NO922028L - Azol-derivater - Google Patents

Azol-derivater

Info

Publication number: NO922028L
Authority: NO; Norway
Prior art keywords: alkyl; phenyl; unsubstituted; substituted; oxygen
Prior art date: 1991-05-23

Application number

NO92922028A

Other languages

English (en)

Norwegian (no)

Other versions

NO922028D0 (no

Inventor

Peter William Rodney Caulkett

Geraint Jones

Simon Martin Poucher

Michael George Collis

Original Assignee

Ici Plc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1991-05-23

Filing date

1992-05-22

Publication date

1992-11-24

1992-05-22 Application filed by Ici Plc filed Critical Ici Plc

1992-05-22 Publication of NO922028D0 publication Critical patent/NO922028D0/no

1992-11-24 Publication of NO922028L publication Critical patent/NO922028L/no

Links

150000007980 azole derivatives Chemical class 0.000 title 1
125000000217 alkyl group Chemical group 0.000 abstract 4
150000001875 compounds Chemical class 0.000 abstract 3
125000004070 6 membered heterocyclic group Chemical group 0.000 abstract 2
QVGXLLKOCUKJST-UHFFFAOYSA-N atomic oxygen Chemical compound [O] QVGXLLKOCUKJST-UHFFFAOYSA-N 0.000 abstract 2
229910052739 hydrogen Inorganic materials 0.000 abstract 2
239000001257 hydrogen Substances 0.000 abstract 2
125000004433 nitrogen atom Chemical group N* 0.000 abstract 2
229910052760 oxygen Inorganic materials 0.000 abstract 2
239000001301 oxygen Substances 0.000 abstract 2
125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 2
229910052717 sulfur Inorganic materials 0.000 abstract 2
125000004434 sulfur atom Chemical group 0.000 abstract 2
UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 abstract 1
125000004423 acyloxy group Chemical group 0.000 abstract 1
125000003342 alkenyl group Chemical group 0.000 abstract 1
125000003545 alkoxy group Chemical group 0.000 abstract 1
125000000304 alkynyl group Chemical group 0.000 abstract 1
125000001589 carboacyl group Chemical group 0.000 abstract 1
229910052736 halogen Inorganic materials 0.000 abstract 1
150000002367 halogens Chemical class 0.000 abstract 1
125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 1
-1 hydroxy, benzyloxy Chemical group 0.000 abstract 1
239000008194 pharmaceutical composition Substances 0.000 abstract 1
239000000296 purinergic P1 receptor antagonist Substances 0.000 abstract 1
150000003839 salts Chemical class 0.000 abstract 1
125000002023 trifluoromethyl group Chemical group FC(F)(F)* 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/08—Vasodilators for multiple indications

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
Engineering & Computer Science (AREA)
Cardiology (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Bioinformatics & Cheminformatics (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Heart & Thoracic Surgery (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)

NO92922028A 1991-05-23 1992-05-22 Azol-derivater NO922028L (no)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
GB919111130A GB9111130D0 (en)	1991-05-23	1991-05-23	Azole derivatives

Publications (2)

Publication Number	Publication Date
NO922028D0 NO922028D0 (no)	1992-05-22
NO922028L true NO922028L (no)	1992-11-24

Family

ID=10695460

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO92922028A NO922028L (no)	1991-05-23	1992-05-22	Azol-derivater

Country Status (16)

