NO20064185L - Pyrazolin derivater nyttige for bahandling av kreft - Google Patents
Pyrazolin derivater nyttige for bahandling av kreftInfo
- Publication number
- NO20064185L NO20064185L NO20064185A NO20064185A NO20064185L NO 20064185 L NO20064185 L NO 20064185L NO 20064185 A NO20064185 A NO 20064185A NO 20064185 A NO20064185 A NO 20064185A NO 20064185 L NO20064185 L NO 20064185L
- Authority
- NO
- Norway
- Prior art keywords
- cancer
- treatment
- compounds
- derivatives useful
- pyrazoline derivatives
- Prior art date
Links
- 206010028980 Neoplasm Diseases 0.000 title abstract 2
- 201000011510 cancer Diseases 0.000 title abstract 2
- 150000003219 pyrazolines Chemical class 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 3
- 206010061902 Pancreatic neoplasm Diseases 0.000 abstract 2
- 208000015486 malignant pancreatic neoplasm Diseases 0.000 abstract 2
- 201000002528 pancreatic cancer Diseases 0.000 abstract 2
- 208000008443 pancreatic carcinoma Diseases 0.000 abstract 2
- 206010005003 Bladder cancer Diseases 0.000 abstract 1
- 206010005949 Bone cancer Diseases 0.000 abstract 1
- 208000018084 Bone neoplasm Diseases 0.000 abstract 1
- 208000003174 Brain Neoplasms Diseases 0.000 abstract 1
- 206010006187 Breast cancer Diseases 0.000 abstract 1
- 208000026310 Breast neoplasm Diseases 0.000 abstract 1
- 208000000461 Esophageal Neoplasms Diseases 0.000 abstract 1
- 201000003741 Gastrointestinal carcinoma Diseases 0.000 abstract 1
- 206010062038 Lip neoplasm Diseases 0.000 abstract 1
- 206010058467 Lung neoplasm malignant Diseases 0.000 abstract 1
- 208000003445 Mouth Neoplasms Diseases 0.000 abstract 1
- 206010030155 Oesophageal carcinoma Diseases 0.000 abstract 1
- 206010060862 Prostate cancer Diseases 0.000 abstract 1
- 208000000236 Prostatic Neoplasms Diseases 0.000 abstract 1
- 208000000453 Skin Neoplasms Diseases 0.000 abstract 1
- 208000005718 Stomach Neoplasms Diseases 0.000 abstract 1
- 208000007097 Urinary Bladder Neoplasms Diseases 0.000 abstract 1
- 210000001072 colon Anatomy 0.000 abstract 1
- 201000004101 esophageal cancer Diseases 0.000 abstract 1
- 206010017758 gastric cancer Diseases 0.000 abstract 1
- 201000002313 intestinal cancer Diseases 0.000 abstract 1
- 208000012987 lip and oral cavity carcinoma Diseases 0.000 abstract 1
- 201000006721 lip cancer Diseases 0.000 abstract 1
- 201000007270 liver cancer Diseases 0.000 abstract 1
- 208000014018 liver neoplasm Diseases 0.000 abstract 1
- 201000005202 lung cancer Diseases 0.000 abstract 1
- 208000020816 lung neoplasm Diseases 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
- 201000000849 skin cancer Diseases 0.000 abstract 1
- 201000011549 stomach cancer Diseases 0.000 abstract 1
- 201000005112 urinary bladder cancer Diseases 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/06—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/415—1,2-Diazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Foreliggende oppfinnels angår nye substituerte prazolinforbindelser, farmasøytiske sammensetninger inneholdende slike forbindelser og anvendelsen av disse forbindelsene for behandling av cancer, spesielt for behandlingen av hjernecancer, bencancer, leppecancer, munncancer, øsofagal cancer, magecancer, levercancer, blærecancer, pancreascancer, ovariecancer, cervical cancer, lungecancer, brystcancer, hudcancer, spesielt for behandlingen av coloncancer og/eller tarmcancer og/eller prostatacancer.
