PL2523666T3 - Kompozycja farmaceutyczna zawierająca 3-beta-hydroksy-5-alfa-pregnan-20-on o ulepszonych właściwościach przechowywania i rozpuszczalności - Google Patents

Kompozycja farmaceutyczna zawierająca 3-beta-hydroksy-5-alfa-pregnan-20-on o ulepszonych właściwościach przechowywania i rozpuszczalności

Info

Publication number
PL2523666T3
PL2523666T3 PL11733156T PL11733156T PL2523666T3 PL 2523666 T3 PL2523666 T3 PL 2523666T3 PL 11733156 T PL11733156 T PL 11733156T PL 11733156 T PL11733156 T PL 11733156T PL 2523666 T3 PL2523666 T3 PL 2523666T3
Authority
PL
Poland
Prior art keywords
pregnan
beta
alpha
hydroxy
pharmaceutical composition
Prior art date
Application number
PL11733156T
Other languages
English (en)
Inventor
Torbjörn Bäckström
Anders Carlsson
Original Assignee
Asarina Pharma Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Asarina Pharma Ab filed Critical Asarina Pharma Ab
Publication of PL2523666T3 publication Critical patent/PL2523666T3/pl

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/57Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/575Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of three or more carbon atoms, e.g. cholane, cholestane, ergosterol, sitosterol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/14Esters of carboxylic acids, e.g. fatty acid monoglycerides, medium-chain triglycerides, parabens or PEG fatty acid esters
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/28Steroids, e.g. cholesterol, bile acids or glycyrrhetinic acid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/44Oils, fats or waxes according to two or more groups of A61K47/02-A61K47/42; Natural or modified natural oils, fats or waxes, e.g. castor oil, polyethoxylated castor oil, montan wax, lignite, shellac, rosin, beeswax or lanolin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/10Dispersions; Emulsions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/10Dispersions; Emulsions
    • A61K9/107Emulsions ; Emulsion preconcentrates; Micelles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/18Feminine contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/06Antimigraine agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/08Antiepileptics; Anticonvulsants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/30Drugs for disorders of the nervous system for treating abuse or dependence
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/30Drugs for disorders of the nervous system for treating abuse or dependence
    • A61P25/32Alcohol-abuse
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/24Drugs for disorders of the endocrine system of the sex hormones
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0034Urogenital system, e.g. vagina, uterus, cervix, penis, scrotum, urethra, bladder; Personal lubricants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0043Nose

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Dispersion Chemistry (AREA)
  • Psychiatry (AREA)
  • Addiction (AREA)
  • Pain & Pain Management (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Gynecology & Obstetrics (AREA)
  • Diabetes (AREA)
  • Anesthesiology (AREA)
  • Hospice & Palliative Care (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
PL11733156T 2010-01-14 2011-01-14 Kompozycja farmaceutyczna zawierająca 3-beta-hydroksy-5-alfa-pregnan-20-on o ulepszonych właściwościach przechowywania i rozpuszczalności PL2523666T3 (pl)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US29502710P 2010-01-14 2010-01-14
SE1050029 2010-01-14
EP11733156.1A EP2523666B8 (en) 2010-01-14 2011-01-14 A pharmaceutical composition comprising 3-beta-hydroxy-5-alpha-pregnan-20-one with improved storage and solubility properties
PCT/SE2011/050036 WO2011087441A1 (en) 2010-01-14 2011-01-14 A pharmaceutical composition comprising 3-beta-hydroxy-5-alpha-pregnan-20-one with improved storage and solubility properties

Publications (1)

Publication Number Publication Date
PL2523666T3 true PL2523666T3 (pl) 2016-06-30

Family

ID=44304503

Family Applications (1)

Application Number Title Priority Date Filing Date
PL11733156T PL2523666T3 (pl) 2010-01-14 2011-01-14 Kompozycja farmaceutyczna zawierająca 3-beta-hydroksy-5-alfa-pregnan-20-on o ulepszonych właściwościach przechowywania i rozpuszczalności

Country Status (15)

