NO842717L - Fremgangsmaate til fremstilling av karboksylsyrederivater og kjemisk forbindelse til utfoerelse av fremgangsmaaten - Google Patents

Fremgangsmaate til fremstilling av karboksylsyrederivater og kjemisk forbindelse til utfoerelse av fremgangsmaaten

Info

Publication number: NO842717L
Authority: NO; Norway
Prior art keywords: procedure; carboxylic acid; preparation; carrying; acid derivatives
Prior art date: 1983-07-06

Application number

NO842717A

Other languages

English (en)

Other versions

NO163329B (no

NO163329C (no

Inventor

Jose Esteve Soler

Original Assignee

Provesan Sa

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1983-07-06

Filing date

1984-07-04

Publication date

1985-01-07

1983-07-06 Priority claimed from FR8311250A external-priority patent/FR2548664B1/fr

1984-07-04 Application filed by Provesan Sa filed Critical Provesan Sa

1985-01-07 Publication of NO842717L publication Critical patent/NO842717L/no

1990-01-29 Publication of NO163329B publication Critical patent/NO163329B/no

1990-05-09 Publication of NO163329C publication Critical patent/NO163329C/no

Links

150000001732 carboxylic acid derivatives Chemical class 0.000 title 1
239000000126 substance Substances 0.000 title 1
-1 alkali metal salts Chemical class 0.000 abstract 2
DJTQLICBCLDMAC-UHFFFAOYSA-N 1-ethyl-4-oxo-7-pyrrol-1-yl-1,8-naphthyridine-3-carboxylic acid Chemical compound N1=C2N(CC)C=C(C(O)=O)C(=O)C2=CC=C1N1C=CC=C1 DJTQLICBCLDMAC-UHFFFAOYSA-N 0.000 abstract 1
FELNOORDZDEBLV-UHFFFAOYSA-N 1-ethyl-4-oxo-7-pyrrol-1-ylquinoline-3-carboxylic acid Chemical class C1=C2N(CC)C=C(C(O)=O)C(=O)C2=CC=C1N1C=CC=C1 FELNOORDZDEBLV-UHFFFAOYSA-N 0.000 abstract 1
229910052783 alkali metal Inorganic materials 0.000 abstract 1
229910052784 alkaline earth metal Inorganic materials 0.000 abstract 1
239000003242 anti bacterial agent Substances 0.000 abstract 1
230000000844 anti-bacterial effect Effects 0.000 abstract 1
239000003429 antifungal agent Substances 0.000 abstract 1
229940121375 antifungal agent Drugs 0.000 abstract 1
239000004599 antimicrobial Substances 0.000 abstract 1
229910052799 carbon Inorganic materials 0.000 abstract 1
125000004432 carbon atom Chemical group C* 0.000 abstract 1
229910052731 fluorine Chemical group 0.000 abstract 1
125000001153 fluoro group Chemical group F* 0.000 abstract 1
125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 1
229910052757 nitrogen Chemical group 0.000 abstract 1
125000004433 nitrogen atom Chemical group N* 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/48—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
- C07D215/54—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3
- C07D215/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3 with oxygen atoms in position 4
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Pyrrole Compounds (AREA)
Medicines Containing Material From Animals Or Micro-Organisms (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)

NO842717A 1983-07-06 1984-07-04 Analogifremgangsmaate til fremstilling av terapeutisk aktive derivater av 7-(pyrrol-1-yl)-1-etyl-1,4-dihydro-4-okso-kinolin-3-karboksylsyre og 7-(pyrrol-1-yl)-1-etyl-1,4-dihydro-4-okso-(1,8-naftyridin)-3-karboksylsyre. NO163329C (no)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
FR8311250A FR2548664B1 (fr)	1983-07-06	1983-07-06	Derives 7-(pyrrol-l-yl) des acides l-ethyl-1,4-dihydro-4-oxoquinoleine-3-carboxyliques et l-ethyl-1,4-dihydro-4-oxo-(1,8-naphtyridine)-3-carboxyliques substitues, leur preparation et leur application en tant que medicaments
FR8402145A FR2559484B2 (fr)	1983-07-06	1984-02-13	Nouveau derive 7-(pyrrol-1-yl) de l'acide 1-ethyl-1,4-dihydro-4-oxo-(1,8-naphtyridin)-3-carboxylique, sa preparation et son application en tant que medicament

Publications (3)

Publication Number	Publication Date
NO842717L true NO842717L (no)	1985-01-07
NO163329B NO163329B (no)	1990-01-29
NO163329C NO163329C (no)	1990-05-09

Family

ID=26223521

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO842717A NO163329C (no)	1983-07-06	1984-07-04	Analogifremgangsmaate til fremstilling av terapeutisk aktive derivater av 7-(pyrrol-1-yl)-1-etyl-1,4-dihydro-4-okso-kinolin-3-karboksylsyre og 7-(pyrrol-1-yl)-1-etyl-1,4-dihydro-4-okso-(1,8-naftyridin)-3-karboksylsyre.

