NO20074055L - Prosesser for a fremstille 4-(fenoksy-5-metylpyrimidin-4-yloksy)piperidin-1-karboksylsyrederivater og relaterte forbindelser - Google Patents
Prosesser for a fremstille 4-(fenoksy-5-metylpyrimidin-4-yloksy)piperidin-1-karboksylsyrederivater og relaterte forbindelserInfo
- Publication number
- NO20074055L NO20074055L NO20074055A NO20074055A NO20074055L NO 20074055 L NO20074055 L NO 20074055L NO 20074055 A NO20074055 A NO 20074055A NO 20074055 A NO20074055 A NO 20074055A NO 20074055 L NO20074055 L NO 20074055L
- Authority
- NO
- Norway
- Prior art keywords
- methylpyrimidin
- yloxy
- piperidine
- phenoxy
- preparing
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 title abstract 5
- LKLZLFOKCZLKDX-UHFFFAOYSA-N 4-(5-methyl-2-phenoxypyrimidin-4-yl)oxypiperidine-1-carboxylic acid Chemical class N1=C(OC2CCN(CC2)C(O)=O)C(C)=CN=C1OC1=CC=CC=C1 LKLZLFOKCZLKDX-UHFFFAOYSA-N 0.000 title 1
- 150000003839 salts Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Diabetes (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Life Sciences & Earth Sciences (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Emergency Medicine (AREA)
- Endocrinology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Hydrogenated Pyridines (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US64262705P | 2005-01-10 | 2005-01-10 | |
| PCT/US2006/000565 WO2006076243A1 (en) | 2005-01-10 | 2006-01-09 | Processes for preparing 4-(phenoxy-5-methyl-pyrimidin-4-yloxy)piperidine-1-carboxylic acid derivatives and related compounds |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| NO20074055L true NO20074055L (no) | 2007-09-25 |
Family
ID=36297260
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO20074055A NO20074055L (no) | 2005-01-10 | 2007-08-06 | Prosesser for a fremstille 4-(fenoksy-5-metylpyrimidin-4-yloksy)piperidin-1-karboksylsyrederivater og relaterte forbindelser |
Country Status (29)
| Country | Link |
|---|---|
| US (1) | US7812159B2 (ru) |
| EP (1) | EP1838697B1 (ru) |
| JP (1) | JP2008526881A (ru) |
| KR (1) | KR20070098906A (ru) |
| CN (1) | CN101115739A (ru) |
| AR (1) | AR056917A1 (ru) |
| AT (1) | ATE462701T1 (ru) |
| AU (1) | AU2006205176A1 (ru) |
| BR (1) | BRPI0606676A2 (ru) |
| CA (1) | CA2593344A1 (ru) |
| CR (1) | CR9221A (ru) |
| DE (1) | DE602006013271D1 (ru) |
| DK (1) | DK1838697T3 (ru) |
| DO (1) | DOP2006000010A (ru) |
| EA (1) | EA014156B1 (ru) |
| ES (1) | ES2341281T3 (ru) |
| GE (1) | GEP20105071B (ru) |
| GT (1) | GT200600007A (ru) |
| HN (1) | HN2006000970A (ru) |
| IL (1) | IL184366A0 (ru) |
| MX (1) | MX2007008377A (ru) |
| NO (1) | NO20074055L (ru) |
| NZ (1) | NZ556218A (ru) |
| PE (2) | PE20091401A1 (ru) |
| SG (1) | SG158864A1 (ru) |
| TW (1) | TW200637844A (ru) |
| UA (1) | UA92733C2 (ru) |
| WO (1) | WO2006076243A1 (ru) |
| ZA (1) | ZA200705473B (ru) |
Families Citing this family (17)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN102558155A (zh) | 2003-01-14 | 2012-07-11 | 阿伦纳药品公司 | 作为代谢调节剂的芳基和杂芳基衍生物及其所涉及的疾病如糖尿病和高血糖症的预防和治疗 |
| AR045047A1 (es) * | 2003-07-11 | 2005-10-12 | Arena Pharm Inc | Derivados arilo y heteroarilo trisustituidos como moduladores del metabolismo y de la profilaxis y tratamiento de desordenes relacionados con los mismos |
