NO20075758L - Polymorfer av 3-0-(3',3'-dimetylsuccinyl) betulin syre di-N-metyl-D-glukamin - Google Patents

Polymorfer av 3-0-(3',3'-dimetylsuccinyl) betulin syre di-N-metyl-D-glukamin

Info

Publication number: NO20075758L
Authority: NO; Norway
Prior art keywords: dimethylsuccinyl; methyl; betulinic acid; glucamine; polymorphs
Prior art date: 2005-04-12

Application number

NO20075758A

Other languages

English (en)

Norwegian (no)

Inventor

Michael O'neil

Gary G Sweetapple

Randall M Walker

Arndt Err

Gunter Koch

David E Martin

Original Assignee

Panacos Pharmaceuticals Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2005-04-12

Filing date

2007-11-09

Publication date

2008-01-10

2007-11-09 Application filed by Panacos Pharmaceuticals Inc filed Critical Panacos Pharmaceuticals Inc

2008-01-10 Publication of NO20075758L publication Critical patent/NO20075758L/no

Links

YJEJKUQEXFSVCJ-WRFMNRASSA-N bevirimat Chemical compound C1C[C@H](OC(=O)CC(C)(C)C(O)=O)C(C)(C)[C@@H]2CC[C@@]3(C)[C@]4(C)CC[C@@]5(C(O)=O)CC[C@@H](C(=C)C)[C@@H]5[C@H]4CC[C@@H]3[C@]21C YJEJKUQEXFSVCJ-WRFMNRASSA-N 0.000 title abstract 2
239000008186 active pharmaceutical agent Substances 0.000 abstract 1
239000008194 pharmaceutical composition Substances 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J17/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, having an oxygen-containing hetero ring not condensed with the cyclopenta(a)hydrophenanthrene skeleton
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A61K31/7028—Compounds having saccharide radicals attached to non-saccharide compounds by glycosidic linkages
- A61K31/7034—Compounds having saccharide radicals attached to non-saccharide compounds by glycosidic linkages attached to a carbocyclic compound, e.g. phloridzin
- A61K31/704—Compounds having saccharide radicals attached to non-saccharide compounds by glycosidic linkages attached to a carbocyclic compound, e.g. phloridzin attached to a condensed carbocyclic ring system, e.g. sennosides, thiocolchicosides, escin, daunorubicin
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/18—Antivirals for RNA viruses for HIV

Landscapes

Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
Molecular Biology (AREA)
Virology (AREA)
Animal Behavior & Ethology (AREA)
Pharmacology & Pharmacy (AREA)
Medicinal Chemistry (AREA)
Communicable Diseases (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Oncology (AREA)
Epidemiology (AREA)
Tropical Medicine & Parasitology (AREA)
AIDS & HIV (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Steroid Compounds (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Preparation Of Compounds By Using Micro-Organisms (AREA)

NO20075758A 2005-04-12 2007-11-09 Polymorfer av 3-0-(3',3'-dimetylsuccinyl) betulin syre di-N-metyl-D-glukamin NO20075758L (no)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US67022705P	2005-04-12	2005-04-12
PCT/US2006/013640 WO2006110810A2 (en)	2005-04-12	2006-04-12	Polymorphs of 3-o-(3',3'-dimethylsuccinyl) betulinic acid di-n-methyl-d-glucamine

Publications (1)

Publication Number	Publication Date
NO20075758L true NO20075758L (no)	2008-01-10

Family

ID=37087667

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO20075758A NO20075758L (no)	2005-04-12	2007-11-09	Polymorfer av 3-0-(3',3'-dimetylsuccinyl) betulin syre di-N-metyl-D-glukamin

Country Status (14)

