PT91203A - Processo para a preparacao de novos derivados de antibioticos bu-3608 e de composicoes farmaceuticas que os contem - Google Patents

Processo para a preparacao de novos derivados de antibioticos bu-3608 e de composicoes farmaceuticas que os contem

Info

Publication number
PT91203A
PT91203A PT91203A PT9120389A PT91203A PT 91203 A PT91203 A PT 91203A PT 91203 A PT91203 A PT 91203A PT 9120389 A PT9120389 A PT 9120389A PT 91203 A PT91203 A PT 91203A
Authority
PT
Portugal
Prior art keywords
antibiotics
contain
preparation
pharmaceutical compositions
new derivatives
Prior art date
Application number
PT91203A
Other languages
English (en)
Other versions
PT91203B (pt
Inventor
Masataka Konishi
Toshikazu Oki
Masatoshi Kakushima
Maki Nishio
Original Assignee
Bristol Myers Squibb Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol Myers Squibb Co filed Critical Bristol Myers Squibb Co
Publication of PT91203A publication Critical patent/PT91203A/pt
Publication of PT91203B publication Critical patent/PT91203B/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20—Carbocyclic rings
    • C07H15/24—Condensed ring systems having three or more rings
    • C—CHEMISTRY; METALLURGY
    • C12—BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
    • C12P—FERMENTATION OR ENZYME-USING PROCESSES TO SYNTHESISE A DESIRED CHEMICAL COMPOUND OR COMPOSITION OR TO SEPARATE OPTICAL ISOMERS FROM A RACEMIC MIXTURE
    • C12P19/00—Preparation of compounds containing saccharide radicals
    • C12P19/44—Preparation of O-glycosides, e.g. glucosides
    • C12P19/56—Preparation of O-glycosides, e.g. glucosides having an oxygen atom of the saccharide radical directly bound to a condensed ring system having three or more carbocyclic rings, e.g. daunomycin, adriamycin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D309/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20—Carbocyclic rings
    • C07H15/24—Condensed ring systems having three or more rings
    • C07H15/244—Anthraquinone radicals, e.g. sennosides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Zoology (AREA)
  • Wood Science & Technology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Molecular Biology (AREA)
  • General Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Microbiology (AREA)
  • Public Health (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Saccharide Compounds (AREA)
  • Peptides Or Proteins (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Cephalosporin Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Steroid Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
PT91203A 1988-07-19 1989-07-18 Processo para a preparacao de novos derivados de antibioticos bu-3608 e de composicoes farmaceuticas que os contem PT91203B (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US07/221,144 US4960755A (en) 1988-07-19 1988-07-19 BU-3608 derivatives

Publications (2)

Publication Number Publication Date
PT91203A true PT91203A (pt) 1990-02-08
PT91203B PT91203B (pt) 1995-03-01

Family

ID=22826542

Family Applications (1)

Application Number Title Priority Date Filing Date
PT91203A PT91203B (pt) 1988-07-19 1989-07-18 Processo para a preparacao de novos derivados de antibioticos bu-3608 e de composicoes farmaceuticas que os contem

Country Status (23)