Country Link
US (4) US20120322781A1 (pl)
EP (1) EP2523666B8 (pl)
JP (1) JP5687287B2 (pl)
CN (1) CN102753181B (pl)
AU (1) AU2011205821B2 (pl)
BR (1) BR112012017136B1 (pl)
CA (1) CA2786330C (pl)
DK (1) DK2523666T3 (pl)
ES (1) ES2566765T3 (pl)
HU (1) HUE027298T2 (pl)
MX (1) MX2012008257A (pl)
PL (1) PL2523666T3 (pl)
RU (1) RU2012133627A (pl)
WO (1) WO2011087441A1 (pl)
ZA (1) ZA201204574B (pl)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2013043985A1 (en) * 2011-09-23 2013-03-28 The Regents Of The University Of California Edible oils to enhance delivery of orally administered steroids
CN106146597A (zh) * 2016-07-05 2016-11-23 浙江海洋大学 一种马尾藻甾醇化合物及其提取方法、应用
CN106146596A (zh) * 2016-07-05 2016-11-23 浙江海洋大学 一种铜藻β‑谷甾醇化合物及其提取方法、应用
KR102185474B1 (ko) * 2016-09-27 2020-12-03 광시 지우푸 바이오테크놀로지 컴퍼니 리미티드 마약중독 치료효과가 있는 추출물 및 그 제조방법
MX393759B (es) 2017-01-09 2025-03-24 Asarina Pharma Ab Suspensiones inyectables
WO2018147792A1 (en) 2017-02-10 2018-08-16 Asarina Pharma Ab 3-beta-hydroxy-5-alpha-pregnan-20-one for use in medical treatment
CN111432805B (zh) 2017-11-27 2023-02-17 梅克里内科尼蒂翁公司 3α-乙炔基-3β-羟基雄甾烷-17-酮肟的药物制剂
WO2020011789A1 (en) 2018-07-09 2020-01-16 Asarina Pharma Ab Injectable suspensions
EP3593789A1 (fr) * 2018-07-11 2020-01-15 Beta Innov Composition contenant un dérivé de 7beta-hydroxycholestérol et un véhicule lipidique, et son utilisation dans le traitement de pathologies néoplasiques
US20220202832A1 (en) * 2019-04-05 2022-06-30 The Regents Of The University Of California Allopregnanolone compositions and uses thereof
CN112341511A (zh) * 2019-08-09 2021-02-09 南京诺瑞特医药科技有限公司 3-羟基-5-孕烷-20-酮衍生物及其用途
CN114907436A (zh) * 2021-02-08 2022-08-16 南京诺瑞特医药科技有限公司 3-羟基-5-孕烷-20-酮衍生物的晶型及其制备方法和用途
US20240180865A1 (en) * 2021-04-08 2024-06-06 Tionlab Therapeutics Sustained-release lipid pre-concentrate

Family Cites Families (29)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS54122719A (en) * 1978-03-16 1979-09-22 Sankyo Co Ltd Carcinostatic agent for oral administration
US5232917A (en) 1987-08-25 1993-08-03 University Of Southern California Methods, compositions, and compounds for allosteric modulation of the GABA receptor by members of the androstane and pregnane series
US5120723A (en) 1987-08-25 1992-06-09 University Of Southern California Method, compositions, and compounds for modulating brain excitability
US5364632A (en) * 1989-04-05 1994-11-15 Yissum Research Development Company Of The Hebrew University Of Jerusalem Medicinal emulsions
JPH02286625A (ja) * 1989-04-27 1990-11-26 Dainippon Pharmaceut Co Ltd 注射用持続性製剤
FR2663224B1 (fr) * 1990-06-14 1995-01-20 Applicationes Farmaceuticas Sa Forme galenique parenterale.
US5449474A (en) 1992-02-21 1995-09-12 Inland Technology, Inc. Low toxicity solvent composition
SE9302295D0 (sv) 1993-07-02 1993-07-02 Kabi Pharmacia Ab New pharmaceutical composition
AU7569194A (en) 1993-08-20 1995-03-21 Meyer B. Jackson Method for regulating neuropeptide hormone secretion
US5763431A (en) 1993-08-20 1998-06-09 Jackson; Meyer B. Method for regulating neuropeptide hormone secretion
GB9405304D0 (en) * 1994-03-16 1994-04-27 Scherer Ltd R P Delivery systems for hydrophobic drugs
CN1171114A (zh) 1994-11-23 1998-01-21 科斯赛斯公司 用于γ-氨基丁酸受体的变构调节的雄甾烷和孕甾烷组系
FR2734418A1 (fr) * 1995-05-16 1996-11-22 Amp France Connecteur, notamment du type jack modulaire
CA2289006A1 (en) * 1997-05-02 1998-11-12 American Home Products Corporation Pregnan-3-ol-20-ones
CN1270718C (zh) * 1998-03-11 2006-08-23 托布乔恩·贝克斯托罗姆 表别孕烷醇酮在制备治疗甾族化合物诱导的疾病的药物中的应用
US6075058A (en) 1998-12-12 2000-06-13 Tufts University Compositions for increased bioavailability of carotenoids
WO2000059945A1 (en) 1999-04-06 2000-10-12 The Horticulture And Food Research Institute Of New Zealand Limited Improvements in or relating to immunoassays for anaesthetics
US20030236236A1 (en) * 1999-06-30 2003-12-25 Feng-Jing Chen Pharmaceutical compositions and dosage forms for administration of hydrophobic drugs
AU6381000A (en) 1999-07-29 2001-02-19 Interneuron Pharmaceuticals, Inc. Methods and compositions for alleviating stuttering
US20040204490A1 (en) 1999-08-31 2004-10-14 Farb David H. Effect of steroids on NMDA receptors depends on subunit composition
DE60041773D1 (de) 1999-08-31 2009-04-23 Univ Boston Der effekt von steroiden auf ndma-rezeptoren beruht auf der zusammensetzung der untereinheiten
US6855721B1 (en) * 2000-07-28 2005-02-15 Indevus Pharmaceuticals, Inc. Methods and compositions for alleviating stuttering
SE0104423D0 (sv) 2001-12-27 2001-12-27 Umecrine Ab Pregnane steroids and their use in the treatment of CNS disorders
US6888721B1 (en) 2002-10-18 2005-05-03 Atec Corporation Electrohydrodynamic (EHD) thin film evaporator with splayed electrodes
US20050096365A1 (en) 2003-11-03 2005-05-05 David Fikstad Pharmaceutical compositions with synchronized solubilizer release
US20060003002A1 (en) 2003-11-03 2006-01-05 Lipocine, Inc. Pharmaceutical compositions with synchronized solubilizer release
WO2006037016A2 (en) * 2004-09-27 2006-04-06 The Regents Of The University Of California Novel therapy for treatment of chronic degenerative brain diseases and nervous system injury
ES2423493T3 (es) 2004-11-18 2013-09-20 Umecrine Ab Antagonistas de los GABA-esteroides y su uso para el tratamiento de trastornos del SNC
IN2014DN02014A (pl) 2006-11-21 2015-07-10 Umecrine Ab

