PL2709988T3 - Proces przygotowania kwasu [4,6-bis-dimetyloamino-2-[4-(4- trifluorometylbenzoyl-amino)benzylo]pyrimidin-5-ylo] octowego - Google Patents

Proces przygotowania kwasu [4,6-bis-dimetyloamino-2-[4-(4- trifluorometylbenzoyl-amino)benzylo]pyrimidin-5-ylo] octowego

Info

Publication number
PL2709988T3
PL2709988T3 PL12718262T PL12718262T PL2709988T3 PL 2709988 T3 PL2709988 T3 PL 2709988T3 PL 12718262 T PL12718262 T PL 12718262T PL 12718262 T PL12718262 T PL 12718262T PL 2709988 T3 PL2709988 T3 PL 2709988T3
Authority
PL
Poland
Prior art keywords
trifluoromethylbenzoyl
pyrimidin
dimethylamino
benzyl
bis
Prior art date
Application number
PL12718262T
Other languages
English (en)
Inventor
Juan M. Rodriguez Dehli
Robert Hagenkoetter
Michael Schul
Christian Stange
Xiao-Jun Wang
Li Zhang
Oriol MASSOT
Original Assignee
Actimis Pharmaceuticals, Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Actimis Pharmaceuticals, Inc. filed Critical Actimis Pharmaceuticals, Inc.
Publication of PL2709988T3 publication Critical patent/PL2709988T3/pl

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48Two nitrogen atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
PL12718262T 2011-05-16 2012-05-07 Proces przygotowania kwasu [4,6-bis-dimetyloamino-2-[4-(4- trifluorometylbenzoyl-amino)benzylo]pyrimidin-5-ylo] octowego PL2709988T3 (pl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201161486363P 2011-05-16 2011-05-16
EP12718262.4A EP2709988B1 (en) 2011-05-16 2012-05-07 Process for preparing [4,6-bis-dimethylamino-2-[4-(4-trifluoromethylbenzoyl-amino)benzyl]pyrimidin-5-yl]acetic acid
PCT/EP2012/058338 WO2012156221A1 (en) 2011-05-16 2012-05-07 Process for preparing [4,6-bis-dimethylamino-2-[4-(4-trifluoromethylbenzoyl-amino)benzyl]pyrimidin-5-yl]acetic acid

Publications (1)

Publication Number Publication Date
PL2709988T3 true PL2709988T3 (pl) 2018-04-30

Family

ID=46025756

Family Applications (1)

Application Number Title Priority Date Filing Date
PL12718262T PL2709988T3 (pl) 2011-05-16 2012-05-07 Proces przygotowania kwasu [4,6-bis-dimetyloamino-2-[4-(4- trifluorometylbenzoyl-amino)benzylo]pyrimidin-5-ylo] octowego

Country Status (16)

Country Link
US (1) US8859770B2 (pl)
EP (2) EP3293180A1 (pl)
JP (1) JP5988253B2 (pl)
CY (1) CY1119348T1 (pl)
DK (1) DK2709988T3 (pl)
ES (1) ES2639045T3 (pl)
HK (1) HK1252529A1 (pl)
HR (1) HRP20171287T1 (pl)
HU (1) HUE034889T2 (pl)
LT (1) LT2709988T (pl)
PL (1) PL2709988T3 (pl)
PT (1) PT2709988T (pl)
RS (1) RS56326B1 (pl)
SI (1) SI2709988T1 (pl)
SM (1) SMT201700432T1 (pl)
WO (1) WO2012156221A1 (pl)

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE316077T1 (de) * 2003-04-25 2006-02-15 Actimis Pharmaceuticals Inc Pyrimidin-essigsäure derivate geeignet zur behandlung von crth2-bedingten krankheiten
US8541419B2 (en) * 2008-09-02 2013-09-24 Actimis Pharmaceuticals, Inc. Isotopically enriched pyrimidin-5-yl acetic acid derivatives as CRTH2 antagonists

Also Published As

Publication number Publication date
US8859770B2 (en) 2014-10-14
EP2709988A1 (en) 2014-03-26
RS56326B1 (sr) 2017-12-29
HK1252529A1 (en) 2019-05-31
US20140187779A1 (en) 2014-07-03
HRP20171287T1 (hr) 2017-11-17
SI2709988T1 (sl) 2017-11-30
CY1119348T1 (el) 2018-03-07
WO2012156221A1 (en) 2012-11-22
EP2709988B1 (en) 2017-07-05
SMT201700432T1 (it) 2017-11-15
EP3293180A1 (en) 2018-03-14
PT2709988T (pt) 2017-09-08
LT2709988T (lt) 2017-10-10
DK2709988T3 (en) 2017-09-18
ES2639045T3 (es) 2017-10-25
JP2014515033A (ja) 2014-06-26
HUE034889T2 (hu) 2018-03-28
JP5988253B2 (ja) 2016-09-07

Similar Documents

Publication Publication Date Title
HUE057571T2 (hu) Eljárás [(5-(3-klór-fenil)-3-hidroxi-piridin-2-karbonil)-amino]-ecetsav elõállítására 5-((3-klór-fenil)-3-klór-piridin-2-il)-nitrilbõl kiindulva, és eljárás 5-(halogén-fenil)-3-halogén-piridin-2-il)-nitril-származékok elõállítására
IL244812B (en) Process for preparing 23(s)-methyl-12α,7α,3α-trihydroxy-6α-ethyl-5β-cholan-24-butyric acid
IL230477A0 (en) Process for preparing 2,2-difluoroethanol
SG11201503291RA (en) Process for producing acetic acid
IL232139A0 (en) A process for the preparation of quinoline hist
IL207526A0 (en) Process for preparing 2-amino-5-cyanobenzoic acid derivatives
EP2667714A1 (en) Process for the preparation of 4-amino-5-fluoro-3-halo-6-(substituted)picolinates
EP2797866A4 (en) PROCESS FOR THE PREPARATION OF 1,6-HEXANEDIOL
EP2562152A4 (en) PROCESS FOR PREPARING 2,5-DIMETHYLPHENYL-ACETIC ACID
IL233282A0 (en) Manufacturing process for pyrimidine history
IL222290A0 (en) Process for preparing aminobenzofuran derivatives
IL222191A0 (en) Process for preparing sulfonamido-benzofuran derivatives
IL201670A0 (en) Process for preparing 2-amino-5-cyanobenzoic acid derivatives
ZA201308894B (en) Process for preparing methacrylic acid
IL227872A0 (en) A process for the preparation of n-converted phenylhydroxylamines
IL227220A (en) A process for preparing a history of 3-alkylsulfinylbenzoyl
TWI562986B (en) Process for preparing 4-amino-5-biphenyl-4-yl-2-hydroxymethyl-2-methyl-pentanoic acid compounds
EP2663546A1 (fr) Procede de production de composes nitrile-acide gras
EP2619174A4 (en) PROCESS FOR THE PREPARATION OF L-PHENYL-3-DIMETHYLAMINOPROPANE DERIVATIVES
ZA201405237B (en) Process for preparing formic acid
PL2771328T3 (pl) Sposób otrzymywania 1,2-benzizotiazolin-3-onu
IL232630A0 (en) A method for the preparation of 6,2-difluoroacetophenones
SMT201700432T1 (it) Procedimento per la preparazione di acido [4,6-bis-dimetilammino-2-[4-(4-trifluorometilbenzoil-ammino)benzil)pirimidin-5-il]acetico
PL2791201T3 (pl) Sposób wytwarzania określonych funkcjonalnych oligomerów kwasu mlekowego
IL218764A0 (en) Crystalline levofolinic acid and process for its preparation