NO309526B1 - Hetero-aromatiske ring-substituerte fenyloksazolidinon- antimikrobielle midler og anvendelse av disse for fremstilling av et medikament - Google Patents

Hetero-aromatiske ring-substituerte fenyloksazolidinon- antimikrobielle midler og anvendelse av disse for fremstilling av et medikament Download PDF

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Publication number
NO309526B1
NO309526B1 NO973550A NO973550A NO309526B1 NO 309526 B1 NO309526 B1 NO 309526B1 NO 973550 A NO973550 A NO 973550A NO 973550 A NO973550 A NO 973550A NO 309526 B1 NO309526 B1 NO 309526B1
Authority
NO
Norway
Prior art keywords
mmol
solution
fluoro
phenyl
treated
Prior art date
Application number
NO973550A
Other languages
English (en)
Norwegian (no)
Other versions
NO973550D0 (no
NO973550L (no
Inventor
Douglas K Hutchinson
Original Assignee
Upjohn Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Upjohn Co filed Critical Upjohn Co
Publication of NO973550D0 publication Critical patent/NO973550D0/no
Publication of NO973550L publication Critical patent/NO973550L/no
Publication of NO309526B1 publication Critical patent/NO309526B1/no

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42—Oxazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Saccharide Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
NO973550A 1995-02-03 1997-08-01 Hetero-aromatiske ring-substituerte fenyloksazolidinon- antimikrobielle midler og anvendelse av disse for fremstilling av et medikament NO309526B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US38427895A 1995-02-03 1995-02-03
PCT/US1996/000718 WO1996023788A1 (fr) 1995-02-03 1996-01-29 Phenyloxazolidinone substituee par un noyau heteroaromatique comme agent antimicrobien

Publications (3)

Publication Number Publication Date
NO973550D0 NO973550D0 (no) 1997-08-01
NO973550L NO973550L (no) 1997-10-03
NO309526B1 true NO309526B1 (no) 2001-02-12

Family

ID=23516681

Family Applications (1)

Application Number Title Priority Date Filing Date
NO973550A NO309526B1 (no) 1995-02-03 1997-08-01 Hetero-aromatiske ring-substituerte fenyloksazolidinon- antimikrobielle midler og anvendelse av disse for fremstilling av et medikament

Country Status (19)

Country Link
US (1) US5910504A (fr)
EP (1) EP0807112B1 (fr)
JP (1) JPH10513446A (fr)
KR (1) KR100441334B1 (fr)
CN (1) CN1075073C (fr)
AT (1) ATE205205T1 (fr)
BR (1) BR9607017A (fr)
CA (1) CA2208603A1 (fr)
CZ (1) CZ231497A3 (fr)
DE (1) DE69615002T2 (fr)
DK (1) DK0807112T3 (fr)
ES (1) ES2163004T3 (fr)
FI (1) FI973217A7 (fr)
NO (1) NO309526B1 (fr)
NZ (1) NZ302844A (fr)
PL (1) PL185872B1 (fr)
PT (1) PT807112E (fr)
RU (1) RU2154645C2 (fr)
WO (1) WO1996023788A1 (fr)

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GB9717804D0 (en) 1997-08-22 1997-10-29 Zeneca Ltd Chemical compounds
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US6608081B2 (en) * 1999-08-12 2003-08-19 Ortho-Mcneil Pharmaceutical, Inc. Bicyclic heterocyclic substituted phenyl oxazolidinone antibacterials, and related compositions and methods
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EP2072514A1 (fr) * 2007-12-17 2009-06-24 Ferrer Internacional, S.A. 1(2)H-Tétrazol-5-yl-phényl-oxazolidinone en tant qu'agents antibactériens
WO2012171479A1 (fr) * 2011-06-17 2012-12-20 四川大学 Composés d'oxazolidinone et leurs utilisations pour la préparation d'antibiotiques oxazolidinone compounds and their uses in preparation of antibiotics
EP2602248A1 (fr) 2011-12-05 2013-06-12 University Of Leicester Nouveaux composés pyrroliques
WO2013182070A1 (fr) * 2012-06-08 2013-12-12 四川贝力克生物技术有限责任公司 Médicament pour la prévention ou le traitement de maladies mycobactériennes
CN104873510B (zh) * 2014-02-28 2019-03-19 四川好医生药业集团有限公司 噁唑烷酮类化合物抗生物膜用途
CN103965183B (zh) * 2014-03-17 2017-05-03 上海应用技术学院 一种含氟噁唑烷酮类化合物及其制备方法和应用
CN105272976B (zh) * 2014-07-22 2018-11-20 四川好医生药业集团有限公司 一种噁唑烷酮类化合物
CN105399737B (zh) * 2014-09-10 2018-09-21 四川好医生药业集团有限公司 噁唑烷酮类化合物及其用途
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EP3541802B1 (fr) 2016-11-16 2025-01-01 Amgen Inc. Composés de triazole substitués par alkyle en tant qu'agonistes du récepteur apj
US11046680B1 (en) 2016-11-16 2021-06-29 Amgen Inc. Heteroaryl-substituted triazoles as APJ receptor agonists
US10906890B2 (en) 2016-11-16 2021-02-02 Amgen Inc. Triazole phenyl compounds as agonists of the APJ receptor
EP3541792B1 (fr) 2016-11-16 2020-12-23 Amgen Inc. Composés de triazole furane utilisés en tant qu'agonistes du récepteur apj
WO2018093577A1 (fr) 2016-11-16 2018-05-24 Amgen Inc. Composés de triazole à substitution cycloalkyle en tant qu'agonistes du récepteur apj
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CN106831615B (zh) * 2017-02-15 2019-02-15 南京农业大学 一类1，2，3－三唑－5－酰胺类化合物作为农用杀菌剂的应用
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Also Published As

Publication number Publication date
EP0807112B1 (fr) 2001-09-05
WO1996023788A1 (fr) 1996-08-08
KR19980701908A (ko) 1998-06-25
JPH10513446A (ja) 1998-12-22
CN1075073C (zh) 2001-11-21
DE69615002T2 (de) 2002-06-13
ATE205205T1 (de) 2001-09-15
DK0807112T3 (da) 2001-12-17
NZ302844A (en) 1999-06-29
BR9607017A (pt) 1997-10-28
EP0807112A1 (fr) 1997-11-19
KR100441334B1 (ko) 2004-10-20
FI973217A0 (fi) 1997-08-04
FI973217A7 (fi) 1997-08-04
PL185872B1 (pl) 2003-08-29
RU2154645C2 (ru) 2000-08-20
PL321663A1 (en) 1997-12-22
AU4899896A (en) 1996-08-21
CA2208603A1 (fr) 1996-08-08
NO973550D0 (no) 1997-08-01
AU703465B2 (en) 1999-03-25
PT807112E (pt) 2002-02-28
ES2163004T3 (es) 2002-01-16
HK1008898A1 (en) 1999-07-23
NO973550L (no) 1997-10-03
DE69615002D1 (de) 2001-10-11
CZ231497A3 (cs) 1998-08-12
CN1172484A (zh) 1998-02-04
US5910504A (en) 1999-06-08

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