NO20065863L - 3-[4-(6-(4,5-dihydroisoksazol-3-yl]pyridin-3-yl)-3-fenyl]-5-(1 H,1,2,3-triazol-1-yl-metyl)-1,3-oksazolidin-2-oner som antibakterielle midler - Google Patents
3-[4-(6-(4,5-dihydroisoksazol-3-yl]pyridin-3-yl)-3-fenyl]-5-(1 H,1,2,3-triazol-1-yl-metyl)-1,3-oksazolidin-2-oner som antibakterielle midlerInfo
- Publication number
- NO20065863L NO20065863L NO20065863A NO20065863A NO20065863L NO 20065863 L NO20065863 L NO 20065863L NO 20065863 A NO20065863 A NO 20065863A NO 20065863 A NO20065863 A NO 20065863A NO 20065863 L NO20065863 L NO 20065863L
- Authority
- NO
- Norway
- Prior art keywords
- methyl
- optionally substituted
- antibacterial agents
- dihydroisoxazol
- oxazolidin
- Prior art date
Links
- 239000003242 anti bacterial agent Substances 0.000 title abstract 2
- -1 6- (4,5-Dihydroisoxazol-3-yl) pyridin-3-yl Chemical group 0.000 title 2
- 150000001875 compounds Chemical class 0.000 abstract 3
- 239000001257 hydrogen Substances 0.000 abstract 3
- 229910052739 hydrogen Inorganic materials 0.000 abstract 3
- 150000002431 hydrogen Chemical class 0.000 abstract 3
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 abstract 2
- ZAMOUSCENKQFHK-UHFFFAOYSA-N Chlorine atom Chemical compound [Cl] ZAMOUSCENKQFHK-UHFFFAOYSA-N 0.000 abstract 1
- PXGOKWXKJXAPGV-UHFFFAOYSA-N Fluorine Chemical compound FF PXGOKWXKJXAPGV-UHFFFAOYSA-N 0.000 abstract 1
- 125000000217 alkyl group Chemical group 0.000 abstract 1
- 229910052801 chlorine Inorganic materials 0.000 abstract 1
- 239000000460 chlorine Substances 0.000 abstract 1
- 229910052731 fluorine Inorganic materials 0.000 abstract 1
- 239000011737 fluorine Substances 0.000 abstract 1
- 229910052736 halogen Inorganic materials 0.000 abstract 1
- 150000002367 halogens Chemical class 0.000 abstract 1
- 125000000623 heterocyclic group Chemical group 0.000 abstract 1
- 125000002883 imidazolyl group Chemical group 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
- 229910052757 nitrogen Inorganic materials 0.000 abstract 1
- 125000004433 nitrogen atom Chemical group N* 0.000 abstract 1
- 229940002612 prodrug Drugs 0.000 abstract 1
- 239000000651 prodrug Substances 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 229920006395 saturated elastomer Polymers 0.000 abstract 1
- 125000002023 trifluoromethyl group Chemical group FC(F)(F)* 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Public Health (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB0411594A GB0411594D0 (en) | 2004-05-25 | 2004-05-25 | Chemical compounds |
| GB0500055A GB0500055D0 (en) | 2005-01-05 | 2005-01-05 | Chemical compounds |
| PCT/GB2005/002040 WO2005116021A1 (en) | 2004-05-25 | 2005-05-24 | 3-[4-(6-{4,5-dihydroisoxazol-3-yl}pyridin-3-yl)-3-phenyl]-5-(1h-1,2,3-triazol-1-ylmethyl)-1,3-oxazolidin-2-ones as antibacterial agents |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| NO20065863L true NO20065863L (no) | 2007-02-20 |
Family
ID=34968779
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO20065863A NO20065863L (no) | 2004-05-25 | 2006-12-19 | 3-[4-(6-(4,5-dihydroisoksazol-3-yl]pyridin-3-yl)-3-fenyl]-5-(1 H,1,2,3-triazol-1-yl-metyl)-1,3-oksazolidin-2-oner som antibakterielle midler |
Country Status (14)
| Country | Link |
|---|---|
| US (1) | US20080064689A1 (pt) |
| EP (1) | EP1753756A1 (pt) |
| JP (1) | JP2008500315A (pt) |
| KR (1) | KR20070027614A (pt) |
| AR (1) | AR049121A1 (pt) |
| AU (1) | AU2005247663A1 (pt) |
| BR (1) | BRPI0511554A (pt) |
| CA (1) | CA2567454A1 (pt) |
| IL (1) | IL179348A0 (pt) |
| MX (1) | MXPA06013539A (pt) |
| NO (1) | NO20065863L (pt) |
| TW (1) | TW200604185A (pt) |
