OA09358A - Dérivés azoliques. - Google Patents

Dérivés azoliques.

Info

Publication number: OA09358A
Authority: OA; OAPI
Prior art keywords: azolic derivatives; azolic; derivatives
Prior art date: 1990-05-29

Application number

OA60010A

Other languages

English (en)

Inventor

Caulkett Peter William Rodney

Jones Geraint

Collis Michael George

Poucher Simon Martin

Original Assignee

Ici Plc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1990-05-29

Filing date

1991-05-29

Publication date

1992-09-15

1990-05-29 Priority claimed from GB909011913A external-priority patent/GB9011913D0/en

1990-05-29 Priority claimed from GB909011914A external-priority patent/GB9011914D0/en

1991-01-22 Priority claimed from GB919101380A external-priority patent/GB9101380D0/en

1991-01-22 Priority claimed from GB919101379A external-priority patent/GB9101379D0/en

1991-02-27 Priority claimed from GB919104125A external-priority patent/GB9104125D0/en

1991-05-29 Application filed by Ici Plc filed Critical Ici Plc

1992-09-15 Publication of OA09358A publication Critical patent/OA09358A/fr

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/06—Antimigraine agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/08—Vasodilators for multiple indications
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Veterinary Medicine (AREA)
Life Sciences & Earth Sciences (AREA)
Public Health (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Health & Medical Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
Heart & Thoracic Surgery (AREA)
Cardiology (AREA)
Pain & Pain Management (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Vascular Medicine (AREA)
Urology & Nephrology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)

OA60010A 1990-05-29 1991-05-29 Dérivés azoliques. OA09358A (fr)

Applications Claiming Priority (5)

Application Number	Priority Date	Filing Date	Title
GB909011913A GB9011913D0 (en)	1990-05-29	1990-05-29	Azole derivatives
GB909011914A GB9011914D0 (en)	1990-05-29	1990-05-29	Heterocyclic compounds
GB919101380A GB9101380D0 (en)	1991-01-22	1991-01-22	Azole derivatives
GB919101379A GB9101379D0 (en)	1991-01-22	1991-01-22	Heterocyclic compounds
GB919104125A GB9104125D0 (en)	1991-02-27	1991-02-27	Azole derivatives

Publications (1)

Publication Number	Publication Date
OA09358A true OA09358A (fr)	1992-09-15

Family

ID=27516979

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
OA60010A OA09358A (fr)	1990-05-29	1991-05-29	Dérivés azoliques.

Country Status (20)

Country	Link
US (1)	US5270311A (fr)
EP (1)	EP0459702A1 (fr)
JP (1)	JP2504879B2 (fr)
KR (1)	KR910020012A (fr)
CN (1)	CN1056879A (fr)
AP (1)	AP248A (fr)
AU (1)	AU642494B2 (fr)
CA (1)	CA2043424A1 (fr)
CS (1)	CS159591A3 (fr)
FI (1)	FI912563A7 (fr)
GB (1)	GB2244487B (fr)
HU (1)	HUT61311A (fr)
IE (1)	IE911818A1 (fr)
IL (1)	IL98316A (fr)
NO (1)	NO178401C (fr)
NZ (1)	NZ238288A (fr)
OA (1)	OA09358A (fr)
PT (1)	PT97776A (fr)
RO (1)	RO109542B1 (fr)
YU (1)	YU47812B (fr)