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ES200400362A ES2238923B1 (es) | 2004-02-16 | 2004-02-16 | Nuevos derivados pirazolinicos sustituidos. |
| US10/804,695 US20050182119A1 (en) | 2004-02-16 | 2004-03-19 | Substituted pyrazoline derivatives |
| PCT/EP2005/001656 WO2005077910A1 (en) | 2004-02-16 | 2005-02-16 | Pyrazoline derivatives useful for the treatment of cancer |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| NO20064185L true NO20064185L (no) | 2006-11-13 |
Family
ID=34863166
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO20064185A NO20064185L (no) | 2004-02-16 | 2006-09-15 | Pyrazolin derivater nyttige for bahandling av kreft |
Country Status (9)
| Country | Link |
|---|---|
| EP (1) | EP1718618A1 (no) |
| JP (1) | JP2007522180A (no) |
| KR (1) | KR20070044799A (no) |
| AU (1) | AU2005212833A1 (no) |
| BR (1) | BRPI0507718A (no) |
| CA (1) | CA2556478A1 (no) |
| NO (1) | NO20064185L (no) |
| RU (1) | RU2006133150A (no) |
| WO (1) | WO2005077910A1 (no) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| RU2304989C2 (ru) * | 2005-08-26 | 2007-08-27 | Государственное образовательное учреждение высшего профессионального образования "Нижегородская государственная медицинская академия Федерального Агентства по здравоохранению и социальному развитию" (ГОУ ВПО "НижГМА Росздрава") | Способ комбинированного лечения операбельного рака желудка |
| JP2008308473A (ja) * | 2007-06-18 | 2008-12-25 | Japan Health Science Foundation | 癌治療剤 |
| CN101735150B (zh) * | 2009-12-16 | 2011-12-28 | 南京大学 | 一类含有吡唑环的硫脲类衍生物及其制法和用途 |
| CN101759695B (zh) * | 2009-12-30 | 2011-09-14 | 南京大学 | 一类含有吡唑环的噻唑类衍生物及其制法和用途 |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6376519B1 (en) * | 1999-06-16 | 2002-04-23 | Temple University-Of The Commonwealth Of Higher Education | 1-(4-sulfamylaryl)-3-substituted-5-aryl-2-pyrazolines and inhibitors of cyclooxygenase-2 |
| ES2174757B1 (es) * | 2001-04-06 | 2003-11-01 | Esteve Labor Dr | Empleo de derivados de firazolinas en la elaboracion de un medicamentopara la prevencion y/o el tratamiento de enfermedades proliferativas celulares. |
-
2005
- 2005-02-16 WO PCT/EP2005/001656 patent/WO2005077910A1/en not_active Ceased
- 2005-02-16 AU AU2005212833A patent/AU2005212833A1/en not_active Abandoned
- 2005-02-16 CA CA002556478A patent/CA2556478A1/en not_active Abandoned
- 2005-02-16 EP EP05707483A patent/EP1718618A1/en not_active Withdrawn
- 2005-02-16 JP JP2006552580A patent/JP2007522180A/ja active Pending
- 2005-02-16 KR KR1020067018161A patent/KR20070044799A/ko not_active Withdrawn
- 2005-02-16 BR BRPI0507718-4A patent/BRPI0507718A/pt not_active IP Right Cessation
- 2005-02-16 RU RU2006133150/04A patent/RU2006133150A/ru unknown
-
2006
- 2006-09-15 NO NO20064185A patent/NO20064185L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| RU2006133150A (ru) | 2008-04-10 |
| KR20070044799A (ko) | 2007-04-30 |
| JP2007522180A (ja) | 2007-08-09 |
| BRPI0507718A (pt) | 2007-07-03 |
| EP1718618A1 (en) | 2006-11-08 |
| CA2556478A1 (en) | 2005-08-25 |
| AU2005212833A1 (en) | 2005-08-25 |
| WO2005077910A1 (en) | 2005-08-25 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FC2A | Withdrawal, rejection or dismissal of laid open patent application |