NO324873B1 - 3-Nitrogen-6,7-dioksygen-steroider, farmasoytiske preparater omfattende slike samt anvendelse av disse for fremstilling av medikamenter for behandling av sykdom - Google Patents

3-Nitrogen-6,7-dioksygen-steroider, farmasoytiske preparater omfattende slike samt anvendelse av disse for fremstilling av medikamenter for behandling av sykdom Download PDF

Info

Publication number: NO324873B1
Authority: NO; Norway
Prior art keywords: compound; compound according; mmol; substituted; solution
Prior art date: 2000-04-28

Application number

NO20025106A

Other languages

English (en)

Norwegian (no)

Other versions

NO20025106D0 (no

NO20025106L (no

Inventor

Jeffery R Raymond

Claudia E Kasserra

Yaning Shen

Original Assignee

Inflazyme Pharm Ltd

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-04-28

Filing date

2002-10-24

Publication date

2007-12-17

2002-10-24 Application filed by Inflazyme Pharm Ltd filed Critical Inflazyme Pharm Ltd

2002-10-24 Publication of NO20025106D0 publication Critical patent/NO20025106D0/no

2002-12-18 Publication of NO20025106L publication Critical patent/NO20025106L/no

2007-12-17 Publication of NO324873B1 publication Critical patent/NO324873B1/no

Links

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Classifications

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- C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
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- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
- C07J41/0005—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring the nitrogen atom being directly linked to the cyclopenta(a)hydro phenanthrene skeleton
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
- C07J41/0005—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring the nitrogen atom being directly linked to the cyclopenta(a)hydro phenanthrene skeleton
- C07J41/0011—Unsubstituted amino radicals
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J43/00—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
- C07J71/0036—Nitrogen-containing hetero ring
- C07J71/0042—Nitrogen only
- C07J71/0047—Nitrogen only at position 2(3)
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
- C07J71/0036—Nitrogen-containing hetero ring
- C07J71/0057—Nitrogen and oxygen
- C07J71/0063—Nitrogen and oxygen at position 2(3)
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

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Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
General Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Pulmonology (AREA)
Virology (AREA)
Cardiology (AREA)
Heart & Thoracic Surgery (AREA)
Communicable Diseases (AREA)
Oncology (AREA)
AIDS & HIV (AREA)
Tropical Medicine & Parasitology (AREA)
Molecular Biology (AREA)
Immunology (AREA)
Urology & Nephrology (AREA)
Vascular Medicine (AREA)
Pain & Pain Management (AREA)
Rheumatology (AREA)
Dermatology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Steroid Compounds (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

NO20025106A 2000-04-28 2002-10-24 3-Nitrogen-6,7-dioksygen-steroider, farmasoytiske preparater omfattende slike samt anvendelse av disse for fremstilling av medikamenter for behandling av sykdom NO324873B1 (no)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US20061700P	2000-04-28	2000-04-28
PCT/CA2001/000581 WO2001083512A1 (en)	2000-04-28	2001-04-30	3-nitrogen-6,7-dioxygen steroids and uses related thereto

Publications (3)

Publication Number	Publication Date
NO20025106D0 NO20025106D0 (no)	2002-10-24
NO20025106L NO20025106L (no)	2002-12-18
NO324873B1 true NO324873B1 (no)	2007-12-17

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NO20025106A NO324873B1 (no)	2000-04-28	2002-10-24	3-Nitrogen-6,7-dioksygen-steroider, farmasoytiske preparater omfattende slike samt anvendelse av disse for fremstilling av medikamenter for behandling av sykdom

Country Status (33)

Country	Link
US (4)	US6635629B2 (de)
EP (1)	EP1278763B1 (de)
JP (1)	JP2003531916A (de)
KR (1)	KR20030045671A (de)
CN (1)	CN1214039C (de)
AP (1)	AP1825A (de)
AT (1)	ATE353909T1 (de)
AU (2)	AU2001252084B2 (de)
BG (1)	BG107289A (de)
BR (1)	BR0110419A (de)
CA (1)	CA2418748A1 (de)
CO (1)	CO5590904A2 (de)
DE (1)	DE60126597T2 (de)
DK (1)	DK1278763T3 (de)
DZ (1)	DZ3355A1 (de)
EE (1)	EE200200613A (de)
ES (1)	ES2282247T3 (de)
HR (1)	HRP20020944A2 (de)
HU (1)	HUP0300908A2 (de)
IL (2)	IL152448A0 (de)
MA (1)	MA25808A1 (de)
MX (1)	MXPA02010645A (de)
NO (1)	NO324873B1 (de)
NZ (1)	NZ522181A (de)
OA (1)	OA12255A (de)
PL (1)	PL365798A1 (de)
PT (1)	PT1278763E (de)
RU (1)	RU2291873C2 (de)
SK (1)	SK15692002A3 (de)
UA (1)	UA79229C2 (de)
WO (1)	WO2001083512A1 (de)
YU (1)	YU88102A (de)
ZA (1)	ZA200208631B (de)

