PH23837A - Phenoxyalkylcarboxylic acids and esters and pharmaceutical formulation containing them - Google Patents
Phenoxyalkylcarboxylic acids and esters and pharmaceutical formulation containing themInfo
- Publication number
- PH23837A PH23837A PH34491A PH34491A PH23837A PH 23837 A PH23837 A PH 23837A PH 34491 A PH34491 A PH 34491A PH 34491 A PH34491 A PH 34491A PH 23837 A PH23837 A PH 23837A
- Authority
- PH
- Philippines
- Prior art keywords
- integer
- esters
- pharmaceutical formulation
- formulation containing
- group
- Prior art date
Links
- 239000002253 acid Substances 0.000 title 1
- 150000007513 acids Chemical class 0.000 title 1
- 150000002148 esters Chemical class 0.000 title 1
- 239000008194 pharmaceutical composition Substances 0.000 title 1
- 125000004178 (C1-C4) alkyl group Chemical group 0.000 abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 2
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 2
- 125000000229 (C1-C4)alkoxy group Chemical group 0.000 abstract 1
- 206010006482 Bronchospasm Diseases 0.000 abstract 1
- 206010047139 Vasoconstriction Diseases 0.000 abstract 1
- 125000003277 amino group Chemical group 0.000 abstract 1
- 208000006673 asthma Diseases 0.000 abstract 1
- 210000001772 blood platelet Anatomy 0.000 abstract 1
- 230000007885 bronchoconstriction Effects 0.000 abstract 1
- 125000005843 halogen group Chemical group 0.000 abstract 1
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 1
- 125000002887 hydroxy group Chemical group [H]O* 0.000 abstract 1
- 125000001624 naphthyl group Chemical group 0.000 abstract 1
- 125000000449 nitro group Chemical group [O-][N+](*)=O 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 208000010110 spontaneous platelet aggregation Diseases 0.000 abstract 1
- 125000001544 thienyl group Chemical group 0.000 abstract 1
- 125000002023 trifluoromethyl group Chemical group FC(F)(F)* 0.000 abstract 1
- 208000019553 vascular disease Diseases 0.000 abstract 1
- 230000025033 vasoconstriction Effects 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D333/30—Hetero atoms other than halogen
- C07D333/34—Sulfur atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/08—Bronchodilators
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/08—Vasodilators for multiple indications
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Pulmonology (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Hydrogenated Pyridines (AREA)
- Indole Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB858528398A GB8528398D0 (en) | 1985-11-19 | 1985-11-19 | Chemical compounds |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| PH23837A true PH23837A (en) | 1989-11-23 |
Family
ID=10588403
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PH34491A PH23837A (en) | 1985-11-19 | 1986-11-18 | Phenoxyalkylcarboxylic acids and esters and pharmaceutical formulation containing them |
Country Status (14)
| Country | Link |
|---|---|
| EP (1) | EP0223593B1 (de) |
| JP (1) | JPS62155250A (de) |
| KR (1) | KR870004950A (de) |
| AT (1) | ATE65992T1 (de) |
| AU (1) | AU593039B2 (de) |
| DE (1) | DE3680753D1 (de) |
| DK (1) | DK550186A (de) |
| FI (1) | FI864692L (de) |
| GB (2) | GB8528398D0 (de) |
| IL (1) | IL80701A0 (de) |
| NO (1) | NO864599L (de) |
| PH (1) | PH23837A (de) |
| PT (1) | PT83762B (de) |
| ZA (1) | ZA868740B (de) |
Families Citing this family (20)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE3610643A1 (de) * | 1986-03-29 | 1987-10-01 | Boehringer Mannheim Gmbh | Neue phenoxyalkylcarbonsaeure-derivate, verfahren zu ihrer herstellung sowie diese verbindungen enthaltende arzneimittel |
| DE3642105A1 (de) * | 1986-12-10 | 1988-06-16 | Bayer Ag | Substituierte aminomethyl-5,6,7,8-tetrahydronaphtyl-oxyessigsaeuren, neue zwischenprodukte, verfahren zu ihrer herstellung sowie ihre verwendung in arzneimitteln |
| AT396235B (de) * | 1987-02-06 | 1993-07-26 | Tanabe Seiyaku Co | Phenoxyessigsaeurederivate und ihre herstellung |
| GB8708233D0 (en) * | 1987-04-07 | 1987-05-13 | Smith Kline French Lab | Pharmaceutically active compounds |
| JPH068274B2 (ja) * | 1988-01-19 | 1994-02-02 | 田辺製薬株式会社 | フェノキシ酢酸誘導体 |
| EP0325245B1 (de) * | 1988-01-19 | 1993-10-20 | Tanabe Seiyaku Co., Ltd. | Phenoxyessigsäure-Derivate, ihre Herstellung, pharmazeutische Zusammensetzungen, die sie enthalten, und deren Verwendung |
| JPH068275B2 (ja) * | 1988-02-04 | 1994-02-02 | 田辺製薬株式会社 | フェノキシ酢酸誘導体 |
| DE3821540A1 (de) * | 1988-06-25 | 1989-12-28 | Boehringer Mannheim Gmbh | Neue sulfonamide, verfahren zu ihrer herstellung sowie solche sulfonamide enthaltende arzneimittel |