Country Status (21)

Country	Link
US (1)	US4552882A (no)
EP (1)	EP0134165B1 (no)
KR (1)	KR880002355B1 (no)
AT (1)	ATE34982T1 (no)
AU (1)	AU564326B2 (no)
BR (1)	BR8403342A (no)
CA (1)	CA1256876A (no)
CS (1)	CS244139B2 (no)
DD (1)	DD223150A5 (no)
DE (1)	DE3471934D1 (no)
DK (1)	DK163126C (no)
ES (1)	ES8503335A1 (no)
FR (1)	FR2559484B2 (no)
GR (1)	GR81646B (no)
HK (1)	HK10491A (no)
HU (1)	HU189916B (no)
MX (1)	MX156436A (no)
NO (1)	NO163329C (no)
PL (1)	PL143730B1 (no)
PT (1)	PT78854B (no)
YU (1)	YU43577B (no)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
FR2574404B1 (fr) *	1984-12-12	1987-04-24	Provesan Sa	Derives 1-substitues de l'acide 6-fluoro-7-(pyrrol-1-yl)-1,4-dihydro-4-oxoquinoleine-3-carboxylique, leur preparation et leur application en tant que medicaments
DE3519286A1 (de) *	1985-05-30	1986-12-04	Bayer Ag, 5090 Leverkusen	7-azolyl-1-cyclopropyl-1,4-dihydro-4-oxo-3- chinolincarbonsaeuren und -1,8-naphthyridin-3-carbonsaeuren, verfahren zu ihrer herstellung sowie diese enthaltende antibakterielle mittel
US4692454A (en) *	1986-02-03	1987-09-08	Warner-Lambert Company	Opthalmic use of quinolone antibiotics
DE3615767A1 (de) *	1986-05-10	1987-11-12	Bayer Ag	Verfahren zur herstellung von 4-hydroxy-chinolin-3-carbonsaeuren
FR2607504B1 (fr) *	1986-12-02	1989-01-27	Rhone Poulenc Sante	Nouveaux derives de l'isoindolinone, leur preparation et les compositions pharmaceutiques qui les contiennent
US5262417A (en) *	1988-12-06	1993-11-16	The Upjohn Company	Antibacterial quinolone compounds
ES2051225B1 (es) *	1992-07-23	1994-12-16	Esteve Quimica Sa	Procedimiento de preparacion del acido 1-etil-6-fluoro-7-(pirrol-1-il) -1,4-dihidro-4-oxo-3-quinoleincarboxilico.
AU2002322720B2 (en)	2001-07-25	2008-11-13	Raptor Pharmaceutical Inc.	Compositions and methods for modulating blood-brain barrier transport
CN102379684B (zh)	2005-04-28	2014-11-19	普罗透斯数字保健公司	药物信息系统
KR20090071598A (ko)	2006-09-18	2009-07-01	랩터 파마슈티컬 인코포레이티드	수용체 결합 단백질(ｒａｐ)-접합체 투여에 의한 간 질환의 치료
EP2398500B1 (en)	2009-02-20	2019-03-13	2-BBB Medicines B.V.	Glutathione-based drug delivery system
ES2942923T3 (es)	2009-05-06	2023-06-07	Laboratory Skin Care Inc	Composiciones de administración dérmica que comprenden complejos de agente activo-partículas de fosfato de calcio y métodos de uso de las mismas
US20120077778A1 (en)	2010-09-29	2012-03-29	Andrea Bourdelais	Ladder-Frame Polyether Conjugates
CN104803975A (zh) *	2015-04-24	2015-07-29	河南大学	一种氨甲基三唑取代的二氟喹诺酮羧酸类衍生物及其制备方法和应用

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
CA1006521A (en) *	1972-12-18	1977-03-08	Minoru Sugita	Piperazine derivatives and process for preparing them
JPS5233694A (en) *	1975-09-09	1977-03-14	Dai Ichi Seiyaku Co Ltd	Process for preparation of 6_nitro-1,8-naphthyridine derivatives
AR223983A1 (es) *	1978-08-25	1981-10-15	Dainippon Pharmaceutical Co	Un procedimiento para-preparar derivados de acido 6-halogeno-4-oxo-7-(1-piperazinil)-1,8-naftiridin-3-carboxilico
JPS5649382A (en) *	1979-09-28	1981-05-02	Dainippon Pharmaceut Co Ltd	6-fluoro-7-cyclic amino-1,8-naphthylidine derivative and its salt

