NO20062090L - Polymorf form av N-[(R)-2,3-dihydroksy-propksy]-3,4-difluor-2-(2-fluor-4-iodfenylamino)-benzamid - Google Patents

Polymorf form av N-[(R)-2,3-dihydroksy-propksy]-3,4-difluor-2-(2-fluor-4-iodfenylamino)-benzamid

Info

Publication number
NO20062090L
NO20062090L NO20062090A NO20062090A NO20062090L NO 20062090 L NO20062090 L NO 20062090L NO 20062090 A NO20062090 A NO 20062090A NO 20062090 A NO20062090 A NO 20062090A NO 20062090 L NO20062090 L NO 20062090L
Authority
NO
Norway
Prior art keywords
polymorphic form
benzamide
difluoro
dihydroxy
propoxy
Prior art date
Application number
NO20062090A
Other languages
English (en)
Inventor
Dainius Mackikenas
Thomas Nanninga
Original Assignee
Warner Lambert Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Warner Lambert Co filed Critical Warner Lambert Co
Publication of NO20062090L publication Critical patent/NO20062090L/no

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    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C259/00—Compounds containing carboxyl groups, an oxygen atom of a carboxyl group being replaced by a nitrogen atom, this nitrogen atom being further bound to an oxygen atom and not being part of nitro or nitroso groups
    • C07C259/04—Compounds containing carboxyl groups, an oxygen atom of a carboxyl group being replaced by a nitrogen atom, this nitrogen atom being further bound to an oxygen atom and not being part of nitro or nitroso groups without replacement of the other oxygen atom of the carboxyl group, e.g. hydroxamic acids
    • C07C259/10—Compounds containing carboxyl groups, an oxygen atom of a carboxyl group being replaced by a nitrogen atom, this nitrogen atom being further bound to an oxygen atom and not being part of nitro or nitroso groups without replacement of the other oxygen atom of the carboxyl group, e.g. hydroxamic acids having carbon atoms of hydroxamic groups bound to carbon atoms of six-membered aromatic rings
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    • A61P11/06—Antiasthmatics
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    • A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
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    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
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    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C237/00—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups
    • C07C237/28—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atom of at least one of the carboxamide groups bound to a carbon atom of a non-condensed six-membered aromatic ring of the carbon skeleton

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Abstract

Det er beskrevet en ny polymorf form av N-[(R)-2,3-dihydroksy-propoksy]-3,4-difluor-2-(2-fluor-4-iod-fenylamino)-benzamid, så vel som farmasøytiske preparater og terapeutiske fremgangsmåter som anvender den polymorfe formen.
NO20062090A 2003-10-21 2006-05-09 Polymorf form av N-[(R)-2,3-dihydroksy-propksy]-3,4-difluor-2-(2-fluor-4-iodfenylamino)-benzamid NO20062090L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US51298003P 2003-10-21 2003-10-21
PCT/IB2004/003309 WO2005040098A1 (en) 2003-10-21 2004-10-11 Polymorphic form of n-[(r)-2,3-dihydroxy-propoxy]-3,4-difluoro-2-(2-fluoro-4-iodophenylamino)-benzamide

Publications (1)

Publication Number Publication Date
NO20062090L true NO20062090L (no) 2006-07-12

Family

ID=34520067

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20062090A NO20062090L (no) 2003-10-21 2006-05-09 Polymorf form av N-[(R)-2,3-dihydroksy-propksy]-3,4-difluor-2-(2-fluor-4-iodfenylamino)-benzamid

Country Status (18)

Country Link
US (1) US7060856B2 (no)
EP (1) EP1682495A1 (no)
JP (1) JP2007509125A (no)
KR (1) KR101013932B1 (no)
CN (1) CN100594212C (no)
AR (1) AR046124A1 (no)
AU (1) AU2004283148A1 (no)
BR (1) BRPI0415710A (no)
CA (1) CA2542210A1 (no)
CO (1) CO5690569A2 (no)
IL (1) IL174367A0 (no)
MX (1) MXPA06004363A (no)
NO (1) NO20062090L (no)
NZ (1) NZ546011A (no)
RU (1) RU2352558C2 (no)
TW (1) TW200524584A (no)
WO (1) WO2005040098A1 (no)
ZA (1) ZA200602250B (no)

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EP1682495A1 (en) 2006-07-26
US20050085550A1 (en) 2005-04-21
KR20060080230A (ko) 2006-07-07
WO2005040098A1 (en) 2005-05-06
RU2006113437A (ru) 2006-08-27
RU2352558C2 (ru) 2009-04-20
MXPA06004363A (es) 2006-06-14
IL174367A0 (en) 2006-08-01
AU2004283148A1 (en) 2005-05-06
CN100594212C (zh) 2010-03-17
KR101013932B1 (ko) 2011-02-14
TW200524584A (en) 2005-08-01
HK1093483A1 (en) 2007-03-02
CO5690569A2 (es) 2006-10-31
US7060856B2 (en) 2006-06-13
CA2542210A1 (en) 2005-05-06
JP2007509125A (ja) 2007-04-12
AR046124A1 (es) 2005-11-23
ZA200602250B (en) 2007-05-30
NZ546011A (en) 2009-09-25
BRPI0415710A (pt) 2006-12-19

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