NO985227L - Alkylaminobenzothiazol og -benzoksazol - derivater - Google Patents

Alkylaminobenzothiazol og -benzoksazol - derivater

Info

Publication number: NO985227L
Authority: NO; Norway
Prior art keywords: alkylaminobenzothiazole; benzoxazole derivatives; benzoxazole; derivatives
Prior art date: 1996-05-10

Application number

NO985227A

Other languages

English (en)

Other versions

NO311027B1 (no

NO985227D0 (no

Inventor

Ludo Edmond Josephine Kennis

Josephus Carolus Mertens

Serge Maria Aloysius Pieters

Original Assignee

Janssen Pharmaceutica Nv

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1996-05-10

Filing date

1998-11-09

Publication date

1999-01-11

1998-11-09 Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv

1998-11-09 Publication of NO985227D0 publication Critical patent/NO985227D0/no

1999-01-11 Publication of NO985227L publication Critical patent/NO985227L/no

2001-10-01 Publication of NO311027B1 publication Critical patent/NO311027B1/no

Links

BCMCBBGGLRIHSE-UHFFFAOYSA-N 1,3-benzoxazole Chemical class C1=CC=C2OC=NC2=C1 BCMCBBGGLRIHSE-UHFFFAOYSA-N 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/52—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings condensed with carbocyclic rings or ring systems
- C07D263/54—Benzoxazoles; Hydrogenated benzoxazoles
- C07D263/58—Benzoxazoles; Hydrogenated benzoxazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/42—Oxazoles
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B59/00—Introduction of isotopes of elements into organic compounds ; Labelled organic compounds per se
- C07B59/002—Heterocyclic compounds
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
- C07D277/62—Benzothiazoles
- C07D277/68—Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- C07D277/82—Nitrogen atoms

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
Medicinal Chemistry (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Neurosurgery (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Psychiatry (AREA)
Epidemiology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
Thiazole And Isothizaole Compounds (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

NO19985227A 1996-05-10 1998-11-09 Alkylaminobenzotiazol og -benzoksazolderivater NO311027B1 (no)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
EP96201282		1996-05-10
PCT/EP1997/002505 WO1997043271A1 (en)	1996-05-10	1997-05-02	Alkylaminobenzothiazole and -benzoxazole derivatives

Publications (3)

Publication Number	Publication Date
NO985227D0 NO985227D0 (no)	1998-11-09
NO985227L true NO985227L (no)	1999-01-11
NO311027B1 NO311027B1 (no)	2001-10-01

Family

ID=8223970

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO19985227A NO311027B1 (no)	1996-05-10	1998-11-09	Alkylaminobenzotiazol og -benzoksazolderivater

Country Status (28)

