NO20044005L - HFA-Suspensjonsformulering inneholdende et anticholinergicum - Google Patents

HFA-Suspensjonsformulering inneholdende et anticholinergicum

Info

Publication number: NO20044005L
Authority: NO; Norway
Prior art keywords: anticholinergic; hfa; formulation containing; suspension formulation; hfa suspension
Prior art date: 2002-03-28

Application number

NO20044005A

Other languages

English (en)

Inventor

Christel Schmelzer

Original Assignee

Boehringer Ingelheim Pharma

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2002-03-28

Filing date

2004-09-23

Publication date

2004-10-05

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=28050989&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO20044005(L) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

2004-09-23 Application filed by Boehringer Ingelheim Pharma filed Critical Boehringer Ingelheim Pharma

2004-10-05 Publication of NO20044005L publication Critical patent/NO20044005L/no

Links

230000001078 anti-cholinergic effect Effects 0.000 title abstract 2
239000000725 suspension Substances 0.000 title abstract 2
238000009472 formulation Methods 0.000 title 1
239000000203 mixture Substances 0.000 title 1
OFBQJSOFQDEBGM-UHFFFAOYSA-N n-pentane Natural products CCCCC OFBQJSOFQDEBGM-UHFFFAOYSA-N 0.000 abstract 3
LCGLNKUTAGEVQW-UHFFFAOYSA-N Dimethyl ether Chemical compound COC LCGLNKUTAGEVQW-UHFFFAOYSA-N 0.000 abstract 2
ATUOYWHBWRKTHZ-UHFFFAOYSA-N Propane Chemical compound CCC ATUOYWHBWRKTHZ-UHFFFAOYSA-N 0.000 abstract 2
RWRIWBAIICGTTQ-UHFFFAOYSA-N difluoromethane Chemical compound FCF RWRIWBAIICGTTQ-UHFFFAOYSA-N 0.000 abstract 2
239000007789 gas Substances 0.000 abstract 2
NNPPMTNAJDCUHE-UHFFFAOYSA-N isobutane Chemical compound CC(C)C NNPPMTNAJDCUHE-UHFFFAOYSA-N 0.000 abstract 2
QWTDNUCVQCZILF-UHFFFAOYSA-N isopentane Chemical compound CCC(C)C QWTDNUCVQCZILF-UHFFFAOYSA-N 0.000 abstract 2
CRSOQBOWXPBRES-UHFFFAOYSA-N neopentane Chemical compound CC(C)(C)C CRSOQBOWXPBRES-UHFFFAOYSA-N 0.000 abstract 2
239000003380 propellant Substances 0.000 abstract 2
YFMFNYKEUDLDTL-UHFFFAOYSA-N 1,1,1,2,3,3,3-heptafluoropropane Chemical compound FC(F)(F)C(F)C(F)(F)F YFMFNYKEUDLDTL-UHFFFAOYSA-N 0.000 abstract 1
LVGUZGTVOIAKKC-UHFFFAOYSA-N 1,1,1,2-tetrafluoroethane Chemical compound FCC(F)(F)F LVGUZGTVOIAKKC-UHFFFAOYSA-N 0.000 abstract 1
VOPWNXZWBYDODV-UHFFFAOYSA-N Chlorodifluoromethane Chemical compound FC(F)Cl VOPWNXZWBYDODV-UHFFFAOYSA-N 0.000 abstract 1
230000001088 anti-asthma Effects 0.000 abstract 1
230000003110 anti-inflammatory effect Effects 0.000 abstract 1
239000000924 antiasthmatic agent Substances 0.000 abstract 1
239000001273 butane Substances 0.000 abstract 1
AFABGHUZZDYHJO-UHFFFAOYSA-N dimethyl butane Natural products CCCC(C)C AFABGHUZZDYHJO-UHFFFAOYSA-N 0.000 abstract 1
230000000694 effects Effects 0.000 abstract 1
239000001282 iso-butane Substances 0.000 abstract 1
230000010534 mechanism of action Effects 0.000 abstract 1
IJDNQMDRQITEOD-UHFFFAOYSA-N n-butane Chemical compound CCCC IJDNQMDRQITEOD-UHFFFAOYSA-N 0.000 abstract 1
239000001294 propane Substances 0.000 abstract 1
MQLXPRBEAHBZTK-SEINRUQRSA-M tiotropium bromide hydrate Chemical compound O.[Br-].C[N+]1(C)[C@H]2C[C@@H](C[C@@H]1[C@H]1O[C@@H]21)OC(=O)C(O)(c1cccs1)c1cccs1 MQLXPRBEAHBZTK-SEINRUQRSA-M 0.000 abstract 1

