PL354809A1 - Pochodne chinolilopropylopiperydyny, sposób ich wytwarzania i zawierające je kompozycje - Google Patents

Pochodne chinolilopropylopiperydyny, sposób ich wytwarzania i zawierające je kompozycje

Info

Publication number: PL354809A1
Authority: PL; Poland
Prior art keywords: piperidine; preparation; compositions containing; containing same; propyl derivatives
Prior art date: 1999-09-17

Application number

PL00354809A

Other languages

English (en)

Inventor

Jean-Luc Malleron

Michel Tabart

Jean-Chistophe Carry

Michel Evers

Ahmad Youssef El

Serge Mignani

Fabrice Viviani

Michel Cheve

Original Assignee

Aventis Pharma S.A.

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1999-09-17

Filing date

2000-09-14

Publication date

2004-02-23

2000-09-14 Application filed by Aventis Pharma S.A. filed Critical Aventis Pharma S.A.

2004-02-23 Publication of PL354809A1 publication Critical patent/PL354809A1/pl

Links

239000000203 mixture Substances 0.000 title 1
238000002360 preparation method Methods 0.000 title 1
NQRYJNQNLNOLGT-UHFFFAOYSA-N tetrahydropyridine hydrochloride Natural products C1CCNCC1 NQRYJNQNLNOLGT-UHFFFAOYSA-N 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Life Sciences & Earth Sciences (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Communicable Diseases (AREA)
Pharmacology & Pharmacy (AREA)
Oncology (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Hydrogenated Pyridines (AREA)

PL00354809A 1999-09-17 2000-09-14 Pochodne chinolilopropylopiperydyny, sposób ich wytwarzania i zawierające je kompozycje PL354809A1 (pl)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
FR9911679A FR2798656B1 (fr)	1999-09-17	1999-09-17	Derives de la quinolyl propyl piperidine, leur preparation et les compositions qui les contiennent
PCT/FR2000/002541 WO2001025227A2 (fr)	1999-09-17	2000-09-14	Derives de la quinolyl propyl piperidine et leur utilisation en tant que antibacteriens

Publications (1)

Publication Number	Publication Date
PL354809A1 true PL354809A1 (pl)	2004-02-23

Family

ID=9549990

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
PL00354809A PL354809A1 (pl)	1999-09-17	2000-09-14	Pochodne chinolilopropylopiperydyny, sposób ich wytwarzania i zawierające je kompozycje

Country Status (30)

Country	Link
EP (2)	EP1218370B1 (pl)
JP (1)	JP2004527448A (pl)
KR (1)	KR20020038757A (pl)
CN (1)	CN1374959A (pl)
AP (1)	AP2002002459A0 (pl)
AT (1)	ATE284399T1 (pl)
AU (1)	AU7429500A (pl)
BG (1)	BG106524A (pl)
BR (1)	BR0014060A (pl)
CA (1)	CA2383836A1 (pl)
CZ (1)	CZ2002940A3 (pl)
DE (2)	DE60034713T2 (pl)
DZ (1)	DZ3195A1 (pl)
EA (1)	EA005183B1 (pl)
EE (1)	EE200200138A (pl)
FR (1)	FR2798656B1 (pl)
GE (1)	GEP20043223B (pl)
HR (1)	HRP20020214A2 (pl)
HU (1)	HUP0204283A3 (pl)
IL (1)	IL148720A0 (pl)
MA (1)	MA26820A1 (pl)
MX (1)	MXPA02001979A (pl)
NO (1)	NO20021253L (pl)
OA (1)	OA12022A (pl)
PL (1)	PL354809A1 (pl)
SK (1)	SK3632002A3 (pl)
TN (1)	TNSN00184A1 (pl)
WO (1)	WO2001025227A2 (pl)
YU (1)	YU19002A (pl)
ZA (1)	ZA200202073B (pl)