Families Citing this family (32)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
EP0459702A1 (fr) *	1990-05-29	1991-12-04	Zeneca Limited	Dérivés d'azoles
GB9226735D0 (en) *	1992-12-22	1993-02-17	Ici Plc	Azole derivatives
US5356894A (en) *	1990-05-29	1994-10-18	Rodney Peter W	Morpholinyl substituted [1,2,4]-triazolo[1,5-a]triazine as antagonist
GB9111131D0 (en) *	1991-05-23	1991-07-17	Ici Plc	Heterocyclic compounds
GB9111130D0 (en) *	1991-05-23	1991-07-17	Ici Plc	Azole derivatives
GB9125001D0 (en) *	1991-11-25	1992-01-22	Ici Plc	Heterocyclic compounds
GB9125002D0 (en) *	1991-11-25	1992-01-22	Ici Plc	Azole derivatives
GB9124968D0 (en) *	1991-11-25	1992-01-22	Ici Plc	Chemical process
WO1995003806A1 (fr) *	1993-07-27	1995-02-09	Kyowa Hakko Kogyo Co., Ltd.	Remede contre la maladie de parkinson
CA2148502A1 (fr) *	1993-09-06	1995-03-16	Fumio Suzuki	Antidepresseurs
DE69820866T2 (de)	1997-03-24	2004-12-30	Kyowa Hakko Kogyo Co., Ltd.	[1,2,4]TRIAZOLO[1,5-c]PYRIMIDIN-DERIVATE
US6060481A (en) *	1998-05-28	2000-05-09	The Penn State Research Foundation	Method for improving insulin sensitivity using an adenosine receptor antagonist
WO2000017201A1 (fr) *	1998-09-22	2000-03-30	Kyowa Hakko Kogyo Co., Ltd.	DERIVES DE [1,2,4]TRIAZOLO[1,5-c]PYRIMIDINE
WO2004029056A1 (fr) *	2002-09-24	2004-04-08	Kyowa Hakko Kogyo Co., Ltd.	Dérivé de [1,2,4]-triazolo[1,5]pyrimidine
US7329658B2 (en) *	2003-02-06	2008-02-12	Pfizer Inc	Cannabinoid receptor ligands and uses thereof
WO2004092173A2 (fr)	2003-04-09	2004-10-28	Biogen Idec Ma Inc.	Antagonistes de recepteur d'adenosine a2a
WO2004092170A2 (fr) *	2003-04-09	2004-10-28	Biogen Idec Ma Inc.	Triazolotriazines et pyrazolotriazines et leurs procedes de fabrication et d'utilisation
WO2004092177A1 (fr)	2003-04-09	2004-10-28	Biogen Idec Ma Inc.	Triazolopyrazines et procedes de preparation et d'utilisation ce celles-ci
WO2004092172A2 (fr) *	2003-04-09	2004-10-28	Biogen Idec Ma Inc.	Triazolo[1,5-c]pyrimidines et pyrazolo[1,5-c]pyrimidines et procedes de preparation et d'utilisation de celles-ci
WO2004110454A1 (fr) *	2003-06-13	2004-12-23	Ishihara Sangyo Kaisha, Ltd.	Composition de traitement ou de prevention de maladies necessitant l'administration d'un agoniste du recepteur a2a de l'adenosine
AU2006204724A1 (en)	2005-01-14	2006-07-20	Millennium Pharmaceuticals, Inc.	Cinnamide and hydrocinnamide derivatives with raf-kinase inhibitory activity
RU2015126797A (ru)	2012-12-06	2017-01-12	Сименс Акциенгезелльшафт	Система и способ введения тепла в геологическую формацию при помощи электромагнитной индукции
CN106916073A (zh) *	2017-01-20	2017-07-04	上海巧坤化工科技有限公司	一种大麦芽碱盐酸盐的合成方法
WO2019154294A1 (fr) *	2018-02-06	2019-08-15	江苏恒瑞医药股份有限公司	Dérivé de pyrazolo[1,5-a][1,3,5]triazine-2-amine, son procédé de préparation et son utilisation médicale
JP7197206B2 (ja) *	2018-06-26	2022-12-27	チョーチヤンビムグリーンファーマシューティカルズ、リミテッド	Ａ２ａ受容体拮抗薬として用いられるトリアゾロトリアジン誘導体
KR102633145B1 (ko) *	2018-06-26	2024-02-05	쩌지앙 빔그린 파머슈티컬스, 엘티디	A2a 수용체 길항제로서의 트리아졸로 트리아진 유도체
BE1026602B1 (fr)	2018-09-27	2020-06-18	Iteos Therapeutics S A	Inhibiteurs d’a2a ne penetrant pas dans le cerveau et methodes d’utilisation dans le traitement de cancers
WO2020103939A1 (fr) *	2018-11-22	2020-05-28	上海科技大学	Composé à cycle triazolo, son procédé de préparation, intermédiaires de celui-ci et utilisation associée
CN112028891B (zh) *	2019-07-30	2022-07-05	厦门宝太生物科技股份有限公司	腺苷受体拮抗剂
WO2021105916A1 (fr) *	2019-11-26	2021-06-03	Aurigene Discovery Technologies Limited	Composés de sulfonamide ciblant cd73 et les récepteurs d'adénosine
JP2023508182A (ja) *	2019-12-26	2023-03-01	チェジンヴィムグリーンファーマシューティカルズリミテッド	トリアゾロトリアジン誘導体の疾患治療への応用
MX2023012338A (es) *	2021-04-23	2023-10-30	Chong Kun Dang Pharmaceutical Corp	Compuesto como antagonista del receptor de adenosina a2a y composicion farmaceutica que comprende al mismo.

