PL1720882T3 - Pochodne pirazolopirymidyny jako inhibitory kinazy zależnej od cyklin - Google Patents

Pochodne pirazolopirymidyny jako inhibitory kinazy zależnej od cyklin

Info

Publication number
PL1720882T3
PL1720882T3 PL05722809T PL05722809T PL1720882T3 PL 1720882 T3 PL1720882 T3 PL 1720882T3 PL 05722809 T PL05722809 T PL 05722809T PL 05722809 T PL05722809 T PL 05722809T PL 1720882 T3 PL1720882 T3 PL 1720882T3
Authority
PL
Poland
Prior art keywords
pyrazolopyrimidine
derivatives
kinase inhibitors
dependent kinase
cyclin dependent
Prior art date
Application number
PL05722809T
Other languages
English (en)
Inventor
Timothy J Guzi
Kamil Paruch
Michael P Dwyer
Ronald J Doll
Viyyoor Moopil Girijavallabhan
Alan Mallams
Carmen S Alvarez
Kartik M Keertikar
Jocelyn Rivera
Tin-Yau Chan
Vincent Madison
Thierry O Fischmann
Lawrence W Dillard
Vinh D Tran
Zhen Min He
Ray Anthony James
Haengsoon Park
Vidyadhar M Paradkar
Douglas Walsh Hobbs
Original Assignee
Pharmacopeia Llc
Merck Sharp & Dohme
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34860861&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PL1720882(T3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pharmacopeia Llc, Merck Sharp & Dohme filed Critical Pharmacopeia Llc
Publication of PL1720882T3 publication Critical patent/PL1720882T3/pl

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Neurology (AREA)
  • Oncology (AREA)
  • Rheumatology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Communicable Diseases (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Hematology (AREA)
  • Immunology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Virology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
PL05722809T 2004-02-11 2005-02-08 Pochodne pirazolopirymidyny jako inhibitory kinazy zależnej od cyklin PL1720882T3 (pl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US10/776,988 US7119200B2 (en) 2002-09-04 2004-02-11 Pyrazolopyrimidines as cyclin dependent kinase inhibitors
EP05722809A EP1720882B1 (en) 2004-02-11 2005-02-08 Pyrazolopyrimidine-derivatives as cyclin dependent kinase inhibitors
PCT/US2005/003859 WO2005077954A2 (en) 2004-02-11 2005-02-08 Pyrazolopyrimidine-derivatives as cyclin dependent kinase inhibitors

Publications (1)

Publication Number Publication Date
PL1720882T3 true PL1720882T3 (pl) 2011-08-31

Family

ID=34860861

Family Applications (1)

Application Number Title Priority Date Filing Date
PL05722809T PL1720882T3 (pl) 2004-02-11 2005-02-08 Pochodne pirazolopirymidyny jako inhibitory kinazy zależnej od cyklin

Country Status (26)

Country Link
US (2) US7119200B2 (pl)
EP (1) EP1720882B1 (pl)
JP (2) JP4845743B2 (pl)
KR (1) KR101196498B1 (pl)
CN (1) CN1946725B (pl)
AR (1) AR047543A1 (pl)
AT (1) ATE494287T1 (pl)
AU (1) AU2005212409C1 (pl)
BR (1) BRPI0507644B8 (pl)
CA (1) CA2555345C (pl)
CY (1) CY1112400T1 (pl)
DE (1) DE602005025733D1 (pl)
DK (1) DK1720882T3 (pl)
ES (1) ES2359410T3 (pl)
HR (1) HRP20110245T1 (pl)
IL (1) IL177283A (pl)
MY (1) MY149044A (pl)
NO (1) NO337520B1 (pl)
NZ (1) NZ590480A (pl)
PE (1) PE20050774A1 (pl)
PL (1) PL1720882T3 (pl)
RU (1) RU2414472C9 (pl)
SI (1) SI1720882T1 (pl)
TW (1) TWI393566B (pl)
WO (1) WO2005077954A2 (pl)
ZA (1) ZA200606573B (pl)

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* Cited by examiner, † Cited by third party
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