
US20050065157A1 (en) 2005-03-24
US7408064B2 (en) 2008-08-05
NZ531678A (en) 2005-09-30

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