Family Cites Families (15)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3846423A (en) *	1972-06-08	1974-11-05	Icn Pharmaceuticals	Pyrazolo (1,5a) 1,3,5-triazines
ZA743316B (en) *	1973-05-22	1976-01-28	Sandoz Ltd	Improvements in or relating to organic compounds
US3995039A (en) *	1975-05-27	1976-11-30	Merck & Co., Inc.	Pyrazolo [1,5-a] [1,3,5] triazines
GB1579932A (en) *	1976-05-12	1980-11-26	Ici Ltd	Herbicidal triazolotriazines
GB2016002B (en) *	1978-01-09	1982-05-06	Aron Sa	Amino derivatives of pyrazolo(1,5-a)s triazine
AU2192683A (en) *	1982-12-30	1984-07-05	Biomeasure Incorporated	Pyrazolo(1,5-alpha)-1,3,5-triazines
CA1267143A (fr) *	1985-06-06	1990-03-27	Sun H. Kim	Derives de 7-phenylpyrazole[1,5-a]-1,3,5-triazine, agents anti-arthrite
DE3677445D1 (de) *	1985-09-30	1991-03-14	Ciba Geigy Ag	2-substituierte-e-kondensierte(1,5-c)-pyrimidine, pharmazeutische zubereitungen und ihre verwendung.
ES2051772T3 (es) *	1986-09-30	1994-07-01	Ciba Geigy Ag	2-sustituido-e-fusionado-(1,2,4)-triazol(1,5-c)pirimidinas, composiciones farmaceuticas y sus usos.
US4824834A (en) *	1986-10-31	1989-04-25	Otsuka Pharmaceutical Company, Limited	Pyrazolotriazine compounds
US4734413A (en) *	1987-03-02	1988-03-29	Riker Laboratories, Inc.	Substituted 1,2,4-triazolo[1,5-A]triazines as bronchodilators
DE3885357T2 (de) *	1987-06-29	1994-03-24	Duphar Int Res	Anellierte Indolderivate.
DE8817122U1 (de) *	1988-12-22	1993-02-04	Boehringer Ingelheim Kg, 55218 Ingelheim	Neue Xanthinderivate mit Adenosinantogenistischer Wirkung
US4970142A (en) *	1989-02-16	1990-11-13	Konica Corporation	Silver halide photographic light-sensitive material containing cyan coupler
EP0459702A1 (fr) *	1990-05-29	1991-12-04	Zeneca Limited	Dérivés d'azoles

1991
- 1991-05-23 EP EP91304665A patent/EP0459702A1/fr not_active Withdrawn
- 1991-05-23 GB GB9111132A patent/GB2244487B/en not_active Expired - Fee Related
- 1991-05-28 IE IE181891A patent/IE911818A1/en unknown
- 1991-05-28 US US07/708,265 patent/US5270311A/en not_active Expired - Lifetime
- 1991-05-28 AU AU77348/91A patent/AU642494B2/en not_active Ceased
- 1991-05-28 FI FI912563A patent/FI912563A7/fi not_active Application Discontinuation
- 1991-05-28 CA CA002043424A patent/CA2043424A1/fr not_active Abandoned
- 1991-05-28 PT PT97776A patent/PT97776A/pt not_active Application Discontinuation
- 1991-05-28 NZ NZ238288A patent/NZ238288A/xx unknown
- 1991-05-28 AP APAP/P/1991/000266A patent/AP248A/en active
- 1991-05-28 RO RO147639A patent/RO109542B1/ro unknown
- 1991-05-28 NO NO912051A patent/NO178401C/no unknown
- 1991-05-28 CS CS911595A patent/CS159591A3/cs unknown
- 1991-05-28 YU YU94791A patent/YU47812B/sh unknown
- 1991-05-28 KR KR1019910008926A patent/KR910020012A/ko not_active Withdrawn
- 1991-05-29 OA OA60010A patent/OA09358A/fr unknown
- 1991-05-29 HU HU911789A patent/HUT61311A/hu unknown
- 1991-05-29 JP JP3235332A patent/JP2504879B2/ja not_active Expired - Fee Related
- 1991-05-29 CN CN91103744A patent/CN1056879A/zh active Pending
- 1991-05-30 IL IL9831691A patent/IL98316A/en not_active IP Right Cessation