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/10—Dispersions; Emulsions
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/007—Pulmonary tract; Aromatherapy
- A61K9/0073—Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy
- A61K9/008—Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy comprising drug dissolved or suspended in liquid propellant for inhalation via a pressurized metered dose inhaler [MDI]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/439—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom the ring forming part of a bridged ring system, e.g. quinuclidine
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/10—Dispersions; Emulsions
- A61K9/12—Aerosols; Foams
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Animal Behavior & Ethology (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Medicinal Chemistry (AREA)
Epidemiology (AREA)
Pulmonology (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Dispersion Chemistry (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Organic Chemistry (AREA)
Otolaryngology (AREA)
Medicinal Preparation (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Agricultural Chemicals And Associated Chemicals (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

NO20044005A 2002-03-28 2004-09-23 HFA-Suspensjonsformulering inneholdende et anticholinergicum NO20044005L (no)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
DE10214263A DE10214263A1 (de)	2002-03-28	2002-03-28	HFA-Suspensionsformulierungen enthaltend ein Anticholinergikum
PCT/EP2003/002898 WO2003082252A1 (de)	2002-03-28	2003-03-20	Hfa-suspensionsformulierungen enthaltend ein anticholinergikum

Publications (1)

Publication Number	Publication Date
NO20044005L true NO20044005L (no)	2004-10-05

Family

ID=28050989

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO20044005A NO20044005L (no)	2002-03-28	2004-09-23	HFA-Suspensjonsformulering inneholdende et anticholinergicum

Country Status (26)

Country	Link
EP (2)	EP1695701B1 (no)
JP (1)	JP4480401B2 (no)
KR (1)	KR101066801B1 (no)
CN (1)	CN1329023C (no)
AT (1)	ATE339953T1 (no)
AU (1)	AU2003209743B2 (no)
BR (1)	BR0308764A (no)
CA (1)	CA2479640C (no)
CY (1)	CY1105543T1 (no)
DE (2)	DE10214263A1 (no)
DK (1)	DK1492513T3 (no)
EA (1)	EA007239B1 (no)
EC (1)	ECSP045321A (no)
ES (1)	ES2273020T3 (no)
HR (1)	HRP20040889B1 (no)
IL (2)	IL163697A0 (no)
ME (1)	ME00247B (no)
MX (1)	MXPA04009337A (no)
NO (1)	NO20044005L (no)
NZ (1)	NZ536043A (no)
PL (1)	PL371296A1 (no)
PT (1)	PT1492513E (no)
RS (1)	RS52178B (no)
UA (1)	UA78557C2 (no)
WO (1)	WO2003082252A1 (no)
ZA (1)	ZA200405638B (no)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
BRPI0512878A (pt) †	2004-07-02	2008-04-15	Boehringer Ingelheim Int	formulações de suspensão de aerossol, com tg 227 ea ou tg 134 a como agente propulsor
US20070086957A1 (en) *	2005-10-10	2007-04-19	Thierry Bouyssou	Combination of medicaments for the treatment of respiratory diseases
GB201200504D0 (en) *	2011-12-19	2012-02-22	Teva Branded Pharmaceutical Prod R & D Inc	An inhaler
GB201200525D0 (en)	2011-12-19	2012-02-29	Teva Branded Pharmaceutical Prod R & D Inc	An inhalable medicament
EP2705838A1 (en) *	2012-09-06	2014-03-12	Xspray Microparticles Ab	Tiotropium preparations
CA2885767A1 (en) *	2012-10-23	2014-05-01	Cipla Limited	Pharmaceutical composition
US10034866B2 (en)	2014-06-19	2018-07-31	Teva Branded Pharmaceutical Products R&D, Inc.	Inhalable medicament comprising tiotropium
CN107056629B (zh) *	2017-04-27	2019-04-30	河北科技大学	一种无水卤化胆碱及其衍生物单晶的制备方法

