PL361993A1 - Sposób syntezy peptydu zawierajacego resztę Trp - Google Patents

Sposób syntezy peptydu zawierajacego resztę Trp

Info

Publication number: PL361993A1
Authority: PL; Poland
Prior art keywords: peptide; synthesis; tryptophan residue; residue; protecting group
Prior art date: 2000-12-22

Application number

PL01361993A

Other languages

English (en)

Other versions

PL205949B1 (pl

Inventor

Steven Allen Jackson

Original Assignee

Ipsen Manufacturing Ireland Limited

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-12-22

Filing date

2001-12-19

Publication date

2004-10-18

2001-12-19 Application filed by Ipsen Manufacturing Ireland Limited filed Critical Ipsen Manufacturing Ireland Limited

2004-10-18 Publication of PL361993A1 publication Critical patent/PL361993A1/pl

2010-06-30 Publication of PL205949B1 publication Critical patent/PL205949B1/pl

Links

238000000034 method Methods 0.000 title abstract 3
108090000765 processed proteins & peptides Proteins 0.000 title abstract 3
125000000430 tryptophan group Chemical group [H]N([H])C(C(=O)O*)C([H])([H])C1=C([H])N([H])C2=C([H])C([H])=C([H])C([H])=C12 0.000 title abstract 2
230000015572 biosynthetic process Effects 0.000 title 1
238000003786 synthesis reaction Methods 0.000 title 1
125000006239 protecting group Chemical group 0.000 abstract 2
238000003776 cleavage reaction Methods 0.000 abstract 1
125000001041 indolyl group Chemical group 0.000 abstract 1
230000007017 scission Effects 0.000 abstract 1
239000007787 solid Substances 0.000 abstract 1
238000010532 solid phase synthesis reaction Methods 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
- C07K1/04—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length on carriers
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
- C07K1/06—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents
- C07K1/061—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents using protecting groups
- C07K1/068—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents using protecting groups for heterocyclic side chains
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
- C07K7/04—Linear peptides containing only normal peptide links
- C07K7/23—Luteinising hormone-releasing hormone [LHRH]; Related peptides
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
Proteomics, Peptides & Aminoacids (AREA)
Biophysics (AREA)
General Health & Medical Sciences (AREA)
Genetics & Genomics (AREA)
Life Sciences & Earth Sciences (AREA)
Molecular Biology (AREA)
Biochemistry (AREA)
Analytical Chemistry (AREA)
Endocrinology (AREA)
Peptides Or Proteins (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Preparation Of Compounds By Using Micro-Organisms (AREA)
Indole Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

PL361993A 2000-12-22 2001-12-19 Sposób wytwarzania peptydu PL205949B1 (pl)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
IE20001079		2000-12-22
PCT/IE2001/000159 WO2002051861A2 (en)	2000-12-22	2001-12-19	Process for the synthesis of a peptide having a tryptophan residue

Publications (2)

Publication Number	Publication Date
PL361993A1 true PL361993A1 (pl)	2004-10-18
PL205949B1 PL205949B1 (pl)	2010-06-30

Family

ID=11042704

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
PL361993A PL205949B1 (pl)	2000-12-22	2001-12-19	Sposób wytwarzania peptydu

Country Status (24)

