PH23736A - Emulsion compositions for the parenteral and/or oral administration of sparingly water soluble ionizable hydrophobic drugs - Google Patents

Emulsion compositions for the parenteral and/or oral administration of sparingly water soluble ionizable hydrophobic drugs

Info

Publication number
PH23736A
PH23736A PH34246A PH34246A PH23736A PH 23736 A PH23736 A PH 23736A PH 34246 A PH34246 A PH 34246A PH 34246 A PH34246 A PH 34246A PH 23736 A PH23736 A PH 23736A
Authority
PH
Philippines
Prior art keywords
parenteral
oral administration
water soluble
emulsion compositions
hydrophobic drugs
Prior art date
Application number
PH34246A
Other languages
English (en)
Inventor
Narendra Raghunathi Desai
Madurai Ganesan
Eugene Albert Carpenter
Edward Charles Shinal
Original Assignee
American Cyanamid Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by American Cyanamid Co filed Critical American Cyanamid Co
Publication of PH23736A publication Critical patent/PH23736A/en

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/10—Dispersions; Emulsions
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/10—Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/44—Oils, fats or waxes according to two or more groups of A61K47/02-A61K47/42; Natural or modified natural oils, fats or waxes, e.g. castor oil, polyethoxylated castor oil, montan wax, lignite, shellac, rosin, beeswax or lanolin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/10—Dispersions; Emulsions
    • A61K9/107—Emulsions ; Emulsion preconcentrates; Micelles

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Dispersion Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Dermatology (AREA)
  • Engineering & Computer Science (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
PH34246A 1985-09-16 1986-09-11 Emulsion compositions for the parenteral and/or oral administration of sparingly water soluble ionizable hydrophobic drugs PH23736A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/776,306 US4784845A (en) 1985-09-16 1985-09-16 Emulsion compostions for the parenteral administration of sparingly water soluble ionizable hydrophobic drugs

Publications (1)

Publication Number Publication Date
PH23736A true PH23736A (en) 1989-11-03

Family

ID=25107019

Family Applications (1)

Application Number Title Priority Date Filing Date
PH34246A PH23736A (en) 1985-09-16 1986-09-11 Emulsion compositions for the parenteral and/or oral administration of sparingly water soluble ionizable hydrophobic drugs

Country Status (18)

Country Link
US (1) US4784845A (de)
EP (1) EP0215313B1 (de)
JP (1) JPS6267018A (de)
KR (1) KR890004684B1 (de)
AR (1) AR242716A1 (de)
AT (1) ATE78683T1 (de)
AU (1) AU591705B2 (de)
CA (1) CA1272447A (de)
DE (1) DE3686221T2 (de)
DK (1) DK165730C (de)
ES (1) ES2002750A6 (de)
FI (1) FI863728L (de)
GR (1) GR862354B (de)
HU (1) HU199282B (de)
NO (1) NO863670L (de)
NZ (1) NZ217484A (de)
PH (1) PH23736A (de)
ZA (1) ZA867009B (de)