Families Citing this family (38)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB9822440D0 (en)	1998-10-14	1998-12-09	Smithkline Beecham Plc	Medicaments
GB9917406D0 (en)	1999-07-23	1999-09-22	Smithkline Beecham Plc	Compounds
GB9917408D0 (en)	1999-07-23	1999-09-22	Smithkline Beecham Plc	Compounds
ES2278778T3 (es)	2000-07-26	2007-08-16	Smithkline Beecham Plc	Aminopiperidin quinolinas y sus analogos azaisostericos con actividad antibacteriana.
GB0031086D0 (en) *	2000-12-20	2001-01-31	Smithkline Beecham Plc	Medicaments
GB0101577D0 (en)	2001-01-22	2001-03-07	Smithkline Beecham Plc	Compounds
GB0112834D0 (en)	2001-05-25	2001-07-18	Smithkline Beecham Plc	Medicaments
GB0112836D0 (en)	2001-05-25	2001-07-18	Smithkline Beecham Plc	Medicaments
TW200406410A (en)	2002-01-29	2004-05-01	Glaxo Group Ltd	Compounds
JP4508650B2 (ja)	2002-01-29	2010-07-21	グラクソグループリミテッド	アミノピペリジン化合物、当該化合物の製法および当該化合物を含有する医薬組成物
AR040336A1 (es)	2002-06-26	2005-03-30	Glaxo Group Ltd	Compuesto de piperidina, uso del mismo para la fabricacion de un medicamento, composicion farmaceutica que lo comprende y procedimiento para preparar dicho compuesto
TW200406413A (en)	2002-06-26	2004-05-01	Glaxo Group Ltd	Compounds
FR2842807A1 (fr) *	2002-07-23	2004-01-30	Aventis Pharma Sa	Derives de la quinolyl propyl piperidine, procede et intermediaires de preparation et compositions les renfermant
FR2844270B1 (fr)	2002-09-11	2006-05-19	Aventis Pharma Sa	Derives de la quinolyl propyl piperidine, leur procede et intermediaires de preparation et les compositions qui les contiennent
FR2844268B1 (fr) *	2002-09-11	2004-10-22	Aventis Pharma Sa	Derives de la quinolyl propyl piperidine, leurs procedes et intermediaires de preparation et les compositions qui les contiennent
KR20050072432A (ko) *	2002-10-10	2005-07-11	모르포켐 악티엥게셀샤프트 퓌르 콤비나토리셰 케미	항균 활성을 갖는 신규한 화합물
ES2340484T3 (es)	2002-11-05	2010-06-04	Glaxo Group Limited	Agentes antibacterianos.
JP4654035B2 (ja)	2002-11-05	2011-03-16	グラクソスミスクライン・リミテッド・ライアビリティ・カンパニー	抗菌剤
US7491714B2 (en)	2002-12-04	2009-02-17	Glaxo Group Limited	Quinolines and nitrogenated derivatives thereof and their use as antibacterial agents
EP1799674B1 (en) *	2004-10-05	2010-05-05	Actelion Pharmaceuticals Ltd.	New piperidine antibiotics
ATE466857T1 (de) *	2004-10-05	2010-05-15	Actelion Pharmaceuticals Ltd	Neue piperidin-antibiotika
WO2006081178A2 (en)	2005-01-25	2006-08-03	Glaxo Group Limited	Antibacterial agents
US7605169B2 (en)	2005-01-25	2009-10-20	Glaxo Group Limited	Antibacterial agents
WO2006081182A2 (en)	2005-01-25	2006-08-03	Glaxo Group Limited	Antibacterial agents
JP2008528587A (ja)	2005-01-25	2008-07-31	グラクソグループリミテッド	抗菌剤
WO2007086016A1 (en)	2006-01-26	2007-08-02	Actelion Pharmaceuticals Ltd	Tetrahydropyrane antibiotics
US7709483B2 (en)	2006-04-06	2010-05-04	Glaxo Group Limited	Pyrrolo-quinoxalinone derivatives as antibacterials
GB0613208D0 (en)	2006-07-03	2006-08-09	Glaxo Group Ltd	Compounds
EP1992628A1 (en)	2007-05-18	2008-11-19	Glaxo Group Limited	Derivatives and analogs of N-ethylquinolones and N-ethylazaquinolones
EP2481735A1 (en) *	2007-05-09	2012-08-01	Pfizer Inc.	Substituted heterocyclic derivatives and compositions and their pharmaceutical use as antibacterials
EP2080761A1 (en)	2008-01-18	2009-07-22	Glaxo Group Limited	Compounds
EP2352734A1 (en)	2008-10-17	2011-08-10	Glaxo Group Limited	Tricyclic nitrogen compounds used as antibacterials
EP2379554B1 (en)	2009-01-15	2015-11-11	Glaxo Group Limited	Naphthyridin-2(1h)-one compounds useful as antibacterials
CN105636945B (zh) *	2013-10-14	2017-11-17	卫材R&D管理有限公司	选择性取代的喹啉化合物
AU2015304847B2 (en)	2014-08-22	2018-10-25	Glaxosmithkline Intellectual Property Development Limited	Tricyclic nitrogen containing compounds for treating Neisseria gonorrhoea infection
TW201722965A (zh)	2015-08-16	2017-07-01	葛蘭素史密斯克藍智慧財產發展有限公司	用於抗菌應用之化合物
PL3889145T3 (pl)	2015-12-17	2024-07-01	Merck Patent Gmbh	8-cyjano-5-piperydyno-chinoliny jako antagoniści TLR7/8 oraz ich zastosowanie w leczeniu zaburzeń immunologicznych
DK3497094T3 (da)	2016-08-08	2023-05-15	Merck Patent Gmbh	Tlr7/8-antagonister og anvendelser deraf

