NO931960L - Nye pilokarpinderivater og fremgangsmaate ved fremstillingav disse - Google Patents
Nye pilokarpinderivater og fremgangsmaate ved fremstillingav disseInfo
- Publication number
- NO931960L NO931960L NO93931960A NO931960A NO931960L NO 931960 L NO931960 L NO 931960L NO 93931960 A NO93931960 A NO 93931960A NO 931960 A NO931960 A NO 931960A NO 931960 L NO931960 L NO 931960L
- Authority
- NO
- Norway
- Prior art keywords
- pilocarpin
- procedures
- derivatives
- same
- new
- Prior art date
Links
- QCHFTSOMWOSFHM-WPRPVWTQSA-N (+)-Pilocarpine Chemical class C1OC(=O)[C@@H](CC)[C@H]1CC1=CN=CN1C QCHFTSOMWOSFHM-WPRPVWTQSA-N 0.000 title 1
- 238000000034 method Methods 0.000 title 1
- 125000002252 acyl group Chemical group 0.000 abstract 2
- 229910052739 hydrogen Inorganic materials 0.000 abstract 2
- 239000001257 hydrogen Substances 0.000 abstract 2
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 2
- 208000010412 Glaucoma Diseases 0.000 abstract 1
- 125000001931 aliphatic group Chemical group 0.000 abstract 1
- 125000003118 aryl group Chemical group 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/64—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/06—Antiglaucoma agents or miotics
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Ophthalmology & Optometry (AREA)
- Pharmacology & Pharmacy (AREA)
- General Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Plural Heterocyclic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FI905930A FI98815C (fi) | 1990-11-30 | 1990-11-30 | Menetelmä uusien, farmakologisesti käyttökelpoisten bispilokarpiinihapon esterijohdannaisten valmistamiseksi |
| PCT/FI1991/000359 WO1992009583A1 (en) | 1990-11-30 | 1991-11-27 | Novel pilocarpine derivatives and process for their preparation |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| NO931960L true NO931960L (no) | 1993-05-28 |
| NO931960D0 NO931960D0 (no) | 1993-05-28 |
| NO304228B1 NO304228B1 (no) | 1998-11-16 |
Family
ID=8531500
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO931960A NO304228B1 (no) | 1990-11-30 | 1993-05-28 | AnalogifremgangsmÕte ved fremstilling av esterderivater av bispilokarpinsyre |
Country Status (19)
| Country | Link |
|---|---|
| EP (1) | EP0559700B1 (no) |
| JP (1) | JP3094232B2 (no) |
| KR (1) | KR930703264A (no) |
| AT (1) | ATE192144T1 (no) |
| AU (1) | AU664958B2 (no) |
| CA (1) | CA2096444A1 (no) |
| CZ (1) | CZ282229B6 (no) |
| DE (1) | DE69132143T2 (no) |
| EE (1) | EE9400143A (no) |
| FI (1) | FI98815C (no) |
| HU (1) | HUT67273A (no) |
| LT (1) | LT3532B (no) |
| LV (1) | LV10094B (no) |
| NO (1) | NO304228B1 (no) |
| NZ (1) | NZ240781A (no) |
| PL (2) | PL168715B1 (no) |
| RU (1) | RU2100352C1 (no) |
| SK (1) | SK52393A3 (no) |
| WO (1) | WO1992009583A1 (no) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO1993024466A1 (en) * | 1992-05-29 | 1993-12-09 | Leiras Oy | Novel pilocarpine derivatives and process for their preparation |
| GB9310965D0 (en) * | 1993-05-27 | 1993-07-14 | Ucb Sa | 2-hydroxy-3-(1h-imidazol-4-yl)alkyl)benzenecarboximidamides |
| AU6973094A (en) * | 1993-06-24 | 1995-01-17 | Leiras Oy | Composition for ophthalmic use |
| SE501482C2 (sv) * | 1993-06-24 | 1995-02-27 | Leiras Oy | Komposition för topisk administration av bispilokarpinsyradiestrar till ögat i form av en vattenlösning |
