PT90843A - Processo para a preparacao de derivados do colestadieno e de composicoes farmaceuticas que os contem, dotadas de actividade de inibicao da redutase de hmg-coa - Google Patents
Processo para a preparacao de derivados do colestadieno e de composicoes farmaceuticas que os contem, dotadas de actividade de inibicao da redutase de hmg-coaInfo
- Publication number
- PT90843A PT90843A PT90843A PT9084389A PT90843A PT 90843 A PT90843 A PT 90843A PT 90843 A PT90843 A PT 90843A PT 9084389 A PT9084389 A PT 9084389A PT 90843 A PT90843 A PT 90843A
- Authority
- PT
- Portugal
- Prior art keywords
- colestadiene
- gifted
- hmg
- derivatives
- contain
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/655—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having oxygen atoms, with or without sulfur, selenium, or tellurium atoms, as the only ring hetero atoms
- C07F9/65515—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having oxygen atoms, with or without sulfur, selenium, or tellurium atoms, as the only ring hetero atoms the oxygen atom being part of a five-membered ring
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J17/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, having an oxygen-containing hetero ring not condensed with the cyclopenta(a)hydrophenanthrene skeleton
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J31/00—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring
- C07J31/006—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring not covered by C07J31/003
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J53/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton has been modified by condensation with a carbocyclic rings or by formation of an additional ring by means of a direct link between two ring carbon atoms, including carboxyclic rings fused to the cyclopenta(a)hydrophenanthrene skeleton are included in this class
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J9/00—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of more than two carbon atoms, e.g. cholane, cholestane, coprostane
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J9/00—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of more than two carbon atoms, e.g. cholane, cholestane, coprostane
- C07J9/005—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of more than two carbon atoms, e.g. cholane, cholestane, coprostane containing a carboxylic function directly attached or attached by a chain containing only carbon atoms to the cyclopenta[a]hydrophenanthrene skeleton
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Vascular Medicine (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Urology & Nephrology (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Biochemistry (AREA)
- Molecular Biology (AREA)
- Steroid Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE3820177A DE3820177A1 (de) | 1988-06-14 | 1988-06-14 | Cholestadienderivate, verfahren zu ihrer herstellung, ihre verwendung als arzneimittel mit hmg-coa-reduktase-hemmender wirkung |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| PT90843A true PT90843A (pt) | 1989-12-29 |
Family
ID=6356493
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PT90843A PT90843A (pt) | 1988-06-14 | 1989-06-14 | Processo para a preparacao de derivados do colestadieno e de composicoes farmaceuticas que os contem, dotadas de actividade de inibicao da redutase de hmg-coa |
Country Status (11)
| Country | Link |
|---|---|
| EP (1) | EP0346759A3 (pt) |
| JP (1) | JPH0236192A (pt) |
| KR (1) | KR910000786A (pt) |
| AU (1) | AU3629189A (pt) |
| DE (1) | DE3820177A1 (pt) |
| DK (1) | DK288989A (pt) |
| FI (1) | FI892867L (pt) |
| IL (1) | IL90572A0 (pt) |
| NO (1) | NO892441L (pt) |
| PT (1) | PT90843A (pt) |
| ZA (1) | ZA894469B (pt) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR20200066690A (ko) | 2017-10-16 | 2020-06-10 | 칭화대학교 | 메발로네이트 경로 억제제 및 이의 약제학적 조성물 |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4107188A (en) * | 1977-04-22 | 1978-08-15 | Hoffmann-La Roche Inc. | Pregnanes |
-
1988
- 1988-06-14 DE DE3820177A patent/DE3820177A1/de not_active Withdrawn
-
1989
- 1989-06-08 EP EP89110349A patent/EP0346759A3/de not_active Withdrawn
- 1989-06-12 IL IL90572A patent/IL90572A0/xx unknown
- 1989-06-12 FI FI892867A patent/FI892867L/fi not_active Application Discontinuation
- 1989-06-13 JP JP1148558A patent/JPH0236192A/ja active Pending
- 1989-06-13 KR KR1019890008086A patent/KR910000786A/ko not_active Withdrawn
- 1989-06-13 NO NO89892441A patent/NO892441L/no unknown
- 1989-06-13 DK DK288989A patent/DK288989A/da not_active Application Discontinuation
- 1989-06-13 ZA ZA894469A patent/ZA894469B/xx unknown
- 1989-06-13 AU AU36291/89A patent/AU3629189A/en not_active Abandoned
- 1989-06-14 PT PT90843A patent/PT90843A/pt not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| DE3820177A1 (de) | 1989-12-21 |
| NO892441L (no) | 1989-12-15 |
| EP0346759A3 (de) | 1990-01-31 |
| FI892867A7 (fi) | 1989-12-15 |
| JPH0236192A (ja) | 1990-02-06 |
| AU3629189A (en) | 1989-12-21 |
| IL90572A0 (en) | 1990-01-18 |
| DK288989D0 (da) | 1989-06-13 |
| KR910000786A (ko) | 1991-01-30 |
| DK288989A (da) | 1989-12-15 |
| ZA894469B (en) | 1990-02-28 |
| EP0346759A2 (de) | 1989-12-20 |
| FI892867A0 (fi) | 1989-06-12 |
| FI892867L (fi) | 1989-12-15 |
| NO892441D0 (no) | 1989-06-13 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FC3A | Refusal |
Effective date: 19940906 |