Country	Link
US (2)	US6103725A (no)
EP (2)	EP1325917B1 (no)
JP (1)	JP3237759B2 (no)
KR (1)	KR100330699B1 (no)
CN (1)	CN1074766C (no)
AR (1)	AR007079A1 (no)
AT (2)	ATE350373T1 (no)
AU (1)	AU710175B2 (no)
BG (1)	BG64097B1 (no)
BR (1)	BR9709065A (no)
CA (1)	CA2253453C (no)
CZ (1)	CZ295639B6 (no)
DE (2)	DE69730962T2 (no)
EA (1)	EA001360B1 (no)
EE (1)	EE03563B1 (no)
ES (2)	ES2279923T3 (no)
HU (1)	HUP9902993A3 (no)
ID (1)	ID16889A (no)
IL (1)	IL126968A0 (no)
MY (1)	MY117852A (no)
NO (1)	NO311027B1 (no)
NZ (1)	NZ332309A (no)
PL (1)	PL190721B1 (no)
SK (1)	SK282919B6 (no)
TR (1)	TR199802253T2 (no)
TW (1)	TW593290B (no)
WO (1)	WO1997043271A1 (no)
ZA (1)	ZA974053B (no)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
IT1293804B1 (it)	1997-08-01	1999-03-10	Recordati Chem Pharm	Diarilalchilpiperazine attive sulle basse vie urinarie
US6281216B1 (en) *	1998-02-09	2001-08-28	Duphar International Research B.V.	2-aminoquinoline derivatives having d4-agonistic activity
EP0982030A3 (en)	1998-08-17	2000-05-10	Pfizer Products Inc.	2,7-substituted octahydro-pyrrolo 1,2-a]pyrazine derivatives as 5ht 1a ligands
AU6280199A (en) *	1998-09-30	2000-04-17	Neurogen Corporation	2-piperazino alkylamino benzoazole derivatives: dopamine receptor subtype specific ligands
US6284759B1 (en)	1998-09-30	2001-09-04	Neurogen Corporation	2-piperazinoalkylaminobenzo-azole derivatives: dopamine receptor subtype specific ligands
US6107313A (en) *	1998-10-02	2000-08-22	Combichem, Inc.	Dopamine receptor antagonists
WO2001000604A1 (fr) *	1999-06-30	2001-01-04	Santen Pharmaceutical Co., Ltd.	Ligand de liaison avec le recepteur sigma-1 du cerveau
AU2001249679A1 (en)	2000-03-31	2001-10-15	Ortho-Mcneil Pharmaceutical, Inc.	Phenyl-substituted imidazopyridines
AU2001251083A1 (en)	2000-03-31	2001-10-15	Ortho-Mcneil Pharmaceutical, Inc.	Method for using 2-aryloxyalkylaminobenzoxazoles and 2-aryloxyalkylaminobenzothiazoles as h3 antagonists
GB0203299D0 (en) *	2002-02-12	2002-03-27	Glaxo Group Ltd	Novel compounds
WO2004022060A2 (en)	2002-09-06	2004-03-18	Janssen Pharmaceutica, N.V.	(1h-benzoimidazol-2-yl)-(piperazinyl)-methanone derivatives and related compounds as histamine h4-receptor antagonists for the treatment of inflammatory and allergic disorders
US9017724B2 (en)	2004-02-24	2015-04-28	The General Hospital Corporation	Catalytic radiofluorination
US8257680B1 (en)	2004-02-24	2012-09-04	The General Hospital Corporation	Catalytic radiofluorination
EP2388017B1 (en) *	2004-02-24	2014-12-24	The General Hospital Corporation	Catalytic radiofluorination
FR2877005A1 (fr) *	2004-10-22	2006-04-28	Bioprojet Soc Civ Ile	Nouveaux derives d'arylpiperazine
US7731940B2 (en)	2006-01-25	2010-06-08	The Regents Of The University Of California	Compositions and methods related to serotonin 5-HT1A receptors
EP3231804B1 (en)	2008-03-21	2021-03-03	The General Hospital Corporation	Compounds and compositions for the detection and treatment of alzheimer's disease and related disorders
KR20190040502A (ko) *	2016-08-26	2019-04-18	브리스톨-마이어스 스큅 컴퍼니	인돌아민 2,3-디옥시게나제의 억제제 및 그의 사용 방법
PT109740B (pt)	2016-11-14	2020-07-30	Hovione Farmaciencia Sa	Processo para a preparação de brometo de umeclidínio
KR102823891B1 (ko) *	2020-01-14	2025-06-20	서울대학교산학협력단	혈관생성 저해 효과를 가지는 n-페닐벤조티아졸-2-아민 화합물 및 그를 포함하는 약제학적 조성물

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE3480340D1 (en) *	1984-05-22	1989-12-07	Sumitomo Chemical Co	Novel radioactive iodospiroperidol and process for its preparation
AU620327B2 (en) *	1987-04-08	1992-02-20	Salutar, Inc.	Amyloidosis and alzheimer's disease diagnostic assay and reagents therefor
US4929618A (en) *	1988-03-25	1990-05-29	Ube Industries, Ltd.	Piperdine and piperazine derivatives, and antihistaminic pharmaceutical compositions containing the same
FR2656609B1 (fr) *	1989-12-28	1992-03-27	Synthelabo	Derives de 2-aminopyrimidine-4-carboxamide, leur preparation et leur application en therapeutique.
US5731438A (en) *	1996-08-01	1998-03-24	Isis Pharmaceuticals, Inc.	N-(aminoalkyl)-and/or N-(amidoalkyl)-dinitrogen heterocycles