| MY148521A (en) * | 2005-01-10 | 2013-04-30 | Arena Pharm Inc | Substituted pyridinyl and pyrimidinyl derivatives as modulators of metabolism and the treatment of disorders related thereto |
| US20110166176A1 (en) * | 2008-02-22 | 2011-07-07 | Irm Llc | Compounds and compositions as modulators of gpr119 activity |
| CA2786994C (en) | 2010-01-27 | 2018-01-16 | Arena Pharmaceuticals, Inc. | Processes for the preparation of (r)-2-(7-(4-cyclopentyl-3-(trifluoromethyl)benzyloxy)-1,2,3,4-tetrahydrocyclopenta[b]indol-3-yl)acetic acid and salts thereof |
| EP2547339A1 (en) | 2010-03-18 | 2013-01-23 | Boehringer Ingelheim International GmbH | Combination of a gpr119 agonist and the dpp-iv inhibitor linagliptin for use in the treatment of diabetes and related conditions |
| WO2012025811A1 (en) | 2010-08-23 | 2012-03-01 | Lupin Limited | Indolylpyrimidines as modulators of gpr119 |
| MX2013003184A (es) | 2010-09-22 | 2013-06-07 | Arena Pharm Inc | Moduladores del receptor gpr119 y el tratamiento de transtornos relacionados con el mismo. |
| EP2643311A1 (en) | 2010-11-26 | 2013-10-02 | Lupin Limited | Bicyclic gpr119 modulators |
| AU2012267556B9 (en) | 2011-06-09 | 2017-05-11 | Rhizen Pharmaceuticals Sa | Novel compounds as modulators of GPR-119 |
| AU2016205361C1 (en) | 2015-01-06 | 2021-04-08 | Arena Pharmaceuticals, Inc. | Methods of treating conditions related to the S1P1 receptor |
| PL3310760T3 (pl) | 2015-06-22 | 2023-03-06 | Arena Pharmaceuticals, Inc. | Krystaliczna sól L-argininy kwasu (R)-2-(7-(4-cyklopentylo-3-(trifluorometylo)benzyloksy)- 1,2,3,4-tetrahydrocyklo-penta[b]indol-3-ilo)octowego do zastosowania w zaburzeniach związanych z receptorem S1P1 |
| TW201825458A (zh) | 2016-09-20 | 2018-07-16 | 英商葛蘭素史克智慧財產（第二）有限公司 | Ｔｒｐｖ４拮抗劑 |
| KR20190049865A (ko) | 2016-09-20 | 2019-05-09 | 글락소스미스클라인 인털렉츄얼 프로퍼티 (넘버 2) 리미티드 | Trpv4 길항제 |
| WO2018055527A1 (en) | 2016-09-20 | 2018-03-29 | Glaxosmithkline Intellectual Property (No.2) Limited | Trpv4 antagonists |
| KR20190116416A (ko) | 2017-02-16 | 2019-10-14 | 아레나 파마슈티칼스, 인크. | 원발 담즙성 담관염을 치료하기 위한 화합물 및 방법 |
| AU2019280822A1 (en) | 2018-06-06 | 2021-01-07 | Arena Pharmaceuticals, Inc. | Methods of treating conditions related to the S1P1 receptor |
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| WO2004076413A2 (en) | 2003-02-24 | 2004-09-10 | Arena Pharmaceuticals, Inc. | Phenyl- and pyridylpiperidine-derivatives as modulators of glucose metabolism |
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| AR045047A1 (es) | 2003-07-11 | 2005-10-12 | Arena Pharm Inc | Derivados arilo y heteroarilo trisustituidos como moduladores del metabolismo y de la profilaxis y tratamiento de desordenes relacionados con los mismos |
| TWI335328B (en) | 2003-07-14 | 2011-01-01 | Arena Pharm Inc | Fused-aryl and heteroaryl derivatives as modulators of metabolism and the prophylaxis and treatment of disorders related hereto |
| MY148521A (en) | 2005-01-10 | 2013-04-30 | Arena Pharm Inc | Substituted pyridinyl and pyrimidinyl derivatives as modulators of metabolism and the treatment of disorders related thereto |
-
2006
- 2006-01-05 DO DO2006000010A patent/DOP2006000010A/es unknown
- 2006-01-06 PE PE2009000963A patent/PE20091401A1/es not_active Application Discontinuation
