NO923079D0 - N-fenyl-n-acetamidoglycinamider, deres fremstilling samt medikamenter inneholdende forbindelsene - Google Patents

N-fenyl-n-acetamidoglycinamider, deres fremstilling samt medikamenter inneholdende forbindelsene

Info

Publication number
NO923079D0
NO923079D0 NO923079A NO923079A NO923079D0 NO 923079 D0 NO923079 D0 NO 923079D0 NO 923079 A NO923079 A NO 923079A NO 923079 A NO923079 A NO 923079A NO 923079 D0 NO923079 D0 NO 923079D0
Authority
NO
Norway
Prior art keywords
unsubstituted
radical
pct
compounds
preparation
Prior art date
Application number
NO923079A
Other languages
English (en)
Other versions
NO923079L (no
Inventor
Jean-Dominique Bourzat
Marc Capet
Claude Cotrel
Claude Guyon
Franco Manfre
Geard Roussel
Original Assignee
Rhone Poulenc Rorer Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from FR9001553A external-priority patent/FR2658196B1/fr
Priority claimed from FR9011916A external-priority patent/FR2667319B2/fr
Priority claimed from FR9012594A external-priority patent/FR2667863B2/fr
Application filed by Rhone Poulenc Rorer Sa filed Critical Rhone Poulenc Rorer Sa
Publication of NO923079D0 publication Critical patent/NO923079D0/no
Publication of NO923079L publication Critical patent/NO923079L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06008—Dipeptides with the first amino acid being neutral
    • C07K5/06017—Dipeptides with the first amino acid being neutral and aliphatic
    • C07K5/06026—Dipeptides with the first amino acid being neutral and aliphatic the side chain containing 0 or 1 carbon atom, i.e. Gly or Ala
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C205/00—Compounds containing nitro groups bound to a carbon skeleton
    • C07C205/13—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by hydroxy groups
    • C07C205/19—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by hydroxy groups having nitro groups bound to carbon atoms of six-membered aromatic rings and hydroxy groups bound to acyclic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C205/00—Compounds containing nitro groups bound to a carbon skeleton
    • C07C205/13—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by hydroxy groups
    • C07C205/20—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by hydroxy groups having nitro groups and hydroxy groups bound to carbon atoms of six-membered aromatic rings
    • C07C205/21—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by hydroxy groups having nitro groups and hydroxy groups bound to carbon atoms of six-membered aromatic rings having nitro groups and hydroxy groups bound to carbon atoms of the same non-condensed six-membered aromatic ring
    • C07C205/22—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by hydroxy groups having nitro groups and hydroxy groups bound to carbon atoms of six-membered aromatic rings having nitro groups and hydroxy groups bound to carbon atoms of the same non-condensed six-membered aromatic ring having one nitro groups bound to the ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C205/00—Compounds containing nitro groups bound to a carbon skeleton
    • C07C205/27—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by etherified hydroxy groups
    • C07C205/35—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by etherified hydroxy groups having nitro groups and etherified hydroxy groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton
    • C07C205/36—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by etherified hydroxy groups having nitro groups and etherified hydroxy groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton to carbon atoms of the same non-condensed six-membered aromatic ring or to carbon atoms of six-membered aromatic rings being part of the same condensed ring system
    • C07C205/37—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by etherified hydroxy groups having nitro groups and etherified hydroxy groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton to carbon atoms of the same non-condensed six-membered aromatic ring or to carbon atoms of six-membered aromatic rings being part of the same condensed ring system the oxygen atom of at least one of the etherified hydroxy groups being further bound to an acyclic carbon atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C205/00—Compounds containing nitro groups bound to a carbon skeleton
    • C07C205/49—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by carboxyl groups
    • C07C205/56—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by carboxyl groups having nitro groups bound to carbon atoms of six-membered aromatic rings and carboxyl groups bound to acyclic carbon atoms of the carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C205/00—Compounds containing nitro groups bound to a carbon skeleton
    • C07C205/49—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by carboxyl groups
    • C07C205/57—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by carboxyl groups having nitro groups and carboxyl groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton
    • C07C205/58—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by carboxyl groups having nitro groups and carboxyl groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton the carbon skeleton being further substituted by halogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C205/00—Compounds containing nitro groups bound to a carbon skeleton
    • C07C205/49—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by carboxyl groups
    • C07C205/57—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by carboxyl groups having nitro groups and carboxyl groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton
    • C07C205/59—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by carboxyl groups having nitro groups and carboxyl groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton the carbon skeleton being further substituted by singly-bound oxygen atoms
    • C07C205/60—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by carboxyl groups having nitro groups and carboxyl groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton the carbon skeleton being further substituted by singly-bound oxygen atoms in ortho-position to the carboxyl group, e.g. nitro-salicylic acids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Medicinal Preparation (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
NO92923079A 1990-02-09 1992-08-05 N-fenyl-n-acetamidoglycinamider, deres fremstilling samt medikamenter inneholdende forbindelsene NO923079L (no)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
FR9001553A FR2658196B1 (fr) 1990-02-09 1990-02-09 N-phenyl n-acetamido glycinamides leur preparation et les medicaments les contenant.
FR9011916A FR2667319B2 (fr) 1990-02-09 1990-09-27 N-phenyl n-acetamido glycinamides, leur preparation et les medicaments les contenant.
FR9012594A FR2667863B2 (fr) 1990-02-09 1990-10-12 N-phenyl n-acetamido glycinamides, leur preparation et les medicaments les contenant.
PCT/FR1991/000087 WO1991012264A1 (fr) 1990-02-09 1991-02-06 N-phenyl n-acetamido glycinamides, leur preparation et les medicaments les contenant