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US5004593A (en) * 1989-04-17 1991-04-02 Mayo Foundation For Medical Education And Research Hexamethylmelamine formulation exhibiting reduced neurotoxicity
CA2017507C (en) 1989-05-25 1996-11-12 Gary Van Nest Adjuvant formulation comprising a submicron oil droplet emulsion
GB8919172D0 (en) * 1989-08-23 1989-10-04 Univ Nottingham Useful composition
US5534502A (en) * 1990-11-06 1996-07-09 Nippon Shinyaku Co. Ltd. Process for producing fat emulsion
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DE4124252A1 (de) * 1991-07-22 1993-01-28 Knoll Ag Verfahren zur herstellung einer sterilfiltrierbaren wirkstoffloesung
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WO1994028872A1 (en) * 1993-06-04 1994-12-22 Warner-Lambert Company Non-alcoholic cold and sinus medication
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US5616330A (en) * 1994-07-19 1997-04-01 Hemagen/Pfc Stable oil-in-water emulsions incorporating a taxine (taxol) and method of making same
US5616342A (en) * 1995-04-11 1997-04-01 Pdt, Inc. Emulsioin suitable for administering a poorly water-soluble photosensitizing compound and use thereof
US5824638A (en) * 1995-05-22 1998-10-20 Shire Laboratories, Inc. Oral insulin delivery
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US6458373B1 (en) * 1997-01-07 2002-10-01 Sonus Pharmaceuticals, Inc. Emulsion vehicle for poorly soluble drugs
US6054421A (en) * 1997-09-23 2000-04-25 Scimed Life Systems, Inc. Medical emulsion lubricant
US6281175B1 (en) 1997-09-23 2001-08-28 Scimed Life Systems, Inc. Medical emulsion for lubrication and delivery of drugs
US6169084B1 (en) * 1997-09-30 2001-01-02 Eli Lilly And Company 2-methyl-thieno-benzodiazepine formulation
US6036946A (en) * 1997-12-24 2000-03-14 Shaklee Corporation Methods for protecting skin from damaging effects of ultraviolet light
WO1999043301A1 (en) * 1998-02-24 1999-09-02 The Board Of Trustees Of The University Of Illinois Lipid emulsions in the treatment of systemic poisoning
US7030155B2 (en) * 1998-06-05 2006-04-18 Sonus Pharmaceuticals, Inc. Emulsion vehicle for poorly soluble drugs
US6146664A (en) * 1998-07-10 2000-11-14 Shaklee Corporation Stable topical ascorbic acid compositions
US6682758B1 (en) 1998-12-22 2004-01-27 The United States Of America As Represented By The Department Of Health And Human Services Water-insoluble drug delivery system
US6777450B1 (en) * 2000-05-26 2004-08-17 Color Access, Inc. Water-thin emulsions with low emulsifier levels
JP2005515996A (ja) * 2001-12-03 2005-06-02 ノバセア インコーポレイティッド 活性型ビタミンｄ化合物を含む薬学的組成物
AU2002353118A1 (en) * 2001-12-11 2003-07-24 Dor Biopharma, Inc. Lipid particles and suspensions and uses thereof
US20040058895A1 (en) * 2002-09-18 2004-03-25 Bone Care International, Inc. Multi-use vessels for vitamin D formulations
US7148211B2 (en) * 2002-09-18 2006-12-12 Genzyme Corporation Formulation for lipophilic agents
US20040053895A1 (en) * 2002-09-18 2004-03-18 Bone Care International, Inc. Multi-use vessels for vitamin D formulations
US20040062779A1 (en) * 2002-09-26 2004-04-01 Jerry Whittemore Dermatologic composition using ultra-fine/micronized 1-ascorbic acid and other antioxidant ingredients in a stabilized anhydrous vehicle
US20060189586A1 (en) * 2003-06-11 2006-08-24 Cleland Jeffrey L Pharmaceutical compositions comprising active vitamin D compounds
US20050186230A1 (en) * 2004-01-23 2005-08-25 Sd Pharmaceuticals, Inc. Elemene compositions containing liquid oil
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ES2375115T3 (es) 2005-03-31 2012-02-24 Suntory Holdings Limited Emulsión de aceite en agua que contiene un compuesto de lignano y composición que comprenden al mismo.
CN101547687A (zh) * 2005-11-17 2009-09-30 生物药效率有限公司 生物相容的潜在乳化剂
KR101425241B1 (ko) * 2006-10-04 2014-08-01 산토리 홀딩스 가부시키가이샤 리그난류 화합물 함유 ｏ/ｗ/ｏ형 에멀션 및 그것을 함유하는 조성물
EP2200613B1 (de) 2007-09-21 2018-09-05 The Johns Hopkins University Phenazin-derivate und ihre verwendungen
NZ590141A (en) * 2008-06-24 2012-05-25 Merial Ltd Anthelminthic formulations including castor oil and another vegetable oil
CN112472699A (zh) 2013-07-26 2021-03-12 种族肿瘤学公司 改善比生群及衍生物的治疗益处的组合方法
EP3079668A1 (de) 2013-12-09 2016-10-19 Durect Corporation Pharmazeutisch aktive wirkstoffkomplexe, polymerkomplexe und zusammensetzungen und verfahren damit
EP4529951A3 (de) 2017-01-08 2025-05-28 The United States Government as Represented by the Department of Veterans Affairs Verfahren zur verminderung von verletzungen im zusammenhang mit intraoperativer hypotonie
CA3073527A1 (en) * 2017-09-12 2019-03-21 Academic Pharmaceuticals, Inc. Metolazone emulsion formulation
WO2020089942A2 (en) * 2018-11-02 2020-05-07 Amaterasu Lifesciences Llp A liquid injectable composition
CN114980896A (zh) * 2019-08-07 2022-08-30 阿克里普斯一有限公司 (6AS)-6-甲基-5,6,6A,7-四氢-4H-二苯并[de,g]喹啉-10,11-二醇的药物组合物
WO2025182691A1 (ja) * 2024-02-29 2025-09-04 株式会社ユニファイジャパン ５－デアザフラビン化合物含有乳剤およびその製造方法

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Also Published As

Publication number Publication date
AU6269686A (en) 1987-03-19
NZ217484A (en) 1990-04-26
DK438286D0 (da) 1986-09-12
GR862354B (en) 1987-01-19
EP0215313A3 (en) 1987-09-09
US4784845A (en) 1988-11-15
HUT43947A (en) 1988-01-28
EP0215313A2 (de) 1987-03-25
DK438286A (da) 1987-03-17
FI863728A7 (fi) 1987-03-17
DE3686221D1 (de) 1992-09-03
DK165730B (da) 1993-01-11
EP0215313B1 (de) 1992-07-29
KR890004684B1 (ko) 1989-11-25
NO863670D0 (no) 1986-09-15
AR242716A1 (es) 1993-05-31
ATE78683T1 (de) 1992-08-15
FI863728L (fi) 1987-03-17
AU591705B2 (en) 1989-12-14
HU199282B (en) 1990-02-28
CA1272447A (en) 1990-08-07
DK165730C (da) 1993-06-07
JPS6267018A (ja) 1987-03-26
DE3686221T2 (de) 1993-02-25
FI863728A0 (fi) 1986-09-15
ES2002750A6 (es) 1988-10-01
KR870002835A (ko) 1987-04-13
ZA867009B (en) 1987-07-29
NO863670L (no) 1987-03-17

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