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
AU2717899A (en) *	1998-01-26	1999-08-09	Smithkline Beecham Plc	Quinoline derivatives as antibacterials
EP1144404A1 (en) *	1999-01-20	2001-10-17	Smithkline Beecham Plc	Piperidinylquinolines as protein tyrosine kinase inhibitors

1999
- 1999-09-17 FR FR9911679A patent/FR2798656B1/fr not_active Expired - Fee Related
2000
- 2000-09-14 YU YU19002A patent/YU19002A/sh unknown
- 2000-09-14 AP APAP/P/2002/002459A patent/AP2002002459A0/en unknown
- 2000-09-14 DE DE60034713T patent/DE60034713T2/de not_active Expired - Fee Related
- 2000-09-14 JP JP2001528171A patent/JP2004527448A/ja active Pending
- 2000-09-14 EE EEP200200138A patent/EE200200138A/xx unknown
- 2000-09-14 OA OA1200200074A patent/OA12022A/fr unknown
- 2000-09-14 HU HU0204283A patent/HUP0204283A3/hu unknown
- 2000-09-14 DE DE60016611T patent/DE60016611T2/de not_active Expired - Fee Related
- 2000-09-14 CN CN00813020A patent/CN1374959A/zh active Pending
- 2000-09-14 KR KR1020027003547A patent/KR20020038757A/ko not_active Ceased
- 2000-09-14 EP EP00962637A patent/EP1218370B1/fr not_active Expired - Lifetime
- 2000-09-14 CZ CZ2002940A patent/CZ2002940A3/cs unknown
- 2000-09-14 GE GEAP20006413A patent/GEP20043223B/en unknown
- 2000-09-14 SK SK363-2002A patent/SK3632002A3/sk unknown
- 2000-09-14 MX MXPA02001979A patent/MXPA02001979A/es unknown
- 2000-09-14 AT AT00962637T patent/ATE284399T1/de not_active IP Right Cessation
- 2000-09-14 EA EA200200374A patent/EA005183B1/ru not_active IP Right Cessation
- 2000-09-14 CA CA002383836A patent/CA2383836A1/fr not_active Abandoned
- 2000-09-14 DZ DZ003195A patent/DZ3195A1/xx active
- 2000-09-14 HR HR20020214A patent/HRP20020214A2/hr not_active Application Discontinuation
- 2000-09-14 IL IL14872000A patent/IL148720A0/xx unknown
- 2000-09-14 BR BR0014060-0A patent/BR0014060A/pt not_active IP Right Cessation
- 2000-09-14 EP EP04019136A patent/EP1484328B1/fr not_active Expired - Lifetime
- 2000-09-14 PL PL00354809A patent/PL354809A1/pl not_active Application Discontinuation
- 2000-09-14 AU AU74295/00A patent/AU7429500A/en not_active Abandoned
- 2000-09-14 WO PCT/FR2000/002541 patent/WO2001025227A2/fr not_active Ceased
- 2000-09-15 TN TNTNSN00184A patent/TNSN00184A1/fr unknown
2002
- 2002-03-13 NO NO20021253A patent/NO20021253L/no not_active Application Discontinuation
- 2002-03-13 ZA ZA200202073A patent/ZA200202073B/en unknown
- 2002-03-14 MA MA26554A patent/MA26820A1/fr unknown
- 2002-03-15 BG BG106524A patent/BG106524A/xx unknown

Also Published As

Publication number	Publication date
BG106524A (en)	2003-01-31
MXPA02001979A (es)	2002-08-20
ZA200202073B (en)	2003-08-27
DE60034713T2 (de)	2008-01-17
EP1484328B1 (fr)	2007-05-02
HUP0204283A2 (hu)	2003-04-28
DE60016611D1 (de)	2005-01-13
OA12022A (fr)	2006-04-19
HUP0204283A3 (en)	2004-07-28
FR2798656A1 (fr)	2001-03-23
GEP20043223B (en)	2004-04-26
WO2001025227A2 (fr)	2001-04-12
IL148720A0 (en)	2002-09-12
CN1374959A (zh)	2002-10-16
HRP20020214A2 (en)	2005-04-30
NO20021253D0 (no)	2002-03-13
KR20020038757A (ko)	2002-05-23
DE60016611T2 (de)	2005-12-22
ATE284399T1 (de)	2004-12-15
CA2383836A1 (fr)	2001-04-12
JP2004527448A (ja)	2004-09-09
EP1218370A2 (fr)	2002-07-03
WO2001025227A3 (fr)	2001-11-22
AU7429500A (en)	2001-05-10
YU19002A (sh)	2005-06-10
EE200200138A (et)	2003-06-16
DE60034713D1 (de)	2007-06-14
SK3632002A3 (en)	2003-04-01
TNSN00184A1 (fr)	2005-11-10
EA005183B1 (ru)	2004-12-30
FR2798656B1 (fr)	2004-12-17
EP1484328A1 (fr)	2004-12-08
NO20021253L (no)	2002-04-24
MA26820A1 (fr)	2004-12-20
EP1218370B1 (fr)	2004-12-08
EA200200374A1 (ru)	2002-10-31
CZ2002940A3 (cs)	2002-07-17
DZ3195A1 (fr)	2001-04-12
BR0014060A (pt)	2002-05-21
AP2002002459A0 (en)	2002-06-30