Also Published As

Publication number Publication date
BR112012017136A2 (pt) 2018-06-12
CN102753181B (zh) 2014-09-17
US20120322781A1 (en) 2012-12-20
US20230117905A1 (en) 2023-04-20
JP5687287B2 (ja) 2015-03-18
BR112012017136B1 (pt) 2021-05-25
CA2786330A1 (en) 2011-07-21
AU2011205821A1 (en) 2012-07-12
HUE027298T2 (en) 2016-10-28
US9687496B2 (en) 2017-06-27
ZA201204574B (en) 2013-08-28
RU2012133627A (ru) 2014-04-20
CN102753181A (zh) 2012-10-24
JP2013517269A (ja) 2013-05-16
US20170258809A1 (en) 2017-09-14
ES2566765T3 (es) 2016-04-15
EP2523666B1 (en) 2016-01-13
US11534446B2 (en) 2022-12-27
EP2523666A4 (en) 2013-07-03
DK2523666T3 (en) 2016-04-04
AU2011205821B2 (en) 2013-07-25
WO2011087441A1 (en) 2011-07-21
EP2523666A1 (en) 2012-11-21
MX2012008257A (es) 2012-11-21
EP2523666B8 (en) 2016-04-06
CA2786330C (en) 2013-11-19
US20150164914A1 (en) 2015-06-18

Similar Documents

Publication Publication Date Title
PL2523666T3 (pl) Kompozycja farmaceutyczna zawierająca 3-beta-hydroksy-5-alfa-pregnan-20-on o ulepszonych właściwościach przechowywania i rozpuszczalności
IL257517B (en) Integrin agonist compounds and medicinal compositions thereof
IL253870B (en) Certain amino-pyrimidines and pharmaceutical preparations containing them
EP2570361A4 (en) ARTICLE STORAGE BOX
IL247079A0 (en) A rapidly dissolving pharmaceutical compound
IL215825A0 (en) Selable storage container
EP2642983A4 (en) DEVICE INGREABLE WITH PHARMACEUTICAL PRODUCT
PL2411025T3 (pl) Stabilna w wysokiej temperaturze kompozycja farmaceutyczna zawierająca nośnik tlenu
TWM388065U (en) Rotary and telescopic storage device
ZA201302120B (en) Biodegradable drug delivery composition
IL222086A (en) A pharmaceutical composition that melts quickly
EP2636666A4 (en) TRANS-2 DECENTRIC ACID DERIVATIVES AND MEDICAMENTS CONTAINING THEREOF
IL239297A0 (en) Tablets with improved reception and good storage stability
IL206739A0 (en) Injectable pharmaceutical composition
GB201019296D0 (en) Storing and retrieving garments
IL223707A0 (en) N-hydroxyformamide derivative and medicament containing same
ZA201208210B (en) A combination composition comprising ibuprofen and paracetamal
IL221501A (en) Medicinal product containing miramistine
ZA201205684B (en) Ester compound and use thereof
AP2788A (en) Simalikalactone E and use thereof as a medicament
SI2415681T1 (sl) Skladiščna in transportna priprava
ZA201300098B (en) Pharmaceutical composition with enhanced solubility characteristics
PL2857014T3 (pl) Kompozycja farmaceutyczna zawierająca aspirynę i bisoprolol
GB201001026D0 (en) Article for storage and play
TWM401636U (en) Display box with storage and display effects