- 2006-01-06 PE PE2006000044A patent/PE20060836A1/es not_active Application Discontinuation
- 2006-01-09 HN HN2006000970A patent/HN2006000970A/es unknown
- 2006-01-09 DK DK06717730.3T patent/DK1838697T3/da active
- 2006-01-09 AT AT06717730T patent/ATE462701T1/de not_active IP Right Cessation
- 2006-01-09 ES ES06717730T patent/ES2341281T3/es not_active Expired - Lifetime
- 2006-01-09 GE GEAP200610222A patent/GEP20105071B/en unknown
- 2006-01-09 JP JP2007550519A patent/JP2008526881A/ja not_active Withdrawn
- 2006-01-09 MX MX2007008377A patent/MX2007008377A/es active IP Right Grant
- 2006-01-09 WO PCT/US2006/000565 patent/WO2006076243A1/en not_active Ceased
- 2006-01-09 UA UAA200709151A patent/UA92733C2/ru unknown
- 2006-01-09 DE DE602006013271T patent/DE602006013271D1/de not_active Expired - Lifetime
- 2006-01-09 SG SG201000106-3A patent/SG158864A1/en unknown
- 2006-01-09 NZ NZ556218A patent/NZ556218A/en not_active IP Right Cessation
- 2006-01-09 EA EA200701470A patent/EA014156B1/ru not_active IP Right Cessation
- 2006-01-09 US US11/327,923 patent/US7812159B2/en not_active Expired - Fee Related
- 2006-01-09 GT GT200600007A patent/GT200600007A/es unknown
- 2006-01-09 EP EP06717730A patent/EP1838697B1/en not_active Expired - Lifetime
- 2006-01-09 AU AU2006205176A patent/AU2006205176A1/en not_active Withdrawn
- 2006-01-09 BR BRPI0606676-3A patent/BRPI0606676A2/pt not_active IP Right Cessation
- 2006-01-09 AR ARP060100070A patent/AR056917A1/es not_active Application Discontinuation
- 2006-01-09 CN CNA2006800018668A patent/CN101115739A/zh not_active Withdrawn
- 2006-01-09 CA CA002593344A patent/CA2593344A1/en not_active Withdrawn
- 2006-01-09 KR KR1020077018267A patent/KR20070098906A/ko not_active Withdrawn
- 2006-01-09 TW TW095100805A patent/TW200637844A/zh unknown
-
2007
- 2007-07-02 CR CR9221A patent/CR9221A/es not_active Application Discontinuation
- 2007-07-02 IL IL184366A patent/IL184366A0/en unknown
- 2007-07-04 ZA ZA200705473A patent/ZA200705473B/xx unknown
- 2007-08-06 NO NO20074055A patent/NO20074055L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| JP2008526881A (ja) | 2008-07-24 |
| US20060155129A1 (en) | 2006-07-13 |
| HN2006000970A (es) | 2010-04-19 |
| DK1838697T3 (da) | 2010-06-28 |
| HK1102810A1 (en) | 2007-12-07 |
| EP1838697B1 (en) | 2010-03-31 |
| PE20060836A1 (es) | 2006-09-02 |
| AU2006205176A1 (en) | 2006-07-20 |
| EA014156B1 (ru) | 2010-10-29 |
| GT200600007A (es) | 2006-08-01 |
| ES2341281T3 (es) | 2010-06-17 |
| GEP20105071B (en) | 2010-09-10 |
| KR20070098906A (ko) | 2007-10-05 |
| EA200701470A1 (ru) | 2008-02-28 |
| UA92733C2 (ru) | 2010-12-10 |
| CR9221A (es) | 2007-10-23 |
| IL184366A0 (en) | 2007-10-31 |
| DE602006013271D1 (de) | 2010-05-12 |
| CA2593344A1 (en) | 2006-07-20 |
| DOP2006000010A (es) | 2006-07-31 |
| TW200637844A (en) | 2006-11-01 |
| ZA200705473B (en) | 2009-07-29 |
| CN101115739A (zh) | 2008-01-30 |
| NZ556218A (en) | 2010-10-29 |
| ATE462701T1 (de) | 2010-04-15 |
| US7812159B2 (en) | 2010-10-12 |
| BRPI0606676A2 (pt) | 2009-07-07 |
| SG158864A1 (en) | 2010-02-26 |
| EP1838697A1 (en) | 2007-10-03 |
| WO2006076243A1 (en) | 2006-07-20 |
| AR056917A1 (es) | 2007-11-07 |
| MX2007008377A (es) | 2007-09-07 |
| PE20091401A1 (es) | 2009-09-18 |
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