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5610163A (en) *	1989-09-16	1997-03-11	Boehringer Ingelheim Gmbh	Esters of thienyl carboxylic acids and amino alcohols and their quaternization products
GB2326334A (en) *	1997-06-13	1998-12-23	Chiesi Farma Spa	Pharmaceutical aerosol compositions
ATE234604T1 (de) *	1998-08-04	2003-04-15	Jago Res Ag	Medizinische aerosolformulierungen
DZ2947A1 (fr) *	1998-11-25	2004-03-15	Chiesi Farma Spa	Inhalateur à compteur de dose sous pression.
DE19921693A1 (de) *	1999-05-12	2000-11-16	Boehringer Ingelheim Pharma	Neuartige Arzneimittelkompositionen auf der Basis von anticholinergisch wirksamen Verbindungen und ß-Mimetika
IT1317846B1 (it) *	2000-02-22	2003-07-15	Chiesi Farma Spa	Formulazioni contenenti un farmaco anticolinergico per il trattamentodella broncopneumopatia cronica ostruttiva.
GB0009605D0 (en) *	2000-04-18	2000-06-07	Glaxo Group Ltd	Medicaments
AU2002214996B2 (en) *	2000-10-12	2007-03-15	Boehringer Ingelheim Pharma Gmbh & Co. Kg	Crystalline monohydrate, method for producing the same and the use thereof in the production of a medicament
CA2733294C (en) *	2000-10-31	2011-12-20	Boehringer Ingelheim Pharma Gmbh & Co. Kg	Pharmaceutical combination of a tiotropium salt and ciclesonide
DE10056104A1 (de) *	2000-11-13	2002-05-23	Boehringer Ingelheim Pharma	Neue Arzneimittelkompositionen auf der Basis von Tiotropiumsalzen und Salzen des Salmeterols

2002
- 2002-03-28 DE DE10214263A patent/DE10214263A1/de not_active Withdrawn
2003
- 2003-03-20 CN CNB038072491A patent/CN1329023C/zh not_active Expired - Lifetime
- 2003-03-20 HR HRP20040889AA patent/HRP20040889B1/hr not_active IP Right Cessation
- 2003-03-20 MX MXPA04009337A patent/MXPA04009337A/es active IP Right Grant
- 2003-03-20 IL IL16369703A patent/IL163697A0/xx active IP Right Grant
- 2003-03-20 UA UA20041008770A patent/UA78557C2/uk unknown
- 2003-03-20 RS YU85904A patent/RS52178B/sr unknown
- 2003-03-20 DE DE50305118T patent/DE50305118D1/de not_active Expired - Lifetime
- 2003-03-20 CA CA2479640A patent/CA2479640C/en not_active Expired - Fee Related
- 2003-03-20 AT AT03745193T patent/ATE339953T1/de active
- 2003-03-20 EA EA200401190A patent/EA007239B1/ru not_active IP Right Cessation
- 2003-03-20 EP EP06115508.1A patent/EP1695701B1/de not_active Expired - Lifetime
- 2003-03-20 PL PL03371296A patent/PL371296A1/xx unknown
- 2003-03-20 KR KR1020047015356A patent/KR101066801B1/ko not_active Expired - Fee Related
- 2003-03-20 ME MEP-2008-474A patent/ME00247B/me unknown
- 2003-03-20 BR BR0308764-6A patent/BR0308764A/pt not_active IP Right Cessation
- 2003-03-20 DK DK03745193T patent/DK1492513T3/da active
- 2003-03-20 NZ NZ536043A patent/NZ536043A/en not_active IP Right Cessation
- 2003-03-20 AU AU2003209743A patent/AU2003209743B2/en not_active Ceased
- 2003-03-20 ES ES03745193T patent/ES2273020T3/es not_active Expired - Lifetime
- 2003-03-20 EP EP03745193A patent/EP1492513B1/de not_active Expired - Lifetime
- 2003-03-20 WO PCT/EP2003/002898 patent/WO2003082252A1/de not_active Ceased
- 2003-03-20 PT PT03745193T patent/PT1492513E/pt unknown
- 2003-03-20 JP JP2003579790A patent/JP4480401B2/ja not_active Expired - Lifetime
2004
- 2004-07-15 ZA ZA2004/05638A patent/ZA200405638B/en unknown
- 2004-08-24 IL IL163697A patent/IL163697A/en unknown
- 2004-09-23 NO NO20044005A patent/NO20044005L/no not_active Application Discontinuation
- 2004-09-28 EC EC2004005321A patent/ECSP045321A/es unknown
2006
- 2006-09-26 CY CY20061101380T patent/CY1105543T1/el unknown

