OA12599A - Tartrate salts of 5,8, 14-triazatetracyclo Ä10.3.1.o2,11.o4.9Ü-hexadeca2(11),3,5,7,9-pentaene and pharmaceutical compositions thereof. - Google Patents

Tartrate salts of 5,8, 14-triazatetracyclo Ä10.3.1.o2,11.o4.9Ü-hexadeca2(11),3,5,7,9-pentaene and pharmaceutical compositions thereof. Download PDF

Info

Publication number: OA12599A
Authority: OA; OAPI
Prior art keywords: tartrate; compound according; pentaene; hexadeca; sait
Prior art date: 2001-05-14

Application number

OA1200300289A

Other languages

English (en)

Inventor

David Everett Bogle

Peter Robert Rose

Glenn Robert Williams

Original Assignee

Pfizer Prod Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2001-05-14

Filing date

2002-04-26

Publication date

2006-06-08

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=23117845&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=OA12599(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

2002-04-26 Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc

2006-06-08 Publication of OA12599A publication Critical patent/OA12599A/en

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102000005962 receptors Human genes 0.000 description 1
108020003175 receptors Proteins 0.000 description 1
230000004044 response Effects 0.000 description 1
238000000646 scanning calorimetry Methods 0.000 description 1
230000035945 sensitivity Effects 0.000 description 1
230000000697 serotonin reuptake Effects 0.000 description 1
150000004760 silicates Chemical class 0.000 description 1
230000000391 smoking effect Effects 0.000 description 1
239000001509 sodium citrate Substances 0.000 description 1
NLJMYIDDQXHKNR-UHFFFAOYSA-K sodium citrate Chemical compound O.O.[Na+].[Na+].[Na+].[O-]C(=O)CC(O)(CC([O-])=O)C([O-])=O NLJMYIDDQXHKNR-UHFFFAOYSA-K 0.000 description 1
235000019333 sodium laurylsulphate Nutrition 0.000 description 1
239000008247 solid mixture Substances 0.000 description 1
239000007921 spray Substances 0.000 description 1
239000005720 sucrose Substances 0.000 description 1
239000000829 suppository Substances 0.000 description 1
239000000375 suspending agent Substances 0.000 description 1
239000003765 sweetening agent Substances 0.000 description 1
238000003786 synthesis reaction Methods 0.000 description 1
235000020357 syrup Nutrition 0.000 description 1
239000006188 syrup Substances 0.000 description 1
239000003826 tablet Substances 0.000 description 1
239000000454 talc Substances 0.000 description 1
229910052623 talc Inorganic materials 0.000 description 1
229960001367 tartaric acid Drugs 0.000 description 1
239000011975 tartaric acid Substances 0.000 description 1
235000002906 tartaric acid Nutrition 0.000 description 1
230000000699 topical effect Effects 0.000 description 1
239000003029 tricyclic antidepressant agent Substances 0.000 description 1
238000005406 washing Methods 0.000 description 1
239000003643 water by type Substances 0.000 description 1
238000002424 x-ray crystallography Methods 0.000 description 1

Classifications

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- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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Pharmacology & Pharmacy (AREA)
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OA1200300289A 2001-05-14 2002-04-26 Tartrate salts of 5,8, 14-triazatetracyclo Ä10.3.1.o2,11.o4.9Ü-hexadeca2(11),3,5,7,9-pentaene and pharmaceutical compositions thereof. OA12599A (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US29086101P	2001-05-14	2001-05-14

Publications (1)

Publication Number	Publication Date
OA12599A true OA12599A (en)	2006-06-08

Family

ID=23117845

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
OA1200300289A OA12599A (en)	2001-05-14	2002-04-26	Tartrate salts of 5,8, 14-triazatetracyclo Ä10.3.1.o2,11.o4.9Ü-hexadeca2(11),3,5,7,9-pentaene and pharmaceutical compositions thereof.

Country Status (47)

Country	Link
US (2)	US6890927B2 (es)
EP (1)	EP1392307B1 (es)
JP (1)	JP3779682B2 (es)
KR (1)	KR100551184B1 (es)
CN (1)	CN100370987C (es)
AP (1)	AP1473A (es)
AR (1)	AR033635A1 (es)
AT (1)	ATE302607T1 (es)
AU (1)	AU2002253482B2 (es)
BG (1)	BG66408B1 (es)
BR (1)	BR0209605A (es)
CA (1)	CA2447405C (es)
CR (1)	CR7080A (es)
CZ (1)	CZ304763B6 (es)
DE (1)	DE60205742T2 (es)
DK (1)	DK1392307T3 (es)
DO (1)	DOP2002000392A (es)
EA (1)	EA005528B1 (es)
EC (2)	ECSP034849A (es)
EE (1)	EE05441B1 (es)
EG (1)	EG24228A (es)
ES (1)	ES2246396T3 (es)
GE (1)	GEP20053712B (es)
GT (1)	GT200200084A (es)
HR (1)	HRP20030910B1 (es)
HU (1)	HU229867B1 (es)
IL (2)	IL157933A0 (es)
IS (1)	IS2217B (es)
MA (1)	MA27020A1 (es)
ME (1)	ME00466B (es)
MX (1)	MXPA03010364A (es)
MY (1)	MY127807A (es)
NO (1)	NO326148B1 (es)
NZ (1)	NZ528210A (es)
OA (1)	OA12599A (es)
PA (1)	PA8545101A1 (es)
PE (1)	PE20021065A1 (es)
PL (1)	PL214876B1 (es)
PT (1)	PT1392307E (es)
RS (1)	RS50814B (es)
SI (1)	SI1392307T1 (es)
SK (1)	SK287170B6 (es)
TN (1)	TNSN03113A1 (es)
TW (1)	TWI262078B (es)
UA (1)	UA73422C2 (es)
WO (1)	WO2002092089A1 (es)
ZA (1)	ZA200307235B (es)