Country	Link
US (1)	US5290776A (cs)
EP (1)	EP0515107A3 (cs)
JP (1)	JPH05155887A (cs)
KR (1)	KR920021547A (cs)
AU (1)	AU654010B2 (cs)
CA (1)	CA2069455A1 (cs)
CS (1)	CS153392A3 (cs)
FI (1)	FI922340A7 (cs)
GB (2)	GB9111130D0 (cs)
HU (1)	HU210764B (cs)
IE (1)	IE921655A1 (cs)
IL (1)	IL101965A0 (cs)
NO (1)	NO922028L (cs)
NZ (1)	NZ242865A (cs)
TW (1)	TW213917B (cs)
ZA (1)	ZA923767B (cs)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5356894A (en) *	1990-05-29	1994-10-18	Rodney Peter W	Morpholinyl substituted [1,2,4]-triazolo[1,5-a]triazine as antagonist
FR2671551B1 (fr) *	1991-01-15	1993-03-12	Adir	Nouveaux composes de structure aryl triazinique, leur procede de preparation et les compositions pharmaceutiques qui les contiennent.
ES2165393T3 (es) *	1993-07-27	2002-03-16	Kyowa Hakko Kogyo Kk	Remedio contra la enfermedad de parkinson.
AU7546794A (en) *	1993-09-06	1995-03-27	Kyowa Hakko Kogyo Co. Ltd.	Depression remedy
US5477857A (en) *	1993-09-10	1995-12-26	Discovery Therapeutics, Inc.	Diagnostic uses of hydrazinoadenosines
US8003705B2 (en) *	1996-09-23	2011-08-23	Incept Llc	Biocompatible hydrogels made with small molecule precursors
US6566406B1 (en) *	1998-12-04	2003-05-20	Incept, Llc	Biocompatible crosslinked polymers
AU2639299A (en) *	1998-02-24	1999-09-15	Kyowa Hakko Kogyo Co. Ltd.	Remedies/preventives for parkinson's disease
WO2003071986A2 (en) *	2002-02-22	2003-09-04	Control Delivery Systems, Inc.	Method for treating otic disorders
FR2842809A1 (fr) *	2002-07-26	2004-01-30	Greenpharma Sas	NOUVELLES PYRAZOLO[1,5-a]-1,3,5-TRIAZINES SUBSTITUEES ET LEURS ANALOGUES, COMPOSITIONS PHARMACEUTIQUES LES CONTENANT, UTILISATION A TITRE DE MEDICAMENT ET PROCEDES POUR LEUR PREPARATION
AU2003272886A1 (en) *	2002-09-24	2004-04-19	Kyowa Hakko Kogyo Co., Ltd.	(1,2,4)-TRIAZOLO(1,5-c)PYRIMIDINE DERIVATIVE
KR100490893B1 (ko) *	2002-10-11	2005-05-23	(주) 비엔씨바이오팜	2-메톡시-1,3,5-트리아진 유도체, 그 제조방법 및 이를 포함하는 항바이러스용 약학적 조성물
US7329658B2 (en) *	2003-02-06	2008-02-12	Pfizer Inc	Cannabinoid receptor ligands and uses thereof
DE602004018637D1 (de)	2003-04-09	2009-02-05	Biogen Idec Inc	A2a-adenosinrezeptorantagonisten
WO2004092171A2 (en) *	2003-04-09	2004-10-28	Biogen Idec Ma Inc.	Triazolo[1,5-a]pyrimidines and pyrazolo[1,5-a]pyrimidines useful as a2a adenosin e receptor antagonists
WO2004092170A2 (en) *	2003-04-09	2004-10-28	Biogen Idec Ma Inc.	Triazolotriazines and pyrazolotriazines useful as a2a adenosine receptor antagon ists
US20070010522A1 (en) *	2003-04-09	2007-01-11	Chi Vu	Triazolo[1,5-c]pyrimidines and pyrazolo[1,5-c]pyrimidines useful as a2a adenosine receptor antagonists
US7674791B2 (en)	2003-04-09	2010-03-09	Biogen Idec Ma Inc.	Triazolopyrazines and methods of making and using the same
WO2004110454A1 (ja) *	2003-06-13	2004-12-23	Ishihara Sangyo Kaisha, Ltd.	アデノシンＡ2ａ受容体アゴニストの投与が必要な疾患を治療又は予防するための組成物
US8067028B2 (en) *	2007-08-13	2011-11-29	Confluent Surgical Inc.	Drug delivery device
KR20250063269A (ko) *	2023-10-30	2025-05-08	현대약품 주식회사	신규한 화합물, 및 이를 포함하는 암의 예방 또는 치료용 약학적 조성물

