DK306586A - Pyridoncarboxylsyre-derivater og fremgangsmaade til fremstilling deraf - Google Patents

Pyridoncarboxylsyre-derivater og fremgangsmaade til fremstilling deraf Download PDF

Info

Publication number: DK306586A
Authority: DK; Denmark
Prior art keywords: sup; acid derivatives; group; pyridon; procedures
Prior art date: 1985-06-28

Application number

DK306586A

Other languages

English (en)

Other versions

DK171330B1 (da

DK306586D0 (da

Inventor

Kuniyoshi Masuzawa

Seigo Suzue

Keiji Hirai

Takayoshi Ishizaki

Original Assignee

Kyorin Seiyaku Kk

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1985-06-28

Filing date

1986-06-27

Publication date

1986-12-29

1986-06-27 Application filed by Kyorin Seiyaku Kk filed Critical Kyorin Seiyaku Kk

1986-06-27 Publication of DK306586D0 publication Critical patent/DK306586D0/da

1986-12-29 Publication of DK306586A publication Critical patent/DK306586A/da

1996-09-09 Application granted granted Critical

1996-09-09 Publication of DK171330B1 publication Critical patent/DK171330B1/da

Links

-1 PYRIDON CARBOXYLIC ACID DERIVATIVES Chemical class 0.000 title 1
238000000034 method Methods 0.000 title 1
125000000217 alkyl group Chemical group 0.000 abstract 3
125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 3
YSLIPUSJNFIFAB-UHFFFAOYSA-N 2-oxopyridine-1-carboxylic acid Chemical class OC(=O)N1C=CC=CC1=O YSLIPUSJNFIFAB-UHFFFAOYSA-N 0.000 abstract 1
125000002252 acyl group Chemical group 0.000 abstract 1
125000004453 alkoxycarbonyl group Chemical group 0.000 abstract 1
239000003242 anti bacterial agent Substances 0.000 abstract 1
125000000753 cycloalkyl group Chemical group 0.000 abstract 1
125000001188 haloalkyl group Chemical group 0.000 abstract 1
125000005843 halogen group Chemical group 0.000 abstract 1
150000004677 hydrates Chemical class 0.000 abstract 1
150000003839 salts Chemical class 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/48—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
- C07D215/54—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3
- C07D215/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3 with oxygen atoms in position 4
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Oncology (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Communicable Diseases (AREA)
Public Health (AREA)
Chemical Kinetics & Catalysis (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Pyridine Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Saccharide Compounds (AREA)
Vessels, Lead-In Wires, Accessory Apparatuses For Cathode-Ray Tubes (AREA)
Photoreceptors In Electrophotography (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

DK306586A 1985-06-28 1986-06-27 Pyridoncarboxylsyre-derivater, fremgangsmåde til fremstilling deraf samt antibakterielt farmaceutisk præparat DK171330B1 (da)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
JP60141813A JPH0635457B2 (ja)	1985-06-28	1985-06-28	ピリドンカルボン酸誘導体およびその製造方法
JP14181385		1985-06-28

Publications (3)

Publication Number	Publication Date
DK306586D0 DK306586D0 (da)	1986-06-27
DK306586A true DK306586A (da)	1986-12-29
DK171330B1 DK171330B1 (da)	1996-09-09

Family

ID=15300723

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK306586A DK171330B1 (da)	1985-06-28	1986-06-27	Pyridoncarboxylsyre-derivater, fremgangsmåde til fremstilling deraf samt antibakterielt farmaceutisk præparat

Country Status (16)

Country	Link
US (1)	US4753953A (da)
EP (1)	EP0208210B1 (da)
JP (1)	JPH0635457B2 (da)
KR (1)	KR930005002B1 (da)
CN (1)	CN1010312B (da)
AT (1)	ATE57699T1 (da)
AU (1)	AU589427B2 (da)
CA (1)	CA1262349A (da)
DE (1)	DE3675087D1 (da)
DK (1)	DK171330B1 (da)
ES (1)	ES2000185A6 (da)
FI (1)	FI85697C (da)
HU (1)	HU208128B (da)
MX (1)	MX162950B (da)
NO (1)	NO166126C (da)
PT (1)	PT82854B (da)