Country	Link
US (1)	US7799768B2 (de)
EP (1)	EP1868613B1 (de)
JP (1)	JP2008535923A (de)
CN (1)	CN101160132A (de)
AT (1)	ATE548043T1 (de)
AU (1)	AU2006235486A1 (de)
BR (1)	BRPI0610668A2 (de)
CA (1)	CA2604720A1 (de)
ES (1)	ES2383534T3 (de)
IL (1)	IL186058A0 (de)
MX (1)	MX2007011981A (de)
NO (1)	NO20075758L (de)
RU (1)	RU2007141631A (de)
WO (1)	WO2006110810A2 (de)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
WO2008057420A2 (en)	2006-11-03	2008-05-15	Panacos Pharmaceuticals, Inc.	Extended triterpene derivatives
WO2008091532A1 (en) *	2007-01-19	2008-07-31	Panacos Pharmaceuticals, Inc.	Salts of 3-o-(3',3'-dimethylsuccinyl)betulinic acid and solid state forms thereof
US20080294115A1 (en) *	2007-05-22	2008-11-27	Chen Raymond H	Microscopic Tumor Injection Treatment
US20080294106A1 (en) *	2007-05-22	2008-11-27	Convergent Medical Solutions, Inc.	Multiple robotic injections of anesthesia based on scanned image
US20080294141A1 (en) *	2007-05-22	2008-11-27	Convergent Medical Solutions, Inc.	Multiple robotic injections of immunosuppressive drugs based on scanned image
US20080294107A1 (en) *	2007-05-22	2008-11-27	Convergent Medical Solutions, Inc.	Multiple robotic injections of prenatal medications based on scanned image
WO2009146240A1 (en) *	2008-05-27	2009-12-03	Convergent Medical Solutions, Inc.	Multiple robotic injections based on scanned image

Family Cites Families (25)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB1415601A (en)	1973-03-14	1975-11-26	Biorex Laboratories Ltd	Dihydrobetulinic acid derivatives
JPH01143832A (ja)	1987-12-01	1989-06-06	Toa Nenryo Kogyo Kk	制癌剤
WO1993007904A1 (en) *	1991-10-16	1993-04-29	Schering Corporation	Lipophilic oligosaccharide antibiotic salt compositions
FR2683531B1 (fr)	1991-11-13	1993-12-31	Rhone Poulenc Rorer Sa	Nouveaux derives du lupane, leur preparation et les compositions pharmaceutiques qui les contiennent.
US5643884A (en)	1993-08-09	1997-07-01	Glycomed Incorporated	Lupane triterpenoid derivatives
US5679828A (en)	1995-06-05	1997-10-21	Biotech Research Labs, Inc.	Betulinic acid and dihydrobetulinic acid derivatives and uses therefor
US5648888A (en) *	1995-12-27	1997-07-15	Hydro-Quebec	Power distribution substation
US5776912A (en) *	1996-12-20	1998-07-07	Schering Corporation	Lipophilic oligosaccharide antibiotic compositions
US6043245A (en)	1997-09-25	2000-03-28	Schering Corporation	Tetrahydrofuran antifungal phosphate
US6670345B1 (en) *	1997-09-30	2003-12-30	Dabur Research Foundation	Betulinic acid derivatives for inhabiting cancer growth and process for the manufacture of betulinic acid
NZ506623A (en) *	1998-03-02	2002-10-25	Univ North Carolina	Acylated betulin and dihydrobetulin derivatives, preparation thereof and use in treatment of retroviral infections
US6043254A (en) *	1998-04-03	2000-03-28	Boehringer Ingelheim Pharma Kg	Indolinones having kinase-inhibiting activity
EP1189607A2 (de)	1999-04-07	2002-03-27	Washington State University Research Foundation	Anti-tumor aktivität von vitamin e, cholesterol, taxol und betulinsäurederivaten
US6147077A (en) *	1999-04-29	2000-11-14	Sepracor Inc.	2R,4S-hydroxyitraconazole isomers
RU2174982C2 (ru)	1999-11-05	2001-10-20	Институт органической химии Уфимского научного центра РАН	3,28-ди-о-никотинат бетулина, проявляющий гепатопротекторную и анти-вич активность
CA2406562C (en) *	2000-05-08	2009-09-15	Janssen Pharmaceutica N.V.	Hiv replication inhibiting pyrimidines and triazines
JP2004509972A (ja)	2000-09-29	2004-04-02	リージェンツ　オブ　ザ　ユニバーシティ　オブ　ミネソタ	酵母に対する殺真菌活性を有するトリテルペン
JP4179768B2 (ja)	2001-10-01	2008-11-12	ポーラ化成工業株式会社	トリテルペン誘導体及びそれを含有する化合物
US7365221B2 (en) *	2002-09-26	2008-04-29	Panacos Pharmaceuticals, Inc.	Monoacylated betulin and dihydrobetulin derivatives, preparation thereof and use thereof
WO2004028455A2 (en) *	2002-09-26	2004-04-08	Panacos Pharmaceuticals, Inc.	Monoacylated betulin and dihydrobetulin derivatives, preparation thereof and use thereof
EP1675866A1 (de) *	2003-09-26	2006-07-05	Panacos Pharmaceuticals, Inc.	Neue triterpenderivate, deren herstellung und deren verwendung
EP1730163A4 (de)	2004-03-17	2009-12-30	Panacos Pharmaceuticals Inc	Pharmazeutische salze von 3-o-(3,3-dimethylsuccinyl)betulinsäure
TW200628161A (en) *	2004-11-12	2006-08-16	Panacos Pharmaceuticals Inc	Novel betulin derivatives, preparation thereof and use thereof
ZA200805703B (en) *	2005-12-16	2009-10-28	Panacos Pharmaceuticals Inc	Preparation of pharmaceutical salts of 3-0-(3',3'-dimethyl-succinyl) betulinic acid
US8180205B2 (en)	2007-01-12	2012-05-15	Guoning Yao	Electrothermal oil radiator

