PL2181988T3 - Kompozycje farmaceutyczne oparte na Krystalicznej Postaci I 5-azacytydyny - Google Patents

Kompozycje farmaceutyczne oparte na Krystalicznej Postaci I 5-azacytydyny

Info

Publication number
PL2181988T3
PL2181988T3 PL10151392.7T PL10151392T PL2181988T3 PL 2181988 T3 PL2181988 T3 PL 2181988T3 PL 10151392 T PL10151392 T PL 10151392T PL 2181988 T3 PL2181988 T3 PL 2181988T3
Authority
PL
Poland
Prior art keywords
azacytidine
pharmaceutical compositions
crystalline form
compositions based
crystalline
Prior art date
Application number
PL10151392.7T
Other languages
English (en)
Inventor
Dumitru Ionescu
Peter Blumbergs
Lee Alani Selvey
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=32987551&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PL2181988(T3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed filed Critical
Publication of PL2181988T3 publication Critical patent/PL2181988T3/pl

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/02Antineoplastic agents specific for leukemia
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H1/00Processes for the preparation of sugar derivatives
    • C07H1/06Separation; Purification
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/12Triazine radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Engineering & Computer Science (AREA)
  • Molecular Biology (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Hematology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Medicinal Preparation (AREA)
PL10151392.7T 2003-03-17 2004-03-16 Kompozycje farmaceutyczne oparte na Krystalicznej Postaci I 5-azacytydyny PL2181988T3 (pl)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US10/390,530 US6943249B2 (en) 2003-03-17 2003-03-17 Methods for isolating crystalline Form I of 5-azacytidine

Publications (1)

Publication Number Publication Date
PL2181988T3 true PL2181988T3 (pl) 2016-11-30

Family

ID=32987551

Family Applications (2)

Application Number Title Priority Date Filing Date
PL04721078T PL1608634T3 (pl) 2003-03-17 2004-03-16 Sposób wyodrębniania krystalicznej formy i 5-azacytydyny
PL10151392.7T PL2181988T3 (pl) 2003-03-17 2004-03-16 Kompozycje farmaceutyczne oparte na Krystalicznej Postaci I 5-azacytydyny

Family Applications Before (1)

Application Number Title Priority Date Filing Date
PL04721078T PL1608634T3 (pl) 2003-03-17 2004-03-16 Sposób wyodrębniania krystalicznej formy i 5-azacytydyny

Country Status (16)

Country Link
US (5) US6943249B2 (pl)
EP (3) EP1608634B1 (pl)
JP (1) JP4792550B2 (pl)
AU (2) AU2004222274B2 (pl)
BR (1) BRPI0408506A (pl)
CA (1) CA2518973A1 (pl)
CY (2) CY1114213T1 (pl)
DK (2) DK2181988T3 (pl)
EC (1) ECSP056023A (pl)
ES (2) ES2575535T3 (pl)
HU (1) HUE028268T2 (pl)
MX (1) MXPA05009969A (pl)
PL (2) PL1608634T3 (pl)
PT (2) PT1608634E (pl)
SI (2) SI1608634T1 (pl)
WO (1) WO2004082822A2 (pl)

