NO20075399L - Benzimidazolerivat og anvendelse derav - Google Patents

Benzimidazolerivat og anvendelse derav

Info

Publication number
NO20075399L
NO20075399L NO20075399A NO20075399A NO20075399L NO 20075399 L NO20075399 L NO 20075399L NO 20075399 A NO20075399 A NO 20075399A NO 20075399 A NO20075399 A NO 20075399A NO 20075399 L NO20075399 L NO 20075399L
Authority
NO
Norway
Prior art keywords
methyl
benzimidazole derivative
oxo
pharmaceutical
benzimidazole
Prior art date
Application number
NO20075399A
Other languages
English (en)
Norwegian (no)
Inventor
Takanobu Kuroita
Mami Ojima
Junko Ban
Original Assignee
Takeda Pharmaceutical
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Takeda Pharmaceutical filed Critical Takeda Pharmaceutical
Publication of NO20075399L publication Critical patent/NO20075399L/no

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    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/10Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
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    • C07D413/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
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    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4245Oxadiazoles
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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/14Vasoprotectives; Antihaemorrhoidals; Drugs for varicose therapy; Capillary stabilisers

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NO20075399A 2005-03-30 2007-10-23 Benzimidazolerivat og anvendelse derav NO20075399L (no)

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WO2007097452A1 (ja) * 2006-02-27 2007-08-30 Takeda Pharmaceutical Company Limited 医薬用ブリスターパッケージ
EP2068812B9 (en) * 2006-09-25 2012-08-08 Takeda Pharmaceutical Company Limited Medicinal package
KR101126383B1 (ko) * 2007-02-07 2012-04-12 교와 핫꼬 기린 가부시키가이샤 3환계 화합물
AR072883A1 (es) 2008-07-31 2010-09-29 Takeda Pharmaceutical COMPOSICIoN FARMACÉUTICA SoLIDA CON EL COMPUESTO (5-METIL-2-OXO-1,3-DIOXOL-4-IL)METIL2-ETOXI-1-{[2' -(5-OXO-4,5-DIHIDRO-1,2,4-OXADIAZOL-3-IL)BIFENIL-4-IL]METIL}-1H-BENCIMIDAZOL-7-CARBOXILATO Y UN DIURÉTICO PARA LA PROFILAXIS O TRATAMIENTO DE ENFERMEDADES DEL APARATO CIRCULATORIO.
EP2327690A4 (en) 2008-08-06 2012-03-28 Kyowa Hakko Kirin Co Ltd TRICYCLIC CONNECTION
TW201014850A (en) 2008-09-25 2010-04-16 Takeda Pharmaceutical Solid pharmaceutical composition
EP2673274B1 (en) * 2011-02-08 2019-07-17 Jubilant Generics Limited An improved process for the preparation of azilsartan medoxomil
CZ304252B6 (cs) * 2011-04-11 2014-01-29 Zentiva, K. S. Způsob výroby 2-ethoxy-1-((2´-(5-oxo-4,5-dihydro-1,2,4-oxadiazol-3-yl)bifenyl-4-yl)methyl)-1H-benzo[d]imidazol-7-karboxylátů a jejich převedení na azilsartan
KR101275092B1 (ko) * 2011-05-19 2013-06-17 한미정밀화학주식회사 아질사르탄의 개선된 제조방법
CN102827153B (zh) * 2011-06-14 2016-10-05 江苏豪森药业集团有限公司 阿齐沙坦的晶型及其制备方法
JP6281735B2 (ja) * 2013-03-19 2018-02-21 トーアエイヨー株式会社 急性心不全治療薬の評価方法、及び、急性心不全モデルの作製方法

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DK1863801T3 (da) 2010-11-15
GEP20115138B (en) 2011-01-10
RU2407742C2 (ru) 2010-12-27
MY146254A (en) 2012-07-31
KR20070116648A (ko) 2007-12-10
PT1863801E (pt) 2010-11-19
IL185726A0 (en) 2008-01-06
SI1863801T1 (sl) 2010-12-31
NZ562887A (en) 2010-10-29
MA29438B1 (fr) 2008-05-02
JP2008534434A (ja) 2008-08-28
AR055755A1 (es) 2007-09-05
BRPI0608944A2 (pt) 2010-11-16
US20120172401A1 (en) 2012-07-05
RS20080510A (sr) 2009-07-15
EP1863801B1 (en) 2010-09-29
HRP20080552A9 (en) 2009-08-31
CY1111168T1 (el) 2015-06-11
JP2011190265A (ja) 2011-09-29
RU2007139928A (ru) 2009-05-10
EP1863801A2 (en) 2007-12-12
JP4795362B2 (ja) 2011-10-19
PL1863801T3 (pl) 2011-03-31
AU2006231418B2 (en) 2011-10-13
WO2006107062A2 (en) 2006-10-12
HK1115584A1 (en) 2008-12-05
DE602006017183D1 (de) 2010-11-11
AU2006231418A1 (en) 2006-10-12
IL185726A (en) 2012-07-31
CR9432A (es) 2008-02-04
TW200724539A (en) 2007-07-01
US20090054502A1 (en) 2009-02-26
PE20061195A1 (es) 2006-12-21
WO2006107062A3 (en) 2006-12-14
HRP20080552A2 (hr) 2009-03-31
CA2602624A1 (en) 2006-10-12

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