Also Published As

Publication number	Publication date
DK1492513T3 (da)	2006-12-18
CN1642534A (zh)	2005-07-20
AU2003209743A1 (en)	2003-10-13
PL371296A1 (en)	2005-06-13
ZA200405638B (en)	2005-07-27
CY1105543T1 (el)	2010-07-28
MEP47408A (en)	2011-02-10
JP2005529087A (ja)	2005-09-29
CA2479640A1 (en)	2003-10-09
UA78557C2 (en)	2007-04-10
HK1079091A1 (en)	2006-03-31
JP4480401B2 (ja)	2010-06-16
EP1492513A1 (de)	2005-01-05
EP1492513B1 (de)	2006-09-20
ME00247B (me)	2011-05-10
PT1492513E (pt)	2006-12-29
WO2003082252A1 (de)	2003-10-09
KR20040098031A (ko)	2004-11-18
IL163697A (en)	2011-03-31
EA200401190A1 (ru)	2005-04-28
NZ536043A (en)	2005-09-30
KR101066801B1 (ko)	2011-09-22
CA2479640C (en)	2010-09-28
CN1329023C (zh)	2007-08-01
DE50305118D1 (de)	2006-11-02
EA007239B1 (ru)	2006-08-25
EP1695701A3 (de)	2010-04-28
BR0308764A (pt)	2005-01-11
AU2003209743B2 (en)	2008-03-06
RS52178B (sr)	2012-10-31
EP1695701B1 (de)	2015-01-07
ECSP045321A (es)	2005-01-28
ES2273020T3 (es)	2007-05-01
EP1695701A2 (de)	2006-08-30
MXPA04009337A (es)	2005-01-25
HRP20040889B1 (hr)	2012-11-30
ATE339953T1 (de)	2006-10-15
HRP20040889A2 (en)	2004-12-31
YU85904A (sh)	2006-08-17
IL163697A0 (en)	2005-12-18
DE10214263A1 (de)	2003-10-16

Legal Events

Date	Code	Title	Description
2016-02-22	FC2A	Withdrawal, rejection or dismissal of laid open patent application

Publication	Publication Date	Title
ATE164864T1 (de)	1998-04-15	Flüssiges kohlendioxid enthaltende treibmittel
JP2008036429A5 (no)	2012-09-27
ATE201033T1 (de)	2001-05-15	Gemische mit 1,1,1,3,3-pentafluorbutan
WO2005048976A3 (en)	2006-10-26	Foams comprising a sclerosing and a viscosity enhancing agent, methods for production thereof
CO4410246A1 (es)	1997-01-09	Proceso para preparar una espuma de poliuretano en presencia de un agente inflador de hidrocarburo
EP2036943A3 (en)	2009-07-22	Compositions containing fluorine substituted olefins
DE69522441D1 (de)	2001-10-04	Zusammensetzungen aus fluorkohlenwasserstoffen
CA2148854A1 (en)	1992-01-27	Near-azeotropic blends for use as refrigerants
AU2001277096A1 (en)	2002-02-05	Monolithic expandable structures, methods of manufacture and composite structures
ATE283033T1 (de)	2004-12-15	Medizinische aerosolformulierungen
ES2178817T3 (es)	2003-01-01	Formulaciones medicinales de aerosol.
ATE339953T1 (de)	2006-10-15	Hfa-suspensionsformulierungen enthaltend ein anticholinergikum
TW200639202A (en)	2006-11-16	Class fiber reinforced polyurethane/polyisocyanurate foam
BRPI0713310A2 (pt)	2012-03-06	aumentadores de tamanho de cÉlula para espumas de poliestireno
BRPI0507524A (pt)	2007-07-03	composição refrigerante
MXPA05005692A (es)	2005-10-18	Refrigerantes para enfriador.
CA2329989A1 (en)	2000-09-28	High productivity, low fugitive emission foams and foam processes
DE69004344D1 (de)	1993-12-09	Azeotrope von Wasserstoff enthaltenden Kohlenstoffen mit Butanen.
BR9808818A (pt)	2000-06-27	Composição constituìda essencialmente de 1, 1, 1, 3, 3-pentafluorobutano e de um hidrocarboneto, utilização de composições azeotrópicas ou pseudo-azeotrópicas, agente espumante para espumas celulares poliméricas e pré-mistura para espuma de poliuretano.
EP0626421A4 (en)	1995-09-13	FUEL COMPOSITION, PRODUCTION OF FOAM BY MEANS OF THIS COMPOSITION AND FOAM PRODUCED THEREOF.
DK0632090T3 (da)	1999-04-12	Fremgangsmåde til opskumning af brandhæmmende styrenpolymerisater
CA2305777A1 (en)	1999-04-08	High productivity, low fugitive voc emission foam process
DK0552075T3 (da)	1995-11-13	Blandinger af 1,1,1-trifluorethan og perfluorpropan og deres anvendelse som kølemedier, drivmidler til aerosoler eller midler til ekspansion af plastskum
NO953675L (no)	1995-09-18	Azeotrop-lignende blandinger av 1,1,1,2,3,3,3-heptafluor propan og 1,1-difluoretan, og anvendelse av slike
MX2007007549A (es)	2007-07-20	Composiciones de espuma de poliestireno retardadoras d ela flama.