Families Citing this family (26)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
JPH089597B2 (ja) *	1986-01-21	1996-01-31	杏林製薬株式会社	選択毒性に優れた８‐アルコキシキノロンカルボン酸およびその塩並びにその製造方法
US4692454A (en) *	1986-02-03	1987-09-08	Warner-Lambert Company	Opthalmic use of quinolone antibiotics
DE3705621C2 (de) *	1986-02-25	1997-01-09	Otsuka Pharma Co Ltd	Heterocyclisch substituierte Chinoloncarbonsäurederivate
JPS62205060A (ja) *	1986-03-04	1987-09-09	Kyorin Pharmaceut Co Ltd	８位置換キノロンカルボン酸誘導体
JPS62215572A (ja) *	1986-03-17	1987-09-22	Kyorin Pharmaceut Co Ltd	キノロンカルボン酸誘導体
US5147871A (en) *	1986-07-03	1992-09-15	Hoffmann La-Roche, Inc.	Anti-bacterial cephalosporin compounds
DE3639465A1 (de) *	1986-11-18	1988-05-19	Hoechst Ag	Optisch aktive gyrasehemmer, ihre herstellung und verwendung als antibiotika
JP2603638B2 (ja) *	1987-07-08	1997-04-23	第一製薬株式会社	光学異性体の分析法及び分取法
CS273349B2 (en) *	1988-03-31	1991-03-12	Hoffmann La Roche	Method of cephalosporin's new derivatives production
US5336768A (en) *	1988-05-24	1994-08-09	Hoffmann-La Roche Inc.	Antibacterial cephalosporin compounds
CA1332605C (en) *	1988-10-03	1994-10-18	Yasuhiro Nishitani	Pyridonecarboxylic acids
DE3918544A1 (de) *	1989-06-07	1990-12-13	Bayer Ag	Verfahren zur herstellung von 7-(3-amino- sowie 3-amino-methyl-1-pyrrolidinyl)-3-chinolon- carbonsaeuren sowie -naphthyridoncarbonsaeuren
US5162523A (en) *	1989-07-21	1992-11-10	Hoffmann-La Roche Inc.	Cephalosporin antibacterial compounds
US5159077A (en) *	1989-07-21	1992-10-27	Hoffmann-La Roche Inc.	Penam antibacterial compounds
MY109714A (en) *	1990-10-18	1997-04-30	Daiichi Seiyaku Co	Process for preparing 8-chloroquinolone derivatives
NO179912C (no) *	1990-11-28	1997-01-08	Daiichi Seiyaku Co	Analogifremgangsmåte for fremstilling av et terapeutisk virksomt optisk aktivt pyridobenzoksazinderivat
KR950014567B1 (ko) *	1991-08-01	1995-12-08	주식회사대웅제약	신규한 퀴놀론 카르복실산 유도체
FR2692577B1 (fr) *	1992-05-26	1996-02-02	Bouchara Sa	Nouvelles quinolones fluorees, leur procede de preparation et les compositions pharmaceutiques en renfermant.
TW252107B (da) *	1993-08-27	1995-07-21	Hokuriku Pharmacetical Co Ltd
EP0806421A4 (en) *	1995-01-24	1998-04-15	Hokuriku Pharmaceutical	DERIVATIVES OF CHINOLINE CARBONIC ACID
PL1666477T3 (pl)	2003-09-10	2013-11-29	Kyorin Seiyaku Kk	Pochodna kwasu 7-(4-podstawionego-3-cyklopropyloaminometylo-1- pirolidynylo)chinolonokarboksylowego
WO2005073238A1 (ja) *	2004-02-02	2005-08-11	Daiichi Pharmaceutical Co., Ltd.	ピリドベンズオキサジン誘導体
US7977327B2 (en)	2004-05-13	2011-07-12	Daiichi Sankyo Company, Limited	Substituted pyrrolidine derivative
US7563805B2 (en) *	2005-05-19	2009-07-21	Daiichi Pharmaceutical Co., Ltd.	Tri-, tetra-substituted-3-aminopyrrolidine derivative
JP5322927B2 (ja)	2007-05-24	2013-10-23	杏林製薬株式会社	１４位置換基に複素芳香環カルボン酸構造を有するムチリン誘導体
FR2961207B1 (fr) *	2010-06-09	2013-01-18	Oreal	Utilisation d'un derive de 4- carboxy 2-pyrrolidinone comme solvant dans les compositions cosmetiques ; compositions cosmetiques les contenant ; nouveaux composes

