PL149903B1 - Method of obtaining novel derivatives of 1h,3h-pyrol/1,2-c/thiazole - Google Patents

Method of obtaining novel derivatives of 1h,3h-pyrol/1,2-c/thiazole

Info

Publication number
PL149903B1
PL149903B1 PL1987279923A PL27992387A PL149903B1 PL 149903 B1 PL149903 B1 PL 149903B1 PL 1987279923 A PL1987279923 A PL 1987279923A PL 27992387 A PL27992387 A PL 27992387A PL 149903 B1 PL149903 B1 PL 149903B1
Authority
PL
Poland
Prior art keywords
formula
pyridyl
pyrrolo
phenyl
thiazole
Prior art date
Application number
PL1987279923A
Other languages
English (en)
Polish (pl)
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of PL149903B1 publication Critical patent/PL149903B1/pl

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Pyrrole Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Medicines Containing Plant Substances (AREA)
  • Steroid Compounds (AREA)
PL1987279923A 1986-07-04 1987-07-02 Method of obtaining novel derivatives of 1h,3h-pyrol/1,2-c/thiazole PL149903B1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR8609728A FR2601015B1 (fr) 1986-07-04 1986-07-04 Nouveaux derives du 1h,3h-pyrrolo (1,2-c) thiazole, leur preparation et les compositions pharmaceutiques qui les contiennent

Publications (1)

Publication Number Publication Date
PL149903B1 true PL149903B1 (en) 1990-03-31

Family

ID=9337075

Family Applications (2)

Application Number Title Priority Date Filing Date
PL1987279923A PL149903B1 (en) 1986-07-04 1987-07-02 Method of obtaining novel derivatives of 1h,3h-pyrol/1,2-c/thiazole
PL1987266582A PL149434B1 (en) 1986-07-04 1987-07-02 The method of manufacture of new derivatives of 1-pyro/2-c/thiazole

Family Applications After (1)

Application Number Title Priority Date Filing Date
PL1987266582A PL149434B1 (en) 1986-07-04 1987-07-02 The method of manufacture of new derivatives of 1-pyro/2-c/thiazole

Country Status (28)

Country Link
US (1) US4783472A (cs)
EP (1) EP0253711B1 (cs)
JP (1) JPS6322589A (cs)
KR (1) KR880001681A (cs)
AT (1) ATE53037T1 (cs)
AU (1) AU597996B2 (cs)
BG (2) BG47498A3 (cs)
CA (1) CA1294966C (cs)
CS (1) CS262692B2 (cs)
DD (1) DD263772A5 (cs)
DE (1) DE3762861D1 (cs)
DK (1) DK340087A (cs)
ES (1) ES2015070B3 (cs)
FI (1) FI84727C (cs)
FR (1) FR2601015B1 (cs)
GR (1) GR3000502T3 (cs)
HU (1) HU198727B (cs)
IE (1) IE60743B1 (cs)
IL (1) IL83066A (cs)
MA (1) MA21027A1 (cs)
MX (1) MX173398B (cs)
NO (1) NO170419C (cs)
NZ (1) NZ220929A (cs)
PL (2) PL149903B1 (cs)
PT (1) PT85235B (cs)
SU (2) SU1528323A3 (cs)
TN (1) TNSN87083A1 (cs)
ZA (1) ZA874814B (cs)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2601016B1 (fr) * 1986-07-04 1988-10-07 Rhone Poulenc Sante Nouveaux derives du 1h,3h-pyrrolo (1,2-c) thiazole, leur preparation et les compositions pharmaceutiques qui les contiennent
FR2617484B1 (fr) * 1987-07-02 1989-10-20 Rhone Poulenc Sante Procede de preparation de l'acide (pyridyl-3)-3 1h-3h-pyrrolo (1,2-c) thiazolecarboxylique-7 dextrogyre
FR2644456B1 (fr) * 1989-03-17 1991-07-05 Rhone Poulenc Sante Nouveaux derives du 1h, 3h-pyrrolo(1,2-c)thiazolecarboxamide-7, leur preparation et les compositions pharmaceutiques qui les contiennent
JP3061631B2 (ja) * 1989-10-11 2000-07-10 山之内製薬株式会社 新規なヘテロ環化合物およびその製造法
FR2662606A1 (fr) * 1990-06-01 1991-12-06 Rhone Poulenc Sante Compositions pharmaceutiques pour le traitement de la fibrillation ventriculaire, du syndrome de menace de l'infarctus du myocarde et de l'angine de poitrine contenant le n-(benzoyl-3 phenyl) (pyridyl-3)-3 1h,3h-pyrrolo[1,2-c]thiazolecarboxamide-7.
FR2687574B1 (fr) * 1992-02-25 1995-05-05 Rhone Poulenc Rorer Sa Nouvelle application therapeutique de derives du pyridylpyrrolothiazole carboxamide.
GB9207645D0 (en) * 1992-04-08 1992-05-27 Smithkline Beecham Corp Methods
AU2002367023A1 (en) * 2001-12-21 2003-07-30 Cytokinetics, Inc. Compositions and methods for treating heart failure
JP2010518014A (ja) 2007-01-31 2010-05-27 バーテックス ファーマシューティカルズ インコーポレイテッド キナーゼ阻害剤として有用な２−アミノピリジン誘導体
US8569337B2 (en) 2008-07-23 2013-10-29 Vertex Pharmaceuticals Incorporated Tri-cyclic pyrazolopyridine kinase inhibitors
JP5631310B2 (ja) 2008-07-23 2014-11-26 バーテックス ファーマシューティカルズ インコーポレイテッドＶｅｒｔｅｘ Ｐｈａｒｍａｃｅｕｔｉｃａｌｓ Ｉｎｃｏｒｐｏｒａｔｅｄ 三環式ピラゾロピリジンキナーゼ阻害剤
EP2318407B1 (en) 2008-07-23 2013-01-02 Vertex Pharmaceuticals Incorporated Pyrazolopyridine kinase inhibitors
CA2732765A1 (en) * 2008-08-06 2010-02-11 Vertex Pharmaceuticals Incorporated Aminopyridine kinase inhibitors
WO2010129668A1 (en) 2009-05-06 2010-11-11 Vertex Pharmaceuticals Incorporated Pyrazolopyridines
MX2012008643A (es) 2010-01-27 2013-02-26 Vertex Pharma Inhibidores de cinasas de pirazolopiridinas.
US9067932B2 (en) 2010-01-27 2015-06-30 Vertex Pharmaceuticals Incorporated Pyrazolopyridine kinase inhibitors
CN102869663A (zh) 2010-01-27 2013-01-09 沃泰克斯药物股份有限公司 吡唑并吡嗪激酶抑制剂
KR102608281B1 (ko) * 2022-07-27 2023-12-01 김규현 감자를 이용한 맥주 제조 방법 및 이에 의해 제조된 감자 맥주