Also Published As

Publication number	Publication date
EP0459702A1 (fr)	1991-12-04
AU642494B2 (en)	1993-10-21
PT97776A (pt)	1992-03-31
GB9111132D0 (en)	1991-07-17
RO109542B1 (ro)	1995-03-30
KR910020012A (ko)	1991-12-19
JP2504879B2 (ja)	1996-06-05
FI912563A7 (fi)	1991-11-30
US5270311A (en)	1993-12-14
YU94791A (sh)	1994-06-24
AP9100266A0 (en)	1991-07-31
AU7734891A (en)	1991-12-05
NO178401C (no)	1996-03-20
CS159591A3 (en)	1992-01-15
FI912563A0 (fi)	1991-05-28
NO912051L (no)	1991-12-02
CN1056879A (zh)	1991-12-11
NO178401B (no)	1995-12-11
AP248A (en)	1993-03-16
NO912051D0 (no)	1991-05-28
JPH0597855A (ja)	1993-04-20
HU911789D0 (en)	1991-12-30
IL98316A (en)	1995-05-26
CA2043424A1 (fr)	1991-11-30
IE911818A1 (en)	1991-12-04
IL98316A0 (en)	1992-06-21
HUT61311A (en)	1992-12-28
GB2244487A (en)	1991-12-04
GB2244487B (en)	1994-02-02
YU47812B (sr)	1996-01-09
NZ238288A (en)	1993-07-27

Publication	Publication Date	Title
OA09358A (fr)	1992-09-15	Dérivés azoliques.
FI915487L (fi)	1992-05-23	4-bensoylisoxazolderivat.
FI915736A7 (fi)	1992-06-08	A-oxoacetamidderivat.
DE59108494D1 (de)	1997-03-06	1-H-3-Aryl-pyrrolidin-2,4-dion-Derivate
NL300250I1 (nl)	2007-02-01	Chinuclidinederivaten.
FI911702L (fi)	1991-11-11	Pollist foer teleteknik.
FI915208A7 (fi)	1992-05-07	Styrrulle.
FI923931A0 (fi)	1992-09-02	Anordning foer granskning av insidan av en foergrenad roerlinje.
FI913865A0 (fi)	1991-08-15	Stabiliserade flytande fiber- och hudbehandlingskompositioner.
FI910473L (fi)	1991-08-02	Naol - suturkombination.
DE69110254D1 (de)	1995-07-13	Hydroxychinolonderivate.
FI911776A7 (fi)	1991-10-14	Benzimidazolinonederivat.
FI913142L (fi)	1991-12-30	Migraenfoerhindrande alkoxipyrimidinderivat.
DE69103503D1 (de)	1994-09-22	Adriamycinderivate.
DZ1514A1 (fr)	2004-09-13	Dérivés de benzèneacetamides.
FI911942L (fi)	1991-10-24	Kolhydratderivat innehaollande en trisackaridenhet.
DE69105856D1 (de)	1995-01-26	Acetamidderivate.
NO911213L (no)	1991-09-27	Undervannsbroenn-koplingsmekanisme.
FI912598L (fi)	1991-12-01	Dioxo-tetrahydrokinolinderivat.
DE69108314D1 (de)	1995-04-27	Dihydro-Campholen-Aldehydderivate.
FI920394L (fi)	1992-08-02	3-kinuklidinderivat.
FI912844L (fi)	1991-12-16	Inloppslaoda.
FI906123L (fi)	1991-07-30	Nytt uttryckningssystem foer svampar.
DE59106761D1 (de)	1995-11-30	N-Acylpyrrolidin-Derivate.
ATE124392T1 (de)	1995-07-15	8-sulfamylmethylen-2-aminotetraline.