2006
- 2006-04-12 BR BRPI0610668-4A patent/BRPI0610668A2/pt not_active IP Right Cessation
- 2006-04-12 RU RU2007141631/04A patent/RU2007141631A/ru not_active Application Discontinuation
- 2006-04-12 JP JP2008506631A patent/JP2008535923A/ja not_active Withdrawn
- 2006-04-12 MX MX2007011981A patent/MX2007011981A/es not_active Application Discontinuation
- 2006-04-12 AT AT06749874T patent/ATE548043T1/de active
- 2006-04-12 ES ES06749874T patent/ES2383534T3/es not_active Expired - Lifetime
- 2006-04-12 CA CA002604720A patent/CA2604720A1/en not_active Abandoned
- 2006-04-12 US US11/401,960 patent/US7799768B2/en not_active Expired - Fee Related
- 2006-04-12 EP EP06749874A patent/EP1868613B1/de not_active Expired - Lifetime
- 2006-04-12 WO PCT/US2006/013640 patent/WO2006110810A2/en not_active Ceased
- 2006-04-12 CN CNA2006800121527A patent/CN101160132A/zh active Pending
- 2006-04-12 AU AU2006235486A patent/AU2006235486A1/en not_active Abandoned
2007
- 2007-09-19 IL IL186058A patent/IL186058A0/en unknown
- 2007-11-09 NO NO20075758A patent/NO20075758L/no not_active Application Discontinuation

Also Published As

Publication number	Publication date
EP1868613A4 (de)	2008-04-30
WO2006110810A2 (en)	2006-10-19
EP1868613A2 (de)	2007-12-26
IL186058A0 (en)	2008-08-07
JP2008535923A (ja)	2008-09-04
EP1868613B1 (de)	2012-03-07
ES2383534T3 (es)	2012-06-22
MX2007011981A (es)	2007-12-05
AU2006235486A1 (en)	2006-10-19
US20060252704A1 (en)	2006-11-09
WO2006110810A3 (en)	2007-03-29
BRPI0610668A2 (pt)	2010-07-13
ATE548043T1 (de)	2012-03-15
CA2604720A1 (en)	2006-10-19
RU2007141631A (ru)	2009-05-20
CN101160132A (zh)	2008-04-09
US7799768B2 (en)	2010-09-21

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Legal Events

Date	Code	Title	Description
2011-11-28	FC2A	Withdrawal, rejection or dismissal of laid open patent application