NO20061818L - Fremgangsmate for a inhibere remnant lipoproteinproduksjon - Google Patents
Fremgangsmate for a inhibere remnant lipoproteinproduksjonInfo
- Publication number
- NO20061818L NO20061818L NO20061818A NO20061818A NO20061818L NO 20061818 L NO20061818 L NO 20061818L NO 20061818 A NO20061818 A NO 20061818A NO 20061818 A NO20061818 A NO 20061818A NO 20061818 L NO20061818 L NO 20061818L
- Authority
- NO
- Norway
- Prior art keywords
- lipoprotein production
- remnant lipoprotein
- inhibiting
- inhibiting remnant
- compound
- Prior art date
Links
- 102000004895 Lipoproteins Human genes 0.000 title abstract 4
- 108090001030 Lipoproteins Proteins 0.000 title abstract 4
- 230000002401 inhibitory effect Effects 0.000 title abstract 4
- 238000000034 method Methods 0.000 title abstract 2
- KEWSCDNULKOKTG-UHFFFAOYSA-N 4-cyano-4-ethylsulfanylcarbothioylsulfanylpentanoic acid Chemical compound CCSC(=S)SC(C)(C#N)CCC(O)=O KEWSCDNULKOKTG-UHFFFAOYSA-N 0.000 abstract 2
- 102100037637 Cholesteryl ester transfer protein Human genes 0.000 abstract 2
- 101000880514 Homo sapiens Cholesteryl ester transfer protein Proteins 0.000 abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 2
- 239000003112 inhibitor Substances 0.000 abstract 2
- 239000004480 active ingredient Substances 0.000 abstract 1
Classifications
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/21—Esters, e.g. nitroglycerine, selenocyanates
- A61K31/255—Esters, e.g. nitroglycerine, selenocyanates of sulfoxy acids or sulfur analogues thereof
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- A—HUMAN NECESSITIES
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- A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
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- A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
- A61K31/167—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide having the nitrogen of a carboxamide group directly attached to the aromatic ring, e.g. lidocaine, paracetamol
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- A61K31/19—Carboxylic acids, e.g. valproic acid
- A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
- A61K31/196—Carboxylic acids, e.g. valproic acid having an amino group the amino group being directly attached to a ring, e.g. anthranilic acid, mefenamic acid, diclofenac, chlorambucil
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Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Emergency Medicine (AREA)
- Diabetes (AREA)
- Pain & Pain Management (AREA)
- Endocrinology (AREA)
- Urology & Nephrology (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Vascular Medicine (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Quinoline Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
- Steroid Compounds (AREA)
Abstract
Den foreliggende oppfinnelse sikter mot frembringelse av en fremgangsmåte for å inhibere resterende lipoproteinproduksjon og en resterende lipoproteinproduksjons-inhibitor, som inkluderer administrering av en forbindelse med en CETP inhibitorisk aktivitet til et administreringssubjekt. Den resterende lipoproteinproduksjonsinhibitor ifølge den foreliggende oppfinnelse inneholder en forbindelse med en CETP inhibitorisk aktivitet som en aktiv bestanddel.
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2003373453 | 2003-09-26 | ||
| US59081104P | 2004-07-23 | 2004-07-23 | |
| PCT/JP2004/014428 WO2005030185A2 (en) | 2003-09-26 | 2004-09-24 | Method of inhibiting remnant lipoprotein production |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| NO20061818L true NO20061818L (no) | 2006-06-26 |
Family
ID=37583964
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO20061818A NO20061818L (no) | 2003-09-26 | 2006-04-25 | Fremgangsmate for a inhibere remnant lipoproteinproduksjon |
Country Status (17)
| Country | Link |
|---|---|
| US (3) | US20070054839A1 (no) |
