PT97992A - Processo de preparacao de analogos polipeptidicos - Google Patents

Processo de preparacao de analogos polipeptidicos

Info

Publication number
PT97992A
PT97992A PT97992A PT9799291A PT97992A PT 97992 A PT97992 A PT 97992A PT 97992 A PT97992 A PT 97992A PT 9799291 A PT9799291 A PT 9799291A PT 97992 A PT97992 A PT 97992A
Authority
PT
Portugal
Prior art keywords
peptoids
designed
methods
libraries
activity
Prior art date
Application number
PT97992A
Other languages
English (en)
Other versions
PT97992B (pt
Original Assignee
Santi Daniel V
Marlowe Charles K
Paul A Bartlett
Reyna J Simon
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Santi Daniel V, Marlowe Charles K, Paul A Bartlett, Reyna J Simon filed Critical Santi Daniel V
Publication of PT97992A publication Critical patent/PT97992A/pt
Publication of PT97992B publication Critical patent/PT97992B/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/001—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof by chemical synthesis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/50—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
    • A61K47/51—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent
    • A61K47/62—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being a protein, peptide or polyamino acid
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
    • C07K1/04—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length on carriers
    • C07K1/047—Simultaneous synthesis of different peptide species; Peptide libraries
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/02—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
    • C07K5/0207—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -NH-(X)4-C(=0), e.g. 'isosters', replacing two amino acids
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/02—Linear peptides containing at least one abnormal peptide link
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Analytical Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Crystallography & Structural Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Treatments For Attaching Organic Compounds To Fibrous Goods (AREA)
  • Macromolecular Compounds Obtained By Forming Nitrogen-Containing Linkages In General (AREA)
  • Treatments Of Macromolecular Shaped Articles (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
PT97992A 1990-06-14 1991-06-14 Processo de preparacao de analogos de um patrimonio peptoide com resistencia a protease, e processo para a sintese de uma mistura de polimeros com eles relacionados PT97992B (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US53833990A 1990-06-14 1990-06-14
US71582391A 1991-06-14 1991-06-14

Publications (2)

Publication Number Publication Date
PT97992A true PT97992A (pt) 1992-04-30
PT97992B PT97992B (pt) 1998-11-30

Family

ID=27065784

Family Applications (1)

Application Number Title Priority Date Filing Date
PT97992A PT97992B (pt) 1990-06-14 1991-06-14 Processo de preparacao de analogos de um patrimonio peptoide com resistencia a protease, e processo para a sintese de uma mistura de polimeros com eles relacionados

Country Status (11)

Country Link
EP (1) EP0535155B1 (pt)
JP (1) JPH06504758A (pt)
AT (1) ATE212641T1 (pt)
AU (2) AU8286891A (pt)
CA (1) CA2085118A1 (pt)
DE (1) DE69132914T2 (pt)
DK (1) DK0535155T3 (pt)
ES (1) ES2167311T3 (pt)
IE (1) IE66205B1 (pt)
PT (1) PT97992B (pt)
WO (1) WO1991019735A1 (pt)

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EP0535155B1 (en) 2002-01-30
EP0535155A4 (en) 1994-08-17
DK0535155T3 (da) 2002-02-25
AU3296495A (en) 1996-03-07
AU683184B2 (en) 1997-10-30
ATE212641T1 (de) 2002-02-15
PT97992B (pt) 1998-11-30
IE66205B1 (en) 1995-12-13
CA2085118A1 (en) 1991-12-15
DE69132914T2 (de) 2002-09-19
IE912021A1 (en) 1991-12-18
JPH06504758A (ja) 1994-06-02
DE69132914D1 (de) 2002-03-14
WO1991019735A1 (en) 1991-12-26
AU8286891A (en) 1992-01-07
EP0535155A1 (en) 1993-04-07
ES2167311T3 (es) 2002-05-16

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