| UY (1) | UY28924A1 (pt) |
| WO (1) | WO2005116021A1 (pt) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR100854211B1 (ko) * | 2003-12-18 | 2008-08-26 | 동아제약주식회사 | 신규한 옥사졸리디논 유도체, 그의 제조방법 및 이를유효성분으로 하는 항생제용 약학 조성물 |
| KR100848232B1 (ko) * | 2007-04-12 | 2008-07-24 | 일동제약주식회사 | 신규 헤테로 고리 또는 알콕시아미노메틸 옥사졸리디논 및그 제조방법 |
| RU2659792C1 (ru) | 2008-10-10 | 2018-07-04 | Мерк Шарп Энд Домэ Корп. | Оксазолидиноны и способ их очистки |
| CN102224151A (zh) | 2008-11-20 | 2011-10-19 | 万能药生物有限公司 | 新的抗微生物剂 |
| MY156354A (en) | 2009-02-03 | 2016-02-15 | Merck Sharp & Dohme | Crystalline form of r)-3-(4-(2-(2-methyltetrazol-5-yl)pyridin-5-yl)-3-fluorophenyl)-5-hydroxymethyl oxazolidin-2-one dihydrogen phosphate |
| US8580767B2 (en) * | 2009-05-28 | 2013-11-12 | Trius Therapeutics, Inc. | Oxazolidinone containing dimer compounds, compositions and methods to make and use |
| KR20120106697A (ko) | 2009-06-26 | 2012-09-26 | 파나세아 바이오테크 리미티드 | 신규 아자비시클로헥산 |
| WO2011130419A2 (en) * | 2010-04-13 | 2011-10-20 | The Regents Of The University Of California | Broad spectrum antiviral and antiparasitic agents |
| JP6610905B2 (ja) * | 2015-02-27 | 2019-11-27 | オーピーバイオファクトリー株式会社 | カケロマイシンおよびその誘導体の製造方法 |
| CN111471041B (zh) * | 2019-01-23 | 2022-09-20 | 中国科学院上海药物研究所 | 一种噁唑烷酮类抗菌药物中间体的合成方法 |
| WO2021000297A1 (en) | 2019-07-03 | 2021-01-07 | Merck Sharp & Dohme Corp. | Compounds and methods of use thereof as antibacterial agents |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SI1427711T1 (sl) * | 2001-09-11 | 2005-12-31 | Astrazeneca Ab | Oksazolidinonski in/ali izoksazolinski derivati kot antibakterijska sredstva |
| MXPA05005651A (es) * | 2002-11-28 | 2005-07-27 | Astrazeneca Ab | Derivados de oxazolidinona y/o isoxazolina como agentes antibacterianos. |
| GB0227701D0 (en) * | 2002-11-28 | 2003-01-08 | Astrazeneca Ab | Chemical compounds |
| TW200500360A (en) * | 2003-03-01 | 2005-01-01 | Astrazeneca Ab | Hydroxymethyl compounds |
-
2004
- 2004-05-24 US US11/569,148 patent/US20080064689A1/en not_active Abandoned
-
2005
- 2005-05-18 TW TW094116025A patent/TW200604185A/zh unknown
- 2005-05-24 BR BRPI0511554-0A patent/BRPI0511554A/pt not_active Application Discontinuation
- 2005-05-24 MX MXPA06013539A patent/MXPA06013539A/es not_active Application Discontinuation
- 2005-05-24 KR KR1020067027174A patent/KR20070027614A/ko not_active Withdrawn
- 2005-05-24 EP EP05746731A patent/EP1753756A1/en not_active Withdrawn
- 2005-05-24 AU AU2005247663A patent/AU2005247663A1/en not_active Abandoned
- 2005-05-24 AR ARP050102159A patent/AR049121A1/es unknown
- 2005-05-24 JP JP2007514084A patent/JP2008500315A/ja active Pending
- 2005-05-24 CA CA002567454A patent/CA2567454A1/en not_active Abandoned
- 2005-05-24 WO PCT/GB2005/002040 patent/WO2005116021A1/en not_active Ceased
- 2005-05-25 UY UY28924A patent/UY28924A1/es not_active Application Discontinuation
-
2006
- 2006-11-16 IL IL179348A patent/IL179348A0/en unknown
- 2006-12-19 NO NO20065863A patent/NO20065863L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| KR20070027614A (ko) | 2007-03-09 |
| JP2008500315A (ja) | 2008-01-10 |
| AR049121A1 (es) | 2006-06-28 |
| IL179348A0 (en) | 2007-03-08 |
| AU2005247663A1 (en) | 2005-12-08 |
| WO2005116021A1 (en) | 2005-12-08 |
| CA2567454A1 (en) | 2005-12-08 |
| EP1753756A1 (en) | 2007-02-21 |
| US20080064689A1 (en) | 2008-03-13 |
| BRPI0511554A (pt) | 2008-01-02 |
| MXPA06013539A (es) | 2007-01-26 |
| TW200604185A (en) | 2006-02-01 |
| UY28924A1 (es) | 2005-12-30 |
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| FC2A | Withdrawal, rejection or dismissal of laid open patent application |