NO20090100L - Kontrollert frigjoringssystem for fremstilling derav - Google Patents

Kontrollert frigjoringssystem for fremstilling derav

Info

Publication number
NO20090100L
NO20090100L NO20090100A NO20090100A NO20090100L NO 20090100 L NO20090100 L NO 20090100L NO 20090100 A NO20090100 A NO 20090100A NO 20090100 A NO20090100 A NO 20090100A NO 20090100 L NO20090100 L NO 20090100L
Authority
NO
Norway
Prior art keywords
layer
pharmaceutically acceptable
controlled release
release system
layer containing
Prior art date
Application number
NO20090100A
Other languages
English (en)
Inventor
Thomas Friedl
Florian Sommer
Nantharat Pearnchob
Karl Gerhard Wagner
Original Assignee
Boehringer Ingelheim Int
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=38596345&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO20090100(L) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Boehringer Ingelheim Int filed Critical Boehringer Ingelheim Int
Publication of NO20090100L publication Critical patent/NO20090100L/no

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5073—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system

Landscapes

  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Oppfinnelsen omhandler et farmasøytisk kontrollert frigjøringssystem for administrering, spesielt oral administrering, av aktive substanser med pH-avhengige løseligheter, som omfatter a) et kjernemateriale inneholdende eller bestående av én eller flere farmasøytisk akseptable pH-modifiserere; b) eventuelt et isolerende lag, c) et første lag som inneholder eller består av én eller flere farmasøytisk akseptable vannuløselige polymerer; d) et andre lag som inneholder eller består av minst én aktiv substans som har en pH-avhengig løselighet; e) et tredje lag som inneholder eller består av én eller flere farmasøytisk akseptable polymerer som har anioniske eller ingen ioniske grupper; og f) eventuelt et fjerde lag, fortrinnsvis i form av en ytre beleggingslag. Det er tilveiebrakt en pH-uavhengig frigjøringsprofil av aktive substanser som har pH-avhengige løseligheter in vitro og vivo.
NO20090100A 2006-08-25 2009-01-08 Kontrollert frigjoringssystem for fremstilling derav NO20090100L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP06017754 2006-08-25
PCT/EP2007/058302 WO2008022932A2 (en) 2006-08-25 2007-08-10 Controlled release system and method for manufacturing the same

Publications (1)

Publication Number Publication Date
NO20090100L true NO20090100L (no) 2009-04-23

Family

ID=38596345

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20090100A NO20090100L (no) 2006-08-25 2009-01-08 Kontrollert frigjoringssystem for fremstilling derav

Country Status (19)

Country Link
US (1) US8512748B2 (no)
EP (1) EP2056797A2 (no)
JP (1) JP5220746B2 (no)
KR (1) KR20090045945A (no)
CN (2) CN104721168A (no)
AR (1) AR062321A1 (no)
AU (1) AU2007287639A1 (no)
BR (1) BRPI0716436B8 (no)
CA (1) CA2661613C (no)
CL (1) CL2007002358A1 (no)
CO (1) CO6150131A2 (no)
EA (1) EA200900270A1 (no)
IL (1) IL197129A (no)
MX (1) MX2009002031A (no)
NO (1) NO20090100L (no)
PE (1) PE20080738A1 (no)
TW (1) TW200817053A (no)
WO (1) WO2008022932A2 (no)
ZA (1) ZA200810781B (no)

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ZA200810781B (en) 2009-10-28
WO2008022932A2 (en) 2008-02-28
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EA200900270A1 (ru) 2009-08-28
CO6150131A2 (es) 2010-04-20
CA2661613C (en) 2016-01-26
PE20080738A1 (es) 2008-08-05
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WO2008022932A3 (en) 2008-07-24
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US8512748B2 (en) 2013-08-20
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