Country Link
US (1) US4960755A (pt)
EP (1) EP0351799B1 (pt)
JP (1) JP2772549B2 (pt)
KR (1) KR970003127B1 (pt)
AT (1) ATE100459T1 (pt)
AU (1) AU622197B2 (pt)
CA (1) CA1337907C (pt)
CS (1) CS274700B2 (pt)
DD (2) DD296081A5 (pt)
DE (1) DE68912438T2 (pt)
DK (1) DK170778B1 (pt)
ES (1) ES2048793T3 (pt)
FI (1) FI92206C (pt)
HU (2) HU205131B (pt)
IE (1) IE62586B1 (pt)
IL (1) IL91001A (pt)
MY (1) MY105128A (pt)
NO (1) NO170544C (pt)
NZ (1) NZ229964A (pt)
PT (1) PT91203B (pt)
RU (2) RU2032693C1 (pt)
YU (1) YU138289A (pt)
ZA (1) ZA895455B (pt)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5114857A (en) * 1988-11-10 1992-05-19 Bristol-Myers Company Actinomadura hibisca microorganism useful for preparing serine analogs of BU-3608 antibiotics
US5183808A (en) * 1988-11-10 1993-02-02 Bristol-Myers Squibb Company Method for treating fungal infections with serine analogs of BU-3608 antibiotics
JP2643404B2 (ja) * 1989-01-13 1997-08-20 財団法人微生物化学研究会 新抗生物質n―アセチルベナノマイシンbならびにその製造法
AU634250B2 (en) * 1989-07-10 1993-02-18 Bristol-Myers Squibb Company Antiviral antibiotic bu-3889v
US5098708A (en) * 1990-06-14 1992-03-24 Bristol-Myers Squibb Company Antiviral antibiotic BU-3889V
FI92207C (fi) * 1989-11-14 1994-10-10 Squibb Bristol Myers Co Menetelmä terapeuttisesti käyttökelpoisten pradimisiinijohdannaisten valmistamiseksi
US5227370A (en) * 1989-11-14 1993-07-13 Bristol-Myers Squibb Company Pradimicin derivatives
CA2030166C (en) * 1989-11-22 1997-10-07 Shimpei Aburaki Pradimicin derivatives
US5696096A (en) * 1990-09-28 1997-12-09 Bristol-Myers Squibb Company Pradimicin derivatives
US5843908A (en) * 1990-09-28 1998-12-01 Bristol-Myers Squibb Company Pradimicins l and fl, and derivatives thereof
US5326867A (en) * 1992-07-16 1994-07-05 Bristol-Myers Squibb Company Pradimic acids, amides, and pradimicin derivatives
US5338728A (en) * 1992-08-14 1994-08-16 Bristol-Myers Squibb Pradimicin compounds
RU2220706C2 (ru) * 2001-11-15 2004-01-10 Научный Центр Здоровья детей РАМН Лекарственное противогрибковое средство

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4591637A (en) * 1985-01-17 1986-05-27 Sri International Open chain-morpholino adriamycins
US4870165A (en) * 1987-02-02 1989-09-26 Bristol-Myers Company Antifungal antibiotics
US5055453A (en) * 1987-11-02 1991-10-08 Zaidan Hojin Biseibutsu Kagaku Kenkyu Kai Benanomicins a and antibiotic compositions
JP2512050B2 (ja) * 1987-12-25 1996-07-03 財団法人微生物化学研究会 新規抗かび性抗生物質デキシロシルベナノマイシンbならびにその製造法
US5696096A (en) * 1990-09-28 1997-12-09 Bristol-Myers Squibb Company Pradimicin derivatives

Also Published As

Publication number Publication date
MY105128A (en) 1994-08-30
HU908256D0 (en) 1991-06-28
AU622197B2 (en) 1992-04-02
US4960755A (en) 1990-10-02
NZ229964A (en) 1991-07-26
JPH0273095A (ja) 1990-03-13
HUT51283A (en) 1990-04-28
HU203112B (en) 1991-05-28
NO892939D0 (no) 1989-07-18
ZA895455B (en) 1991-12-24
YU138289A (en) 1991-02-28
DE68912438D1 (de) 1994-03-03
RU2032693C1 (ru) 1995-04-10
DD287509A5 (de) 1991-02-28
HU205131B (en) 1992-03-30
EP0351799B1 (en) 1994-01-19
IE892325L (en) 1990-01-19
ES2048793T3 (es) 1994-04-01
CS274700B2 (en) 1991-09-15
DK170778B1 (da) 1996-01-15
FI893426L (fi) 1990-01-20
DK354689A (da) 1990-01-20
EP0351799A2 (en) 1990-01-24
RU2026302C1 (ru) 1995-01-09
ATE100459T1 (de) 1994-02-15
KR970003127B1 (ko) 1997-03-14
DK354689D0 (da) 1989-07-18
KR900001715A (ko) 1990-02-27
PT91203B (pt) 1995-03-01
NO170544B (no) 1992-07-20
DD296081A5 (de) 1991-11-21
FI893426A0 (fi) 1989-07-14
DE68912438T2 (de) 1994-06-01
FI92206C (fi) 1994-10-10
JP2772549B2 (ja) 1998-07-02
IL91001A0 (en) 1990-02-09
EP0351799A3 (en) 1991-04-24
IE62586B1 (en) 1995-02-08
NO892939L (no) 1990-01-22
IL91001A (en) 1995-06-29
FI92206B (fi) 1994-06-30
CS440889A2 (en) 1990-11-14
NO170544C (no) 1992-10-28
AU3827489A (en) 1990-01-25
CA1337907C (en) 1996-01-09