Legal Events

Date	Code	Title	Description
2007-11-30	REFS	Decisions on refusal to grant patents (taken after the publication of the particulars of the applications)

Publication	Publication Date	Title
PL354809A1 (pl)	2004-02-23	Pochodne chinolilopropylopiperydyny, sposób ich wytwarzania i zawierające je kompozycje
AU1836502A (en)	2002-05-27	Heterocyclylalkyl piperidine derivatives, their preparation and compositions containing same
IL150539A0 (en)	2003-02-12	Novel 1,3-dihydro-2h-indol-2-one derivatives, preparation method and pharmaceutical compositions containing them
HUP0204515A3 (en)	2005-04-28	4-aminopiperidine derivatives, process for their preparation, pharmaceutical compositions containing them and their use
HUP0201953A3 (en)	2006-03-28	Benzene derivatives, preparation method and pharmaceutical compositions containing same
IL157850A0 (en)	2004-03-28	Quinolyl propyl piperidine derivatives, the preparation thereof and compositions containing same
AU2002253219A1 (en)	2003-03-20	Quinolyl propyl piperidine derivatives, the preparation thereof and compositions containing same
HUP0203821A3 (en)	2003-10-28	Novel oligosaccharides, preparation method and pharmaceutical compositions containing same
HUP0303118A3 (en)	2007-08-28	Novel 1,3-dihydro-2h-indol-one derivatives, method for preparing same and pharmaceutical compositions containing them
IL153632A0 (en)	2003-07-06	Aminoalkylbenzoyl-benzofuran or benzothiophene derivatives, method for preparing same and compositions containing same
IL146441A0 (en)	2002-07-25	Purine derivatives, preparation method and pharmaceutical compositions containing same
PL356911A1 (pl)	2004-07-12	Skondensowane związki azolowe i ich stosowanie jako środki hipoglikemiczne
IL146185A0 (en)	2002-07-25	Streptogramin derivatives, preparation and compositions containing them
HUP0204154A3 (en)	2006-01-30	Novel benzothiadiazine derivatives, preparation method and pharmaceutical compositions containing same
IL180579A0 (en)	2007-06-03	Piperidine derivatives, process for obtaining them and pharmaceutical compositions containing them
PL352432A1 (en)	2003-08-25	Neurothrophic pyrolydines and piperidines, their affinite composition and methods of using them
HUP0203839A3 (en)	2004-07-28	4-phenyl-1-piperazinyl, -piperidinyl and -tetrahydropyridyl derivatives, pharmaceutical compositions containing them and their use
AU3560601A (en)	2001-08-07	Novel isoquinoline derivatives, preparation method and pharmaceutical compositions containing them
HUP0204572A3 (en)	2004-07-28	Substituierte bisindolylmaleinimide derivatives, process for their preparation and use and pharmaceutcial compositions containing them
IL154986A0 (en)	2003-10-31	Triazolo-epothilone derivatives, pharmaceutical compositions containing the same and methods for the preparation thereof
AU2003267528A8 (en)	2004-02-16	Quinolyl propyl piperidine derivatives, preparation method and intermediates and compositions containing same
HUP0302892A3 (en)	2005-02-28	Aminoalkenylbenzoyl-benzofuran or benzothiophene derivatives, method for preparing same and compositions containing same
SI1370550T1 (sl)	2007-10-31	Derivati kinolil propil piperidina, njihova priprava in sestavki, ki jih vsebujejo
IL147540A0 (en)	2002-08-14	OXATHIEPINO [6,5-b] DIHYDROPYRIDINES, AND RELATED COMPOSITIONS AND METHODS
SI1252150T1 (en)	2003-10-31	Heterocyclic derivatives, preparation method and pharmaceutical compositions containing same