PL2089382T3 - Podstawione związki diazepanowe jako antagoniści receptora oreksyny - Google Patents
Podstawione związki diazepanowe jako antagoniści receptora oreksynyInfo
- Publication number
- PL2089382T3 PL2089382T3 PL07862400T PL07862400T PL2089382T3 PL 2089382 T3 PL2089382 T3 PL 2089382T3 PL 07862400 T PL07862400 T PL 07862400T PL 07862400 T PL07862400 T PL 07862400T PL 2089382 T3 PL2089382 T3 PL 2089382T3
- Authority
- PL
- Poland
- Prior art keywords
- receptor antagonists
- orexin receptor
- diazepan compounds
- substituted diazepan
- substituted
- Prior art date
Links
- 229940123730 Orexin receptor antagonist Drugs 0.000 title 1
- QPMLSUSACCOBDK-UHFFFAOYSA-N diazepane Chemical class C1CCNNCC1 QPMLSUSACCOBDK-UHFFFAOYSA-N 0.000 title 1
Classifications
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
- A61K31/551—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
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- C07D491/052—Ortho-condensed systems with only one oxygen atom as ring hetero atom in the oxygen-containing ring the oxygen-containing ring being six-membered
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- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
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| US87239306P | 2006-12-01 | 2006-12-01 | |
| US95974207P | 2007-07-16 | 2007-07-16 | |
| EP07862400A EP2089382B1 (en) | 2006-12-01 | 2007-11-30 | Substituted diazepan compounds as orexin receptor antagonists |
| PCT/US2007/024690 WO2008069997A1 (en) | 2006-12-01 | 2007-11-30 | Substituted diazepan compounds as orexin receptor antagonists |
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