NO931679L - Nye heterocykliske forbindelser som antagonister for eksitatoriske aminosyrereseptorer, fremgangsmaater for deres fremstilling og deres anvendelse - Google Patents

Nye heterocykliske forbindelser som antagonister for eksitatoriske aminosyrereseptorer, fremgangsmaater for deres fremstilling og deres anvendelse

Info

Publication number
NO931679L
NO931679L NO93931679A NO931679A NO931679L NO 931679 L NO931679 L NO 931679L NO 93931679 A NO93931679 A NO 93931679A NO 931679 A NO931679 A NO 931679A NO 931679 L NO931679 L NO 931679L
Authority
NO
Norway
Prior art keywords
antagonists
procedures
preparation
amino acid
heterocyclic compounds
Prior art date
Application number
NO93931679A
Other languages
English (en)
Other versions
NO931679D0 (no
Inventor
Alf Claesson
Britt-Marie Swahn
Original Assignee
Astra Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astra Ab filed Critical Astra Ab
Publication of NO931679D0 publication Critical patent/NO931679D0/no
Publication of NO931679L publication Critical patent/NO931679L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/645—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having two nitrogen atoms as the only ring hetero atoms
    • C07F9/6509—Six-membered rings
    • C07F9/650952—Six-membered rings having the nitrogen atoms in the positions 1 and 4
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/553—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having one nitrogen atom as the only ring hetero atom
    • C07F9/576—Six-membered rings
    • C07F9/59—Hydrogenated pyridine rings

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pain & Pain Management (AREA)
  • Anesthesiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Injection Moulding Of Plastics Or The Like (AREA)
  • Plural Heterocyclic Compounds (AREA)
NO93931679A 1990-11-15 1993-05-07 Nye heterocykliske forbindelser som antagonister for eksitatoriske aminosyrereseptorer, fremgangsmaater for deres fremstilling og deres anvendelse NO931679L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
SE9003652A SE9003652D0 (sv) 1990-11-15 1990-11-15 New heterocyclic compounds
PCT/SE1991/000753 WO1992008724A1 (en) 1990-11-15 1991-11-07 New heterocyclic compounds as antagonists of excitatory amino acid receptors, processes for their preparation and their use

Publications (2)

Publication Number Publication Date
NO931679D0 NO931679D0 (no) 1993-05-07
NO931679L true NO931679L (no) 1993-05-07

Family

ID=20380925

Family Applications (1)

Application Number Title Priority Date Filing Date
NO93931679A NO931679L (no) 1990-11-15 1993-05-07 Nye heterocykliske forbindelser som antagonister for eksitatoriske aminosyrereseptorer, fremgangsmaater for deres fremstilling og deres anvendelse

Country Status (17)

Country Link
EP (1) EP0557375A1 (no)
JP (1) JPH06502421A (no)
CN (1) CN1061595A (no)
AU (1) AU652399B2 (no)
CA (1) CA2095224A1 (no)
CZ (1) CZ80993A3 (no)
FI (1) FI932206A7 (no)
HU (1) HU9301417D0 (no)
IE (1) IE913922A1 (no)
IS (1) IS3782A7 (no)
LT (1) LTIP1718A (no)
MX (1) MX9101979A (no)
NO (1) NO931679L (no)
PT (1) PT99515A (no)
SE (1) SE9003652D0 (no)
SK (1) SK46993A3 (no)
WO (1) WO1992008724A1 (no)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5194430A (en) * 1990-05-17 1993-03-16 Merrell Dow Pharmaceuticals Inc. Heterocyclic-nmda antagonists
TW281670B (no) * 1993-09-02 1996-07-21 Hoffmann La Roche
US5491241A (en) * 1993-10-18 1996-02-13 Eli Lilly And Company Bicyclic intermediates for excitatory amino acid receptor antagonists
LT3984994T (lt) 2016-02-04 2024-10-10 Takeda Pharmaceutical Company Limited Pakeistas piperidino junginys kaip 2 tipo oreksino agonistas narkolepsijai gydyti

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1248531A (en) * 1984-04-17 1989-01-10 Jeffrey C. Watkins 4-substituted piperazine-2-carboxylic acids
JPS612519A (ja) * 1984-04-24 1986-01-08 Aron Kasei Co Ltd 射出成形法
US4906621A (en) * 1985-05-24 1990-03-06 Ciba-Geigy Corporation Certain 2-carboxypiperidyl-alkylene phosphonic acids and esters thereof useful for the treatment of disorders responsive to N-methyl-D-aspartate receptor blockade
US4740346A (en) * 1986-02-26 1988-04-26 The Budd Company Perimeter resin feeding of composite structures
JPS63112129A (ja) * 1986-10-30 1988-05-17 Toyoda Gosei Co Ltd 多色樹脂成形用金型
ATE60776T1 (de) * 1986-11-21 1991-02-15 Ciba Geigy Ag Ungesaettigte phosphonsaeure und derivate.

Also Published As

Publication number Publication date
FI932206A0 (fi) 1993-05-14
IS3782A7 (is) 1992-05-16
FI932206L (fi) 1993-05-14
LTIP1718A (en) 1995-07-25
IE913922A1 (en) 1992-05-20
EP0557375A1 (en) 1993-09-01
HU9301417D0 (en) 1993-09-28
JPH06502421A (ja) 1994-03-17
NO931679D0 (no) 1993-05-07
AU8939191A (en) 1992-06-11
CZ80993A3 (en) 1994-02-16
SE9003652D0 (sv) 1990-11-15
PT99515A (pt) 1992-09-30
MX9101979A (es) 1992-07-08
WO1992008724A1 (en) 1992-05-29
CN1061595A (zh) 1992-06-03
FI932206A7 (fi) 1993-05-14
AU652399B2 (en) 1994-08-25
SK46993A3 (en) 1993-10-06
CA2095224A1 (en) 1992-05-16

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