| DE3829431A1 (de) * | 1988-08-31 | 1990-03-01 | Boehringer Mannheim Gmbh | Sulfonamide mit tetrazolylrest, verfahren zur ihrer herstellung sowie arzneimittel |
| US5280043A (en) * | 1988-10-10 | 1994-01-18 | Smith Kline & French Laboratories Ltd. | Sulphonamido containing phenylalkanoic acids as thromboxane A2 antagonists |
| US5070099A (en) * | 1988-10-31 | 1991-12-03 | E. R. Squibb & Sons, Inc. | Arylthioalkylphenyl carboxylic acids, derivatives thereof, compositions containing same method of use |
| US4959383A (en) * | 1988-10-31 | 1990-09-25 | E. R. Squibb & Sons, Inc. | Phenylsulfone alkenoic acids, derivatives thereof, compositions containing same and method of use |
| US5006542A (en) * | 1988-10-31 | 1991-04-09 | E. R. Squibb & Sons, Inc. | Arylthioalkylphenyl carboxylic acids, derivatives thereof, compositions containing same and method of use |
| DE3942923A1 (de) * | 1989-12-23 | 1991-06-27 | Boehringer Mannheim Gmbh | Neue phenoxyalkylcarbonsaeure-amide, verfahren zu ihrer herstellung sowie diese verbindungen enthaltende arzneimittel |
| DE4031821A1 (de) * | 1990-10-08 | 1992-04-09 | Boehringer Mannheim Gmbh | Verwendung von thromboxan-a2-rezeptoren-antagonisten gegen proliferative veraenderungen in der gefaesswand |
| AU688756B2 (en) * | 1993-03-17 | 1998-03-19 | Meiji Seika Kabushiki Kaisha | Novel compound with platelet aggregation inhibitor activity |
| WO1999047497A2 (en) * | 1998-03-13 | 1999-09-23 | Merck Frosst Canada & Co. | Carboxylic acids and acylsulfonamides, compositions containing such compounds and methods of treatment |
| US6242493B1 (en) | 1998-03-13 | 2001-06-05 | Merck Frosst Canada & Co. | Carboxylic acids and acylsulfonamides, compositions containing such compounds and methods of treatment |
| JP4879433B2 (ja) * | 2000-01-13 | 2012-02-22 | エミスフェアー・テクノロジーズ・インク | 活性剤を送達するための化合物および組成物 |
| WO2007008541A2 (en) * | 2005-07-08 | 2007-01-18 | Kalypsys, Inc. | Cellular cholesterol absorption modifiers |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE2809377A1 (de) * | 1978-03-04 | 1979-09-13 | Boehringer Mannheim Gmbh | Phenoxyalkylcarbonsaeure-derivate, verfahren zu deren herstellung sowie diese verbindungen enthaltende arzneimittel |
| DE3535167A1 (de) * | 1985-10-02 | 1987-04-09 | Boehringer Mannheim Gmbh | Neue sulfonyl-phenyl(alkyl)amine, verfahren zu ihrer herstellung sowie arzneimittel |
| DE3610643A1 (de) * | 1986-03-29 | 1987-10-01 | Boehringer Mannheim Gmbh | Neue phenoxyalkylcarbonsaeure-derivate, verfahren zu ihrer herstellung sowie diese verbindungen enthaltende arzneimittel |
-
1985
- 1985-11-19 GB GB858528398A patent/GB8528398D0/en active Pending
-
1986
- 1986-11-18 DE DE8686308992T patent/DE3680753D1/de not_active Expired - Fee Related
- 1986-11-18 PT PT83762A patent/PT83762B/pt unknown
- 1986-11-18 KR KR860009720A patent/KR870004950A/ko not_active Withdrawn
- 1986-11-18 PH PH34491A patent/PH23837A/en unknown
- 1986-11-18 EP EP86308992A patent/EP0223593B1/de not_active Expired - Lifetime
- 1986-11-18 JP JP61273062A patent/JPS62155250A/ja active Pending
- 1986-11-18 FI FI864692A patent/FI864692L/fi not_active IP Right Cessation
- 1986-11-18 AU AU65505/86A patent/AU593039B2/en not_active Ceased
- 1986-11-18 NO NO864599A patent/NO864599L/no unknown
- 1986-11-18 GB GB8627512A patent/GB2183234B/en not_active Expired
- 1986-11-18 DK DK550186A patent/DK550186A/da not_active Application Discontinuation
- 1986-11-18 ZA ZA868740A patent/ZA868740B/xx unknown
- 1986-11-18 AT AT86308992T patent/ATE65992T1/de active
- 1986-11-19 IL IL80701A patent/IL80701A0/xx unknown
Also Published As
| Publication number | Publication date |
|---|---|
| FI864692A7 (fi) | 1987-05-20 |
| AU6550586A (en) | 1987-05-21 |
| DK550186A (da) | 1987-05-20 |
| EP0223593A3 (en) | 1989-01-18 |
| FI864692A0 (fi) | 1986-11-18 |
| EP0223593B1 (de) | 1991-08-07 |
| GB2183234A (en) | 1987-06-03 |
| GB8528398D0 (en) | 1985-12-24 |
| NO864599D0 (no) | 1986-11-18 |
| PT83762B (en) | 1988-12-07 |
| GB8627512D0 (en) | 1986-12-17 |
| JPS62155250A (ja) | 1987-07-10 |
| ATE65992T1 (de) | 1991-08-15 |
| IL80701A0 (en) | 1987-02-27 |
| DE3680753D1 (de) | 1991-09-12 |
| KR870004950A (ko) | 1987-06-02 |
| ZA868740B (en) | 1987-07-29 |
| NO864599L (no) | 1987-05-20 |
| FI864692L (fi) | 1987-05-20 |
| PT83762A (en) | 1986-12-01 |
| GB2183234B (en) | 1989-10-04 |
| DK550186D0 (da) | 1986-11-18 |
| AU593039B2 (en) | 1990-02-01 |
| EP0223593A2 (de) | 1987-05-27 |
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