1997
- 1997-05-01 TW TW086105767A patent/TW593290B/zh not_active IP Right Cessation
- 1997-05-02 IL IL12696897A patent/IL126968A0/xx not_active IP Right Cessation
- 1997-05-02 ES ES03075959T patent/ES2279923T3/es not_active Expired - Lifetime
- 1997-05-02 AT AT03075959T patent/ATE350373T1/de not_active IP Right Cessation
- 1997-05-02 BR BR9709065A patent/BR9709065A/pt not_active IP Right Cessation
- 1997-05-02 DE DE69730962T patent/DE69730962T2/de not_active Expired - Lifetime
- 1997-05-02 TR TR1998/02253T patent/TR199802253T2/xx unknown
- 1997-05-02 CN CN97194515A patent/CN1074766C/zh not_active Expired - Lifetime
- 1997-05-02 AU AU29560/97A patent/AU710175B2/en not_active Ceased
- 1997-05-02 WO PCT/EP1997/002505 patent/WO1997043271A1/en not_active Ceased
- 1997-05-02 EP EP03075959A patent/EP1325917B1/en not_active Expired - Lifetime
- 1997-05-02 EA EA199801000A patent/EA001360B1/ru not_active IP Right Cessation
- 1997-05-02 AT AT97923913T patent/ATE277917T1/de not_active IP Right Cessation
- 1997-05-02 ES ES97923913T patent/ES2230605T3/es not_active Expired - Lifetime
- 1997-05-02 EE EE9800378A patent/EE03563B1/xx not_active IP Right Cessation
- 1997-05-02 CZ CZ19983553A patent/CZ295639B6/cs not_active IP Right Cessation
- 1997-05-02 PL PL97329849A patent/PL190721B1/pl not_active IP Right Cessation
- 1997-05-02 NZ NZ332309A patent/NZ332309A/xx unknown
- 1997-05-02 EP EP97923913A patent/EP0912533B1/en not_active Expired - Lifetime
- 1997-05-02 JP JP54053597A patent/JP3237759B2/ja not_active Expired - Lifetime
- 1997-05-02 US US09/180,369 patent/US6103725A/en not_active Expired - Lifetime
- 1997-05-02 CA CA002253453A patent/CA2253453C/en not_active Expired - Fee Related
- 1997-05-02 SK SK1532-98A patent/SK282919B6/sk not_active IP Right Cessation
- 1997-05-02 HU HU9902993A patent/HUP9902993A3/hu unknown
- 1997-05-02 KR KR1019980707914A patent/KR100330699B1/ko not_active Expired - Fee Related
- 1997-05-02 DE DE69737217T patent/DE69737217T2/de not_active Expired - Lifetime
- 1997-05-07 MY MYPI97002022A patent/MY117852A/en unknown
- 1997-05-09 ZA ZA974053A patent/ZA974053B/xx unknown
- 1997-05-09 AR ARP970101955A patent/AR007079A1/es active IP Right Grant
- 1997-05-09 ID IDP971546A patent/ID16889A/id unknown
1998
- 1998-10-07 BG BG102819A patent/BG64097B1/bg unknown
- 1998-11-09 NO NO19985227A patent/NO311027B1/no unknown
2000
- 2000-06-27 US US09/604,427 patent/US6224849B1/en not_active Expired - Lifetime