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2541280B1 (fr) * 1983-01-13 1985-06-21 Rhone Poulenc Sante Nouveaux derives du 1h, 3h-pyrrolo (1,2c) thiazolecarboxamide-7, leur preparation et les medicaments qui les contiennent
US4500532A (en) * 1983-03-03 1985-02-19 Usv Pharmaceutical Corporation 1-(Substituted aminoalkyl)-1,4-dihydropyridines
FR2601016B1 (fr) * 1986-07-04 1988-10-07 Rhone Poulenc Sante Nouveaux derives du 1h,3h-pyrrolo (1,2-c) thiazole, leur preparation et les compositions pharmaceutiques qui les contiennent

Also Published As

Publication number Publication date
IL83066A (en) 1991-01-31
FI84727C (fi) 1992-01-10
PL266582A1 (en) 1988-09-01
NO170419B (no) 1992-07-06
IE60743B1 (en) 1994-08-10
MA21027A1 (fr) 1988-04-01
CA1294966C (fr) 1992-01-28
ES2015070B3 (es) 1990-08-01
FR2601015B1 (fr) 1988-08-05
FI872931A0 (fi) 1987-07-02
CS501387A2 (en) 1988-08-16
SU1528323A3 (ru) 1989-12-07
NO872779D0 (no) 1987-07-02
ATE53037T1 (de) 1990-06-15
DE3762861D1 (de) 1990-06-28
ZA874814B (en) 1988-03-30
SU1588284A3 (ru) 1990-08-23
PT85235B (pt) 1990-03-30
IL83066A0 (en) 1987-12-31
BG47498A3 (bg) 1990-07-16
EP0253711B1 (fr) 1990-05-23
BG47038A3 (bg) 1990-04-16
PT85235A (fr) 1987-08-01
US4783472A (en) 1988-11-08
IE871767L (en) 1988-01-04
DD263772A5 (de) 1989-01-11
HU198727B (en) 1989-11-28
PL149434B1 (en) 1990-02-28
TNSN87083A1 (fr) 1990-01-01
AU597996B2 (en) 1990-06-14
MX173398B (es) 1994-02-28
NO170419C (no) 1992-10-14
NZ220929A (en) 1989-09-27
FI872931A7 (fi) 1988-01-05
MX7191A (es) 1993-10-01
GR3000502T3 (en) 1991-07-31
AU7504787A (en) 1988-01-07
DK340087D0 (da) 1987-07-02
JPS6322589A (ja) 1988-01-30
HUT44791A (en) 1988-04-28
DK340087A (da) 1988-01-05
KR880001681A (ko) 1988-04-26
FR2601015A1 (fr) 1988-01-08
CS262692B2 (en) 1989-03-14
NO872779L (no) 1988-01-05
FI84727B (fi) 1991-09-30
EP0253711A1 (fr) 1988-01-20

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