Similar Documents

Publication Publication Date Title
AU617918B2 (en) 2-aminopyrimidinone derivatives
PT92935A (pt) Processo para a preparacao de um composto de pirazolo-piridina e de composicoes farmaceuticas que o contem
PT96145A (pt) Processo para a preparacao de novos derivados de aminoacidos e de composicoes farmaceuticas que os contem
NO942953L (no) 11-benzaldoksimestradienderivater, fremgangsmåte for deres fremstilling smat legemddel inneholdende slike
FI894477A0 (fi) Menetelmä terapeuttisesti aktiivisten 7-substituoitujen 3,5-dihydroksihept-6-yynihappojen ja niiden johdannaisten valmistamiseksi ja välituotteina käyttökelpoiset yhdisteet
PT89502A (pt) Processo para a preparacao de derivados de 2-(2-hidroxi-3-fenoxi-metilo e de composicoes farmaceuticas que os contem
PT91364A (pt) Processo para a preparacao de derivados de 3-piperazinil-benzazol e de composicoes farmaceuticas que os contem
PT90022A (pt) Processo para a preparacao de derivados cefem e dos intermediarios correspondentes
FI893426A0 (fi) Analogiamenetelmä terapeuttisesti käyttökelpoisten BU-3608-johdannaisten ja niiden suolojen valmistamiseksi
PT96226A (pt) Processo para a preparacao de derivados morfolinilicos de doxorubicina e de composicoes farmaceuticas que os contem
RU94014256A (ru) Производные 4-хинолиндигидропиридина, смесь их изомеров или отдельные изомеры и их соли
ES2045067T3 (es) Procedimiento para preparar nuevos compuestos de tiazol.
DE69330601D1 (de) Serotoninergische ergolin derivate
DK240889D0 (da) S-enantiomere glutaramidderivater og deres anvendelse som laegemidler samt farmaceutiske praeparater indeholdende disse forbindelser
BR9502079A (pt) Composto,formulação farmaceutica e processo para preparar um composto
IL93594A0 (en) Pharmaceutical compositions containing an imidazopyrimidone derivative
AU581856B2 (en) 1-(4'-alkylthiophenyl)-2-amino-1, 3-propanediol N-substituted derivatives
ATE237619T1 (de) Sesquiterpen-derivate mit antiviraler aktivität
BR9302809A (pt) Composto,processo para sua preparacao,processo de purificacao dos compostos,medicmanto,emprego e processo para a preparacao de um agente anti-tumoral
FI893121L (fi) Menetelmä farmakologisesti aktiivisten 6,21-dimetyyli-19-norprogesteronijohdannaisten valmistamiseksi
DE68918298D1 (de) Antibiotikum-Derivat.
NO931112L (no) Krystallinske former av endo-2,3-dihydro n-(8-metyl/hydrogen-8-azabicyklo-(3.2.1)okt-3-yl)-2-okso-1h-benzimidazol-1-karboksamid-hydroklorid-monohydrat
PT91259A (pt) Processo para a preparacao de composicoes microbicidas, contendo derivados de halogeno-vinil-azol
ATE79259T1 (de) Prophylaktische und heilende zusammensetzung enthaltende eine 8-chlorbenzothiazepin-verbindung und dessen verwendung.

Legal Events

Date Code Title Description
FG3A Patent granted, date of granting

Effective date: 19940822