OA11570A - 4-Benzyl piperidine alkylsulfoxide heterocycles and their use as subtype-selective NMDA receptor antagonists. - Google Patents
4-Benzyl piperidine alkylsulfoxide heterocycles and their use as subtype-selective NMDA receptor antagonists. Download PDFInfo
- Publication number
- OA11570A OA11570A OA1200000347A OA1200000347A OA11570A OA 11570 A OA11570 A OA 11570A OA 1200000347 A OA1200000347 A OA 1200000347A OA 1200000347 A OA1200000347 A OA 1200000347A OA 11570 A OA11570 A OA 11570A
- Authority
- OA
- OAPI
- Prior art keywords
- benzooxazol
- piperidin
- ethanesulfinyl
- compound
- benzyl
- Prior art date
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Classifications
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
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Landscapes
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- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
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- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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- Psychiatry (AREA)
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- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Epidemiology (AREA)
- Urology & Nephrology (AREA)
- Pulmonology (AREA)
- Hospice & Palliative Care (AREA)
- Vascular Medicine (AREA)
- Psychology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US9091498P | 1998-06-26 | 1998-06-26 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| OA11570A true OA11570A (en) | 2004-07-01 |
Family
ID=22224939
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| OA1200000347A OA11570A (en) | 1998-06-26 | 1999-06-25 | 4-Benzyl piperidine alkylsulfoxide heterocycles and their use as subtype-selective NMDA receptor antagonists. |
Country Status (28)
| Country | Link |
|---|---|
| US (1) | US6284774B1 (de) |
| EP (1) | EP1089735B1 (de) |
| JP (1) | JP2002519322A (de) |
| KR (1) | KR20010053170A (de) |
| CN (1) | CN1304307A (de) |
| AP (1) | AP2000001949A0 (de) |
| AT (1) | ATE297207T1 (de) |
| AU (1) | AU769650B2 (de) |
| BG (1) | BG105082A (de) |
| BR (1) | BR9911575A (de) |
| CA (1) | CA2327888A1 (de) |
| DE (1) | DE69925730T2 (de) |
| EA (1) | EA200100058A1 (de) |
| EE (1) | EE200000778A (de) |
| ES (1) | ES2244201T3 (de) |
| HU (1) | HUP0102471A2 (de) |
| ID (1) | ID28005A (de) |
| IL (1) | IL138949A0 (de) |
| IS (1) | IS5667A (de) |
| NO (1) | NO20006482D0 (de) |
| NZ (1) | NZ508808A (de) |
| OA (1) | OA11570A (de) |
| PE (1) | PE20000728A1 (de) |
| PL (1) | PL345024A1 (de) |
| SK (1) | SK19512000A3 (de) |
| TR (1) | TR200003888T2 (de) |
| WO (1) | WO2000000197A1 (de) |
| ZA (1) | ZA200005848B (de) |
Families Citing this family (55)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6476041B1 (en) | 1999-10-29 | 2002-11-05 | Merck & Co., Inc. | 1,4 substituted piperidinyl NMDA/NR2B antagonists |
| UA73749C2 (en) * | 1999-11-01 | 2005-09-15 | Diarylenines | |
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-
1999
- 1999-06-24 PE PE1999000567A patent/PE20000728A1/es not_active Application Discontinuation
- 1999-06-25 NZ NZ508808A patent/NZ508808A/xx unknown
- 1999-06-25 EA EA200100058A patent/EA200100058A1/ru unknown
- 1999-06-25 HU HU0102471A patent/HUP0102471A2/hu unknown
- 1999-06-25 AU AU48303/99A patent/AU769650B2/en not_active Ceased
- 1999-06-25 ID IDW20002514A patent/ID28005A/id unknown
- 1999-06-25 JP JP2000556782A patent/JP2002519322A/ja active Pending
- 1999-06-25 AP APAP/P/2000/001949A patent/AP2000001949A0/en unknown
- 1999-06-25 OA OA1200000347A patent/OA11570A/en unknown
- 1999-06-25 IL IL13894999A patent/IL138949A0/xx unknown
- 1999-06-25 WO PCT/US1999/014291 patent/WO2000000197A1/en not_active Ceased
- 1999-06-25 CN CN99807087A patent/CN1304307A/zh active Pending
- 1999-06-25 ES ES99931887T patent/ES2244201T3/es not_active Expired - Lifetime
- 1999-06-25 KR KR1020007014745A patent/KR20010053170A/ko not_active Withdrawn
- 1999-06-25 PL PL99345024A patent/PL345024A1/xx unknown
- 1999-06-25 BR BR9911575-1A patent/BR9911575A/pt not_active Application Discontinuation
- 1999-06-25 TR TR2000/03888T patent/TR200003888T2/xx unknown
- 1999-06-25 CA CA002327888A patent/CA2327888A1/en not_active Abandoned
- 1999-06-25 DE DE69925730T patent/DE69925730T2/de not_active Expired - Fee Related
- 1999-06-25 SK SK1951-2000A patent/SK19512000A3/sk unknown
- 1999-06-25 EP EP99931887A patent/EP1089735B1/de not_active Expired - Lifetime
- 1999-06-25 EE EEP200000778A patent/EE200000778A/xx unknown
- 1999-06-25 US US09/674,298 patent/US6284774B1/en not_active Expired - Fee Related
- 1999-06-25 AT AT99931887T patent/ATE297207T1/de not_active IP Right Cessation
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2000
- 2000-10-16 IS IS5667A patent/IS5667A/is unknown
- 2000-10-19 ZA ZA200005848A patent/ZA200005848B/en unknown
- 2000-12-19 NO NO20006482A patent/NO20006482D0/no not_active Application Discontinuation
- 2000-12-21 BG BG105082A patent/BG105082A/xx unknown
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|---|---|
| ATE297207T1 (de) | 2005-06-15 |
| DE69925730D1 (de) | 2005-07-14 |
| PL345024A1 (en) | 2001-11-19 |
| US6284774B1 (en) | 2001-09-04 |
| ID28005A (id) | 2001-05-03 |
| ES2244201T3 (es) | 2005-12-01 |
| EA200100058A1 (ru) | 2001-08-27 |
| IL138949A0 (en) | 2001-11-25 |
| SK19512000A3 (sk) | 2001-08-06 |
| PE20000728A1 (es) | 2000-08-21 |
| NO20006482L (no) | 2000-12-19 |
| AU769650B2 (en) | 2004-01-29 |
| JP2002519322A (ja) | 2002-07-02 |
| AP2000001949A0 (en) | 2000-12-31 |
| IS5667A (is) | 2000-10-16 |
| KR20010053170A (ko) | 2001-06-25 |
| NZ508808A (en) | 2002-12-20 |
| BG105082A (en) | 2001-09-28 |
| DE69925730T2 (de) | 2006-03-23 |
| EP1089735A1 (de) | 2001-04-11 |
| EP1089735B1 (de) | 2005-06-08 |
| AU4830399A (en) | 2000-01-17 |
| NO20006482D0 (no) | 2000-12-19 |
| ZA200005848B (en) | 2001-12-18 |
| EP1089735A4 (de) | 2002-12-18 |
| EE200000778A (et) | 2002-04-15 |
| TR200003888T2 (tr) | 2001-06-21 |
| CN1304307A (zh) | 2001-07-18 |
| CA2327888A1 (en) | 2000-01-06 |
| HUP0102471A2 (hu) | 2002-05-29 |
| WO2000000197A1 (en) | 2000-01-06 |
| BR9911575A (pt) | 2001-03-20 |
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