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2001
- 2001-04-30 RU RU2002131941/04A patent/RU2291873C2/ru not_active IP Right Cessation
- 2001-04-30 DZ DZ013355A patent/DZ3355A1/fr active
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- 2001-04-30 MX MXPA02010645A patent/MXPA02010645A/es active IP Right Grant
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- 2001-04-30 DK DK01925262T patent/DK1278763T3/da active
- 2001-04-30 AU AU2001252084A patent/AU2001252084B2/en not_active Ceased
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- 2001-04-30 UA UA2002119460A patent/UA79229C2/uk unknown
- 2001-04-30 HR HR20020944A patent/HRP20020944A2/xx not_active Application Discontinuation
- 2001-04-30 IL IL15244801A patent/IL152448A0/xx active IP Right Grant
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- 2001-04-30 EE EEP200200613A patent/EE200200613A/xx unknown
- 2001-04-30 DE DE60126597T patent/DE60126597T2/de not_active Expired - Lifetime
- 2001-04-30 US US10/258,950 patent/US20040034216A1/en not_active Abandoned
- 2001-04-30 PL PL01365798A patent/PL365798A1/xx not_active Application Discontinuation
- 2001-04-30 EP EP01925262A patent/EP1278763B1/de not_active Expired - Lifetime
- 2001-04-30 NZ NZ522181A patent/NZ522181A/en unknown
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- 2001-04-30 KR KR1020027014524A patent/KR20030045671A/ko not_active Ceased
- 2001-04-30 JP JP2001580936A patent/JP2003531916A/ja active Pending
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2002
- 2002-10-24 ZA ZA200208631A patent/ZA200208631B/en unknown
- 2002-10-24 NO NO20025106A patent/NO324873B1/no unknown
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- 2002-11-19 BG BG107289A patent/BG107289A/bg unknown
- 2002-11-20 MA MA26916A patent/MA25808A1/fr unknown
- 2002-11-22 CO CO02106292A patent/CO5590904A2/es not_active Application Discontinuation
2003
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Also Published As

Publication number	Publication date
AP2002002659A0 (en)	2002-12-31
PL365798A1 (en)	2005-01-10
DE60126597D1 (de)	2007-03-29
OA12255A (en)	2006-05-11
US20070060553A1 (en)	2007-03-15
CO5590904A2 (es)	2005-12-30
AU5208401A (en)	2001-11-12
SK15692002A3 (sk)	2003-11-04
CN1214039C (zh)	2005-08-10
UA79229C2 (en)	2007-06-11
YU88102A (sh)	2006-01-16
EP1278763A1 (de)	2003-01-29
HRP20020944A2 (en)	2004-02-29
CN1430625A (zh)	2003-07-16
HUP0300908A2 (hu)	2003-07-28
NO20025106D0 (no)	2002-10-24
HK1050694A1 (en)	2003-07-04
US7112580B2 (en)	2006-09-26
MXPA02010645A (es)	2004-04-20
AU2001252084B2 (en)	2006-07-06
US20040138186A1 (en)	2004-07-15
US6635629B2 (en)	2003-10-21
DK1278763T3 (da)	2007-06-11
CA2418748A1 (en)	2001-11-08
AP1825A (en)	2008-02-03
BG107289A (bg)	2003-07-31
NO20025106L (no)	2002-12-18
KR20030045671A (ko)	2003-06-11
WO2001083512A1 (en)	2001-11-08
US20050215534A9 (en)	2005-09-29
IL152448A (en)	2006-12-31
JP2003531916A (ja)	2003-10-28
NZ522181A (en)	2005-04-29
DZ3355A1 (fr)	2001-11-08
PT1278763E (pt)	2007-05-31
RU2291873C2 (ru)	2007-01-20
DE60126597T2 (de)	2007-10-31
ES2282247T3 (es)	2007-10-16
IL152448A0 (en)	2003-05-29
BR0110419A (pt)	2004-02-25
ZA200208631B (en)	2004-02-23
US20040034216A1 (en)	2004-02-19
MA25808A1 (fr)	2003-07-01
EE200200613A (et)	2004-04-15
ATE353909T1 (de)	2007-03-15
EP1278763B1 (de)	2007-02-14
US20020072510A1 (en)	2002-06-13

Publication	Publication Date	Title
US6635629B2 (en)	2003-10-21	3-nitrogen-6,7-dioxygen steroids and uses related thereto
AU2001252084A1 (en)	2002-01-31	3-nitrogen-6,7-dioxygen steroids and uses related thereto
CN103242192B (zh)	2016-05-04	11-β-羟甾类脱氢酶1型酶的抑制剂
EP0404283B1 (de)	1996-05-08	11-Beta-aryl-4-estrene, Verfahren zu ihrer Herstellung sowie deren Verwendung als Arzneimittel
KR20130130784A (ko)	2013-12-02	산화방지성 염증 조절제로서의 피라졸릴 및 피리미디닐 트리사이클릭 엔온
KR20130112026A (ko)	2013-10-11	벤즈아미드 유도체 및 hsp90 억제제로서의 이의 용도
DE69703228T2 (de)	2001-02-22	Neue 6-Hydroxy und 6-Oxo-Androstan Verbindungen mit Kardioaktivität und pharmazeutische Präparate davon
EP1599201B1 (de)	2010-04-14	Selektive nichtsteroidale glucocorticoid-rezeptor- modulatoren
WO2022133480A1 (en)	2022-06-23	Aryl hydrocarbon receptor (ahr) agonists and uses thereof
US7662846B2 (en)	2010-02-16	Selective spirocyclic glucocorticoid receptor modulators
NO334964B1 (no)	2014-08-11	Indenderivater samt anvendelse derav og farmasøytisk preparat
CN101296914A (zh)	2008-10-29	具有ppar激动活性的衍生物
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HK1050694B (en)	2007-09-28	3-nitrogen-6,7-dioxygen steroids and uses related thereto
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