MA30291B1 - Derives de l'azolopyridin-3-one en tant qu'inhibiteurs de la lipase endotheliale - Google Patents

Derives de l'azolopyridin-3-one en tant qu'inhibiteurs de la lipase endotheliale

Info

Publication number
MA30291B1
MA30291B1 MA31257A MA31257A MA30291B1 MA 30291 B1 MA30291 B1 MA 30291B1 MA 31257 A MA31257 A MA 31257A MA 31257 A MA31257 A MA 31257A MA 30291 B1 MA30291 B1 MA 30291B1
Authority
MA
Morocco
Prior art keywords
azolopyridin
inhibitors
derivatives
endothelial lipase
lipase
Prior art date
Application number
MA31257A
Other languages
English (en)
Inventor
Gerhard Zoller
Stefan Petry
Guenter Mueller
Norbert Tennagels
Original Assignee
Sanofi Aventis
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=38190768&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MA30291(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Sanofi Aventis filed Critical Sanofi Aventis
Publication of MA30291B1 publication Critical patent/MA30291B1/fr

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
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    • C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/04—Ortho-condensed systems

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Abstract

Titre : Dérivés de l'azolopyridin-3-one en tant qu'inhibiteurs de la lipase endothéliale La présente invention concerne des dérivés de l'azolopyridin-3-one de formule générale I avec les significations indiquées dans la description, leurs sels pharmaceutiquement utilisables et leur utilisation comme substances médicinales. Les composés sont des inhibiteurs de la lipase endothéliale.
MA31257A 2006-03-28 2008-09-25 Derives de l'azolopyridin-3-one en tant qu'inhibiteurs de la lipase endotheliale MA30291B1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE102006014688A DE102006014688A1 (de) 2006-03-28 2006-03-28 Azolopyridin-3-on-derivate als Inhibitoren von Lipasen und Phospholipasen

Publications (1)

Publication Number Publication Date
MA30291B1 true MA30291B1 (fr) 2009-03-02

Family

ID=38190768

Family Applications (1)

Application Number Title Priority Date Filing Date
MA31257A MA30291B1 (fr) 2006-03-28 2008-09-25 Derives de l'azolopyridin-3-one en tant qu'inhibiteurs de la lipase endotheliale

Country Status (17)

Country Link
US (1) US8148395B2 (fr)
EP (1) EP2001879B1 (fr)
JP (1) JP2009531357A (fr)
KR (1) KR20080104032A (fr)
CN (1) CN101415706A (fr)
AR (1) AR060158A1 (fr)
AU (1) AU2007229709A1 (fr)
BR (1) BRPI0709217A2 (fr)
CA (1) CA2647425A1 (fr)
DE (1) DE102006014688A1 (fr)
MA (1) MA30291B1 (fr)
MX (1) MX2008012127A (fr)
NO (1) NO20084418L (fr)
RU (1) RU2008142535A (fr)
TW (1) TW200813049A (fr)
WO (1) WO2007110216A1 (fr)
ZA (1) ZA200807135B (fr)

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US7217727B2 (en) * 2003-04-01 2007-05-15 Eli Lilly And Company Phospholipase inhibitors
DE102004005172A1 (de) * 2004-02-02 2005-08-18 Aventis Pharma Deutschland Gmbh Indazolderivate als Inhibitoren der Hormon Sensitiven Lipase

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AR060158A1 (es) 2008-05-28
US8148395B2 (en) 2012-04-03
EP2001879A1 (fr) 2008-12-17
NO20084418L (no) 2008-12-23
KR20080104032A (ko) 2008-11-28
AU2007229709A1 (en) 2007-10-04
EP2001879B1 (fr) 2013-08-21
BRPI0709217A2 (pt) 2011-07-12
RU2008142535A (ru) 2010-05-10
CN101415706A (zh) 2009-04-22
JP2009531357A (ja) 2009-09-03
TW200813049A (en) 2008-03-16
US20090054478A1 (en) 2009-02-26
MX2008012127A (es) 2008-10-03
DE102006014688A1 (de) 2007-10-04
CA2647425A1 (fr) 2007-10-04
WO2007110216A1 (fr) 2007-10-04

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