PT90843A - Processo para a preparacao de derivados do colestadieno e de composicoes farmaceuticas que os contem, dotadas de actividade de inibicao da redutase de hmg-coa - Google Patents

Processo para a preparacao de derivados do colestadieno e de composicoes farmaceuticas que os contem, dotadas de actividade de inibicao da redutase de hmg-coa

Info

Publication number
PT90843A
PT90843A PT90843A PT9084389A PT90843A PT 90843 A PT90843 A PT 90843A PT 90843 A PT90843 A PT 90843A PT 9084389 A PT9084389 A PT 9084389A PT 90843 A PT90843 A PT 90843A
Authority
PT
Portugal
Prior art keywords
colestadiene
gifted
hmg
derivatives
contain
Prior art date
Application number
PT90843A
Other languages
English (en)
Inventor
Ernold Granzer
Wolfgang Hermann Kraiser
Peter Scharein
Original Assignee
Hoechst Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoechst Ag filed Critical Hoechst Ag
Publication of PT90843A publication Critical patent/PT90843A/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/547Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/655Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having oxygen atoms, with or without sulfur, selenium, or tellurium atoms, as the only ring hetero atoms
    • C07F9/65515Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having oxygen atoms, with or without sulfur, selenium, or tellurium atoms, as the only ring hetero atoms the oxygen atom being part of a five-membered ring
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/06Antihyperlipidemics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J17/00Normal steroids containing carbon, hydrogen, halogen or oxygen, having an oxygen-containing hetero ring not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J31/00Normal steroids containing one or more sulfur atoms not belonging to a hetero ring
    • C07J31/006Normal steroids containing one or more sulfur atoms not belonging to a hetero ring not covered by C07J31/003
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J53/00Steroids in which the cyclopenta(a)hydrophenanthrene skeleton has been modified by condensation with a carbocyclic rings or by formation of an additional ring by means of a direct link between two ring carbon atoms, including carboxyclic rings fused to the cyclopenta(a)hydrophenanthrene skeleton are included in this class
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J9/00Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of more than two carbon atoms, e.g. cholane, cholestane, coprostane
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J9/00Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of more than two carbon atoms, e.g. cholane, cholestane, coprostane
    • C07J9/005Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of more than two carbon atoms, e.g. cholane, cholestane, coprostane containing a carboxylic function directly attached or attached by a chain containing only carbon atoms to the cyclopenta[a]hydrophenanthrene skeleton

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Vascular Medicine (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
PT90843A 1988-06-14 1989-06-14 Processo para a preparacao de derivados do colestadieno e de composicoes farmaceuticas que os contem, dotadas de actividade de inibicao da redutase de hmg-coa PT90843A (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE3820177A DE3820177A1 (de) 1988-06-14 1988-06-14 Cholestadienderivate, verfahren zu ihrer herstellung, ihre verwendung als arzneimittel mit hmg-coa-reduktase-hemmender wirkung

Publications (1)

Publication Number Publication Date
PT90843A true PT90843A (pt) 1989-12-29

Family

ID=6356493

Family Applications (1)

Application Number Title Priority Date Filing Date
PT90843A PT90843A (pt) 1988-06-14 1989-06-14 Processo para a preparacao de derivados do colestadieno e de composicoes farmaceuticas que os contem, dotadas de actividade de inibicao da redutase de hmg-coa

Country Status (11)

Country Link
EP (1) EP0346759A3 (pt)
JP (1) JPH0236192A (pt)
KR (1) KR910000786A (pt)
AU (1) AU3629189A (pt)
DE (1) DE3820177A1 (pt)
DK (1) DK288989A (pt)
FI (1) FI892867L (pt)
IL (1) IL90572A0 (pt)
NO (1) NO892441L (pt)
PT (1) PT90843A (pt)
ZA (1) ZA894469B (pt)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR20200066690A (ko) 2017-10-16 2020-06-10 칭화대학교 메발로네이트 경로 억제제 및 이의 약제학적 조성물

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4107188A (en) * 1977-04-22 1978-08-15 Hoffmann-La Roche Inc. Pregnanes

Also Published As

Publication number Publication date
DE3820177A1 (de) 1989-12-21
NO892441L (no) 1989-12-15
EP0346759A3 (de) 1990-01-31
FI892867A7 (fi) 1989-12-15
JPH0236192A (ja) 1990-02-06
AU3629189A (en) 1989-12-21
IL90572A0 (en) 1990-01-18
DK288989D0 (da) 1989-06-13
KR910000786A (ko) 1991-01-30
DK288989A (da) 1989-12-15
ZA894469B (en) 1990-02-28
EP0346759A2 (de) 1989-12-20
FI892867A0 (fi) 1989-06-12
FI892867L (fi) 1989-12-15
NO892441D0 (no) 1989-06-13

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Legal Events

Date Code Title Description
FC3A Refusal

Effective date: 19940906