Family Cites Families (21)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
CA1175836A (en) *	1977-09-20	1984-10-09	Marcel Pesson	Production of 1,4-dihydroquinoline-3-carboxylic acid derivatives
US4620007A (en) *	1980-09-03	1986-10-28	Bayer Aktiengesellschaft	6-fluoro-7-chloro-1-cyclopropyl-4-oxo-1,4-dihydro-quinoline-3-carboxylic acid
JPS5788183A (en) *	1980-11-21	1982-06-01	Dai Ichi Seiyaku Co Ltd	Pyridobenzoxazine derivative
JPS5872589A (ja) *	1981-10-28	1983-04-30	Dai Ichi Seiyaku Co Ltd	ピリド〔１，２，３−ｄｅ〕〔１，４〕ベンゾオキサジン誘導体
PH22140A (en) *	1982-06-29	1988-06-01	Daiichi Seiyaku Co	Tricyclic compounds
US4665079A (en) *	1984-02-17	1987-05-12	Warner-Lambert Company	Antibacterial agents
IE55898B1 (en) *	1982-09-09	1991-02-14	Warner Lambert Co	Antibacterial agents
DE3318145A1 (de) *	1983-05-18	1984-11-22	Bayer Ag, 5090 Leverkusen	7-amino-1-cyclopropyl-6,8-difluor-1,4-dihydro-4-oxo-3-chinolincarbonsaeuren, verfahren zu ihrer herstellung sowie diese enthaltende antibakterielle mittel
JPS60260577A (ja) *	1984-06-06	1985-12-23	Dainippon Pharmaceut Co Ltd	１，８−ナフチリジン誘導体
CS274601B2 (en) *	1983-07-27	1991-09-15	Dainippon Pharmaceutical Co	Method of 1,8-naphthyridine derivative production
US4571396A (en) *	1984-04-16	1986-02-18	Warner-Lambert Company	Antibacterial agents
US4542133A (en) *	1984-04-26	1985-09-17	Abbott Laboratories	Methylenedioxy quino-benoxazine derivatives and antibacterial use
EP0160284B1 (en) *	1984-04-26	1990-10-24	Abbott Laboratories	Quino-benoxazine antibacterial compounds
DE3420743A1 (de) *	1984-06-04	1985-12-05	Bayer Ag, 5090 Leverkusen	7-amino-1-cyclopropyl-6,8-dihalogen-1,4-dihydro-4-oxo-3-chinolincarbonsaeuren, verfahren zu ihrer herstellung sowie diese enthaltende antibakterielle mittel
US4604401A (en) *	1984-07-20	1986-08-05	Warner-Lambert Company	Antibacterial agents III
JPH0670032B2 (ja) *	1984-11-22	1994-09-07	大日本製薬株式会社	アミノピロリジン誘導体、そのエステルおよびその塩
JPS61137885A (ja) *	1984-12-08	1986-06-25	Dainippon Pharmaceut Co Ltd	１，８−ナフチリジン誘導体、そのエステルおよびその塩
JPS61148179A (ja) *	1984-12-20	1986-07-05	Dainippon Pharmaceut Co Ltd	新規ナフチリジン誘導体、そのエステルおよびその塩
US4578473A (en) *	1985-04-15	1986-03-25	Warner-Lambert Company	Process for quinoline-3-carboxylic acid antibacterial agents
AU585995B2 (en) *	1985-06-20	1989-06-29	Daiichi Pharmaceutical Co., Ltd.	Optically active pyridobenzoxazine derivatives and intermediates thereof
JPS62205060A (ja) *	1986-03-04	1987-09-09	Kyorin Pharmaceut Co Ltd	８位置換キノロンカルボン酸誘導体