| SE9302201D0 (sv) | 1993-06-24 | 1993-06-24 | Leiras Oy | Composition for ophthalmic use |
| DE4334135A1 (de) * | 1993-10-07 | 1995-04-13 | Merck Patent Gmbh | Verfahren zur Herstellung von Pilocarpin-Derivaten |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4061722A (en) | 1976-04-26 | 1977-12-06 | Interx Research Corporation | Selected quaternary ammonium salts of pilocarpine useful in reducing intraocular pressure in warm-blooded animals |
| IL69593A (en) * | 1982-09-17 | 1988-09-30 | Bundegaard Hans | Pilocarpine prodrugs,their preparation and pharmaceutical compositions containing them |
-
1990
- 1990-11-30 FI FI905930A patent/FI98815C/fi not_active IP Right Cessation
-
1991
- 1991-11-27 HU HU9301569A patent/HUT67273A/hu unknown
- 1991-11-27 JP JP04500392A patent/JP3094232B2/ja not_active Expired - Fee Related
- 1991-11-27 PL PL91308270A patent/PL168715B1/pl unknown
- 1991-11-27 SK SK523-93A patent/SK52393A3/sk unknown
- 1991-11-27 PL PL91299375A patent/PL167773B1/pl unknown
- 1991-11-27 CZ CS931025A patent/CZ282229B6/cs not_active IP Right Cessation
- 1991-11-27 AU AU89398/91A patent/AU664958B2/en not_active Ceased
- 1991-11-27 KR KR1019930701611A patent/KR930703264A/ko not_active Withdrawn
- 1991-11-27 WO PCT/FI1991/000359 patent/WO1992009583A1/en not_active Ceased
- 1991-11-27 AT AT91920512T patent/ATE192144T1/de not_active IP Right Cessation
- 1991-11-27 RU RU93041054/04A patent/RU2100352C1/ru not_active IP Right Cessation
- 1991-11-27 EP EP91920512A patent/EP0559700B1/en not_active Expired - Lifetime
- 1991-11-27 CA CA002096444A patent/CA2096444A1/en not_active Abandoned
- 1991-11-27 DE DE69132143T patent/DE69132143T2/de not_active Expired - Fee Related
- 1991-11-28 NZ NZ240781A patent/NZ240781A/xx unknown
-
1993
- 1993-05-28 NO NO931960A patent/NO304228B1/no not_active IP Right Cessation
- 1993-05-28 LT LTIP577A patent/LT3532B/lt not_active IP Right Cessation
- 1993-05-28 LV LVP-93-436A patent/LV10094B/en unknown
-
1994
- 1994-11-16 EE EE9400143A patent/EE9400143A/xx unknown
Also Published As
| Publication number | Publication date |
|---|---|
| CA2096444A1 (en) | 1992-05-31 |
| LT3532B (en) | 1995-11-27 |
| SK52393A3 (en) | 1994-01-12 |
| DE69132143T2 (de) | 2000-12-14 |
| EE9400143A (et) | 1995-12-15 |
| HU9301569D0 (en) | 1993-09-28 |
| FI905930A7 (fi) | 1992-05-31 |
| FI905930A0 (fi) | 1990-11-30 |
| EP0559700A1 (en) | 1993-09-15 |
| PL168715B1 (pl) | 1996-03-29 |
| CZ102593A3 (en) | 1994-04-13 |
| LV10094A (lv) | 1994-05-10 |
| NO931960D0 (no) | 1993-05-28 |
| FI98815C (fi) | 1997-08-25 |
| DE69132143D1 (de) | 2000-05-31 |
| WO1992009583A1 (en) | 1992-06-11 |
| AU8939891A (en) | 1992-06-25 |
| NO304228B1 (no) | 1998-11-16 |
| ATE192144T1 (de) | 2000-05-15 |
| JPH06504270A (ja) | 1994-05-19 |
| FI98815B (fi) | 1997-05-15 |
| EP0559700B1 (en) | 2000-04-26 |
| KR930703264A (ko) | 1993-11-29 |
| NZ240781A (en) | 1993-12-23 |
| JP3094232B2 (ja) | 2000-10-03 |
| LTIP577A (en) | 1994-12-27 |
| AU664958B2 (en) | 1995-12-07 |
| LV10094B (en) | 1995-02-20 |
| RU2100352C1 (ru) | 1997-12-27 |
| CZ282229B6 (cs) | 1997-06-11 |
| PL167773B1 (pl) | 1995-11-30 |
| HUT67273A (en) | 1995-03-28 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| MM1K | Lapsed by not paying the annual fees |