OA12718A - Benzamide and heteroarylamide as P2X7 receptor antagonists. - Google Patents
Benzamide and heteroarylamide as P2X7 receptor antagonists. Download PDFInfo
- Publication number
- OA12718A OA12718A OA1200400127A OA1200400127A OA12718A OA 12718 A OA12718 A OA 12718A OA 1200400127 A OA1200400127 A OA 1200400127A OA 1200400127 A OA1200400127 A OA 1200400127A OA 12718 A OA12718 A OA 12718A
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- alkyl
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- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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- C07D253/02—Heterocyclic compounds containing six-membered rings having three nitrogen atoms as the only ring hetero atoms, not provided for by group C07D251/00 not condensed with other rings
- C07D253/06—1,2,4-Triazines
- C07D253/065—1,2,4-Triazines having three double bonds between ring members or between ring members and non-ring members
- C07D253/07—1,2,4-Triazines having three double bonds between ring members or between ring members and non-ring members with hetero atoms, or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D253/075—Two hetero atoms, in positions 3 and 5
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- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
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- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/62—Oxygen or sulfur atoms
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- C07D241/06—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having one or two double bonds between ring members or between ring members and non-ring members
- C07D241/08—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having one or two double bonds between ring members or between ring members and non-ring members with oxygen atoms directly attached to ring carbon atoms
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- C07D249/10—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
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- C07D263/18—Oxygen atoms
- C07D263/20—Oxygen atoms attached in position 2
- C07D263/24—Oxygen atoms attached in position 2 with hydrocarbon radicals, substituted by oxygen atoms, attached to other ring carbon atoms
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- C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
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- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
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- Engineering & Computer Science (AREA)
- Neurology (AREA)
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- Neurosurgery (AREA)
- Immunology (AREA)
- Physical Education & Sports Medicine (AREA)
- Diabetes (AREA)
- Rheumatology (AREA)
- Cardiology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Heart & Thoracic Surgery (AREA)
- Pain & Pain Management (AREA)
- Oncology (AREA)
- Pulmonology (AREA)
- Tropical Medicine & Parasitology (AREA)
- Communicable Diseases (AREA)
- Hematology (AREA)
- Psychology (AREA)
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Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US33678101P | 2001-11-12 | 2001-11-12 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| OA12718A true OA12718A (en) | 2006-06-27 |
Family
ID=23317638
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| OA1200400127A OA12718A (en) | 2001-11-12 | 2002-11-04 | Benzamide and heteroarylamide as P2X7 receptor antagonists. |
Country Status (35)
| Country | Link |
|---|---|
| US (2) | US7214677B2 (is) |
| EP (1) | EP1448535B1 (is) |
| JP (1) | JP4365218B2 (is) |
| KR (1) | KR20050043785A (is) |
| CN (1) | CN1585755A (is) |
| AP (1) | AP2004003028A0 (is) |
| AR (1) | AR038365A1 (is) |
| AT (1) | ATE502020T1 (is) |
| BR (1) | BR0214044A (is) |
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| CY (1) | CY1111405T1 (is) |
| DE (1) | DE60239485D1 (is) |
| DK (1) | DK1448535T3 (is) |
| EA (1) | EA200400488A1 (is) |
| EC (1) | ECSP045097A (is) |
| ES (1) | ES2358988T3 (is) |
| GT (1) | GT200200224A (is) |
| HN (1) | HN2002000319A (is) |
| HU (1) | HUP0401936A3 (is) |
| IL (1) | IL161329A0 (is) |
| IS (1) | IS7216A (is) |
| MA (1) | MA27144A1 (is) |
| MX (1) | MXPA04004465A (is) |
| NO (1) | NO20041922L (is) |
| OA (1) | OA12718A (is) |
| PA (1) | PA8557501A1 (is) |
| PE (1) | PE20030537A1 (is) |
| PL (1) | PL370762A1 (is) |
| PT (1) | PT1448535E (is) |
| PY (1) | PY0227300A (is) |
| SV (1) | SV2004001393A (is) |
| TN (1) | TNSN04083A1 (is) |
| UY (1) | UY27535A1 (is) |
| WO (1) | WO2003042191A1 (is) |
| ZA (1) | ZA200402754B (is) |
Families Citing this family (76)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| PA8557501A1 (es) * | 2001-11-12 | 2003-06-30 | Pfizer Prod Inc | Benzamida, heteroarilamida y amidas inversas |
| PA8591801A1 (es) * | 2002-12-31 | 2004-07-26 | Pfizer Prod Inc | Inhibidores benzamidicos del receptor p2x7. |
| BR0317844A (pt) * | 2002-12-31 | 2005-12-06 | Pfizer Prod Inc | Inibidores de benzamida do receptor p2x7 |
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- 2002-11-04 PL PL02370762A patent/PL370762A1/xx not_active Application Discontinuation
- 2002-11-04 AT AT02783358T patent/ATE502020T1/de active
- 2002-11-04 ES ES02783358T patent/ES2358988T3/es not_active Expired - Lifetime
- 2002-11-04 IL IL16132902A patent/IL161329A0/xx unknown
- 2002-11-04 DK DK02783358.1T patent/DK1448535T3/da active
- 2002-11-04 CN CNA028224752A patent/CN1585755A/zh active Pending
- 2002-11-05 PE PE2002001077A patent/PE20030537A1/es not_active Application Discontinuation
- 2002-11-08 UY UY27535A patent/UY27535A1/es not_active Application Discontinuation
- 2002-11-11 HN HN2002000319A patent/HN2002000319A/es unknown
- 2002-11-11 SV SV2002001393A patent/SV2004001393A/es not_active Application Discontinuation
- 2002-11-11 AR ARP020104318A patent/AR038365A1/es unknown
- 2002-11-12 US US10/292,887 patent/US7214677B2/en not_active Expired - Fee Related
-
2004
- 2004-04-07 IS IS7216A patent/IS7216A/is unknown
- 2004-04-08 ZA ZA200402754A patent/ZA200402754B/en unknown
- 2004-04-28 MA MA27660A patent/MA27144A1/fr unknown
- 2004-05-06 EC EC2004005097A patent/ECSP045097A/es unknown
- 2004-05-11 NO NO20041922A patent/NO20041922L/no not_active Application Discontinuation
- 2004-05-11 TN TNP2004000083A patent/TNSN04083A1/fr unknown
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2005
- 2005-10-18 US US11/253,112 patent/US7235549B2/en not_active Expired - Fee Related
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2011
- 2011-04-26 CY CY20111100413T patent/CY1111405T1/el unknown
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