NO20041975L - Bicyklisk oksopyridin og oksopyrimidinderivater - Google Patents

Bicyklisk oksopyridin og oksopyrimidinderivater

Info

Publication number: NO20041975L
Authority: NO; Norway
Prior art keywords: oxopyridine; bicyclic; oxopyrimidine; derivatives; oxopyrimidine derivatives
Prior art date: 2001-10-16

Application number

NO20041975A

Other languages

English (en)

Norwegian (no)

Other versions

NO20041975D0 (no

Inventor

Jeremy Martin Davis

Daniel Christopher Brookings

Barry John Langham

Original Assignee

Celltech R&D Ltd

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2001-10-16

Filing date

2004-05-13

Publication date

2005-07-16

2004-05-13 Application filed by Celltech R&D Ltd filed Critical Celltech R&D Ltd

2004-05-13 Publication of NO20041975D0 publication Critical patent/NO20041975D0/no

2005-07-16 Publication of NO20041975L publication Critical patent/NO20041975L/no

Links

125000002619 bicyclic group Chemical group 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
- A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
- A—HUMAN NECESSITIES
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- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
Public Health (AREA)
Pharmacology & Pharmacy (AREA)
Veterinary Medicine (AREA)
Animal Behavior & Ethology (AREA)
Medicinal Chemistry (AREA)
General Health & Medical Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Immunology (AREA)
Physical Education & Sports Medicine (AREA)
Oncology (AREA)
Virology (AREA)
Neurology (AREA)
Diabetes (AREA)
Communicable Diseases (AREA)
Rheumatology (AREA)
Orthopedic Medicine & Surgery (AREA)
Neurosurgery (AREA)
Biomedical Technology (AREA)
Cardiology (AREA)
Pulmonology (AREA)
Hematology (AREA)
Molecular Biology (AREA)
Heart & Thoracic Surgery (AREA)
Endocrinology (AREA)
Hospice & Palliative Care (AREA)
Dermatology (AREA)
Urology & Nephrology (AREA)
Psychology (AREA)
Tropical Medicine & Parasitology (AREA)
Pain & Pain Management (AREA)
Biotechnology (AREA)
Vascular Medicine (AREA)

NO20041975A 2001-10-16 2004-05-13 Bicyklisk oksopyridin og oksopyrimidinderivater NO20041975L (no)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
GBGB0124848.3A GB0124848D0 (en)	2001-10-16	2001-10-16	Chemical compounds
PCT/GB2002/004680 WO2003033502A1 (en)	2001-10-16	2002-10-16	Bicyclic oxopyridine and oxopyrimidine derivatives

Publications (2)

Publication Number	Publication Date
NO20041975D0 NO20041975D0 (no)	2004-05-13
NO20041975L true NO20041975L (no)	2005-07-16

Family

ID=9923964

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO20041975A NO20041975L (no)	2001-10-16	2004-05-13	Bicyklisk oksopyridin og oksopyrimidinderivater

Country Status (17)

Country	Link
US (1)	US7176215B2 (pl)
EP (1)	EP1438313A1 (pl)
JP (1)	JP2005505627A (pl)
KR (1)	KR20040062565A (pl)
CN (1)	CN1310921C (pl)
AU (1)	AU2002336172B2 (pl)
CA (1)	CA2462147A1 (pl)
EA (1)	EA007957B1 (pl)
GB (1)	GB0124848D0 (pl)
HU (1)	HUP0401718A3 (pl)
IL (1)	IL161384A0 (pl)
MX (1)	MXPA04003450A (pl)
NO (1)	NO20041975L (pl)
NZ (1)	NZ532713A (pl)
PL (1)	PL369867A1 (pl)
WO (1)	WO2003033502A1 (pl)
ZA (1)	ZA200402803B (pl)

