NO20062389L - Fremgangsmate for spray-storkning ved anvendelse av en ekstruder for fremstilling av multipartikkulaere azitromycinmaterialer - Google Patents

Fremgangsmate for spray-storkning ved anvendelse av en ekstruder for fremstilling av multipartikkulaere azitromycinmaterialer

Info

Publication number: NO20062389L
Authority: NO; Norway
Prior art keywords: extruder; prepare; materials; azithromycin; spray solidification
Prior art date: 2003-12-04

Application number

NO20062389A

Other languages

English (en)

Norwegian (no)

Inventor

Scott Max Herbig

Julian Belknap Lo

Leah Elizabeth Appel

Marshall David Crew

Dwayne Thomas Friesen

David Keith Lyon

Scott Baldwin Mccray

Roderick Jack Ray

James Blair West

David Dixon Newbold

Steven Ross Lemott

Original Assignee

Pfizer Prod Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2003-12-04

Filing date

2006-05-24

Publication date

2006-06-16

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34652484&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO20062389(L) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

2006-05-24 Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc

2006-06-16 Publication of NO20062389L publication Critical patent/NO20062389L/no

Links

MQTOSJVFKKJCRP-BICOPXKESA-N azithromycin Chemical compound O([C@@H]1[C@@H](C)C(=O)O[C@@H]([C@@]([C@H](O)[C@@H](C)N(C)C[C@H](C)C[C@@](C)(O)[C@H](O[C@H]2[C@@H]([C@H](C[C@@H](C)O2)N(C)C)O)[C@H]1C)(C)O)CC)[C@H]1C[C@@](C)(OC)[C@@H](O)[C@H](C)O1 MQTOSJVFKKJCRP-BICOPXKESA-N 0.000 title abstract 3
229960004099 azithromycin Drugs 0.000 title abstract 2
238000000034 method Methods 0.000 title abstract 2
238000007711 solidification Methods 0.000 title abstract 2
239000000463 material Substances 0.000 title 1
230000008023 solidification Effects 0.000 title 1
239000007921 spray Substances 0.000 title 1

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/141—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
- A61K9/145—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with organic compounds
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A61K31/7028—Compounds having saccharide radicals attached to non-saccharide compounds by glycosidic linkages
- A61K31/7032—Compounds having saccharide radicals attached to non-saccharide compounds by glycosidic linkages attached to a polyol, i.e. compounds having two or more free or esterified hydroxy groups, including the hydroxy group involved in the glycosidic linkage, e.g. monoglucosyldiacylglycerides, lactobionic acid, gangliosides
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
- A61K31/7052—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1617—Organic compounds, e.g. phospholipids, fats
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1629—Organic macromolecular compounds
- A61K9/1641—Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, poloxamers
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1682—Processes
- A61K9/1694—Processes resulting in granules or microspheres of the matrix type containing more than 5% of excipient
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0087—Galenical forms not covered by A61K9/02 - A61K9/7023
- A61K9/0095—Drinks; Beverages; Syrups; Compositions for reconstitution thereof, e.g. powders or tablets to be dispersed in a glass of water; Veterinary drenches

Landscapes

Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Public Health (AREA)
Medicinal Chemistry (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Veterinary Medicine (AREA)
Pharmacology & Pharmacy (AREA)
Epidemiology (AREA)
Molecular Biology (AREA)
Biophysics (AREA)
Communicable Diseases (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Organic Chemistry (AREA)
Oncology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Medicinal Preparation (AREA)
Glanulating (AREA)

NO20062389A 2003-12-04 2006-05-24 Fremgangsmate for spray-storkning ved anvendelse av en ekstruder for fremstilling av multipartikkulaere azitromycinmaterialer NO20062389L (no)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US52724403P	2003-12-04	2003-12-04
PCT/IB2004/003839 WO2005053653A1 (en)	2003-12-04	2004-11-22	Spray-congeal process using an extruder for preparing multiparticulate azithromycin compositions containing preferably a poloxamer and a glyceride

Publications (1)

