PT94075A - Processo para a preparacao de derivados de milbemicina - Google Patents
Processo para a preparacao de derivados de milbemicinaInfo
- Publication number
- PT94075A PT94075A PT94075A PT9407590A PT94075A PT 94075 A PT94075 A PT 94075A PT 94075 A PT94075 A PT 94075A PT 9407590 A PT9407590 A PT 9407590A PT 94075 A PT94075 A PT 94075A
- Authority
- PT
- Portugal
- Prior art keywords
- preparation
- milbemycin derivatives
- milbemycin
- derivatives
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
- C07H19/01—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/10—Anthelmintics
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
Landscapes
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Molecular Biology (AREA)
- Genetics & Genomics (AREA)
- Biotechnology (AREA)
- Biochemistry (AREA)
- Environmental Sciences (AREA)
- Wood Science & Technology (AREA)
- Veterinary Medicine (AREA)
- Zoology (AREA)
- Agronomy & Crop Science (AREA)
- Pest Control & Pesticides (AREA)
- Plant Pathology (AREA)
- Dentistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Tropical Medicine & Parasitology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Saccharide Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB898911281A GB8911281D0 (en) | 1989-05-17 | 1989-05-17 | Novel compounds |
| GB898929041A GB8929041D0 (en) | 1989-12-22 | 1989-12-22 | Novel compounds |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| PT94075A true PT94075A (pt) | 1991-02-08 |
| PT94075B PT94075B (pt) | 1997-04-30 |
Family
ID=26295361
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PT94075A PT94075B (pt) | 1989-05-17 | 1990-05-17 | Processo para a preparacao de derivados de milbemicina |
Country Status (7)
| Country | Link |
|---|---|
| US (1) | US5962659A (pt) |
| EP (1) | EP0421568A1 (pt) |
| JP (1) | JP2859372B2 (pt) |
| AU (1) | AU640373B2 (pt) |
| CA (1) | CA2017030A1 (pt) |
| NZ (1) | NZ233680A (pt) |
| PT (1) | PT94075B (pt) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5830875A (en) * | 1989-10-30 | 1998-11-03 | Merck & Co., Inc. | 24-and 25-substituted avermectin and milbemycin derivatives |
| GB9024927D0 (en) * | 1990-11-16 | 1991-01-02 | Beecham Group Plc | Novel treatment |
| GB9024928D0 (en) * | 1990-11-16 | 1991-01-02 | Beecham Group Plc | Novel treatment |
| US5411946A (en) * | 1993-02-24 | 1995-05-02 | Merck & Co., Inc. | Avermectin derivatives |
| US5478951A (en) * | 1994-06-22 | 1995-12-26 | American Cyanamid Company | Method for the purification of 23-E isomers of 23-imino derivatives of LL-F28249 compounds |
| GB9716567D0 (en) * | 1997-08-05 | 1997-10-08 | Pfizer | Process |
| JP4373080B2 (ja) * | 2002-12-24 | 2009-11-25 | 三井化学アグロ株式会社 | ミルベマイシン類の精製法 |
| DE102004053964A1 (de) * | 2004-11-09 | 2006-05-11 | Bayer Healthcare Ag | Mittel gegen Demodikose |
Family Cites Families (23)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4408059A (en) * | 1981-12-04 | 1983-10-04 | University Patents, Inc. | Spiroketals useful as intermediates in the synthesis of milbemycin and avermectin macrolides |
| US4668696A (en) * | 1985-07-29 | 1987-05-26 | Merck & Co., Inc. | Novel averonectin fermentation product of a microorganism with anthelmintic activity |
| GB8606107D0 (en) * | 1986-03-12 | 1986-04-16 | Glaxo Group Ltd | Chemical compounds |