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GB0217757D0 (en)	2002-07-31	2002-09-11	Glaxo Group Ltd	Novel compounds
GB0218800D0 (en) *	2002-08-13	2002-09-18	Celltech R&D Ltd	Chemical compounds
GB0222743D0 (en) *	2002-10-01	2002-11-06	Celltech R&D Ltd	Chemical compounds
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WO2005042540A1 (en) *	2003-10-24	2005-05-12	Celltech R & D Limited	Thieno-pyridinone derivatives as kinase inhibitors
JP2007517052A (ja) *	2003-12-23	2007-06-28	ノバルティスアクチエンゲゼルシャフト	二環式ヘテロ環式ｐ−３８キナーゼ阻害剤
GB0402138D0 (en)	2004-01-30	2004-03-03	Smithkline Beecham Corp	Novel compounds
GB0402140D0 (en)	2004-01-30	2004-03-03	Smithkline Beecham Corp	Novel compounds
GB0402143D0 (en) *	2004-01-30	2004-03-03	Smithkline Beecham Corp	Novel compounds
GB0402137D0 (en)	2004-01-30	2004-03-03	Smithkline Beecham Corp	Novel compounds
WO2006010082A1 (en)	2004-07-08	2006-01-26	Arqule, Inc.	1,4-disubstituted naphtalenes as inhibitors of p38 map kinase
CA2584368A1 (en)	2004-10-19	2006-04-27	Arqule, Inc.	Synthesis of imidazooxazole and imidazothiazole inhibitors of p38 map kinase
ATE476434T1 (de) *	2004-12-09	2010-08-15	Xention Ltd	Thienopyridinderivate als kaliumkanalinhibitoren
AP2007004244A0 (en)	2005-05-10	2007-12-31	Intermune Inc	Method of modulating stress-activated protein kinase system
GB0512429D0 (en) *	2005-06-17	2005-07-27	Smithkline Beecham Corp	Novel compound
US20110034495A1 (en) *	2005-11-23	2011-02-10	Intermune, Inc.	Method of Modulating Stress-Activated Protein Kinase System
JP2009520015A (ja) *	2005-12-20	2009-05-21	リヒターゲデオンニュルト	新規な化合物
HUP0501168A3 (en) *	2005-12-20	2007-10-29	Richter Gedeon Nyrt	2-(acyl, oxycarbonyl or aminocarbonyl)-3-phenyl-thieno[2,3-b]pyridines, process for their preparation, their use and pharmaceutical composition containing them
ES2301380B1 (es)	2006-08-09	2009-06-08	Laboratorios Almirall S.A.	Nuevos derivados de 1,7-naftiridina.
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EP2113503A1 (en)	2008-04-28	2009-11-04	Laboratorios Almirall, S.A.	New substituted indolin-2-one derivatives and their use as p39 mitogen-activated kinase inhibitors
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US5219864A (en) *	1991-03-12	1993-06-15	Kyowa Hakko Kogyo Co., Ltd.	Thienopyridine derivatives
CA2121148A1 (en) *	1992-08-19	1994-03-03	Otsuka Pharmaceutical Co., Ltd.	Apoptosis regulator
JPH0776586A (ja) *	1993-07-16	1995-03-20	Yoshitomi Pharmaceut Ind Ltd	ピリジン化合物
DE4444815A1 (de) *	1994-12-15	1996-06-20	Merck Patent Gmbh	Thienopyridone
JPH0959276A (ja) *	1995-08-11	1997-03-04	Kumiai Chem Ind Co Ltd	縮合ヘテロ環誘導体及び除草剤
AU4429799A (en) *	1998-06-12	1999-12-30	Vertex Pharmaceuticals Incorporated	Inhibitors of p38
GB2350111A (en) *	1999-05-17	2000-11-22	Bayer Ag	Oligohydroxyl substituted 3-urea-benzofuran and pyridofuran derivatives
AU778042B2 (en) *	1999-10-19	2004-11-11	Merck & Co., Inc.	Tyrosine kinase inhibitors
WO2001037837A1 (en)	1999-11-23	2001-05-31	Smithkline Beecham Corporation	3,4-DIHYDRO-(1H)-QUINAZOLIN-2-ONES AND THEIR USE AS CSBP/p38 KINASE INHIBITORS
AR030053A1 (es)	2000-03-02	2003-08-13	Smithkline Beecham Corp	1h-pirimido [4,5-d] pirimidin-2-onas y sales, composiciones farmaceuticas, uso para la fabricacion de un medicamento y procedimiento para producirlas
AR030273A1 (es) *	2000-03-10	2003-08-20	Smithkline Beecham Corp	Compuestos de hidroxifenil urea sustituidos con sulfonamidas, composiciones farmaceuticas que los comprenden, y uso de los mismos en la fabricacion de medicamentos para tratar una enfermedad mediada por una quimioquina

2001
- 2001-10-16 GB GBGB0124848.3A patent/GB0124848D0/en not_active Ceased
2002
- 2002-10-16 JP JP2003536241A patent/JP2005505627A/ja not_active Abandoned
- 2002-10-16 CN CNB02825094XA patent/CN1310921C/zh not_active Expired - Fee Related
- 2002-10-16 EP EP02770072A patent/EP1438313A1/en not_active Withdrawn
- 2002-10-16 HU HU0401718A patent/HUP0401718A3/hu unknown
- 2002-10-16 KR KR10-2004-7005544A patent/KR20040062565A/ko not_active Ceased
- 2002-10-16 MX MXPA04003450A patent/MXPA04003450A/es not_active Application Discontinuation
- 2002-10-16 EA EA200400550A patent/EA007957B1/ru not_active IP Right Cessation
- 2002-10-16 WO PCT/GB2002/004680 patent/WO2003033502A1/en not_active Ceased
- 2002-10-16 PL PL02369867A patent/PL369867A1/pl not_active Application Discontinuation
- 2002-10-16 NZ NZ532713A patent/NZ532713A/en unknown
- 2002-10-16 US US10/492,466 patent/US7176215B2/en not_active Expired - Fee Related
- 2002-10-16 IL IL16138402A patent/IL161384A0/xx unknown
- 2002-10-16 CA CA002462147A patent/CA2462147A1/en not_active Abandoned
- 2002-10-16 AU AU2002336172A patent/AU2002336172B2/en not_active Ceased
2004
- 2004-04-13 ZA ZA200402803A patent/ZA200402803B/en unknown
- 2004-05-13 NO NO20041975A patent/NO20041975L/no not_active Application Discontinuation

Also Published As

Publication number	Publication date
US7176215B2 (en)	2007-02-13
MXPA04003450A (es)	2004-07-16
EA200400550A1 (ru)	2004-10-28
HUP0401718A2 (hu)	2004-12-28
HUP0401718A3 (en)	2008-07-28
ZA200402803B (en)	2006-06-28
US20040254200A1 (en)	2004-12-16
EA007957B1 (ru)	2007-02-27
JP2005505627A (ja)	2005-02-24
KR20040062565A (ko)	2004-07-07
NO20041975D0 (no)	2004-05-13
NZ532713A (en)	2005-10-28
EP1438313A1 (en)	2004-07-21
CA2462147A1 (en)	2003-04-24
PL369867A1 (pl)	2005-05-02
IL161384A0 (en)	2004-09-27
GB0124848D0 (en)	2001-12-05
WO2003033502A1 (en)	2003-04-24
AU2002336172B2 (en)	2007-09-13
CN1604901A (zh)	2005-04-06
CN1310921C (zh)	2007-04-18

Legal Events

Date	Code	Title	Description
2009-05-25	FC2A	Withdrawal, rejection or dismissal of laid open patent application

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