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WO2009042767A1 (en) * 2007-09-26 2009-04-02 Mount Sinai School Of Medicine Azacytidine analogues and uses thereof
EP2211870A1 (en) * 2007-11-01 2010-08-04 Celgene Corporation Cytidine analogs for treatment of myelodysplastic syndromes
PL3692983T3 (pl) * 2008-05-15 2021-12-27 Celgene Corporation Doustne formulacje analogów cytydyny i sposoby ich zastosowania
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JP2014503597A (ja) 2011-01-31 2014-02-13 セルジーン コーポレイション シチジンアナログの医薬組成物及びその使用方法
CN103619864A (zh) * 2011-03-31 2014-03-05 细胞基因国际有限公司 5-氮杂胞苷的合成
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CA2849708A1 (en) 2011-09-23 2013-03-28 Celgene Corporation Romidepsin and 5 - azacitidine for use in treating lymphoma
CA2849903A1 (en) 2011-09-26 2013-04-04 Celgene Corporation Combination therapy for chemoresistant cancers
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WO2013080221A2 (en) * 2011-12-01 2013-06-06 Hetero Research Foundation Process for alvimopan
US9669048B2 (en) * 2012-10-25 2017-06-06 Fresenius Kabi Oncology Limited Stable pharmaceutical composition of 5-aza-2′-deoxycitidine
WO2014076616A2 (en) * 2012-11-19 2014-05-22 Shilpa Medicare Limited Formulations of 5-azacytidine
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WO2014160698A1 (en) 2013-03-26 2014-10-02 Celgene Corporation SOLID FORMS COMPRISING 4-AMINO-I-β-D-RIBOFURANOSYL-1,3,5-TRIAZIN-2(1H)-ONE AND A COFORMER, COMPOSITIONS AND METHODS OF USE THEREOF
CN103450303A (zh) * 2013-09-04 2013-12-18 重庆泰濠制药有限公司 阿扎胞苷晶型a、阿扎胞苷晶型b及其制备方法
AU2015305449B2 (en) 2014-08-22 2021-05-06 Celgene Corporation Methods of treating multiple myeloma with immunomodulatory compounds in combination with antibodies
US20160095925A1 (en) * 2014-10-01 2016-04-07 Cadila Healthcare Limited Stable formulation of azacitidine or salts thereof and their process for preparation
US10695352B2 (en) 2015-10-15 2020-06-30 Celgene Corporation Combination therapy for treating malignancies
KR102699521B1 (ko) 2015-10-15 2024-08-26 르 라보레또레 쎄르비에르 악성 종양의 치료를 위한 조합물 요법
EP3527226A4 (en) * 2016-10-17 2020-06-17 Daiichi Sankyo Company, Limited COMBINATION THERAPY PROCEDURE WITH MDM2 INHIBITOR AND DNA METHYL TRANSFERASE INHIBITOR
CN109988207B (zh) * 2017-12-29 2022-01-04 江苏豪森药业集团有限公司 阿扎胞苷晶型的制备方法
US10632211B2 (en) 2018-06-11 2020-04-28 The Regents Of The University Of California Demethylation to treat eye disease
CN110642901A (zh) * 2019-11-11 2020-01-03 扬子江药业集团有限公司 阿扎胞苷甲醇化物及其制备方法和药物组合物、用途
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Also Published As

Publication number Publication date
WO2004082822A2 (en) 2004-09-30
PL1608634T3 (pl) 2013-10-31
MXPA05009969A (es) 2006-02-17
EP1608634A2 (en) 2005-12-28
DK2181988T3 (en) 2016-06-06
EP2181988A1 (en) 2010-05-05
HUE028268T2 (en) 2016-12-28
US20130274459A1 (en) 2013-10-17
DK1608634T3 (da) 2013-08-12
JP2006523210A (ja) 2006-10-12
US20120245342A1 (en) 2012-09-27
AU2010241198B2 (en) 2012-05-10
SI1608634T1 (sl) 2013-09-30
AU2004222274B2 (en) 2010-11-04
US7700770B2 (en) 2010-04-20
US8975392B2 (en) 2015-03-10
US8211862B2 (en) 2012-07-03
EP2181988B1 (en) 2016-05-11
CY1114213T1 (el) 2016-08-31
CY1117639T1 (el) 2017-04-26
EP1608634B1 (en) 2013-05-22
PT1608634E (pt) 2013-08-27
US20100292180A1 (en) 2010-11-18
US20040186284A1 (en) 2004-09-23
AU2010241198A1 (en) 2010-11-25
US6943249B2 (en) 2005-09-13
BRPI0408506A (pt) 2006-03-14
ECSP056023A (es) 2006-01-27
AU2004222274A1 (en) 2004-09-30
WO2004082822A3 (en) 2005-07-07
EP1608634A4 (en) 2006-03-15
PT2181988E (pt) 2016-06-15
ES2425474T3 (es) 2013-10-15
CA2518973A1 (en) 2004-09-30
EP2266965A1 (en) 2010-12-29
ES2575535T3 (es) 2016-06-29
US8481715B2 (en) 2013-07-09
US20050272675A1 (en) 2005-12-08
SI2181988T1 (sl) 2016-09-30
JP4792550B2 (ja) 2011-10-12

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