| BR8701119A (pt) * | 1986-03-12 | 1988-01-05 | Glaxo Group Ltd | Processo para a preparacao de compostos,composicao para o controle de pragas e processo para combater pragas na agricultura |
| GB8606123D0 (en) * | 1986-03-12 | 1986-04-16 | Glaxo Group Ltd | Chemical compounds |
| ZA872140B (en) * | 1986-03-25 | 1988-11-30 | Sankyo Co | Microlide compounds,their preparation and their use |
| DE3785936T2 (de) * | 1986-03-25 | 1993-08-26 | Sankyo Co | Makrolid-derivate, ihre herstellung und ihre verwendung. |
| CA1296329C (en) * | 1986-06-06 | 1992-02-25 | Derek R. Sutherland | Macrolide compounds |
| JPH0826026B2 (ja) * | 1986-06-13 | 1996-03-13 | 三共株式会社 | ミルベマイシン類の13−エステル誘導体およびその用途 |
| EP0260537A1 (en) * | 1986-09-12 | 1988-03-23 | American Cyanamid Company | 13-Deoxy-23-oxo(keto) and 23-imino derivatives of 13-deoxy C-076-aglycone compounds |
| ATE109783T1 (de) * | 1986-09-12 | 1994-08-15 | American Cyanamid Co | 23-oxo(keto) und 23-imino-derivate von ll-f28249- verbindungen. |
| US4849446A (en) * | 1986-09-12 | 1989-07-18 | American Cyanamid Company | 23-imino derivatives of 23-keto compounds |
| US4831016A (en) * | 1986-10-31 | 1989-05-16 | Merck & Co., Inc. | Reduced avermectin derivatives |
| JPH0672145B2 (ja) * | 1986-12-11 | 1994-09-14 | 三共株式会社 | ミルベマイシン化合物、その製法及び用途 |
| AR243528A1 (es) * | 1986-12-11 | 1993-08-31 | Sankyo Co | Procedimiento para preparar compuestos de macrolida y un procedimiento para producir con los mismos una composicion parasiticida. |
| GB8721371D0 (en) * | 1987-09-11 | 1987-10-21 | Glaxo Group Ltd | Chemical compounds |
| GB8721377D0 (en) * | 1987-09-11 | 1987-10-21 | Glaxo Group Ltd | Chemical compounds |
| GB8721647D0 (en) * | 1987-09-15 | 1987-10-21 | Pfizer Ltd | Antiparasitic agents |
| JP2752083B2 (ja) * | 1988-03-24 | 1998-05-18 | 三共株式会社 | マクロライド化合物の製造法 |
| GB8809232D0 (en) * | 1988-04-19 | 1988-05-25 | Pfizer Ltd | Antiparasitic agents |
| GB8811037D0 (en) * | 1988-05-10 | 1988-06-15 | Glaxo Group Ltd | Chemical compounds |
| NZ229052A (en) * | 1988-05-10 | 1991-03-26 | American Cyanamid Co | Milbemycin derivatives, use for combating pests |
| GB8811036D0 (en) * | 1988-05-10 | 1988-06-15 | Glaxo Group Ltd | Chemical compounds |
-
1990
- 1990-05-15 NZ NZ233680A patent/NZ233680A/en unknown
- 1990-05-17 JP JP2125638A patent/JP2859372B2/ja not_active Expired - Lifetime
- 1990-05-17 EP EP90305367A patent/EP0421568A1/en not_active Ceased
- 1990-05-17 CA CA002017030A patent/CA2017030A1/en not_active Abandoned
- 1990-05-17 AU AU55140/90A patent/AU640373B2/en not_active Ceased
- 1990-05-17 PT PT94075A patent/PT94075B/pt not_active IP Right Cessation
-
1991
- 1991-11-29 US US07/798,971 patent/US5962659A/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| CA2017030A1 (en) | 1990-11-17 |
| PT94075B (pt) | 1997-04-30 |
| AU5514090A (en) | 1990-11-22 |
| JP2859372B2 (ja) | 1999-02-17 |
| NZ233680A (en) | 1995-02-24 |
| JPH02311480A (ja) | 1990-12-27 |
| US5962659A (en) | 1999-10-05 |
| AU640373B2 (en) | 1993-08-26 |
| EP0421568A1 (en) | 1991-04-10 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PC3A | Transfer or assignment |
Free format text: 970218 PFIZER INC. US |
|
| MM3A | Annulment or lapse |
Free format text: LAPSE DUE TO NON-PAYMENT OF FEES Effective date: 20010731 |