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3846423A (en) *	1972-06-08	1974-11-05	Icn Pharmaceuticals	Pyrazolo (1,5a) 1,3,5-triazines
BE815405A (en) *	1973-05-22	1974-11-22		Pyrazolo(1,5-a)-s-triazines - and their salts, with bronchospasmolytic activity
US3995039A (en) *	1975-05-27	1976-11-30	Merck & Co., Inc.	Pyrazolo [1,5-a] [1,3,5] triazines
GB1579932A (en) *	1976-05-12	1980-11-26	Ici Ltd	Herbicidal triazolotriazines
GB2016002B (en) *	1978-01-09	1982-05-06	Aron Sa	Amino derivatives of pyrazolo(1,5-a)s triazine
US4565815A (en) *	1982-12-30	1986-01-21	Biomeasure, Inc.	Pyrazolo[1,5-a]-1,3,5-triazines
AU2192683A (en) *	1982-12-30	1984-07-05	Biomeasure Incorporated	Pyrazolo(1,5-alpha)-1,3,5-triazines
US4560689A (en) *	1983-01-10	1985-12-24	Ciba-Geigy Corporation	Heterocyclic-fused pyrazolo-[3,4-d]pyridin-3-ones as benzodiazepine receptor modulators
US4713383A (en) *	1984-10-01	1987-12-15	Ciba-Geigy Corporation	Triazoloquinazoline compounds, and their methods of preparation, pharmaceutical compositions, and uses
CA1267143A (en) *	1985-06-06	1990-03-27	Sun H. Kim	Anti-arthritic 7-phenylpyrazole[1,5-a]-1,3,5- triazine derivatives
DE3677445D1 (de) *	1985-09-30	1991-03-14	Ciba Geigy Ag	2-substituierte-e-kondensierte(1,5-c)-pyrimidine, pharmazeutische zubereitungen und ihre verwendung.
DE3781080T2 (de) *	1986-09-30	1992-12-24	Ciba Geigy Ag	2-substituierte-e-kondensierte(1,2,4)triazolo-(1,5-c)pyrimidine, pharmazeutische zubereitungen und ihre verwendung.
US4734413A (en) *	1987-03-02	1988-03-29	Riker Laboratories, Inc.	Substituted 1,2,4-triazolo[1,5-A]triazines as bronchodilators
DE8817122U1 (de) *	1988-12-22	1993-02-04	Boehringer Ingelheim Kg, 55218 Ingelheim	Neue Xanthinderivate mit Adenosinantogenistischer Wirkung
US4970142A (en) *	1989-02-16	1990-11-13	Konica Corporation	Silver halide photographic light-sensitive material containing cyan coupler
GB2244487B (en) *	1990-05-29	1994-02-02	Ici Plc	Azole derivatives

1991
- 1991-05-23 GB GB919111130A patent/GB9111130D0/en active Pending
1992
- 1992-05-05 GB GB929209622A patent/GB9209622D0/en active Pending
- 1992-05-15 EP EP19920304409 patent/EP0515107A3/en not_active Withdrawn
- 1992-05-21 US US07/886,798 patent/US5290776A/en not_active Expired - Fee Related
- 1992-05-22 NZ NZ242865A patent/NZ242865A/en unknown
- 1992-05-22 CA CA002069455A patent/CA2069455A1/en not_active Abandoned
- 1992-05-22 AU AU17093/92A patent/AU654010B2/en not_active Ceased
- 1992-05-22 ZA ZA923767A patent/ZA923767B/xx unknown
- 1992-05-22 IL IL92101965A patent/IL101965A0/xx unknown
- 1992-05-22 CS CS921533A patent/CS153392A3/cs unknown
- 1992-05-22 FI FI922340A patent/FI922340A7/fi unknown
- 1992-05-22 NO NO92922028A patent/NO922028L/no unknown
- 1992-05-22 HU HU9201704A patent/HU210764B/hu not_active IP Right Cessation
- 1992-05-23 KR KR1019920008803A patent/KR920021547A/ko not_active Withdrawn
- 1992-05-25 JP JP4132526A patent/JPH05155887A/ja active Pending
- 1992-06-04 TW TW081104402A patent/TW213917B/zh active
- 1992-07-01 IE IE165592A patent/IE921655A1/en not_active Application Discontinuation