Publication Number	Publication Date
NO20062389L true NO20062389L (no)	2006-06-16

Family

ID=34652484

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO20062389A NO20062389L (no)	2003-12-04	2006-05-24	Fremgangsmate for spray-storkning ved anvendelse av en ekstruder for fremstilling av multipartikkulaere azitromycinmaterialer

Country Status (15)

Country	Link
US (1)	US20050158391A1 (pt)
EP (1)	EP1701702A1 (pt)
JP (1)	JP2007513143A (pt)
KR (2)	KR20060109481A (pt)
CN (1)	CN1889931A (pt)
AR (1)	AR046468A1 (pt)
AU (1)	AU2004294813A1 (pt)
BR (1)	BRPI0416535A (pt)
CA (1)	CA2547773A1 (pt)
IL (1)	IL175745A0 (pt)
NO (1)	NO20062389L (pt)
RU (1)	RU2006119464A (pt)
TW (1)	TW200528138A (pt)
WO (1)	WO2005053653A1 (pt)
ZA (1)	ZA200604495B (pt)

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CN109288798A (zh) *	2018-12-08	2019-02-01	海南医学院	一种阿奇霉素掩味微球的制备方法
WO2021014360A1 (en)	2019-07-23	2021-01-28	Pfizer Inc.	Oral modified release dosage forms
CA3161153A1 (en)	2019-11-14	2021-05-20	Pfizer Inc.	1-(((2s,3s,4s)-3-ethyl-4-fluoro-5-oxopyrrolidin-2-yl)methoxy)-7-methoxyisoquinoline-6-carboxamide combinations and oral dosage forms
US20230181463A1 (en) *	2020-05-15	2023-06-15	Massachusetts Institute Of Technology	Oleogel and oleopaste compositions and uses thereof

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2004
- 2004-11-22 CN CNA2004800358177A patent/CN1889931A/zh active Pending
- 2004-11-22 CA CA002547773A patent/CA2547773A1/en not_active Abandoned
- 2004-11-22 RU RU2006119464/15A patent/RU2006119464A/ru unknown
- 2004-11-22 EP EP04798952A patent/EP1701702A1/en not_active Withdrawn
- 2004-11-22 BR BRPI0416535-7A patent/BRPI0416535A/pt not_active IP Right Cessation
- 2004-11-22 JP JP2006542040A patent/JP2007513143A/ja not_active Abandoned
- 2004-11-22 AU AU2004294813A patent/AU2004294813A1/en not_active Abandoned
- 2004-11-22 KR KR1020067011027A patent/KR20060109481A/ko not_active Ceased
- 2004-11-22 WO PCT/IB2004/003839 patent/WO2005053653A1/en not_active Ceased
- 2004-11-22 KR KR1020087015425A patent/KR20080064209A/ko not_active Withdrawn
- 2004-12-01 TW TW093137051A patent/TW200528138A/zh unknown
- 2004-12-03 AR ARP040104514A patent/AR046468A1/es unknown
- 2004-12-03 US US11/003,856 patent/US20050158391A1/en not_active Abandoned
2006
- 2006-05-18 IL IL175745A patent/IL175745A0/en unknown
- 2006-05-24 NO NO20062389A patent/NO20062389L/no not_active Application Discontinuation
- 2006-06-01 ZA ZA200604495A patent/ZA200604495B/en unknown

Also Published As

Publication number	Publication date
KR20060109481A (ko)	2006-10-20
AR046468A1 (es)	2005-12-07
AU2004294813A1 (en)	2005-06-16
IL175745A0 (en)	2006-09-05
JP2007513143A (ja)	2007-05-24
US20050158391A1 (en)	2005-07-21
RU2006119464A (ru)	2007-12-20
TW200528138A (en)	2005-09-01
KR20080064209A (ko)	2008-07-08
BRPI0416535A (pt)	2007-01-09
CN1889931A (zh)	2007-01-03
CA2547773A1 (en)	2005-06-16
ZA200604495B (en)	2008-03-26
WO2005053653A1 (en)	2005-06-16
EP1701702A1 (en)	2006-09-20

Legal Events

Date	Code	Title	Description
2010-06-28	FC2A	Withdrawal, rejection or dismissal of laid open patent application

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