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Also Published As

Publication number	Publication date
AR033635A1 (es)	2003-12-26
EG24228A (en)	2008-11-10
DE60205742D1 (de)	2005-09-29
HU229867B1 (en)	2014-10-28
US20050148591A1 (en)	2005-07-07
SK13362003A3 (en)	2004-11-03
AU2002253482B2 (en)	2007-09-06
JP2004533446A (ja)	2004-11-04
BG66408B1 (bg)	2014-01-31
KR100551184B1 (ko)	2006-02-13
CN1509174A (zh)	2004-06-30
EE05441B1 (et)	2011-08-15
SI1392307T1 (sl)	2005-12-31
CA2447405A1 (en)	2002-11-21
TNSN03113A1 (fr)	2005-12-23
IS6957A (is)	2003-09-15
DK1392307T3 (da)	2005-11-07
NO20035036L (no)	2003-11-13
DOP2002000392A (es)	2002-11-15
WO2002092089A1 (en)	2002-11-21
EE200300556A (et)	2004-04-15
NO326148B1 (no)	2008-10-06
MA27020A1 (fr)	2004-12-20
US20030166701A1 (en)	2003-09-04
TWI262078B (en)	2006-09-21
EA200301121A1 (ru)	2004-02-26
ZA200307235B (en)	2004-09-16
US6890927B2 (en)	2005-05-10
AP1473A (en)	2005-09-30
US7265119B2 (en)	2007-09-04
UA73422C2 (en)	2005-07-15
EP1392307B1 (en)	2005-08-24
ME00466B (me)	2011-10-10
MY127807A (en)	2006-12-29
HRP20030910B1 (hr)	2011-11-30
EA005528B1 (ru)	2005-04-28
HRP20030910A2 (en)	2004-02-29
PT1392307E (pt)	2005-11-30
CN100370987C (zh)	2008-02-27
CA2447405C (en)	2006-10-17
EP1392307A1 (en)	2004-03-03
AP2002002523A0 (en)	2002-06-30
GT200200084A (es)	2003-09-12
PA8545101A1 (es)	2003-09-05
JP3779682B2 (ja)	2006-05-31
ES2246396T3 (es)	2006-02-16
PE20021065A1 (es)	2002-11-21
PL214876B1 (pl)	2013-09-30
IS2217B (is)	2007-03-15
DE60205742T2 (de)	2006-05-11
CR7080A (es)	2006-08-09
ECSP034849A (es)	2003-12-24
KR20040010638A (ko)	2004-01-31
CZ20032916A3 (cs)	2004-09-15
RS50814B (sr)	2010-08-31
IL157933A0 (en)	2004-03-28
YU86703A (sh)	2006-05-25
BG108343A (bg)	2004-12-30
ECSP034850A (es)	2003-12-24
NZ528210A (en)	2005-04-29
MXPA03010364A (es)	2004-03-16
HUP0304088A3 (en)	2011-11-28
ATE302607T1 (de)	2005-09-15
HK1062645A1 (en)	2004-11-19
IL157933A (en)	2013-07-31
HUP0304088A2 (hu)	2004-04-28
NO20035036D0 (no)	2003-11-13
SK287170B6 (sk)	2010-02-08
GEP20053712B (en)	2005-12-26
BR0209605A (pt)	2004-03-23
CZ304763B6 (cs)	2014-10-01
PL366551A1 (en)	2005-02-07

Publication	Publication Date	Title
OA12599A (en)	2006-06-08	Tartrate salts of 5,8, 14-triazatetracyclo Ä10.3.1.o2,11.o4.9Ü-hexadeca2(11),3,5,7,9-pentaene and pharmaceutical compositions thereof.
AU2002253482A1 (en)	2003-05-01	Tartrate salts of 5,8,14-triazatetracyclo (10.3.102,11.04.9)-hexadeca-2(11),3,5,7,9-pentaene and pharmaceutical compositions thereof
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CN118791505A (zh)	2024-10-18	一种含肟结构的杂环化合物及其制备方法与用途
KR100572430B1 (ko)	2006-04-18	치료적 화합물의 시트르산 염 및 그의 약제학적 조성물
JP7434273B2 (ja)	2024-02-20	アゼチジン誘導体のボレート
AU2002255219A1 (en)	2002-11-25	The citrate salt of 5, 8, 14-triazatetracyclo(10.3.1.02,11,04.9)-hexadeca-2(11),3,5,7,9-pentaene and pharmaceutical compositions thereof
HK1062645B (en)	2008-08-01	Tartrate salts of 5,8,14-triazatetracyclo[10.3.1.02,11.04,9]-hexadeca-2(11),3,5,7,9-pentaene