PL354481A1 - Tienoizoksazolo-fenoksy-niepodstawione etylo-i propylopochodne użyteczne jako antagoniści D 4 - Google Patents
Tienoizoksazolo-fenoksy-niepodstawione etylo-i propylopochodne użyteczne jako antagoniści D 4Info
- Publication number
- PL354481A1 PL354481A1 PL00354481A PL35448100A PL354481A1 PL 354481 A1 PL354481 A1 PL 354481A1 PL 00354481 A PL00354481 A PL 00354481A PL 35448100 A PL35448100 A PL 35448100A PL 354481 A1 PL354481 A1 PL 354481A1
- Authority
- PL
- Poland
- Prior art keywords
- thienoisoxazole
- derivatives useful
- unsubstituted ethyl
- propyl derivatives
- phenoxy unsubstituted
- Prior art date
Links
- 125000001495 ethyl group Chemical group [H]C([H])([H])C([H])([H])* 0.000 title 1
- 125000001436 propyl group Chemical group [H]C([*])([H])C([H])([H])C([H])([H])[H] 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Psychology (AREA)
- Psychiatry (AREA)
- Addiction (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US39615699A | 1999-09-14 | 1999-09-14 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| PL354481A1 true PL354481A1 (pl) | 2004-01-26 |
Family
ID=23566087
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PL00354481A PL354481A1 (pl) | 1999-09-14 | 2000-09-13 | Tienoizoksazolo-fenoksy-niepodstawione etylo-i propylopochodne użyteczne jako antagoniści D 4 |
Country Status (23)
| Country | Link |
|---|---|
| EP (1) | EP1216249B1 (pl) |
| JP (1) | JP4717306B2 (pl) |
| KR (1) | KR20020027644A (pl) |
| AR (1) | AR032135A1 (pl) |
| AT (1) | ATE254620T1 (pl) |
| AU (1) | AU7577200A (pl) |
| BR (1) | BR0014513A (pl) |
| CA (1) | CA2383327C (pl) |
| CZ (1) | CZ2002896A3 (pl) |
| DE (1) | DE60006698T2 (pl) |
| DK (1) | DK1216249T3 (pl) |
| EA (1) | EA004177B1 (pl) |
| EE (1) | EE200200133A (pl) |
| ES (1) | ES2206305T3 (pl) |
| HU (1) | HUP0202712A3 (pl) |
| IL (1) | IL148522A0 (pl) |
| MX (1) | MXPA02002690A (pl) |
| NO (1) | NO20021249L (pl) |
| PL (1) | PL354481A1 (pl) |
| PT (1) | PT1216249E (pl) |
| SK (1) | SK3502002A3 (pl) |
| WO (1) | WO2001019832A2 (pl) |
| ZA (1) | ZA200201760B (pl) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB0207449D0 (en) * | 2002-03-28 | 2002-05-08 | Glaxo Group Ltd | Novel compounds |
| WO2018166855A1 (en) | 2017-03-16 | 2018-09-20 | Basf Se | Heterobicyclic substituted dihydroisoxazoles |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4728651A (en) * | 1985-10-24 | 1988-03-01 | Hoechst-Roussel Pharmaceuticals Inc. | Antihypertensive thieno-isoxazoles and -pyrazoles |
| US6187774B1 (en) * | 1996-03-04 | 2001-02-13 | Yoshitomi Pharmaceutical Industries, Ltd. | Fused heterocyclic compounds and pharmaceutical applications thereof |
| HUP9603001A3 (en) * | 1996-10-30 | 1999-07-28 | Richter Gedeon Vegyeszet | Heterocycle compounds comprising nitrogen, process for producing them and pharmaceutical compositions containing the same |
