NO20074823L - Rasagilin-formuleringer med forbedret innholdsensartethet - Google Patents

Rasagilin-formuleringer med forbedret innholdsensartethet

Info

Publication number
NO20074823L
NO20074823L NO20074823A NO20074823A NO20074823L NO 20074823 L NO20074823 L NO 20074823L NO 20074823 A NO20074823 A NO 20074823A NO 20074823 A NO20074823 A NO 20074823A NO 20074823 L NO20074823 L NO 20074823L
Authority
NO
Norway
Prior art keywords
formulations
rasagilin
content uniformity
improved content
amino
Prior art date
Application number
NO20074823A
Other languages
English (en)
Inventor
Berger Tirtza Peskin
Original Assignee
Teva Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=36927751&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO20074823(L) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Teva Pharma filed Critical Teva Pharma
Publication of NO20074823L publication Critical patent/NO20074823L/no

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/205—Amine addition salts of organic acids; Inner quaternary ammonium salts, e.g. betaine, carnitine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16—Anti-Parkinson drugs
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2059—Starch, including chemically or physically modified derivatives; Amylose; Amylopectin; Dextrin

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Molecular Biology (AREA)
  • Biophysics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Psychology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

Oppfinnelsen angår farmasøytiske formuleringer av R(+)-N-propargyl- 1 -aminoindansalter med økt innholdsensartethet, fremgangsmåte for fremstilling av sammensetningene og deres anvendelse.
NO20074823A 2005-02-23 2007-09-21 Rasagilin-formuleringer med forbedret innholdsensartethet NO20074823L (no)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US65562205P 2005-02-23 2005-02-23
US72090805P 2005-09-27 2005-09-27
PCT/US2006/006252 WO2006091657A1 (en) 2005-02-23 2006-02-22 Rasagiline formulations of improved content uniformity

Publications (1)

Publication Number Publication Date
NO20074823L true NO20074823L (no) 2007-11-16

Family

ID=36927751

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20074823A NO20074823L (no) 2005-02-23 2007-09-21 Rasagilin-formuleringer med forbedret innholdsensartethet

Country Status (15)

Country Link
US (1) US7815942B2 (no)
EP (1) EP1848402B2 (no)
JP (2) JP5738509B2 (no)
KR (5) KR20070111534A (no)
AU (1) AU2006216696B2 (no)
BR (1) BRPI0608209A2 (no)
CA (2) CA2901244A1 (no)
ES (1) ES2586412T5 (no)
IL (2) IL184033A0 (no)
IS (1) IS8669A (no)
MX (1) MX2007010233A (no)
NO (1) NO20074823L (no)
NZ (1) NZ560660A (no)
RU (1) RU2404746C2 (no)
WO (1) WO2006091657A1 (no)

