NO20065863L - 3-[4-(6-(4,5-dihydroisoksazol-3-yl]pyridin-3-yl)-3-fenyl]-5-(1 H,1,2,3-triazol-1-yl-metyl)-1,3-oksazolidin-2-oner som antibakterielle midler - Google Patents

3-[4-(6-(4,5-dihydroisoksazol-3-yl]pyridin-3-yl)-3-fenyl]-5-(1 H,1,2,3-triazol-1-yl-metyl)-1,3-oksazolidin-2-oner som antibakterielle midler

Info

Publication number
NO20065863L
NO20065863L NO20065863A NO20065863A NO20065863L NO 20065863 L NO20065863 L NO 20065863L NO 20065863 A NO20065863 A NO 20065863A NO 20065863 A NO20065863 A NO 20065863A NO 20065863 L NO20065863 L NO 20065863L
Authority
NO
Norway
Prior art keywords
methyl
optionally substituted
antibacterial agents
dihydroisoxazol
oxazolidin
Prior art date
Application number
NO20065863A
Other languages
English (en)
Norwegian (no)
Inventor
Daniel Robert Carcanague
Michael Barry Gravenstock
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB0411594A external-priority patent/GB0411594D0/en
Priority claimed from GB0500055A external-priority patent/GB0500055D0/en
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of NO20065863L publication Critical patent/NO20065863L/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
NO20065863A 2004-05-25 2006-12-19 3-[4-(6-(4,5-dihydroisoksazol-3-yl]pyridin-3-yl)-3-fenyl]-5-(1 H,1,2,3-triazol-1-yl-metyl)-1,3-oksazolidin-2-oner som antibakterielle midler NO20065863L (no)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB0411594A GB0411594D0 (en) 2004-05-25 2004-05-25 Chemical compounds
GB0500055A GB0500055D0 (en) 2005-01-05 2005-01-05 Chemical compounds
PCT/GB2005/002040 WO2005116021A1 (en) 2004-05-25 2005-05-24 3-[4-(6-{4,5-dihydroisoxazol-3-yl}pyridin-3-yl)-3-phenyl]-5-(1h-1,2,3-triazol-1-ylmethyl)-1,3-oxazolidin-2-ones as antibacterial agents

Publications (1)

Publication Number Publication Date
NO20065863L true NO20065863L (no) 2007-02-20

Family

ID=34968779

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20065863A NO20065863L (no) 2004-05-25 2006-12-19 3-[4-(6-(4,5-dihydroisoksazol-3-yl]pyridin-3-yl)-3-fenyl]-5-(1 H,1,2,3-triazol-1-yl-metyl)-1,3-oksazolidin-2-oner som antibakterielle midler

Country Status (14)

Country Link
US (1) US20080064689A1 (pt)
EP (1) EP1753756A1 (pt)
JP (1) JP2008500315A (pt)
KR (1) KR20070027614A (pt)
AR (1) AR049121A1 (pt)
AU (1) AU2005247663A1 (pt)
BR (1) BRPI0511554A (pt)
CA (1) CA2567454A1 (pt)
IL (1) IL179348A0 (pt)
MX (1) MXPA06013539A (pt)
NO (1) NO20065863L (pt)
TW (1) TW200604185A (pt)
UY (1) UY28924A1 (pt)
WO (1) WO2005116021A1 (pt)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR100854211B1 (ko) * 2003-12-18 2008-08-26 동아제약주식회사 신규한 옥사졸리디논 유도체, 그의 제조방법 및 이를유효성분으로 하는 항생제용 약학 조성물
KR100848232B1 (ko) * 2007-04-12 2008-07-24 일동제약주식회사 신규 헤테로 고리 또는 알콕시아미노메틸 옥사졸리디논 및그 제조방법
RU2659792C1 (ru) 2008-10-10 2018-07-04 Мерк Шарп Энд Домэ Корп. Оксазолидиноны и способ их очистки
CN102224151A (zh) 2008-11-20 2011-10-19 万能药生物有限公司 新的抗微生物剂
MY156354A (en) 2009-02-03 2016-02-15 Merck Sharp & Dohme Crystalline form of r)-3-(4-(2-(2-methyltetrazol-5-yl)pyridin-5-yl)-3-fluorophenyl)-5-hydroxymethyl oxazolidin-2-one dihydrogen phosphate
US8580767B2 (en) * 2009-05-28 2013-11-12 Trius Therapeutics, Inc. Oxazolidinone containing dimer compounds, compositions and methods to make and use
KR20120106697A (ko) 2009-06-26 2012-09-26 파나세아 바이오테크 리미티드 신규 아자비시클로헥산
WO2011130419A2 (en) * 2010-04-13 2011-10-20 The Regents Of The University Of California Broad spectrum antiviral and antiparasitic agents
JP6610905B2 (ja) * 2015-02-27 2019-11-27 オーピーバイオファクトリー株式会社 カケロマイシンおよびその誘導体の製造方法
CN111471041B (zh) * 2019-01-23 2022-09-20 中国科学院上海药物研究所 一种噁唑烷酮类抗菌药物中间体的合成方法
WO2021000297A1 (en) 2019-07-03 2021-01-07 Merck Sharp & Dohme Corp. Compounds and methods of use thereof as antibacterial agents

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SI1427711T1 (sl) * 2001-09-11 2005-12-31 Astrazeneca Ab Oksazolidinonski in/ali izoksazolinski derivati kot antibakterijska sredstva
MXPA05005651A (es) * 2002-11-28 2005-07-27 Astrazeneca Ab Derivados de oxazolidinona y/o isoxazolina como agentes antibacterianos.
GB0227701D0 (en) * 2002-11-28 2003-01-08 Astrazeneca Ab Chemical compounds
TW200500360A (en) * 2003-03-01 2005-01-01 Astrazeneca Ab Hydroxymethyl compounds

Also Published As

Publication number Publication date
KR20070027614A (ko) 2007-03-09
JP2008500315A (ja) 2008-01-10
AR049121A1 (es) 2006-06-28
IL179348A0 (en) 2007-03-08
AU2005247663A1 (en) 2005-12-08
WO2005116021A1 (en) 2005-12-08
CA2567454A1 (en) 2005-12-08
EP1753756A1 (en) 2007-02-21
US20080064689A1 (en) 2008-03-13
BRPI0511554A (pt) 2008-01-02
MXPA06013539A (es) 2007-01-26
TW200604185A (en) 2006-02-01
UY28924A1 (es) 2005-12-30

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