Publications (2)

Publication Number Publication Date
NO923079D0 true NO923079D0 (no) 1992-08-05
NO923079L NO923079L (no) 1992-08-05

Family

ID=27252134

Family Applications (1)

Application Number Title Priority Date Filing Date
NO92923079A NO923079L (no) 1990-02-09 1992-08-05 N-fenyl-n-acetamidoglycinamider, deres fremstilling samt medikamenter inneholdende forbindelsene

Country Status (17)

Country Link
US (1) US5382590A (no)
EP (1) EP0514442B1 (no)
JP (1) JPH05506643A (no)
KR (1) KR927003625A (no)
AT (1) ATE104989T1 (no)
AU (1) AU639081B2 (no)
CA (1) CA2072981A1 (no)
DE (1) DE69101835T2 (no)
DK (1) DK0514442T3 (no)
ES (1) ES2052372T3 (no)
HU (1) HUT61575A (no)
IE (1) IE910428A1 (no)
IL (1) IL97180A0 (no)
NO (1) NO923079L (no)
NZ (1) NZ237052A (no)
PT (1) PT96712A (no)
WO (1) WO1991012264A1 (no)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2658518B1 (fr) * 1990-02-19 1992-04-30 Rhone Poulenc Sante N-phenyl n-alcoxycarbonylalkyle glycinamides, leur preparation et les medicaments les contenant.
GB9206757D0 (en) * 1992-03-27 1992-05-13 Ferring Bv Novel peptide receptor ligands
FR2695643B1 (fr) * 1992-09-11 1994-11-25 Rhone Poulenc Rorer Sa Dérivés d'uréido-acétamide, leur préparation et les médicaments les contenant.
FR2695641B1 (fr) * 1992-09-11 1994-11-25 Rhone Poulenc Rorer Sa (Amino-3 phényl)-1 éthanesulfonate d'hydroquinine optiquement actif, sa préparation et son utilisation.
EP0739903B1 (en) * 1994-02-09 2002-01-23 Shionogi & Co., Ltd. Carbamoylmethylurea derivative
GB9420763D0 (en) * 1994-10-14 1994-11-30 Glaxo Inc Acetamide derivatives
AU4891396A (en) * 1995-03-14 1996-10-02 Daiichi Pharmaceutical Co., Ltd. Aminophenol derivatives
FI974437A7 (fi) 1995-06-06 1997-12-05 Pfizer Substituoituja N-(indoli-2-karbonyyli)amideja ja johdannaisia glykogee nifosforylaasi-inhibiittoreina
KR100241643B1 (ko) 1995-06-06 2000-03-02 디. 제이. 우드 당뇨병치료제인 치환된 N-(인돌-2-카르보닐)-β-알라님아미드 및 그의 유도체
CA2224062C (en) * 1995-06-06 2001-09-04 Pfizer Limited Substituted n-(indole-2-carbonyl)-glycinamides and derivatives as glycogen phosphorylase inhibitors
CA2228622A1 (en) * 1995-08-07 1997-02-20 Haruo Koike Process for producing carbamoylmethylurea derivatives