| EP (3) | EP2316447A1 (no) |
| JP (2) | JP4536061B2 (no) |
| KR (2) | KR20070087197A (no) |
| CN (3) | CN101342162A (no) |
| AU (1) | AU2004275637C1 (no) |
| BR (1) | BRPI0414822A (no) |
| CA (1) | CA2554982A1 (no) |
| CO (1) | CO5690566A2 (no) |
| IL (2) | IL174310A (no) |
| MX (1) | MXPA06003357A (no) |
| NO (1) | NO20061818L (no) |
| NZ (2) | NZ569469A (no) |
| RU (1) | RU2330682C2 (no) |
| SG (1) | SG146695A1 (no) |
| WO (1) | WO2005030185A2 (no) |
| ZA (2) | ZA200603280B (no) |
Families Citing this family (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7700774B2 (en) | 2004-12-20 | 2010-04-20 | Dr. Reddy's Laboratories Ltd. | Heterocyclic compounds and their pharmaceutical compositions |
| US8604055B2 (en) | 2004-12-31 | 2013-12-10 | Dr. Reddy's Laboratories Ltd. | Substituted benzylamino quinolines as cholesterol ester-transfer protein inhibitors |
| CA2605214C (en) | 2004-12-31 | 2016-07-12 | Reddy Us Therapeutics, Inc. | Benzylamine derivatives as cetp inhibitors |
| US7888376B2 (en) | 2005-11-23 | 2011-02-15 | Bristol-Myers Squibb Company | Heterocyclic CETP inhibitors |
| US7790770B2 (en) | 2005-11-23 | 2010-09-07 | Bristol-Myers Squibb Company | Heterocyclic CETP inhibitors |
| US7652023B2 (en) | 2005-11-23 | 2010-01-26 | Bristol-Myers Squibb Company | Heterocyclic CETP inhibitors |
| UY30118A1 (es) * | 2006-01-31 | 2007-06-29 | Tanabe Seiyaku Co | Compueto amina trisustituido |
| CN101663262B (zh) | 2006-12-01 | 2014-03-26 | 百时美施贵宝公司 | 用于治疗动脉粥样硬化和心血管疾病的作为cetp抑制剂的n-(3-苄基)-2,2-(二苯基)-丙-1胺衍生物 |
| EP2744803A2 (en) | 2011-08-18 | 2014-06-25 | Dr. Reddy's Laboratories Ltd. | Substituted heterocyclic amine compounds as cholestryl ester-transfer protein (cetp) inhibitors |
| MX352074B (es) | 2011-09-27 | 2017-11-08 | Dr Reddys Laboratories Ltd | Derivados de 5-bencilaminometil-6-aminopirazolo [3,4-b] piridina como inhibidores de proteina de transferencia de ester de colesterilo (cetp) utiles para el tratamiento de aterosclerosis. |
| JPWO2014017569A1 (ja) * | 2012-07-26 | 2016-07-11 | 興和株式会社 | 血中ldlを低下させるための医薬 |
| SI2978859T1 (sl) | 2013-03-27 | 2018-10-30 | F. Hoffmann-La Roche Ag | Genetski označevalci za napovedovanje odzivnosti na terapijo |
| EP2981522A4 (en) * | 2013-04-05 | 2016-08-31 | Salk Inst For Biological Studi | PPAR AGONISTS |
| MX384679B (es) | 2014-07-30 | 2025-03-14 | Hoffmann La Roche | Marcadores genéticos para predecir la reactividad a terapia con agente que eleva la lipoproteína de alta densidad (hdl) o que imita la lipoproteína de alta densidad (hdl). |
| EA037371B1 (ru) | 2015-10-07 | 2021-03-19 | Митобридж, Инк. | Агонисты ppar, соединения, фармацевтические композиции и способы их применения |
| US11358954B2 (en) | 2016-04-13 | 2022-06-14 | Mitobridge, Inc. | PPAR agonists, compounds, pharmaceutical compositions, and methods of use thereof |
Family Cites Families (73)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US43341A (en) * | 1864-06-28 | Improved vegetable ointment or salve | ||
| US120011A (en) * | 1871-10-17 | Improvement in sad-iron handles | ||
| US40545A (en) * | 1863-11-10 | Joseph h | ||
| US59810A (en) * | 1866-11-20 | babtlett | ||
| US127574A (en) * | 1872-06-04 | Improvement in machinery for breaking and crushing stones | ||
| US18446A (en) * | 1857-10-20 | Improvement in steam-plows | ||
| US32644A (en) * | 1861-06-25 | Tub and pail machine | ||
| US165231A (en) * | 1875-07-06 | Improvement in knuckle-couplings for tumbling-shafts | ||
| US177708A (en) * | 1876-05-23 | Improvement in hinges | ||
| US27826A (en) * | 1860-04-10 | Improvement in harvesters | ||
| JPH01149743A (ja) | 1987-12-04 | 1989-06-12 | Japan Atom Energy Res Inst | エチレングリコールの製造方法 |
| FI941166A7 (fi) * | 1991-09-13 | 1994-03-25 | Sankyo Co | Trisyklinen heterosyklyyliyhdiste |
| JPH05194475A (ja) * | 1991-09-13 | 1993-08-03 | Sankyo Co Ltd | 三環性ヘテロシクリル化合物 |
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