PL353588A1 - Pochodne arylometylo-karbonyloamino-tiazolu i ichPochodne arylometylo-karbonyloamino-tiazolu i ichzastosowanie jako środków przeciwnowotworowychzastosowanie jako środków przeciwnowotworowych - Google Patents

Pochodne arylometylo-karbonyloamino-tiazolu i ichPochodne arylometylo-karbonyloamino-tiazolu i ichzastosowanie jako środków przeciwnowotworowychzastosowanie jako środków przeciwnowotworowych

Info

Publication number
PL353588A1
PL353588A1 PL00353588A PL35358800A PL353588A1 PL 353588 A1 PL353588 A1 PL 353588A1 PL 00353588 A PL00353588 A PL 00353588A PL 35358800 A PL35358800 A PL 35358800A PL 353588 A1 PL353588 A1 PL 353588A1
Authority
PL
Poland
Prior art keywords
arylmethyl
carbonylamino
antitumor agents
thiazole derivatives
thiazole
Prior art date
Application number
PL00353588A
Other languages
English (en)
Other versions
PL203424B1 (pl
Inventor
PaoloPevarello Paolo Pevarello
RaffaellaAmici Raffaella Amici
ManuelaVilla Manuela Villa
BarbaraSalom Barbara Salom
AnnaVulpetti Anna Vulpetti
MarioVarasi Mario Varasi
Original Assignee
Pharmacia Italia S.P.A.Pharmacia Italia S.P.A.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pharmacia Italia S.P.A.Pharmacia Italia S.P.A. filed Critical Pharmacia Italia S.P.A.Pharmacia Italia S.P.A.
Publication of PL353588A1 publication Critical patent/PL353588A1/pl
Publication of PL203424B1 publication Critical patent/PL203424B1/pl

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • A61K31/4261,3-Thiazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/12Drugs for disorders of the urinary system of the kidneys
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/06Antipsoriatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/08Antiseborrheics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/02Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D277/00Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/38Nitrogen atoms
    • C07D277/44Acylated amino or imino radicals
    • C07D277/46Acylated amino or imino radicals by carboxylic acids, or sulfur or nitrogen analogues thereof

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Epidemiology (AREA)
  • Immunology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Urology & Nephrology (AREA)
  • Dermatology (AREA)
  • Neurosurgery (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pulmonology (AREA)
  • Hospice & Palliative Care (AREA)
  • Virology (AREA)
  • Cardiology (AREA)
  • Psychiatry (AREA)
  • Vascular Medicine (AREA)
  • Communicable Diseases (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Rheumatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
PL353588A 1999-08-12 2000-08-11 Pochodne 2-amino-1,3-tiazolu, sposoby ich wytwarzania, ich zastosowanie oraz ich kompozycje farmaceutyczne PL203424B1 (pl)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US09/372,832 US6114365A (en) 1999-08-12 1999-08-12 Arylmethyl-carbonylamino-thiazole derivatives, process for their preparation, and their use as antitumor agents
US09/372,832 1999-08-12

Publications (2)

Publication Number Publication Date
PL353588A1 true PL353588A1 (pl) 2003-12-01
PL203424B1 PL203424B1 (pl) 2009-10-30

Family

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Also Published As

Publication number Publication date
SK1802002A3 (en) 2003-05-02
CN100410245C (zh) 2008-08-13
BG65484B1 (bg) 2008-09-30
US6114365A (en) 2000-09-05
MA25433A1 (fr) 2002-04-01
AP2002002441A0 (en) 2002-03-31
AP1853A (en) 2008-05-29
HRP20020127A2 (en) 2003-04-30
IS6264A (is) 2002-02-11
CZ303138B6 (cs) 2012-04-25
US6784198B1 (en) 2004-08-31
EP1204649A1 (en) 2002-05-15
UA72538C2 (en) 2005-03-15
HUP0202492A3 (en) 2004-12-28
HRP20020127B1 (en) 2010-08-31
CN1425009A (zh) 2003-06-18
IL147924A (en) 2008-03-20
YU9702A (sh) 2004-11-25
AU782882B2 (en) 2005-09-08
ZA200201117B (en) 2003-04-30
ATE375987T1 (de) 2007-11-15
EP1204649B1 (en) 2007-10-17
HK1054233B (zh) 2009-05-29
BR0013281A (pt) 2002-06-18
GEP20053475B (en) 2005-03-25
EE200200064A (et) 2003-04-15
HK1054233A1 (zh) 2003-11-21
NO20020683D0 (no) 2002-02-11
KR20020060159A (ko) 2002-07-16
KR100773709B1 (ko) 2007-11-09
IL147924A0 (en) 2002-08-14
MXPA02001508A (es) 2003-07-21
AU7440000A (en) 2001-03-19
NO323576B1 (no) 2007-06-11
SK287373B6 (sk) 2010-08-09
WO2001014353A1 (en) 2001-03-01
BG106481A (en) 2002-09-30
OA12047A (en) 2006-05-02
JP2003507461A (ja) 2003-02-25
HUP0202492A2 (hu) 2002-11-28
CY1107108T1 (el) 2012-10-24
ES2295056T3 (es) 2008-04-16
DE60036803D1 (de) 2007-11-29
DE60036803T2 (de) 2008-07-24
EA200200247A1 (ru) 2002-08-29
NZ517236A (en) 2004-11-26
RS50300B (sr) 2009-09-08
SI1204649T1 (sl) 2008-02-29
PT1204649E (pt) 2008-01-10
EA005375B1 (ru) 2005-02-24
NO20020683L (no) 2002-04-10
CZ2002486A3 (cs) 2002-11-13
DK1204649T3 (da) 2007-12-03
KR20070074003A (ko) 2007-07-10
EE04939B1 (et) 2007-12-17
IS2594B (is) 2010-03-15
JP4864260B2 (ja) 2012-02-01
KR100827563B1 (ko) 2008-05-07
CA2381097C (en) 2009-06-16
US20050004120A1 (en) 2005-01-06
CA2381097A1 (en) 2001-03-01

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