FR2744364B1 (fr) * 1996-02-07 1998-02-27 Rhone Poulenc Rorer Sa Application d'ureidoacetamides a la preparation de medicaments destines au traitement de l'abus de drogues ou de substances donnant lieu a des pharmacomanies ou a un usage excessif
US6277877B1 (en) 2000-08-15 2001-08-21 Pfizer, Inc. Substituted n-(indole-2-carbonyl)glycinamides and derivates as glycogen phosphorylase inhibitors
MX2010013192A (es) * 2008-06-16 2010-12-17 Hoffmann La Roche Monoamidas heteroaromaticas como antagonistas de receptor orexinina.
WO2011044327A1 (en) * 2009-10-07 2011-04-14 Medivation Prostate Therapeutics, Inc. Substituted phenylcarbamoyl alkylamino arene compounds and n,n'-bis-arylurea compounds
CN107789354B (zh) * 2016-08-31 2022-02-25 中国科学院上海药物研究所 预防和治疗抑郁症的化合物及其应用
CN109020887B (zh) * 2017-06-10 2022-03-01 绍兴从零医药科技有限公司 作为防治精神障碍疾病的酰胺类化合物
CN108689877B (zh) * 2018-07-06 2021-08-03 浙江工业大学 一种含手性碳的双酰胺类化合物及其制备方法与应用
US11596612B1 (en) 2022-03-08 2023-03-07 PTC Innovations, LLC Topical anesthetics

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2533210A1 (fr) * 1982-09-17 1984-03-23 Lyon I Universite Claude Edulcorants de synthese
EP0166355A2 (en) * 1984-06-26 1986-01-02 Merck & Co. Inc. Substituted aminophenyl compounds and acylaminophenyl compounds and pharmaceutical compositions containing them
EP0175498A2 (en) * 1984-08-23 1986-03-26 The Administrators Of The Tulane University Educational Fund Peptides, their use in medicine and methods for their preparation
FR2646847B1 (fr) * 1989-05-12 1991-07-12 Rhone Poulenc Sante N-phenyl amides, leurs procedes de preparation et les medicaments les contenant

Also Published As

Publication number Publication date
IE910428A1 (en) 1991-08-14
CA2072981A1 (fr) 1991-08-10
AU7329591A (en) 1991-09-03
PT96712A (pt) 1991-10-31
AU639081B2 (en) 1993-07-15
EP0514442B1 (fr) 1994-04-27
NZ237052A (en) 1992-12-23
ES2052372T3 (es) 1994-07-01
IL97180A0 (en) 1992-05-25
DE69101835D1 (de) 1994-06-01
KR927003625A (ko) 1992-12-18
EP0514442A1 (fr) 1992-11-25
JPH05506643A (ja) 1993-09-30
US5382590A (en) 1995-01-17
HUT61575A (en) 1993-01-28
WO1991012264A1 (fr) 1991-08-22
NO923079L (no) 1992-08-05
DE69101835T2 (de) 1994-08-18
DK0514442T3 (da) 1994-09-26
ATE104989T1 (de) 1994-05-15

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