Also Published As

Publication number	Publication date
TW213917B (cs)	1993-10-01
GB9111130D0 (en)	1991-07-17
AU1709392A (en)	1992-11-26
IE921655A1 (en)	1992-12-02
CA2069455A1 (en)	1992-11-24
US5290776A (en)	1994-03-01
ZA923767B (en)	1993-04-28
CS153392A3 (en)	1992-12-16
GB9209622D0 (en)	1992-06-17
AU654010B2 (en)	1994-10-20
FI922340A7 (fi)	1992-11-24
FI922340A0 (fi)	1992-05-22
NZ242865A (en)	1995-05-26
HU210764B (en)	1995-07-28
EP0515107A3 (en)	1993-01-13
HU9201704D0 (en)	1992-08-28
JPH05155887A (ja)	1993-06-22
IL101965A0 (en)	1992-12-30
HUT62898A (en)	1993-06-28
KR920021547A (ko)	1992-12-18
EP0515107A2 (en)	1992-11-25
NO922028D0 (no)	1992-05-22

Publication	Publication Date	Title
NO922028L (no)	1992-11-24	Azol-derivater
DE60103754D1 (de)	2004-07-15	Oxazolidinonderivate mit antibiotischer aktivität
AU631466B2 (en)	1992-11-26	New 1,2-benzisoxazole derivatives, processes for preparing them and pharmaceutical compositions containing them
IL97049A0 (en)	1992-03-29	Aryl-and heteroarylethenylene derivatives,their preparation and pharmaceutical compositions containing them
KR890000467A (ko)	1989-03-14	피리딘 유도체 및 그것을 함유하는 궤양 치료제
DE3660258D1 (en)	1988-07-07	Pristinamycine iib derivatives, their preparation and pharmaceutical compositions containing them
AU2636988A (en)	1989-06-01	New 2-(piperazinyl)-2-substituted flavonoid derivatives, processes for preparing them and pharmaceutical compositions containing them
DE3367215D1 (en)	1986-12-04	Pyridobenzodiazepinones, process for their preparation and pharmaceutical compositions containing them
ES2016017A6 (es)	1990-10-01	Procedimiento para preparar derivados de acido 1,1-dioxocefem-4-carbotiolico.
ES8403129A1 (es)	1984-03-01	Procedimiento para la preparacion de nuevas tienobenzodiazepinonas sustituidas.
YU158385A (en)	1988-04-30	Process for obtaining derivatives of 2-pyridine thioles
ES8609330A1 (es)	1986-08-01	Un procedimiento para preparar nuevos derivados de 1,3-dihi-dro-6-1-ciano-1-isopropil-n-fenetil-n-metil-omega-aminoal- quil-7--hidroxi-furo-(3,4-c)-piridina
ES8801637A1 (es)	1988-02-16	Un procedimiento para la preparacion de benzimidazoles.
MX9806341A (es)	1998-10-31	Derivados de ergolina heterociclica.
ZA83771B (en)	1984-10-31	Substituted thienobenzodiazepinones and acid addition salts thereof,processes for the preparation thereof and pharmaceutical compositions containing these compounds
PT87790A (pt)	1988-07-01	A process for the preparation of ergoline derivatives and of pharmaceutical compositions containing the same
HUT50833A (en)	1990-03-28	Process for producing indolo/3,2-1-de/ /1,4/-oxazino/2,3,4-ij/ /1,5/-naphthyridine derivatives
SE8804696L (sv)	1989-07-01	Dioxazocin- derivat, deras framstaellning och beredningar innehaallande desamma
HU895651D0 (en)	1990-01-28	Process for the preparation of substituted 3-amino-nonimine derivatives and pharmaceutical compositions containing said compounds
KR930700507A (ko)	1993-03-15	살생물성 헤테로폴리시클릭 화합물, 그것의 합성방법 및 그 중간체, 그것들을 포함한 제제, 및 의약품으로서 그것의 사용방법