Country	Link
US (1)	US7122628B2 (pl)
EP (1)	EP1343808B1 (pl)
JP (1)	JP4064817B2 (pl)
KR (1)	KR100591832B1 (pl)
CN (2)	CN101003563A (pl)
AT (1)	ATE339442T1 (pl)
AU (1)	AU2002222439C1 (pl)
BR (1)	BR0116447B1 (pl)
CA (1)	CA2432708C (pl)
CZ (1)	CZ299141B6 (pl)
DE (1)	DE60123115T2 (pl)
DK (1)	DK1343808T3 (pl)
ES (1)	ES2266104T3 (pl)
HU (2)	HU229701B1 (pl)
IE (1)	IES20011090A2 (pl)
IL (2)	IL156258A0 (pl)
MX (1)	MXPA03005678A (pl)
NO (1)	NO325038B1 (pl)
NZ (1)	NZ526990A (pl)
PL (1)	PL205949B1 (pl)
PT (1)	PT1343808E (pl)
RU (1)	RU2276156C2 (pl)
WO (1)	WO2002051861A2 (pl)
ZA (1)	ZA200304809B (pl)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US7091311B2 (en)	1996-06-07	2006-08-15	Smithkline Beecham Corporation	Peptides and compounds that bind to a receptor
CA2499625A1 (en)	2002-09-18	2004-04-01	Ortho-Mcneil Pharmaceutical, Inc.	Methods of increasing platelet and hematopoietic stem cell production
UA82710C2 (uk) *	2003-08-28	2008-05-12	Орто-Макнейл Фармацевтикал, Инк.	Пептид, що зв'язується з тромбопоетиновим рецептором (варіанти), та спосіб лікування тромбоциторенії (варіанти)
WO2007077112A1 (en) *	2005-12-30	2007-07-12	F. Hoffmann-La Roche Ag	Methods for the synthesis of arginine-containing peptides
WO2014047822A1 (zh) *	2012-09-27	2014-04-03	深圳翰宇药业股份有限公司	一种制备布舍瑞林的方法
US10308677B2 (en)	2014-12-19	2019-06-04	Cem Corporation	Coupling method for peptide synthesis at elevated temperatures
US9969769B2 (en)	2014-12-19	2018-05-15	Cem Corporation	Coupling method for peptide synthesis at elevated temperatures

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4211693A (en) *	1977-09-20	1980-07-08	The Salk Institute For Biological Studies	Peptides with para-substituted phenylalanine
US4569927A (en) *	1984-02-23	1986-02-11	The Salk Institute For Biological Studies	GnRH Antagonists IV
IL74827A (en)	1984-05-21	1989-06-30	Salk Inst For Biological Studi	Peptides active as gnrh antagonists and pharmaceutical compositions containing them
IT1203600B (it)	1985-12-06	1989-02-15	Phidea Srl	Metodo per preparare il (d-trp6)-lhrh
GB8822502D0 (en)	1988-09-24	1988-10-26	Expansia Sa	New peptide synthesis method
US5175254A (en) *	1988-09-24	1992-12-29	Societe D'expansion Scientifque Expansia	Solid phase peptide synthesis using a polyacrylic support in aqueous solution
RU2043362C1 (ru) *	1991-08-12	1995-09-10	Синтекс (Ю-Эс-Эй) Инк.	Способ твердофазного синтеза пептидов
JPH05331188A (ja)	1992-05-28	1993-12-14	Nippon Chemiphar Co Ltd	トリペプチド、その製造方法及びエンドセリン拮抗剤
RU2086561C1 (ru) *	1995-09-25	1997-08-10	Тихонов Александр Васильевич	Способ получения нонапептидэтиламида

2001
- 2001-12-19 AT AT01272223T patent/ATE339442T1/de active
- 2001-12-19 PT PT01272223T patent/PT1343808E/pt unknown
- 2001-12-19 EP EP01272223A patent/EP1343808B1/en not_active Expired - Lifetime
- 2001-12-19 HU HU0302633A patent/HU229701B1/hu unknown
- 2001-12-19 JP JP2002552954A patent/JP4064817B2/ja not_active Expired - Lifetime
- 2001-12-19 CN CNA2007100047879A patent/CN101003563A/zh active Pending
- 2001-12-19 DK DK01272223T patent/DK1343808T3/da active
- 2001-12-19 US US10/451,486 patent/US7122628B2/en not_active Expired - Lifetime
- 2001-12-19 CN CNA018210384A patent/CN1481389A/zh active Pending
- 2001-12-19 NZ NZ526990A patent/NZ526990A/xx not_active IP Right Cessation
- 2001-12-19 ES ES01272223T patent/ES2266104T3/es not_active Expired - Lifetime
- 2001-12-19 AU AU2002222439A patent/AU2002222439C1/en not_active Expired
- 2001-12-19 KR KR1020037008232A patent/KR100591832B1/ko not_active Expired - Lifetime
- 2001-12-19 DE DE60123115T patent/DE60123115T2/de not_active Expired - Lifetime
- 2001-12-19 CZ CZ20031634A patent/CZ299141B6/cs not_active IP Right Cessation
- 2001-12-19 RU RU2003122779/04A patent/RU2276156C2/ru not_active IP Right Cessation
- 2001-12-19 IL IL15625801A patent/IL156258A0/xx active IP Right Grant
- 2001-12-19 BR BRPI0116447-3B1A patent/BR0116447B1/pt active IP Right Grant
- 2001-12-19 CA CA2432708A patent/CA2432708C/en not_active Expired - Lifetime
- 2001-12-19 WO PCT/IE2001/000159 patent/WO2002051861A2/en not_active Ceased
- 2001-12-19 PL PL361993A patent/PL205949B1/pl unknown
- 2001-12-19 HU HUP1400157A patent/HU230601B1/hu unknown
- 2001-12-19 MX MXPA03005678A patent/MXPA03005678A/es active IP Right Grant
- 2001-12-20 IE IE20011090A patent/IES20011090A2/en not_active IP Right Cessation
2003
- 2003-06-02 IL IL156258A patent/IL156258A/en unknown
- 2003-06-20 ZA ZA200304809A patent/ZA200304809B/en unknown
- 2003-06-20 NO NO20032852A patent/NO325038B1/no not_active IP Right Cessation