| JP4627882B2 (ja) * | 1998-02-09 | 2011-02-09 | デユフアー・インターナシヨナル・リサーチ・ベー・ブイ | D4−アンタゴニスト活性を有するベンズイソキサゾール誘導体 |
-
2000
- 2000-09-13 HU HU0202712A patent/HUP0202712A3/hu unknown
- 2000-09-13 MX MXPA02002690A patent/MXPA02002690A/es active IP Right Grant
- 2000-09-13 JP JP2001523409A patent/JP4717306B2/ja not_active Expired - Fee Related
- 2000-09-13 SK SK350-2002A patent/SK3502002A3/sk unknown
- 2000-09-13 AR ARP000104794A patent/AR032135A1/es not_active Application Discontinuation
- 2000-09-13 IL IL14852200A patent/IL148522A0/xx unknown
- 2000-09-13 EA EA200200357A patent/EA004177B1/ru not_active IP Right Cessation
- 2000-09-13 ES ES00964967T patent/ES2206305T3/es not_active Expired - Lifetime
- 2000-09-13 PT PT00964967T patent/PT1216249E/pt unknown
- 2000-09-13 KR KR1020027003354A patent/KR20020027644A/ko not_active Withdrawn
- 2000-09-13 CZ CZ2002896A patent/CZ2002896A3/cs unknown
- 2000-09-13 EE EEP200200133A patent/EE200200133A/xx unknown
- 2000-09-13 AU AU75772/00A patent/AU7577200A/en not_active Abandoned
- 2000-09-13 CA CA002383327A patent/CA2383327C/en not_active Expired - Fee Related
- 2000-09-13 PL PL00354481A patent/PL354481A1/pl unknown
- 2000-09-13 AT AT00964967T patent/ATE254620T1/de not_active IP Right Cessation
- 2000-09-13 DK DK00964967T patent/DK1216249T3/da active
- 2000-09-13 WO PCT/US2000/024949 patent/WO2001019832A2/en not_active Ceased
- 2000-09-13 BR BR0014513-0A patent/BR0014513A/pt not_active IP Right Cessation
- 2000-09-13 EP EP00964967A patent/EP1216249B1/en not_active Expired - Lifetime
- 2000-09-13 DE DE60006698T patent/DE60006698T2/de not_active Expired - Lifetime
-
2002
- 2002-03-01 ZA ZA200201760A patent/ZA200201760B/en unknown
- 2002-03-13 NO NO20021249A patent/NO20021249L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| IL148522A0 (en) | 2002-09-12 |
| CA2383327A1 (en) | 2001-03-22 |
| CZ2002896A3 (cs) | 2002-08-14 |
| AU7577200A (en) | 2001-04-17 |
| JP2003509431A (ja) | 2003-03-11 |
| EA200200357A1 (ru) | 2002-10-31 |
| EP1216249A2 (en) | 2002-06-26 |
| HUP0202712A3 (en) | 2004-12-28 |
| EE200200133A (et) | 2003-04-15 |
| SK3502002A3 (en) | 2002-09-10 |
| EA004177B1 (ru) | 2004-02-26 |
| DE60006698T2 (de) | 2004-09-23 |
| NO20021249D0 (no) | 2002-03-13 |
| MXPA02002690A (es) | 2004-09-10 |
| ZA200201760B (en) | 2003-08-27 |
| JP4717306B2 (ja) | 2011-07-06 |
| DE60006698D1 (de) | 2003-12-24 |
| AR032135A1 (es) | 2003-10-29 |
| ATE254620T1 (de) | 2003-12-15 |
| WO2001019832A3 (en) | 2001-10-04 |
| CA2383327C (en) | 2009-11-03 |
| BR0014513A (pt) | 2002-07-02 |
| NO20021249L (no) | 2002-05-10 |
| ES2206305T3 (es) | 2004-05-16 |
| EP1216249B1 (en) | 2003-11-19 |
| PT1216249E (pt) | 2004-04-30 |
| KR20020027644A (ko) | 2002-04-13 |
| DK1216249T3 (da) | 2004-03-15 |
| HUP0202712A2 (hu) | 2002-12-28 |
| WO2001019832A2 (en) | 2001-03-22 |
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