NO814138L - Analogifremgangsmaate for fremstilling av terapeutisk aktive n-pyrimidyl-karbaminsyreestere - Google Patents

Analogifremgangsmaate for fremstilling av terapeutisk aktive n-pyrimidyl-karbaminsyreestere

Info

Publication number
NO814138L
NO814138L NO814138A NO814138A NO814138L NO 814138 L NO814138 L NO 814138L NO 814138 A NO814138 A NO 814138A NO 814138 A NO814138 A NO 814138A NO 814138 L NO814138 L NO 814138L
Authority
NO
Norway
Prior art keywords
carbamic acid
trimethoxybenzyl
ester
acid
pharmacologically acceptable
Prior art date
Application number
NO814138A
Other languages
English (en)
Norwegian (no)
Inventor
Peter Scharwaechter
Klaus Gutsche
Friedrich-Wilhelm Kohlmann
Hinrich Beck
Original Assignee
Basf Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Basf Ag filed Critical Basf Ag
Publication of NO814138L publication Critical patent/NO814138L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48—Two nitrogen atoms
    • C07D239/49—Two nitrogen atoms with an aralkyl radical, or substituted aralkyl radical, attached in position 5, e.g. trimethoprim
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/63—Compounds containing para-N-benzenesulfonyl-N-groups, e.g. sulfanilamide, p-nitrobenzenesulfonyl hydrazide
    • A61K31/635—Compounds containing para-N-benzenesulfonyl-N-groups, e.g. sulfanilamide, p-nitrobenzenesulfonyl hydrazide having a heterocyclic ring, e.g. sulfadiazine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Oncology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)
NO814138A 1980-12-04 1981-12-03 Analogifremgangsmaate for fremstilling av terapeutisk aktive n-pyrimidyl-karbaminsyreestere NO814138L (no)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19803045720 DE3045720A1 (de) 1980-12-04 1980-12-04 N-pyrimidinyl-carbaminsaeureester, verfahren zu ihrer herstellung und diese enthaltende arzneimittel

Publications (1)

Publication Number Publication Date
NO814138L true NO814138L (no) 1982-06-07

Family

ID=6118292

Family Applications (1)

Application Number Title Priority Date Filing Date
NO814138A NO814138L (no) 1980-12-04 1981-12-03 Analogifremgangsmaate for fremstilling av terapeutisk aktive n-pyrimidyl-karbaminsyreestere

Country Status (12)

Country Link
US (1) US4386084A (fr)
EP (1) EP0053695A3 (fr)
JP (1) JPS57122068A (fr)
AU (1) AU7821981A (fr)
DE (1) DE3045720A1 (fr)
DK (1) DK535781A (fr)
ES (1) ES8300099A1 (fr)
FI (1) FI813845L (fr)
GR (1) GR75115B (fr)
NO (1) NO814138L (fr)
PT (1) PT74077B (fr)
ZA (1) ZA818370B (fr)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5707996A (en) * 1995-11-06 1998-01-13 Macleod Pharmaceuticals, Inc. Pharmaceutical solution and methods for preparation thereof
WO2004005472A2 (fr) * 2002-07-02 2004-01-15 Southern Research Institute Inhibiteurs de ftsz et leurs utilisations
PL1725540T3 (pl) 2004-03-05 2013-02-28 Hoffmann La Roche Diaminopirymidyny jako antagoniści p2x3 i p2x2/3
BRPI0615613A2 (pt) * 2005-09-01 2009-05-19 Hoffmann La Roche diaminopirimidinas como moduladores de p2x3 e p3x2/3
ES2612890T3 (es) * 2005-09-01 2017-05-19 F. Hoffmann-La Roche Ag Diaminopirimidinas como moduladores de P2X3 y P2X2/3
JP4850913B2 (ja) * 2005-09-01 2012-01-11 エフ．ホフマン−ラ ロシュ アーゲー Ｐ２ｘ３及びｐ２ｘ２／３調節因子としてのジアミノピリジン

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3919229A (en) * 1973-07-19 1975-11-11 Labaz Pyrimidine derivatives and process for preparing the same
BE850974A (fr) * 1977-02-01 1977-05-31 Andreu Sa Dr Nouveaux imides de trimethoprim et leur obtention
DE2709634A1 (de) * 1977-03-05 1978-09-07 Basf Ag Benzylpyrimidine, verfahren zu ihrer herstellung und diese enthaltende arzneimittel
DE2730468A1 (de) * 1977-07-06 1979-01-18 Basf Ag Neue n-pyrimidinyl-imidsaeureester, verfahren zu ihrer herstellung und diese enthaltende arzneimittel
DE2730467A1 (de) * 1977-07-06 1979-01-18 Basf Ag Benzylpyrimidine, verfahren zu ihrer herstellung und diese enthaltende arzneimittel
DE2732029A1 (de) * 1977-07-15 1979-02-01 Basf Ag Neue amidino-benzylpyrimidine, verfahren zu ihrer herstellung und diese enthaltende arzneimittel

Also Published As

Publication number Publication date
EP0053695A3 (fr) 1982-12-15
PT74077A (de) 1982-01-01
PT74077B (de) 1983-05-11
DK535781A (da) 1982-06-05
AU7821981A (en) 1982-06-10
FI813845A7 (fi) 1982-06-05
JPS57122068A (en) 1982-07-29
EP0053695A2 (fr) 1982-06-16
US4386084A (en) 1983-05-31
FI813845L (fi) 1982-06-05
DE3045720A1 (de) 1982-07-08
GR75115B (fr) 1984-07-13
ES507682A0 (es) 1982-10-01
ZA818370B (en) 1982-11-24
ES8300099A1 (es) 1982-10-01

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