Also Published As

Publication number	Publication date
NO20032852D0 (no)	2003-06-20
AU2002222439B2 (en)	2005-04-07
WO2002051861A3 (en)	2002-10-10
BR0116447B1 (pt)	2014-04-29
IL156258A (en)	2008-06-05
EP1343808B1 (en)	2006-09-13
ATE339442T1 (de)	2006-10-15
CZ20031634A3 (cs)	2003-09-17
ZA200304809B (en)	2004-04-20
NO325038B1 (no)	2008-01-21
PT1343808E (pt)	2007-01-31
AU2002222439C1 (en)	2005-10-27
DE60123115D1 (de)	2006-10-26
IES20011090A2 (en)	2002-12-30
IL156258A0 (en)	2004-01-04
EP1343808A2 (en)	2003-09-17
CN1481389A (zh)	2004-03-10
NZ526990A (en)	2005-04-29
US20040077827A1 (en)	2004-04-22
MXPA03005678A (es)	2003-10-06
PL205949B1 (pl)	2010-06-30
HU230601B1 (hu)	2017-02-28
RU2276156C2 (ru)	2006-05-10
HU229701B1 (en)	2014-05-28
HUP0302633A2 (hu)	2003-12-29
KR100591832B1 (ko)	2006-06-20
JP4064817B2 (ja)	2008-03-19
DE60123115T2 (de)	2007-03-29
JP2004516330A (ja)	2004-06-03
RU2003122779A (ru)	2005-02-20
WO2002051861A2 (en)	2002-07-04
HUP1400157A2 (en)	2003-12-29
CA2432708C (en)	2011-07-12
HUP0302633A3 (en)	2008-04-28
ES2266104T3 (es)	2007-03-01
HK1055749A1 (en)	2004-01-21
BR0116447A (pt)	2003-10-07
CA2432708A1 (en)	2002-07-04
CZ299141B6 (cs)	2008-04-30
US7122628B2 (en)	2006-10-17
CN101003563A (zh)	2007-07-25
KR20030081355A (ko)	2003-10-17
DK1343808T3 (da)	2006-12-11
NO20032852L (no)	2003-08-22

Legal Events

Date	Code	Title	Description
2011-04-29	RECP	Rectifications of patent specification

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FI19992802L (fi)	2001-06-30	Parannettu menetelmä tärpätin talteenottamiseksi nykyaikaista keittämöistä
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MY149837A (en)	2013-10-31	New process for the synthesis of perindopril and pharmaceutically acceptable salts thereof
TW200420553A (en)	2004-10-16	Process for the synthesis of 3, 3a, 6, 6a-tetrahydro-2H-cyclopentan[b]furan-2-one
MXPA01004626A (es)	2004-09-10	Resolucion enzimatica de moduladores selectivos de receptores de estrogenos.
ECSP992910A (es)	1999-06-11	Procedimiento para alquilar sulfonamidas impedidas estericamente