1984
- 1984-02-13 FR FR8402145A patent/FR2559484B2/fr not_active Expired
- 1984-06-15 AU AU29425/84A patent/AU564326B2/en not_active Ceased
- 1984-06-20 US US06/622,647 patent/US4552882A/en not_active Expired - Fee Related
- 1984-06-26 CA CA000457471A patent/CA1256876A/en not_active Expired
- 1984-06-27 ES ES533749A patent/ES8503335A1/es not_active Expired
- 1984-06-28 MX MX201827A patent/MX156436A/es unknown
- 1984-06-29 DE DE8484401391T patent/DE3471934D1/de not_active Expired
- 1984-06-29 EP EP84401391A patent/EP0134165B1/fr not_active Expired
- 1984-06-29 AT AT84401391T patent/ATE34982T1/de active
- 1984-07-03 PL PL1984248545A patent/PL143730B1/pl unknown
- 1984-07-03 GR GR75174A patent/GR81646B/el unknown
- 1984-07-04 NO NO842717A patent/NO163329C/no unknown
- 1984-07-05 PT PT78854A patent/PT78854B/pt unknown
- 1984-07-05 DK DK331384A patent/DK163126C/da not_active IP Right Cessation
- 1984-07-05 DD DD84264967A patent/DD223150A5/de not_active IP Right Cessation
- 1984-07-05 HU HU842641A patent/HU189916B/hu not_active IP Right Cessation
- 1984-07-05 BR BR8403342A patent/BR8403342A/pt unknown
- 1984-07-06 CS CS845285A patent/CS244139B2/cs unknown
- 1984-07-06 KR KR1019840003918A patent/KR880002355B1/ko not_active Expired
- 1984-07-06 YU YU1190/84A patent/YU43577B/xx unknown
1991
- 1991-02-06 HK HK104/91A patent/HK10491A/xx unknown

Also Published As

Publication number	Publication date
KR850001198A (ko)	1985-03-16
HK10491A (en)	1991-02-13
HU189916B (en)	1986-08-28
DK163126C (da)	1992-06-15
ATE34982T1 (de)	1988-06-15
PT78854B (fr)	1986-10-23
DK331384A (da)	1985-01-07
FR2559484B2 (fr)	1986-09-26
PL248545A1 (en)	1985-07-16
YU119084A (en)	1986-12-31
EP0134165B1 (fr)	1988-06-08
DD223150A5 (de)	1985-06-05
CS244139B2 (en)	1986-07-17
GR81646B (no)	1984-12-11
NO163329B (no)	1990-01-29
US4552882A (en)	1985-11-12
KR880002355B1 (ko)	1988-10-29
CA1256876A (en)	1989-07-04
PL143730B1 (en)	1988-03-31
AU2942584A (en)	1985-01-10
ES533749A0 (es)	1985-03-01
ES8503335A1 (es)	1985-03-01
DE3471934D1 (en)	1988-07-14
FR2559484A2 (fr)	1985-08-16
DK331384D0 (da)	1984-07-05
CS528584A2 (en)	1985-08-31
EP0134165A2 (fr)	1985-03-13
AU564326B2 (en)	1987-08-06
YU43577B (en)	1989-08-31
BR8403342A (pt)	1985-06-18
PT78854A (fr)	1984-08-01
NO163329C (no)	1990-05-09
MX156436A (es)	1988-08-22
DK163126B (da)	1992-01-20
EP0134165A3 (en)	1985-10-09
HUT34482A (en)	1985-03-28

Publication	Publication Date	Title
ES533749A0 (es)	1985-03-01	Procedimiento de preparar derivados de acidos carboxilicos
DK306586A (da)	1986-12-29	Pyridoncarboxylsyre-derivater og fremgangsmaade til fremstilling deraf
DK163240C (da)	1992-06-29	Analogifremgangsmaade til fremstilling af hidtil ukendte i 8-stilling nitrogensubstituerede ergolinylforbindelser og farmaceutisk acceptable salte heraf
DK519985A (da)	1986-07-01	Quinoloncarboxylsyrederivater, fremgangsmaade til fremstilling deraf og antibakterielt middel indeholdende saadanne derivater
KR860005818A (ko)	1986-08-13	6,7-이치환 1-시클로프로필-1,4-디히드로-4-옥소-1,8-나프티리딘-3-카르복실산의 제조방법
BR8502227A (pt)	1986-01-14	Processos para a obtencao de derivados de acido piridino-2,3-dicarboxilico e de derivados de acido 1-amino-1,4-dihidropiridino-2,3-dicarboxilico
NO885445D0 (no)	1988-12-07	Kinolincarboxylsyre-borsyreanhydrider og fremgangsmaate for fremstilling derav.
HUT43943A (en)	1988-01-28	Herbicide compositions comprising urea derivatives as active substance and process for preparing such compounds
ES8505993A1 (es)	1985-06-16	Un metodo para preparar un derivado de 3-indolcarboxamida
YU42307B (en)	1988-08-31	Process for preparing imidazo (1,2-a)imidazoles
DK412487D0 (da)	1987-08-07	Quinolinderivater og disses fremstilling
SE8405002D0 (sv)	1984-10-05	Framstellning av bensotiazindioxid