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EP1838326A4 (en) * 2005-02-02 2009-09-30 Teva Pharma PROCESS FOR PREPARING POLYPEPTIDE MIXTURES BY HYDROGENOLYSIS
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JP5738509B2 (ja) 2005-02-23 2015-06-24 テバ ファーマシューティカル インダストリーズ リミティド 内容物均一性が改善されたラサギリン製剤
CN101622225B (zh) * 2005-11-17 2015-04-15 泰华制药工业有限公司 炔丙基氨基茚分离方法
US7572834B1 (en) 2005-12-06 2009-08-11 Teva Pharmaceutical Industries, Ltd. Rasagiline formulations and processes for their preparation
JP5701485B2 (ja) 2006-02-21 2015-04-15 テバ ファーマシューティカル インダストリーズ リミティド 多系統萎縮症の治療のためのラサギリンの使用
WO2007117431A2 (en) 2006-04-03 2007-10-18 Teva Pharmaceutical Industries, Ltd. Use of rasagiline for the treatment of restless legs syndrome
EP1892233A1 (de) 2006-08-18 2008-02-27 Ratiopharm GmbH Neue Salze des Wirkstoffs Rasagilin
CN101557706B (zh) * 2006-12-14 2013-08-07 泰华制药工业有限公司 雷沙吉兰碱结晶固体
NZ577623A (en) * 2006-12-14 2011-05-27 Teva Pharma Tannate salt of rasagiline
EP1987816A1 (de) * 2007-04-30 2008-11-05 Ratiopharm GmbH Adsorbate eines Rasagilinsalzes mit einem wasserlöslichen Hilfsstoff
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MX2010007601A (es) * 2008-01-11 2010-08-03 Teva Pharma Formulaciones de rasagilina, su preparacion y uso.
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CN102065853A (zh) * 2008-06-19 2011-05-18 泰华制药工业有限公司 制备和干燥固体雷沙吉兰碱的方法
EP2299993A4 (en) 2008-06-19 2014-08-20 Teva Pharma PROCESS FOR PURIFYING THE BASE OF RASAGILINE
EP2358658A4 (en) * 2008-11-20 2012-11-14 Reddys Lab Ltd Dr PREPARATION OF RASAGILIN AND ITS SALTS
DE102008064061A1 (de) 2008-12-19 2010-06-24 Ratiopharm Gmbh Feste Zusammensetzung mit dem Wirkstoff Rasagilin
US8080584B2 (en) * 2009-01-23 2011-12-20 Teva Pharmaceuticals Industries, Ltd. Delayed release rasagiline citrate formulation
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WO2010111264A2 (en) * 2009-03-24 2010-09-30 Dr. Reddy's Laboratories Ltd. Rasagiline formulations
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CN101622225B (zh) * 2005-11-17 2015-04-15 泰华制药工业有限公司 炔丙基氨基茚分离方法
US7572834B1 (en) * 2005-12-06 2009-08-11 Teva Pharmaceutical Industries, Ltd. Rasagiline formulations and processes for their preparation
JP5701485B2 (ja) 2006-02-21 2015-04-15 テバ ファーマシューティカル インダストリーズ リミティド 多系統萎縮症の治療のためのラサギリンの使用
WO2007117431A2 (en) 2006-04-03 2007-10-18 Teva Pharmaceutical Industries, Ltd. Use of rasagiline for the treatment of restless legs syndrome
EP1892233A1 (de) 2006-08-18 2008-02-27 Ratiopharm GmbH Neue Salze des Wirkstoffs Rasagilin
NZ577623A (en) * 2006-12-14 2011-05-27 Teva Pharma Tannate salt of rasagiline
CN101557706B (zh) 2006-12-14 2013-08-07 泰华制药工业有限公司 雷沙吉兰碱结晶固体
EP1987816A1 (de) 2007-04-30 2008-11-05 Ratiopharm GmbH Adsorbate eines Rasagilinsalzes mit einem wasserlöslichen Hilfsstoff
MX2010007601A (es) * 2008-01-11 2010-08-03 Teva Pharma Formulaciones de rasagilina, su preparacion y uso.

Also Published As

Publication number Publication date
BRPI0608209A2 (pt) 2010-11-09
HK1103366A1 (zh) 2007-12-21
EP1848402A4 (en) 2012-01-18
IL244802A0 (en) 2016-04-21
KR20070111534A (ko) 2007-11-21
US20060188581A1 (en) 2006-08-24
IL244802A (en) 2016-08-31
JP5738509B2 (ja) 2015-06-24
RU2404746C2 (ru) 2010-11-27
KR20170023211A (ko) 2017-03-02
MX2007010233A (es) 2007-11-07
IL184033A0 (en) 2007-10-31
EP1848402A1 (en) 2007-10-31
NZ560660A (en) 2010-11-26
IS8669A (is) 2007-08-15
CA2600011C (en) 2015-11-10
KR20140103356A (ko) 2014-08-26
EP1848402B2 (en) 2019-02-20
WO2006091657A1 (en) 2006-08-31
JP2013139452A (ja) 2013-07-18
CA2600011A1 (en) 2006-08-31
KR20130129300A (ko) 2013-11-27
JP2008531572A (ja) 2008-08-14
CA2901244A1 (en) 2006-08-31
RU2007135169A (ru) 2009-03-27
ES2586412T3 (es) 2016-10-14
ES2586412T5 (es) 2019-05-16
US7815942B2 (en) 2010-10-19
EP1848402B1 (en) 2016-05-11
AU2006216696A1 (en) 2006-08-31
AU2006216696B2 (en) 2011-08-18
KR20180026580A (ko) 2018-03-12

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