NO309190B1 - Neurobeskyttende kromanforbindelser og farmasöytisk blanding - Google Patents

Neurobeskyttende kromanforbindelser og farmasöytisk blanding Download PDF

Info

Publication number: NO309190B1
Authority: NO; Norway
Prior art keywords: hydroxy; fluorophenyl; piperidin; chroman; acid
Prior art date: 1994-01-31

Application number

NO963186A

Other languages

English (en)

Norwegian (no)

Other versions

NO963186D0 (no

NO963186L (no

Inventor

Todd W Butler

Bertrand Leo Chenard

Original Assignee

Pfizer

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1994-01-31

Filing date

1996-07-30

Publication date

2000-12-27

1996-07-30 Application filed by Pfizer filed Critical Pfizer

1996-07-30 Publication of NO963186D0 publication Critical patent/NO963186D0/no

1996-07-30 Publication of NO963186L publication Critical patent/NO963186L/no

2000-12-27 Publication of NO309190B1 publication Critical patent/NO309190B1/no

Links

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Classifications

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- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/04—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
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- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A61P25/06—Antimigraine agents
- A—HUMAN NECESSITIES
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- A61P25/08—Antiepileptics; Anticonvulsants
- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
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- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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Landscapes

Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Chemical Kinetics & Catalysis (AREA)
Animal Behavior & Ethology (AREA)
Medicinal Chemistry (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Neurosurgery (AREA)
Neurology (AREA)
Biomedical Technology (AREA)
Pain & Pain Management (AREA)
Diabetes (AREA)
Toxicology (AREA)
Obesity (AREA)
Hematology (AREA)
Endocrinology (AREA)
Emergency Medicine (AREA)
Psychology (AREA)
Hospice & Palliative Care (AREA)
Psychiatry (AREA)
Anesthesiology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Cosmetics (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Saccharide Compounds (AREA)
Medicines Containing Material From Animals Or Micro-Organisms (AREA)
Medicines Containing Plant Substances (AREA)
Hydrogenated Pyridines (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)

NO963186A 1994-01-31 1996-07-30 Neurobeskyttende kromanforbindelser og farmasöytisk blanding NO309190B1 (no)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US18947994A	1994-01-31	1994-01-31
PCT/IB1994/000365 WO1995020587A1 (en)	1994-01-31	1994-11-21	Neuroprotective chroman compounds

Publications (3)

Publication Number	Publication Date
NO963186D0 NO963186D0 (no)	1996-07-30
NO963186L NO963186L (no)	1996-07-30
NO309190B1 true NO309190B1 (no)	2000-12-27

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ID=22697514

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Application Number	Title	Priority Date	Filing Date
NO963186A NO309190B1 (no)	1994-01-31	1996-07-30	Neurobeskyttende kromanforbindelser og farmasöytisk blanding

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US (1)	US5744483A (pl)
EP (1)	EP0741724B1 (pl)
JP (1)	JP2866743B2 (pl)
CN (1)	CN1048247C (pl)
AT (1)	ATE183184T1 (pl)
AU (1)	AU684568B2 (pl)
BR (2)	BR9408506A (pl)
CA (1)	CA2182101C (pl)
CO (1)	CO4230161A1 (pl)
CZ (1)	CZ286757B6 (pl)
DE (1)	DE69420053T2 (pl)
DK (1)	DK0741724T3 (pl)
EG (1)	EG20672A (pl)
ES (1)	ES2134361T3 (pl)
FI (1)	FI113769B (pl)
GR (1)	GR3031356T3 (pl)
HU (1)	HU221633B1 (pl)
IL (1)	IL112415A (pl)
MY (1)	MY111623A (pl)
NO (1)	NO309190B1 (pl)
NZ (1)	NZ275151A (pl)
PE (1)	PE43795A1 (pl)
PL (1)	PL179448B1 (pl)
RU (1)	RU2126404C1 (pl)
TW (1)	TW449591B (pl)
WO (1)	WO1995020587A1 (pl)
ZA (1)	ZA95692B (pl)

