PT94036A - Processo para a preparacao de piridazinaminas anti-rinovirais - Google Patents
Processo para a preparacao de piridazinaminas anti-rinoviraisInfo
- Publication number
- PT94036A PT94036A PT94036A PT9403690A PT94036A PT 94036 A PT94036 A PT 94036A PT 94036 A PT94036 A PT 94036A PT 9403690 A PT9403690 A PT 9403690A PT 94036 A PT94036 A PT 94036A
- Authority
- PT
- Portugal
- Prior art keywords
- 4alkyl
- chem
- compounds
- pyridazinamins
- antirinoviral
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 abstract 3
- 239000008194 pharmaceutical composition Substances 0.000 abstract 2
- 125000004178 (C1-C4) alkyl group Chemical group 0.000 abstract 1
- 239000004480 active ingredient Substances 0.000 abstract 1
- 230000002128 anti-rhinoviral effect Effects 0.000 abstract 1
- 125000004093 cyano group Chemical group *C#N 0.000 abstract 1
- 229910052739 hydrogen Inorganic materials 0.000 abstract 1
- 239000001257 hydrogen Substances 0.000 abstract 1
- 125000004435 hydrogen atom Chemical class [H]* 0.000 abstract 1
- LETVJWLLIMJADE-UHFFFAOYSA-N pyridazin-3-amine Chemical class NC1=CC=CN=N1 LETVJWLLIMJADE-UHFFFAOYSA-N 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Health & Medical Sciences (AREA)
- Oncology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Virology (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Communicable Diseases (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pyridine Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US35175489A | 1989-05-15 | 1989-05-15 | |
| GB898911158A GB8911158D0 (en) | 1989-05-16 | 1989-05-16 | Antiviral pyridazinamines |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| PT94036A true PT94036A (pt) | 1991-01-08 |
| PT94036B PT94036B (pt) | 1996-11-29 |
Family
ID=26295357
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PT94036A PT94036B (pt) | 1989-05-15 | 1990-05-14 | Processo para a preparacao de piridazinaminas anti-rinovirais |
Country Status (13)
| Country | Link |
|---|---|
| EP (1) | EP0398427B1 (pt) |
| JP (1) | JP2851921B2 (pt) |
| KR (1) | KR900018077A (pt) |
| AT (1) | ATE102942T1 (pt) |
| AU (1) | AU617612B2 (pt) |
| CA (1) | CA2016747A1 (pt) |
| DE (1) | DE69007331T2 (pt) |
| DK (1) | DK0398427T3 (pt) |
| ES (1) | ES2053079T3 (pt) |
| IE (1) | IE63538B1 (pt) |
| IL (1) | IL94384A0 (pt) |
| NZ (1) | NZ233526A (pt) |
| PT (1) | PT94036B (pt) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JO1645B1 (en) * | 1989-12-26 | 1991-11-27 | شركة جانسين فارماسوتيكا ان. في | Pyridazine compounds are antibacterial viruses |
| AU717744B2 (en) * | 1996-01-15 | 2000-03-30 | Janssen Pharmaceutica N.V. | Angiogenesis inhibiting pyridazinamines |
| KR100607838B1 (ko) * | 1997-10-27 | 2006-08-04 | 뉴로서치 에이/에스 | 니코틴 작용성 아세틸콜린 수용체상의 콜린 작용성 리간드로서의 호모피페라진 유도체 및 이를 포함하는 약제학적 조성물 |
| AUPR213700A0 (en) | 2000-12-18 | 2001-01-25 | Biota Scientific Management Pty Ltd | Antiviral agents |
| WO2007046867A2 (en) * | 2005-05-19 | 2007-04-26 | Xenon Pharmaceuticals Inc. | Piperidine derivatives and their uses as therapeutic agents |
| CN1887875B (zh) * | 2005-06-30 | 2011-04-06 | 深圳市东阳光实业发展有限公司 | 哒嗪胺衍生物及其用于制备小rna病毒抑制剂的用途 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4089965A (en) * | 1976-03-26 | 1978-05-16 | American Cyanamid Company | Thiazolylphenylguanidines as antirhinovirus agents |
| US4140785A (en) * | 1978-05-08 | 1979-02-20 | E. I. Du Pont De Nemours And Company | N-(benzothienopyrazol)amide antirhinoviral agents |
| US5001125A (en) * | 1984-03-26 | 1991-03-19 | Janssen Pharmaceutica N.V. | Anti-virally active pyridazinamines |
-
1990
- 1990-05-01 NZ NZ233526A patent/NZ233526A/xx unknown
- 1990-05-10 DK DK90201186.5T patent/DK0398427T3/da active
- 1990-05-10 AU AU54942/90A patent/AU617612B2/en not_active Ceased
- 1990-05-10 AT AT90201186T patent/ATE102942T1/de not_active IP Right Cessation
- 1990-05-10 ES ES90201186T patent/ES2053079T3/es not_active Expired - Lifetime
- 1990-05-10 EP EP90201186A patent/EP0398427B1/en not_active Expired - Lifetime
- 1990-05-10 DE DE69007331T patent/DE69007331T2/de not_active Expired - Fee Related
- 1990-05-12 KR KR1019900006778A patent/KR900018077A/ko not_active Ceased
- 1990-05-14 IE IE172990A patent/IE63538B1/en not_active IP Right Cessation
- 1990-05-14 CA CA002016747A patent/CA2016747A1/en not_active Abandoned
- 1990-05-14 IL IL94384A patent/IL94384A0/xx not_active IP Right Cessation
- 1990-05-14 PT PT94036A patent/PT94036B/pt not_active IP Right Cessation
- 1990-05-15 JP JP2125262A patent/JP2851921B2/ja not_active Expired - Lifetime
Also Published As
| Publication number | Publication date |
|---|---|
| AU5494290A (en) | 1990-11-15 |
| DK0398427T3 (da) | 1994-04-05 |
| CA2016747A1 (en) | 1990-11-15 |
| IL94384A0 (en) | 1991-03-10 |
| PT94036B (pt) | 1996-11-29 |
| ES2053079T3 (es) | 1994-07-16 |
| NZ233526A (en) | 1991-09-25 |
| DE69007331D1 (de) | 1994-04-21 |
| JPH0356484A (ja) | 1991-03-12 |
| KR900018077A (ko) | 1990-12-20 |
| IE901729L (en) | 1990-11-15 |
| EP0398427B1 (en) | 1994-03-16 |
| DE69007331T2 (de) | 1994-07-07 |
| EP0398427A1 (en) | 1990-11-22 |
| IE63538B1 (en) | 1995-05-17 |
| ATE102942T1 (de) | 1994-04-15 |
| JP2851921B2 (ja) | 1999-01-27 |
| AU617612B2 (en) | 1991-11-28 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FG3A | Patent granted, date of granting |
Effective date: 19960829 |
|
| MM3A | Annulment or lapse |
Free format text: LAPSE DUE TO NON-PAYMENT OF FEES Effective date: 19990228 |