NO20081983L - Nye azetidinforbindelser nyttige i behandlingen av funksjonelle gastrointestinale forstyrrelser, IBS og funksjonell dyspepsi - Google Patents

Nye azetidinforbindelser nyttige i behandlingen av funksjonelle gastrointestinale forstyrrelser, IBS og funksjonell dyspepsi

Info

Publication number
NO20081983L
NO20081983L NO20081983A NO20081983A NO20081983L NO 20081983 L NO20081983 L NO 20081983L NO 20081983 A NO20081983 A NO 20081983A NO 20081983 A NO20081983 A NO 20081983A NO 20081983 L NO20081983 L NO 20081983L
Authority
NO
Norway
Prior art keywords
functional
ibs
treatment
gastrointestinal disorders
compounds useful
Prior art date
Application number
NO20081983A
Other languages
English (en)
Inventor
Sverker Von Unge
Sara Holmqvist
Rolf Bergman
Original Assignee
Albireo Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
Application filed by Albireo Ab filed Critical Albireo Ab
Publication of NO20081983L publication Critical patent/NO20081983L/no

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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/04—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/397—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having four-membered rings, e.g. azetidine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/06—Anti-spasmodics, e.g. drugs for colics, esophagic dyskinesia
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    • A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
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    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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    • C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/04—Ortho-condensed systems

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  • Chemical & Material Sciences (AREA)
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  • Pharmacology & Pharmacy (AREA)
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  • Neurology (AREA)
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Abstract

Foreliggende oppfinnelse angår nye acetidinforbindelser, farmasøytiske sammensetninger som inneholder dem og anvendelse av nevnte forbindelser ved behandling av funksjonelle gastrointestinale forstyrrelser, IBS og funksjonell dyspepsi. Forbindelsene er neurokinin (NK) antagonister. Foreliggende oppfinnelse angår videre fremgangsmåte for fremstilling av forbindelsene
NO20081983A 2005-09-29 2008-04-25 Nye azetidinforbindelser nyttige i behandlingen av funksjonelle gastrointestinale forstyrrelser, IBS og funksjonell dyspepsi NO20081983L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
SE0502150 2005-09-29
PCT/SE2006/001092 WO2007037743A1 (en) 2005-09-29 2006-09-27 Novel azetidine compounds useful in the treatment of functional gastrointestinal disorders, ibs and functional dyspepsia

Publications (1)

Publication Number Publication Date
NO20081983L true NO20081983L (no) 2008-06-27

Family

ID=37900052

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20081983A NO20081983L (no) 2005-09-29 2008-04-25 Nye azetidinforbindelser nyttige i behandlingen av funksjonelle gastrointestinale forstyrrelser, IBS og funksjonell dyspepsi

Country Status (15)

Country Link
US (1) US8288370B2 (no)
EP (1) EP1940845B1 (no)
JP (1) JP5139985B2 (no)
KR (1) KR20080077096A (no)
CN (1) CN101316846A (no)
AR (1) AR057828A1 (no)
AU (1) AU2006295473B2 (no)
BR (1) BRPI0616581A2 (no)
CA (1) CA2624491C (no)
ES (1) ES2426259T3 (no)
NO (1) NO20081983L (no)
TW (1) TW200745122A (no)
UY (1) UY29818A1 (no)
WO (1) WO2007037743A1 (no)
ZA (1) ZA200802645B (no)

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CN104958297A (zh) * 2015-06-03 2015-10-07 周玉梅 一种用于麻醉镇静催眠的药物组合物及其应用
CN105663133B (zh) * 2016-03-07 2019-06-25 青岛市肿瘤医院 一种抑制淋巴瘤细胞增殖的药物组合物及其应用
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US8288370B2 (en) 2012-10-16
AR057828A1 (es) 2007-12-19
KR20080077096A (ko) 2008-08-21
EP1940845A4 (en) 2010-11-17
HK1121142A1 (en) 2009-04-17
US20100311713A1 (en) 2010-12-09
CA2624491C (en) 2014-01-14
BRPI0616581A2 (pt) 2011-06-21
AU2006295473B2 (en) 2011-11-10
JP2009510055A (ja) 2009-03-12
CA2624491A1 (en) 2007-04-05
EP1940845B1 (en) 2013-06-12
AU2006295473A1 (en) 2007-04-05
WO2007037743A1 (en) 2007-04-05
ZA200802645B (en) 2008-12-31
UY29818A1 (es) 2007-04-30
JP5139985B2 (ja) 2013-02-06
CN101316846A (zh) 2008-12-03
TW200745122A (en) 2007-12-16
ES2426259T3 (es) 2013-10-22

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