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WO1997010240A1 (en) *	1995-09-15	1997-03-20	Pfizer Inc.	Phenol derivatives with pharmaceutical activity
TW498067B (en) *	1996-07-19	2002-08-11	Hoffmann La Roche	4-hydroxy-piperidine derivatives
UA73981C2 (en) *	2000-03-10	2005-10-17	Merck Patent Gmbh	(r)-(-)-2-[5-(4-fluorophenyl)-3-pyridylmethylaminomethyl]-chromane for treatment of extrapyramidal movement disorders (variants), pharmaceutical composition and kit
PA8525601A1 (es) *	2000-08-21	2002-04-25	Hoffmann La Roche	Profarmacos de (3s,4s)-4-bencil-1-[2-(4-hidroxi-bencenosulfonil)-etil]-piperidin-3-ol
EP1674087A1 (en)	2000-10-02	2006-06-28	Pfizer Products Inc.	Prophylactic use of n-methyl-d-aspartate (NMDA) antagonists
ZA200108038B (en) *	2000-10-02	2003-04-01	Pfizer Prod Inc	Prophylactic use of n-methyl-d-asparrate (NMDA) antagonists.
SE0100902D0 (sv)	2001-03-15	2001-03-15	Astrazeneca Ab	Compounds
ATE352302T1 (de) *	2001-07-26	2007-02-15	Merck Patent Gmbh	Verwendung von 2- 5-(4-fluorphenyl)-3- pyridylmethylaminomethyl-chroman und seiner physiologisch annehmbaren salze
RU2240113C1 (ru) *	2003-01-23	2004-11-20	Государственное образовательное учреждение высшего профессионального образования Московская медицинская академия им. И.М.Сеченова	Способ экстренной медикаментозной помощи при острой травме спинного мозга
CA2547283C (en) *	2003-11-26	2010-11-09	Pfizer Products Inc.	Aminopyrazole derivatives as gsk-3 inhibitors
CN101300246A (zh)	2005-11-03	2008-11-05	弗·哈夫曼-拉罗切有限公司	作为5－ht6抑制剂的芳基磺酰基色满类化合物作为蛋白激酶抑制剂的吲哚基马来酰亚胺衍生物
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1994
- 1994-11-21 BR BR9408506A patent/BR9408506A/pt not_active Application Discontinuation
- 1994-11-21 HU HU9602100A patent/HU221633B1/hu not_active IP Right Cessation
- 1994-11-21 WO PCT/IB1994/000365 patent/WO1995020587A1/en not_active Ceased
- 1994-11-21 NZ NZ275151A patent/NZ275151A/en unknown
- 1994-11-21 AU AU80663/94A patent/AU684568B2/en not_active Ceased
- 1994-11-21 EP EP94931668A patent/EP0741724B1/en not_active Expired - Lifetime
- 1994-11-21 CZ CZ19962256A patent/CZ286757B6/cs not_active IP Right Cessation
- 1994-11-21 JP JP7519959A patent/JP2866743B2/ja not_active Expired - Lifetime
- 1994-11-21 ES ES94931668T patent/ES2134361T3/es not_active Expired - Lifetime
- 1994-11-21 US US08/687,542 patent/US5744483A/en not_active Expired - Fee Related
- 1994-11-21 RU RU96117381A patent/RU2126404C1/ru not_active IP Right Cessation
- 1994-11-21 CN CN94194940A patent/CN1048247C/zh not_active Expired - Fee Related
- 1994-11-21 AT AT94931668T patent/ATE183184T1/de not_active IP Right Cessation
- 1994-11-21 PL PL94315681A patent/PL179448B1/pl unknown
- 1994-11-21 CA CA002182101A patent/CA2182101C/en not_active Expired - Fee Related
- 1994-11-21 DE DE69420053T patent/DE69420053T2/de not_active Expired - Fee Related
- 1994-11-21 DK DK94931668T patent/DK0741724T3/da active
- 1994-11-22 TW TW083110873A patent/TW449591B/zh active
1995
- 1995-01-18 PE PE1995259688A patent/PE43795A1/es not_active Application Discontinuation
- 1995-01-23 IL IL11241595A patent/IL112415A/xx not_active IP Right Cessation
- 1995-01-27 MY MYPI95000224A patent/MY111623A/en unknown
- 1995-01-27 CO CO95003001A patent/CO4230161A1/es unknown
- 1995-01-28 EG EG6795A patent/EG20672A/xx active
- 1995-01-30 ZA ZA95692A patent/ZA95692B/xx unknown
- 1995-01-30 FI FI950403A patent/FI113769B/fi not_active IP Right Cessation
- 1995-01-30 BR BR9500380A patent/BR9500380A/pt not_active IP Right Cessation
1996
- 1996-07-30 NO NO963186A patent/NO309190B1/no unknown
1999
- 1999-09-29 GR GR990402449T patent/GR3031356T3/el unknown

Also Published As

Publication number	Publication date
ZA95692B (en)	1996-07-30
CN1048247C (zh)	2000-01-12
RU2126404C1 (ru)	1999-02-20
PL179448B1 (pl)	2000-09-29
MY111623A (en)	2000-09-27
GR3031356T3 (en)	2000-01-31
CA2182101C (en)	1999-08-03
BR9408506A (pt)	1997-08-05
DK0741724T3 (da)	1999-12-20
NZ275151A (en)	1998-02-26
BR9500380A (pt)	1995-10-17
US5744483A (en)	1998-04-28
IL112415A (en)	1999-07-14
AU684568B2 (en)	1997-12-18
DE69420053T2 (de)	1999-11-25
NO963186D0 (no)	1996-07-30
WO1995020587A1 (en)	1995-08-03
HUT75942A (en)	1997-05-28
JPH09501698A (ja)	1997-02-18
JP2866743B2 (ja)	1999-03-08
CN1142825A (zh)	1997-02-12
NO963186L (no)	1996-07-30
CO4230161A1 (es)	1995-10-19
PE43795A1 (es)	1995-12-09
HU221633B1 (hu)	2002-12-28
FI113769B (fi)	2004-06-15
EP0741724B1 (en)	1999-08-11
CA2182101A1 (en)	1995-08-03
CZ286757B6 (en)	2000-06-14
FI950403A0 (fi)	1995-01-30
CZ225696A3 (en)	1997-01-15
IL112415A0 (en)	1995-03-30
PL315681A1 (en)	1996-11-25
ATE183184T1 (de)	1999-08-15
HU9602100D0 (en)	1996-09-30
FI950403L (fi)	1995-08-01
TW449591B (en)	2001-08-11
ES2134361T3 (es)	1999-10-01
EG20672A (en)	1999-11-30
EP0741724A1 (en)	1996-11-13
AU8066394A (en)	1995-08-15
DE69420053D1 (de)	1999-09-16

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