1985
- 1985-06-28 JP JP60141813A patent/JPH0635457B2/ja not_active Expired - Fee Related
1986
- 1986-06-20 US US06/876,420 patent/US4753953A/en not_active Expired - Lifetime
- 1986-06-23 AU AU59190/86A patent/AU589427B2/en not_active Ceased
- 1986-06-23 HU HU862626A patent/HU208128B/hu not_active IP Right Cessation
- 1986-06-25 CA CA000512440A patent/CA1262349A/en not_active Expired
- 1986-06-26 DE DE8686108728T patent/DE3675087D1/de not_active Expired - Lifetime
- 1986-06-26 AT AT86108728T patent/ATE57699T1/de not_active IP Right Cessation
- 1986-06-26 PT PT82854A patent/PT82854B/pt not_active IP Right Cessation
- 1986-06-26 EP EP86108728A patent/EP0208210B1/en not_active Expired - Lifetime
- 1986-06-27 DK DK306586A patent/DK171330B1/da not_active IP Right Cessation
- 1986-06-27 FI FI862757A patent/FI85697C/fi active IP Right Grant
- 1986-06-27 ES ES8600048A patent/ES2000185A6/es not_active Expired
- 1986-06-27 MX MX2967A patent/MX162950B/es unknown
- 1986-06-27 CN CN86104479A patent/CN1010312B/zh not_active Expired
- 1986-06-27 NO NO862621A patent/NO166126C/no not_active IP Right Cessation
- 1986-06-28 KR KR1019860005232A patent/KR930005002B1/ko not_active Expired - Fee Related

Also Published As

Publication number	Publication date
FI85697B (fi)	1992-02-14
NO166126B (no)	1991-02-25
JPS624284A (ja)	1987-01-10
PT82854A (en)	1986-07-01
DE3675087D1 (de)	1990-11-29
DK171330B1 (da)	1996-09-09
EP0208210B1 (en)	1990-10-24
NO166126C (no)	1991-06-05
CN86104479A (zh)	1987-02-04
FI862757L (fi)	1986-12-29
JPH0635457B2 (ja)	1994-05-11
EP0208210A1 (en)	1987-01-14
FI85697C (fi)	1992-05-25
HUT43051A (en)	1987-09-28
NO862621D0 (no)	1986-06-27
HU208128B (en)	1993-08-30
ATE57699T1 (de)	1990-11-15
MX162950B (es)	1991-07-22
AU589427B2 (en)	1989-10-12
FI862757A0 (fi)	1986-06-27
PT82854B (pt)	1988-05-27
KR870000322A (ko)	1987-02-17
ES2000185A6 (es)	1988-01-01
KR930005002B1 (ko)	1993-06-11
DK306586D0 (da)	1986-06-27
CA1262349A (en)	1989-10-17
NO862621L (no)	1986-12-29
AU5919086A (en)	1987-01-08
CN1010312B (zh)	1990-11-07
US4753953A (en)	1988-06-28

Legal Events

Date	Code	Title	Description
1996-09-09	B1	Patent granted (law 1993)
2005-01-31	PBP	Patent lapsed	Country of ref document: DK

Publication	Publication Date	Title
DK306586D0 (da)	1986-06-27	Pyridoncarboxylsyre-derivater og fremgangsmaade til fremstilling deraf
AU591640B2 (en)	1989-12-14	Quinolonecarboxylic acid derivatives
DK359289D0 (da)	1989-07-19	4-oxoquinolin-3-carboxylsyrederivater og fremgangsmaade til fremstilling deraf samt deres anvendelse
NO892851D0 (no)	1989-07-10	Fremstilling og anvendelse av quinolinderivater.
NO934536D0 (no)	1993-12-10	Fenoksy- og fenoksyalkyl-pepiridiner som antivirale midler
DE3665711D1 (de)	1989-10-26	Novel guanidinomethylbenzoic acid derivatives
NO163329C (no)	1990-05-09	Analogifremgangsmaate til fremstilling av terapeutisk aktive derivater av 7-(pyrrol-1-yl)-1-etyl-1,4-dihydro-4-okso-kinolin-3-karboksylsyre og 7-(pyrrol-1-yl)-1-etyl-1,4-dihydro-4-okso-(1,8-naftyridin)-3-karboksylsyre.
ES2046229T3 (es)	1994-02-01	Composicion antiulcerosa.
ES8801211A1 (es)	1987-12-16	Un procedimiento para preparar derivados de quinolona
ES8307818A1 (es)	1983-08-16	Procedimiento para preparar derivados de cefalosporina.
ES2042727T3 (es)	1993-12-16	Acidos 1,3,4,9-tetrahidropirano(3,4-b)indol-1-acetico.
GB9022821D0 (en)	1990-12-05	Piperazine derivatives
GEP19960472B (en)	1996-05-27	Method of producing derivative of quinoline or its pharmaceutically acceptable ester, or their salts
ES8402303A1 (es)	1984-01-16	Un procedimiento para la preparacion de nuevos derivados de 7-oxo-1-azabiciclo (3.2.0) hepteno.