Also Published As

Publication number	Publication date
CN1218461A (zh)	1999-06-02
NZ332309A (en)	1999-08-30
TR199802253T2 (xx)	1999-02-22
ES2230605T3 (es)	2005-05-01
NO311027B1 (no)	2001-10-01
US6103725A (en)	2000-08-15
EA001360B1 (ru)	2001-02-26
ATE277917T1 (de)	2004-10-15
BG102819A (en)	1999-08-31
AR007079A1 (es)	1999-10-13
EE03563B1 (et)	2001-12-17
HK1018457A1 (en)	1999-12-24
SK282919B6 (sk)	2003-01-09
EA199801000A1 (ru)	1999-04-29
SK153298A3 (en)	1999-03-12
DE69737217D1 (de)	2007-02-15
BG64097B1 (bg)	2003-12-31
ES2279923T3 (es)	2007-09-01
BR9709065A (pt)	1999-08-03
JP3237759B2 (ja)	2001-12-10
CZ295639B6 (cs)	2005-09-14
HUP9902993A2 (hu)	2000-05-28
IL126968A0 (en)	1999-09-22
EP1325917B1 (en)	2007-01-03
NO985227D0 (no)	1998-11-09
ZA974053B (en)	1998-11-09
DE69730962D1 (de)	2004-11-04
US6224849B1 (en)	2001-05-01
CN1074766C (zh)	2001-11-14
ATE350373T1 (de)	2007-01-15
KR100330699B1 (ko)	2002-08-27
ID16889A (id)	1997-11-20
EP1325917A1 (en)	2003-07-09
AU710175B2 (en)	1999-09-16
EP0912533A1 (en)	1999-05-06
DE69730962T2 (de)	2006-03-30
EP0912533B1 (en)	2004-09-29
WO1997043271A1 (en)	1997-11-20
PL329849A1 (en)	1999-04-12
HUP9902993A3 (en)	2002-01-28
TW593290B (en)	2004-06-21
CA2253453C (en)	2007-01-16
AU2956097A (en)	1997-12-05
CZ355398A3 (cs)	1999-02-17
HK1057044A1 (en)	2004-03-12
MY117852A (en)	2004-08-30
KR20000005227A (ko)	2000-01-25
PL190721B1 (pl)	2005-12-30
EE9800378A (et)	1999-04-15
CA2253453A1 (en)	1997-11-20
DE69737217T2 (de)	2007-11-08
JP2000503667A (ja)	2000-03-28

Publication	Publication Date	Title
ATE323682T1 (de)	2006-05-15	Aryl-pyrimidin-derivate
DK0891332T3 (da)	2004-07-05	6-phenylpyridyl-2-aminderivater
FI954681A7 (fi)	1996-04-05	Sykloalkano-indoli- ja azaindolijohdannaisia
FR11C0020I2 (fr)	2012-03-16	Dérives difluoroprostaglandines et leur application
FI954829L (fi)	1996-04-15	Aroyylipiperidiinijohdannaiset
NO952854D0 (no)	1995-07-18	1-arylpyrimidin-derivater
DE59508427D1 (de)	2000-07-06	3-aryl-4-hydroxy-delta 3 -dihydrothiophenon-derivate
NO981946D0 (no)	1998-04-29	Imidazoquinazolin-derivater
EE9800219A (xx)	1998-12-15	Uued 19-nor-pregneeni derivaadid
NO985227L (no)	1999-01-11	Alkylaminobenzothiazol og -benzoksazol - derivater
BR9506832A (pt)	1997-10-14	N-pirazolilanilinas e n-pirazolilaminopiridinas
DE69732576D1 (de)	2005-03-31	Tetrahydrobenzindolon-derivate
DE69430587D1 (de)	2002-06-13	Pyrimidin-acyclonukleosid-derivate
FI971227L (fi)	1997-05-23	Pyramidinyylipyratsolijohdannaisia
IS5026A (is)	1999-04-15	2-metoxýfenýlpíperasín afleiður
DK0826679T3 (da)	2002-05-21	Naphthylforbindelser og -præparater
DE69527786D1 (de)	2002-09-19	Diaminomethyliden-derivate
FI964853L (fi)	1997-02-07	Deasetoksitaksolijohdannaiset
DE59509209D1 (de)	2001-05-23	Diphenyloxazolin-derivate
DE69510792D1 (de)	1999-08-19	Naphtochinonderivate
FI955026A7 (fi)	1996-04-23	Alkyyli-5-metyylisulfonyylibentsoyyliguanidiinijohdannaisia
FI965181A7 (fi)	1998-06-21	Polyalkoholi-peptidijohdannaiset
FI963122L (fi)	1996-08-09	Karbamoyylimetyyliureajohdannaiset
DE59812220D1 (de)	2009-06-04	Halte- und trageband
BR7603138U (pt)	1998-09-22	Prática e única